ES2189784T3 - Procedimiento para el tratamiento de enfermedades relacionadas con adrogenos. - Google Patents

Procedimiento para el tratamiento de enfermedades relacionadas con adrogenos.

Info

Publication number
ES2189784T3
ES2189784T3 ES90909601T ES90909601T ES2189784T3 ES 2189784 T3 ES2189784 T3 ES 2189784T3 ES 90909601 T ES90909601 T ES 90909601T ES 90909601 T ES90909601 T ES 90909601T ES 2189784 T3 ES2189784 T3 ES 2189784T3
Authority
ES
Spain
Prior art keywords
treatment
combination
antiandrogens
biosynthesis inhibitors
novel
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES90909601T
Other languages
English (en)
Inventor
Fernand Labrie
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Endorecherche Inc
Original Assignee
Endorecherche Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=23486146&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ES2189784(T3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Endorecherche Inc filed Critical Endorecherche Inc
Application granted granted Critical
Publication of ES2189784T3 publication Critical patent/ES2189784T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/575—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of three or more carbon atoms, e.g. cholane, cholestane, ergosterol, sitosterol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/57—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Medicines Containing Plant Substances (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

SE PRESENTA UN METODO DE TRATAMIENTO DE ENFERMEDADES RELACIONADAS CON LOS ANDROGENOS TALES COMO EL CANCER DE PROSTATA EN ANIMALES MACHOS SUSCEPTIBLES, INCLUYENDO LOS HUMANOS, EL METODO COMPRENDE LA ADMINISTRACION DE NUEVOS ANTIANDROGENOS Y/O NUEVOS INHIBIDORES DE LA BIOSINTESIS DE LOS ESTEROIDES DEL SEXO COMO PARTE DE UNA TERAPIA DE COMBINACION. LOS INHIBIDORES DE LA BIOSINTESIS DE LOS ESTEROIDES DEL SEXO, ESPECIALMENTE AQUELLOS CAPACES DE INHIBIR LA CONVERSION DE LA DEHIDROEPIANDROESTERONA (DHEA) O DE LA 4-ANDROESTENODIONA (ALFA4DIONA) EN ESTEROIDES NATURALES DEL SEXO (Y TESTOSTERONA EN DIHIDROTESTOSTERONA) EN LOS TEJIDOS PERIFERICOS, SE UTILIZAN EN COMBINACION CON ANTIANDROGENOS USUALMENTE DESPUES DEL BLOQUEO DE LAS SECRECIONES HORMONALES TESTICULARES. LOS ANTIESTROGENOS PUEDEN TAMBIEN FORMAR PARTE DE LA TERAPIA DE COMBINACION. COMPOSICIONES FARMACEUTICAS Y 2,3,4 Y 5 EQUIPOS DE COMPONENTES SON UTILES PARA DICHO TRATAMIENTO DE COMBINACION.
ES90909601T 1989-07-07 1990-07-05 Procedimiento para el tratamiento de enfermedades relacionadas con adrogenos. Expired - Lifetime ES2189784T3 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US37671089A 1989-07-07 1989-07-07

Publications (1)

Publication Number Publication Date
ES2189784T3 true ES2189784T3 (es) 2003-07-16

Family

ID=23486146

Family Applications (1)

Application Number Title Priority Date Filing Date
ES90909601T Expired - Lifetime ES2189784T3 (es) 1989-07-07 1990-07-05 Procedimiento para el tratamiento de enfermedades relacionadas con adrogenos.

Country Status (17)

Country Link
US (2) US5593981A (es)
EP (1) EP0595796B1 (es)
JP (1) JP3350048B2 (es)
KR (1) KR920703065A (es)
AT (1) ATE230994T1 (es)
AU (1) AU5851690A (es)
CA (1) CA2062792C (es)
DE (1) DE69034035T2 (es)
DK (1) DK0595796T3 (es)
ES (1) ES2189784T3 (es)
HU (1) HUT60139A (es)
IE (1) IE902458A1 (es)
IL (1) IL94991A (es)
MY (1) MY106725A (es)
NZ (2) NZ272841A (es)
WO (1) WO1991000733A1 (es)
ZA (1) ZA905313B (es)

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Also Published As

Publication number Publication date
JP3350048B2 (ja) 2002-11-25
AU665311B2 (en) 1995-12-21
CA2062792C (en) 2006-03-21
EP0595796A1 (en) 1994-05-11
US5593981A (en) 1997-01-14
DE69034035T2 (de) 2004-01-22
AU5851690A (en) 1991-02-06
IL94991A0 (en) 1991-06-10
JPH04506799A (ja) 1992-11-26
ZA905313B (en) 1992-02-26
WO1991000733A1 (en) 1991-01-24
KR920703065A (ko) 1992-12-17
ATE230994T1 (de) 2003-02-15
CA2062792A1 (en) 1991-01-08
US5610150A (en) 1997-03-11
EP0595796B1 (en) 2003-01-15
DE69034035D1 (de) 2003-02-20
NZ234417A (en) 1995-10-26
AU6342594A (en) 1994-07-21
HU9200048D0 (en) 1992-06-29
NZ272841A (en) 1999-06-29
HUT60139A (en) 1992-08-28
IE902458A1 (en) 1991-02-13
MY106725A (en) 1995-07-31
DK0595796T3 (da) 2003-05-05
IL94991A (en) 1999-11-30

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