DK0719779T3 - Substituerede thiazolo[3,2-alpha]azepinderivater - Google Patents

Substituerede thiazolo[3,2-alpha]azepinderivater

Info

Publication number: DK0719779T3
Authority: DK; Denmark
Prior art keywords: group; hydrogen atom; lower alkyl; alpha; substituted
Prior art date: 1994-07-18

Application number

DK95921127T

Other languages

Danish (da)

English (en)

Inventor

Hideyuki Adachi

Hitoshi Oinuma

Kazutoshi Miyake

Mamoru Saito

Takeshi Sudo

Shinji Suda

Naoki Yoneda

Makoto Kotake

Masanori Mizuno

Tomohiro Matsushima

Yoshio Fukuda

Toshiyuki Matsuoka

Masayuki Namiki

Makoto Okita

Original Assignee

Eisai Co Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1994-07-18

Filing date

1995-06-07

Publication date

2004-03-22

1994-07-18 Priority claimed from JP6165481A external-priority patent/JPH0827156A/ja

1994-08-24 Priority claimed from JP19918094A external-priority patent/JP3444666B2/ja

1994-12-09 Priority claimed from JP6306468A external-priority patent/JPH08165293A/ja

1995-06-07 Application filed by Eisai Co Ltd filed Critical Eisai Co Ltd

2004-03-22 Application granted granted Critical

2004-03-22 Publication of DK0719779T3 publication Critical patent/DK0719779T3/da

Links

150000001538 azepines Chemical class 0.000 title 1
125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 6
125000000217 alkyl group Chemical group 0.000 abstract 3
125000003545 alkoxy group Chemical group 0.000 abstract 2
125000004414 alkyl thio group Chemical group 0.000 abstract 2
125000006239 protecting group Chemical group 0.000 abstract 2
125000001424 substituent group Chemical group 0.000 abstract 2
102000004270 Peptidyl-Dipeptidase A Human genes 0.000 abstract 1
108090000882 Peptidyl-Dipeptidase A Proteins 0.000 abstract 1
125000003118 aryl group Chemical group 0.000 abstract 1
125000003178 carboxy group Chemical group [H]OC(*)=O 0.000 abstract 1
230000002401 inhibitory effect Effects 0.000 abstract 1
230000007935 neutral effect Effects 0.000 abstract 1
125000003396 thiol group Chemical group [H]S* 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06139—Dipeptides with the first amino acid being heterocyclic
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Proteomics, Peptides & Aminoacids (AREA)
Molecular Biology (AREA)
Genetics & Genomics (AREA)
Biophysics (AREA)
Biochemistry (AREA)
Immunology (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Animal Behavior & Ethology (AREA)
Epidemiology (AREA)
Pharmacology & Pharmacy (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Thiazole And Isothizaole Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)

DK95921127T 1994-07-18 1995-06-07 Substituerede thiazolo[3,2-alpha]azepinderivater DK0719779T3 (da)

Applications Claiming Priority (4)

Application Number	Priority Date	Filing Date	Title
JP6165481A JPH0827156A (ja)	1994-07-18	1994-07-18	アミノ酸誘導体の製造方法
JP19918094A JP3444666B2 (ja)	1994-08-24	1994-08-24	（２ｓ，３ｓ）−３− メチル−２− チオペンタン酸誘導体の製造方法
JP6306468A JPH08165293A (ja)	1994-12-09	1994-12-09	置換チアゾロ［３，２−ａ］アゼピン誘導体
PCT/JP1995/001139 WO1996002549A1 (fr)	1994-07-18	1995-06-07	DERIVE DE THIAZOLO[3,2-α]AZEPINE A SUBSTITUTION

Publications (1)

Publication Number	Publication Date
DK0719779T3 true DK0719779T3 (da)	2004-03-22

Family

ID=27322514

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK95921127T DK0719779T3 (da)	1994-07-18	1995-06-07	Substituerede thiazolo[3,2-alpha]azepinderivater

Country Status (17)

Country	Link
US (2)	US5789403A (fr)
EP (1)	EP0719779B1 (fr)
KR (1)	KR100284247B1 (fr)
CN (2)	CN1053908C (fr)
AT (1)	ATE254622T1 (fr)
AU (1)	AU694233B2 (fr)
CA (1)	CA2171334C (fr)
DE (1)	DE69532155T2 (fr)
DK (1)	DK0719779T3 (fr)
ES (1)	ES2210292T3 (fr)
FI (2)	FI110001B (fr)
HU (1)	HU225916B1 (fr)
MX (1)	MX9601017A (fr)
NO (1)	NO308077B1 (fr)
NZ (1)	NZ287557A (fr)
PT (1)	PT719779E (fr)
WO (1)	WO1996002549A1 (fr)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5650408A (en) *	1995-06-07	1997-07-22	Karanewsky; Donald S.	Thiazolo benzazepine containing dual action inhibitors
CA2251155A1 (fr) *	1997-02-05	1998-08-13	Suntory Limited	Compositions medicinales pour traiter les cardiopathies induites par l'hypertrophie cardiaque
US9823092B2 (en)	2014-10-31	2017-11-21	Allegro Microsystems, Llc	Magnetic field sensor providing a movement detector

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
ZA821904B (en) *	1981-03-23	1983-01-26	Merck & Co Inc	Bicyclic lactams as anthihypertensives
US4415496A (en) *	1981-03-23	1983-11-15	Merck & Co., Inc.	Bicyclic lactams
US4617301A (en) *	1983-06-22	1986-10-14	Merck & Co., Inc.	Sulfoxide and sulfone derivatives of bicyclic lactams as antihypertensives
JPS6056790A (ja) *	1983-09-03	1985-04-02	山陽科学株式会社	荷役用マット
RU2124503C1 (ru) *	1992-05-18	1999-01-10	И.Р.Сквибб энд Санз, Инк.	Гетероциклические азотсодержащие производные карбоновой кислоты, способ их получения и фармацевтическая композиция
DE69329701T2 (de) *	1992-10-30	2001-05-10	Merrell Pharmaceuticals Inc., Cincinnati	Mercaptoacetylamid substituiertes bizyclisches laktam zur verwendung als enkephalinase und ace-hemmer
US5650408A (en) *	1995-06-07	1997-07-22	Karanewsky; Donald S.	Thiazolo benzazepine containing dual action inhibitors

1995
- 1995-06-07 ES ES95921127T patent/ES2210292T3/es not_active Expired - Lifetime
- 1995-06-07 EP EP95921127A patent/EP0719779B1/fr not_active Expired - Lifetime
- 1995-06-07 AT AT95921127T patent/ATE254622T1/de not_active IP Right Cessation
- 1995-06-07 KR KR1019960701358A patent/KR100284247B1/ko not_active Expired - Fee Related
- 1995-06-07 CN CN95190779A patent/CN1053908C/zh not_active Expired - Fee Related
- 1995-06-07 MX MX9601017A patent/MX9601017A/es not_active IP Right Cessation
- 1995-06-07 DE DE69532155T patent/DE69532155T2/de not_active Expired - Fee Related
- 1995-06-07 WO PCT/JP1995/001139 patent/WO1996002549A1/fr not_active Ceased
- 1995-06-07 PT PT95921127T patent/PT719779E/pt unknown
- 1995-06-07 HU HU9600679A patent/HU225916B1/hu not_active IP Right Cessation
- 1995-06-07 AU AU26301/95A patent/AU694233B2/en not_active Ceased
- 1995-06-07 DK DK95921127T patent/DK0719779T3/da active
- 1995-06-07 NZ NZ287557A patent/NZ287557A/en not_active IP Right Cessation
- 1995-06-07 CA CA002171334A patent/CA2171334C/fr not_active Expired - Fee Related
- 1995-06-07 US US08/612,864 patent/US5789403A/en not_active Expired - Lifetime
1996
- 1996-03-14 NO NO19961051A patent/NO308077B1/no not_active IP Right Cessation
- 1996-03-14 FI FI961199A patent/FI110001B/fi active
1998
- 1998-05-27 US US09/085,729 patent/US6051705A/en not_active Expired - Fee Related
1999
- 1999-10-28 CN CNB991236092A patent/CN1170832C/zh not_active Expired - Fee Related
2001
- 2001-06-01 FI FI20011154A patent/FI113656B/fi not_active IP Right Cessation

Also Published As

Publication number	Publication date
CN1134152A (zh)	1996-10-23
WO1996002549A1 (fr)	1996-02-01
FI113656B (fi)	2004-05-31
EP0719779A4 (fr)	1996-12-18
PT719779E (pt)	2004-04-30
CN1053908C (zh)	2000-06-28
FI961199A0 (fi)	1996-03-14
HU225916B1 (en)	2007-12-28
CA2171334C (fr)	2008-10-21
DE69532155T2 (de)	2004-08-19
US6051705A (en)	2000-04-18
NZ287557A (en)	1997-04-24
AU2630195A (en)	1996-02-16
FI20011154L (fi)	2001-06-01
NO961051D0 (no)	1996-03-14
AU694233B2 (en)	1998-07-16
FI110001B (fi)	2002-11-15
KR100284247B1 (ko)	2001-10-24
EP0719779A1 (fr)	1996-07-03
CN1262275A (zh)	2000-08-09
EP0719779B1 (fr)	2003-11-19
KR960704898A (ko)	1996-10-09
MX9601017A (es)	1997-10-31
HUT76477A (en)	1997-09-29
ES2210292T3 (es)	2004-07-01
US5789403A (en)	1998-08-04
FI961199A7 (fi)	1996-05-13
CN1170832C (zh)	2004-10-13
DE69532155D1 (de)	2003-12-24
NO308077B1 (no)	2000-07-17
HU9600679D0 (en)	1996-05-28
CA2171334A1 (fr)	1996-02-01
NO961051L (no)	1996-05-10
ATE254622T1 (de)	2003-12-15

Publication	Publication Date	Title
NO994582D0 (no)	1999-09-21	Fremgangsmaate for fremstilling av piperidinderivater
AU1163492A (en)	1992-08-27	3-benzylidene-1-carbamoyl-2-pyrrolidone analog
ATE194610T1 (de)	2000-07-15	Derivate des radicicols
FI935830A0 (fi)	1993-12-23	Bicykliska aminderivat
NO974588D0 (no)	1997-10-03	Triazol-antifungaltmiddel
DK0806413T3 (da)	2002-01-28	2-substituerede viatmin D3-derivater
DE69532155D1 (de)	2003-12-24	Substituierte thiazolo [3,2-alpha]azepinderivate
DE69930383D1 (de)	2006-05-11	Naphthimidobenzamid-derivate
DE69416683D1 (de)	1999-04-01	Benzolactam-derivate
DE69714841D1 (de)	2002-09-26	Ein 1-methylcarbapenem-derivat
ATE253070T1 (de)	2003-11-15	Penem-derivate und sie enthaltende anti- mikrobische mittel
NO20004477L (no)	2001-03-12	Anvendelse av organiske karbonater for vasking av metalloverflater
MX9710432A (es)	1998-06-28	Composiciones de pigmentos organicos.