DD296916A5 - Neue aromatase inhibierende 4(5)-substituierte imidazol-derivate - Google Patents

Neue aromatase inhibierende 4(5)-substituierte imidazol-derivate Download PDF

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Publication number
DD296916A5
DD296916A5 DD90339203A DD33920390A DD296916A5 DD 296916 A5 DD296916 A5 DD 296916A5 DD 90339203 A DD90339203 A DD 90339203A DD 33920390 A DD33920390 A DD 33920390A DD 296916 A5 DD296916 A5 DD 296916A5
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DD
German Democratic Republic
Prior art keywords
compound
formula
defined above
pharmaceutically acceptable
acid addition
Prior art date
Application number
DD90339203A
Other languages
German (de)
English (en)
Inventor
Arto J Karjalainen
Reino O Pelkonen
Marja-Liisa Soedervall
Matti A Laehde
Risto A S Lammintausta
Arja L Karjalainen
Arja M Kalapudas
Original Assignee
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Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
Application filed by ����`��@���k�� filed Critical ����`��@���k��
Publication of DD296916A5 publication Critical patent/DD296916A5/de

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/64—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
DD90339203A 1989-03-30 1990-03-29 Neue aromatase inhibierende 4(5)-substituierte imidazol-derivate DD296916A5 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB8907218A GB2229719B (en) 1989-03-30 1989-03-30 Novel aromatase inhibiting 4(5)-imidazoles

Publications (1)

Publication Number Publication Date
DD296916A5 true DD296916A5 (de) 1991-12-19

Family

ID=10654204

Family Applications (1)

Application Number Title Priority Date Filing Date
DD90339203A DD296916A5 (de) 1989-03-30 1990-03-29 Neue aromatase inhibierende 4(5)-substituierte imidazol-derivate

Country Status (9)

Country Link
CA (1) CA2013395A1 (pl)
DD (1) DD296916A5 (pl)
FI (1) FI901316A7 (pl)
GB (1) GB2229719B (pl)
LT (1) LT3657B (pl)
PL (1) PL162554B1 (pl)
RU (2) RU2021263C1 (pl)
UA (1) UA19310A1 (pl)
ZA (1) ZA902479B (pl)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2248058B (en) * 1990-09-21 1994-09-14 Orion Yhtymae Oy Aromatase inhibiting 4(5)-imidazoles
EP0943333A1 (de) * 1998-03-18 1999-09-22 S.W. Patentverwertungs GmbH Medikament zur Prophylaxe und/oder Behandlung des Mammakarzinoms enthaltend einen Hemmer der Bildung von Oestrogenen
DE102006019906A1 (de) * 2006-04-28 2007-10-31 Müller-Enoch, Dieter, Prof. Dr. Verwendung von Verbindungen der Formel A-R-X oder deren pharmazeutisch akzeptable Salze zur Herstellung einer pharmazeutischen Zubereitung
US20080146523A1 (en) * 2006-12-18 2008-06-19 Guido Galley Imidazole derivatives

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3759944A (en) 1970-10-14 1973-09-18 Smith Kline French Lab Isothioureas and their derivatives
GB2101114B (en) * 1981-07-10 1985-05-22 Farmos Group Ltd Substituted imidazole derivatives and their preparation and use
CA1238640A (en) * 1984-06-18 1988-06-28 Kenneth S. Hirsch 4(5)-substituted imidazoles
LU85747A1 (fr) * 1985-01-28 1986-08-04 Continental Pharma Derives d'imidazole leur preparation et utilisation ainsi que les compositions pharmaceutiques contenant des derives
GB2210875B (en) 1987-10-09 1991-05-29 Farmos Oy Aromatase inhibiting 4(5)-imidazoles
AU627559B2 (en) 1989-03-30 1992-08-27 Farmos-Yhtyma Oy Novel aromatase inhibiting 4(5)-imidazoles

Also Published As

Publication number Publication date
LTIP847A (en) 1995-02-27
GB2229719B (en) 1992-04-29
UA19310A1 (uk) 1997-12-25
ZA902479B (en) 1990-12-28
RU1836355C (ru) 1993-08-23
GB8907218D0 (en) 1989-05-10
FI901316A0 (fi) 1990-03-16
RU2021263C1 (ru) 1994-10-15
FI901316A7 (fi) 1990-10-01
GB2229719A (en) 1990-10-03
LT3657B (en) 1996-01-25
PL162554B1 (pl) 1993-12-31
CA2013395A1 (en) 1991-09-29
PL288962A1 (en) 1991-10-21

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