DK0595796T3 - Fremgangsmåde til behandling af androgen-relaterede sygdomme - Google Patents

Fremgangsmåde til behandling af androgen-relaterede sygdomme

Info

Publication number: DK0595796T3
Authority: DK; Denmark
Prior art keywords: combination; related diseases; antiandrogens; treatment; biosynthesis inhibitors
Prior art date: 1989-07-07

Application number

DK90909601T

Other languages

English (en)

Inventor

Fernand Labrie

Original Assignee

Endorech Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1989-07-07

Filing date

1990-07-05

Publication date

2003-05-05

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=23486146&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DK0595796(T3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

1990-07-05 Application filed by Endorech Inc filed Critical Endorech Inc

2003-05-05 Application granted granted Critical

2003-05-05 Publication of DK0595796T3 publication Critical patent/DK0595796T3/da

Links

239000003098 androgen Substances 0.000 title abstract 2
201000010099 disease Diseases 0.000 title abstract 2
208000037265 diseases, disorders, signs and symptoms Diseases 0.000 title abstract 2
238000000034 method Methods 0.000 title abstract 2
MUMGGOZAMZWBJJ-DYKIIFRCSA-N Testostosterone Chemical compound O=C1CC[C@]2(C)[C@H]3CC[C@](C)([C@H](CC4)O)[C@@H]4[C@@H]3CCC2=C1 MUMGGOZAMZWBJJ-DYKIIFRCSA-N 0.000 abstract 2
230000002280 anti-androgenic effect Effects 0.000 abstract 2
239000000051 antiandrogen Substances 0.000 abstract 2
229940030495 antiandrogen sex hormone and modulator of the genital system Drugs 0.000 abstract 2
230000015572 biosynthetic process Effects 0.000 abstract 2
238000002648 combination therapy Methods 0.000 abstract 2
239000003163 gonadal steroid hormone Substances 0.000 abstract 2
239000003112 inhibitor Substances 0.000 abstract 2
NVKAWKQGWWIWPM-ABEVXSGRSA-N 17-β-hydroxy-5-α-Androstan-3-one Chemical compound C1C(=O)CC[C@]2(C)[C@H]3CC[C@](C)([C@H](CC4)O)[C@@H]4[C@@H]3CC[C@H]21 NVKAWKQGWWIWPM-ABEVXSGRSA-N 0.000 abstract 1
241001465754 Metazoa Species 0.000 abstract 1
206010060862 Prostate cancer Diseases 0.000 abstract 1
208000000236 Prostatic Neoplasms Diseases 0.000 abstract 1
AEMFNILZOJDQLW-QAGGRKNESA-N androst-4-ene-3,17-dione Chemical compound O=C1CC[C@]2(C)[C@H]3CC[C@](C)(C(CC4)=O)[C@@H]4[C@@H]3CCC2=C1 AEMFNILZOJDQLW-QAGGRKNESA-N 0.000 abstract 1
229960003473 androstanolone Drugs 0.000 abstract 1
AEMFNILZOJDQLW-UHFFFAOYSA-N androstenedione Natural products O=C1CCC2(C)C3CCC(C)(C(CC4)=O)C4C3CCC2=C1 AEMFNILZOJDQLW-UHFFFAOYSA-N 0.000 abstract 1
229940046836 anti-estrogen Drugs 0.000 abstract 1
230000001833 anti-estrogenic effect Effects 0.000 abstract 1
238000006243 chemical reaction Methods 0.000 abstract 1
238000011284 combination treatment Methods 0.000 abstract 1
FMGSKLZLMKYGDP-USOAJAOKSA-N dehydroepiandrosterone Chemical compound C1[C@@H](O)CC[C@]2(C)[C@H]3CC[C@](C)(C(CC4)=O)[C@@H]4[C@@H]3CC=C21 FMGSKLZLMKYGDP-USOAJAOKSA-N 0.000 abstract 1
239000000328 estrogen antagonist Substances 0.000 abstract 1
230000003054 hormonal effect Effects 0.000 abstract 1
230000002401 inhibitory effect Effects 0.000 abstract 1
230000002093 peripheral effect Effects 0.000 abstract 1
239000008194 pharmaceutical composition Substances 0.000 abstract 1
230000028327 secretion Effects 0.000 abstract 1
230000002381 testicular Effects 0.000 abstract 1
229960003604 testosterone Drugs 0.000 abstract 1
210000001519 tissue Anatomy 0.000 abstract 1
238000011282 treatment Methods 0.000 abstract 1

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/575—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of three or more carbon atoms, e.g. cholane, cholestane, ergosterol, sitosterol
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/57—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Epidemiology (AREA)
Organic Chemistry (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Steroid Compounds (AREA)
Medicines Containing Plant Substances (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

DK90909601T 1989-07-07 1990-07-05 Fremgangsmåde til behandling af androgen-relaterede sygdomme DK0595796T3 (da)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US37671089A	1989-07-07	1989-07-07
PCT/CA1990/000212 WO1991000733A1 (en)	1989-07-07	1990-07-05	Method of treatment of androgen-related diseases

Publications (1)

Publication Number	Publication Date
DK0595796T3 true DK0595796T3 (da)	2003-05-05

Family

ID=23486146

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK90909601T DK0595796T3 (da)	1989-07-07	1990-07-05	Fremgangsmåde til behandling af androgen-relaterede sygdomme

Country Status (17)

Country	Link
US (2)	US5593981A (da)
EP (1)	EP0595796B1 (da)
JP (1)	JP3350048B2 (da)
KR (1)	KR920703065A (da)
AT (1)	ATE230994T1 (da)
AU (1)	AU5851690A (da)
CA (1)	CA2062792C (da)
DE (1)	DE69034035T2 (da)
DK (1)	DK0595796T3 (da)
ES (1)	ES2189784T3 (da)
HU (1)	HUT60139A (da)
IE (1)	IE902458A1 (da)
IL (1)	IL94991A (da)
MY (1)	MY106725A (da)
NZ (2)	NZ234417A (da)
WO (1)	WO1991000733A1 (da)
ZA (1)	ZA905313B (da)

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1990
- 1990-07-05 DK DK90909601T patent/DK0595796T3/da active
- 1990-07-05 CA CA002062792A patent/CA2062792C/en not_active Expired - Lifetime
- 1990-07-05 AU AU58516/90A patent/AU5851690A/en not_active Abandoned
- 1990-07-05 JP JP50926390A patent/JP3350048B2/ja not_active Expired - Fee Related
- 1990-07-05 KR KR1019920700028A patent/KR920703065A/ko not_active Ceased
- 1990-07-05 ES ES90909601T patent/ES2189784T3/es not_active Expired - Lifetime
- 1990-07-05 HU HU9248A patent/HUT60139A/hu unknown
- 1990-07-05 DE DE69034035T patent/DE69034035T2/de not_active Expired - Fee Related
- 1990-07-05 WO PCT/CA1990/000212 patent/WO1991000733A1/en not_active Ceased
- 1990-07-05 AT AT90909601T patent/ATE230994T1/de not_active IP Right Cessation
- 1990-07-05 EP EP90909601A patent/EP0595796B1/en not_active Expired - Lifetime
- 1990-07-06 IE IE245890A patent/IE902458A1/en not_active IP Right Cessation
- 1990-07-06 ZA ZA905313A patent/ZA905313B/xx unknown
- 1990-07-06 IL IL9499190A patent/IL94991A/en active IP Right Grant
- 1990-07-07 MY MYPI90001140A patent/MY106725A/en unknown
- 1990-07-09 NZ NZ234417A patent/NZ234417A/en unknown
- 1990-07-09 NZ NZ272841A patent/NZ272841A/xx unknown
1993
- 1993-09-10 US US08/098,607 patent/US5593981A/en not_active Expired - Fee Related
1995
- 1995-06-07 US US08/472,512 patent/US5610150A/en not_active Expired - Fee Related

Also Published As

Publication number	Publication date
NZ272841A (en)	1999-06-29
NZ234417A (en)	1995-10-26
HU9200048D0 (en)	1992-06-29
MY106725A (en)	1995-07-31
AU6342594A (en)	1994-07-21
WO1991000733A1 (en)	1991-01-24
HUT60139A (en)	1992-08-28
DE69034035D1 (de)	2003-02-20
US5610150A (en)	1997-03-11
IE902458A1 (en)	1991-02-13
IL94991A (en)	1999-11-30
AU5851690A (en)	1991-02-06
US5593981A (en)	1997-01-14
ATE230994T1 (de)	2003-02-15
KR920703065A (ko)	1992-12-17
CA2062792C (en)	2006-03-21
ES2189784T3 (es)	2003-07-16
JP3350048B2 (ja)	2002-11-25
EP0595796A1 (en)	1994-05-11
IL94991A0 (en)	1991-06-10
ZA905313B (en)	1992-02-26
AU665311B2 (en)	1995-12-21
DE69034035T2 (de)	2004-01-22
CA2062792A1 (en)	1991-01-08
EP0595796B1 (en)	2003-01-15
JPH04506799A (ja)	1992-11-26

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