DK0730598T3 - Hindrede estere af rapamycin samt deres anvendelse som lægemidler - Google Patents

Hindrede estere af rapamycin samt deres anvendelse som lægemidler

Info

Publication number
DK0730598T3
DK0730598T3 DK95903559T DK95903559T DK0730598T3 DK 0730598 T3 DK0730598 T3 DK 0730598T3 DK 95903559 T DK95903559 T DK 95903559T DK 95903559 T DK95903559 T DK 95903559T DK 0730598 T3 DK0730598 T3 DK 0730598T3
Authority
DK
Denmark
Prior art keywords
rapamycin
obstructed
drugs
esters
well
Prior art date
Application number
DK95903559T
Other languages
English (en)
Inventor
Frances Christy Nelson
Guy Alan Schiehser
Original Assignee
American Home Prod
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by American Home Prod filed Critical American Home Prod
Application granted granted Critical
Publication of DK0730598T3 publication Critical patent/DK0730598T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D498/18—Bridged systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Immunology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Rheumatology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Pain & Pain Management (AREA)
  • Transplantation (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
DK95903559T 1993-11-22 1994-11-18 Hindrede estere af rapamycin samt deres anvendelse som lægemidler DK0730598T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US08/156,206 US5385908A (en) 1993-11-22 1993-11-22 Hindered esters of rapamycin
PCT/US1994/013310 WO1995014696A1 (en) 1993-11-22 1994-11-18 Hindered esters of rapamycin and their use as pharmaceuticals

Publications (1)

Publication Number Publication Date
DK0730598T3 true DK0730598T3 (da) 1999-11-15

Family

ID=22558566

Family Applications (1)

Application Number Title Priority Date Filing Date
DK95903559T DK0730598T3 (da) 1993-11-22 1994-11-18 Hindrede estere af rapamycin samt deres anvendelse som lægemidler

Country Status (13)

Country Link
US (1) US5385908A (da)
EP (1) EP0730598B1 (da)
JP (1) JP3710140B2 (da)
AT (1) ATE181076T1 (da)
AU (1) AU1257595A (da)
CA (1) CA2176955A1 (da)
DE (1) DE69419032T2 (da)
DK (1) DK0730598T3 (da)
ES (1) ES2133715T3 (da)
GR (1) GR3031018T3 (da)
SG (1) SG80525A1 (da)
TW (1) TW342391B (da)
WO (1) WO1995014696A1 (da)

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WO1995014696A1 (en) 1995-06-01
ATE181076T1 (de) 1999-06-15
EP0730598A1 (en) 1996-09-11
GR3031018T3 (en) 1999-12-31
US5385908A (en) 1995-01-31
ES2133715T3 (es) 1999-09-16
EP0730598B1 (en) 1999-06-09
CA2176955A1 (en) 1995-06-01
DE69419032D1 (de) 1999-07-15
HK1013063A1 (en) 1999-08-13
SG80525A1 (en) 2001-05-22
TW342391B (en) 1998-10-11
AU1257595A (en) 1995-06-13
JPH09505592A (ja) 1997-06-03
JP3710140B2 (ja) 2005-10-26
DE69419032T2 (de) 1999-10-07

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