DK1283838T3 - Piperazin- og piperidinforbindelser - Google Patents

Piperazin- og piperidinforbindelser

Info

Publication number: DK1283838T3
Authority: DK; Denmark
Prior art keywords: piperazine; piperidine compounds; piperidine; compounds
Prior art date: 2000-05-12

Application number

DK01938214T

Other languages

English (en)

Inventor

Stephen K Long

Roelof W Feenstra

Der Heijden Johannes A M Van

Cornelis G Kruse

Scharrenburg Gustaaf J M Van

Original Assignee

Solvay Pharm Bv

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-05-12

Filing date

2001-05-10

Publication date

2004-03-22

2001-05-10 Application filed by Solvay Pharm Bv filed Critical Solvay Pharm Bv

2004-03-22 Application granted granted Critical

2004-03-22 Publication of DK1283838T3 publication Critical patent/DK1283838T3/da

Links

GLUUGHFHXGJENI-UHFFFAOYSA-N Piperazine Chemical compound C1CNCCN1 GLUUGHFHXGJENI-UHFFFAOYSA-N 0.000 title 2
150000003053 piperidines Chemical class 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/52—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings condensed with carbocyclic rings or ring systems
- C07D263/54—Benzoxazoles; Hydrogenated benzoxazoles
- C07D263/58—Benzoxazoles; Hydrogenated benzoxazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
General Health & Medical Sciences (AREA)
Neurology (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Chemical Kinetics & Catalysis (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Biomedical Technology (AREA)
Medicinal Chemistry (AREA)
Neurosurgery (AREA)
Psychiatry (AREA)
Psychology (AREA)
Addiction (AREA)
Pain & Pain Management (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Hydrogenated Pyridines (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

DK01938214T 2000-05-12 2001-05-10 Piperazin- og piperidinforbindelser DK1283838T3 (da)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
EP00201699		2000-05-12
PCT/EP2001/005320 WO2001085725A1 (en)	2000-05-12	2001-05-10	Piperazine and piperidine compounds

Publications (1)

Publication Number	Publication Date
DK1283838T3 true DK1283838T3 (da)	2004-03-22

Family

ID=8171488

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK01938214T DK1283838T3 (da)	2000-05-12	2001-05-10	Piperazin- og piperidinforbindelser

Country Status (27)

Country	Link
US (2)	US6911448B2 (da)
EP (1)	EP1283838B1 (da)
JP (1)	JP2003532729A (da)
CN (1)	CN1174979C (da)
AR (1)	AR028443A1 (da)
AT (1)	ATE255578T1 (da)
AU (2)	AU2001263927B2 (da)
BR (1)	BR0110592A (da)
CA (1)	CA2405971C (da)
CZ (1)	CZ301464B6 (da)
DE (1)	DE60101386T2 (da)
DK (1)	DK1283838T3 (da)
DZ (1)	DZ3370A1 (da)
ES (1)	ES2211809T3 (da)
HU (1)	HUP0302016A2 (da)
IL (2)	IL152177A0 (da)
MX (1)	MXPA02011084A (da)
NO (1)	NO323778B1 (da)
NZ (1)	NZ522116A (da)
PL (1)	PL198857B1 (da)
PT (1)	PT1283838E (da)
RU (1)	RU2261250C2 (da)
SK (1)	SK286778B6 (da)
TR (1)	TR200302294T4 (da)
UA (1)	UA72337C2 (da)
WO (1)	WO2001085725A1 (da)
ZA (1)	ZA200208537B (da)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
ES2211809T3 (es) *	2000-05-12	2004-07-16	Solvay Pharmaceuticals B.V.	Compuesto de piperazina y piperidina.
ATE424825T1 (de)	2001-07-20	2009-03-15	Psychogenics Inc	Behandlung von hyperaktivitätsstörungen und aufmerksamkeitsdefiziten
AU2003244160A1 (en) *	2002-06-25	2004-01-06	Sumitomo Pharmaceuticals Co., Ltd.	Novel benzoxazolinone derivative
ES2232292B1 (es) *	2003-07-30	2006-11-01	Laboratorios Del Dr. Esteve, S.A.	Compuestos sulfonamidicos derivados de benzoxazinona, su preparacion y uso como medicamentos.
US7596407B2 (en)	2004-03-26	2009-09-29	Solvay Pharmaceuticals, B.V.	Transdermal iontophoretic delivery of piperazinyl-2(3H)-benzoxazolone compounds
EP1595542A1 (en) *	2004-03-26	2005-11-16	Solvay Pharmaceuticals B.V.	Transdermal iontophoretic delivery of piperazinyl-2(3H)-benzoxazolone compounds
KR20080046205A (ko) *	2005-08-22	2008-05-26	솔베이 파마슈티칼스 비. 브이	프로드럭으로서 피페라진 및 피페리딘 유도체의 ｎ-산화물
AR058022A1 (es) *	2005-08-22	2008-01-23	Solvay Pharm Bv	Derivados de benzooxazoles, composiciones farmaceuticas y su uso para el tratamiento de desordenes del sistema nervioso.
US7750013B2 (en)	2005-08-22	2010-07-06	Solvay Pharmaceuticals, B.V.	N-oxides as prodrugs of piperazine and piperidine derivatives
US20070275977A1 (en) *	2006-05-02	2007-11-29	Van Aar Marcel P	N-oxides of pyridylmethyl -piperazine and -piperidine derivatives
US8106056B2 (en)	2006-06-16	2012-01-31	Solvay Pharmaceuticals B.V.	Combination preparations comprising bifeprunox and a dopamine agonist
BRPI0720246A2 (pt)	2006-12-07	2013-12-31	Hoffmann La Roche	Derivados de espiro-piperidina
EP2102207B1 (en)	2006-12-07	2010-06-02	F.Hoffmann-La Roche Ag	Spiro-piperidine derivatives as via receptor antagonists
CA2670139A1 (en)	2006-12-08	2008-06-12	F. Hoffmann-La Roche Ag	Indoles
US8071622B2 (en)	2006-12-08	2011-12-06	Hoffman-La Roche Inc.	Indoles
EP2097376A2 (en)	2006-12-22	2009-09-09	F. Hoffmann-Roche AG	Spiro-piperidine derivatives
US20110105523A1 (en) *	2008-01-15	2011-05-05	Van Stuivenberg Herman H	Bifeprunox derivatives
US11103499B2 (en)	2016-08-26	2021-08-31	EXCIVA (UG) (haftungsbeschränkt)	Compositions and methods thereof
SG11202100680WA (en) *	2018-07-27	2021-02-25	Chugoku Marine Paints	Antifouling paint composition, antifouling coating, substrate with antifouling coating, production method thereof, and repair method

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
JPS60126275A (ja) *	1983-12-13	1985-07-05	Otsuka Pharmaceut Co Ltd	ベンゾチアゾ−ル誘導体
FR2567884B1 (fr) *	1984-07-19	1987-03-06	Roussel Uclaf	Nouveaux derives de l'indole, leur preparation, leur application comme medicaments et les compositions les renfermant
EP0185429A1 (en)	1984-12-21	1986-06-25	Duphar International Research B.V	New bicyclic heteroaryl piperazines
DE3586794T2 (de) *	1984-12-21	1993-05-27	Duphar Int Res	Arzneimittel mit psychotroper wirkung.
DE4127849A1 (de) *	1991-08-22	1993-02-25	Merck Patent Gmbh	Benzodioxanderivate
DE69736704T2 (de) *	1996-03-29	2007-09-13	Duphar International Research B.V.	Piperazin- und piperidin- derivate
TW530054B (en) *	1997-09-24	2003-05-01	Duphar Int Res	New piperazine and piperidine compounds
GB9811879D0 (en) *	1998-06-03	1998-07-29	Knoll Ag	Therapeutic agents
UA71590C2 (en) *	1998-11-13	2004-12-15	Duphar Int Res	Piperazine and piperidine derivatives
ES2211809T3 (es) *	2000-05-12	2004-07-16	Solvay Pharmaceuticals B.V.	Compuesto de piperazina y piperidina.
EP1284731A1 (en) *	2000-05-12	2003-02-26	Solvay Pharmaceuticals B.V.	Use of compounds having combined dopamine d2, 5-ht1a and alpha adrenoreceptor agonistic action for treating cns disorders

2001
- 2001-05-10 ES ES01938214T patent/ES2211809T3/es not_active Expired - Lifetime
- 2001-05-10 AU AU2001263927A patent/AU2001263927B2/en not_active Ceased
- 2001-05-10 BR BR0110592-2A patent/BR0110592A/pt not_active IP Right Cessation
- 2001-05-10 IL IL15217701A patent/IL152177A0/xx unknown
- 2001-05-10 PT PT01938214T patent/PT1283838E/pt unknown
- 2001-05-10 PL PL358201A patent/PL198857B1/pl not_active IP Right Cessation
- 2001-05-10 TR TR2003/02294T patent/TR200302294T4/xx unknown
- 2001-05-10 AU AU6392701A patent/AU6392701A/xx active Pending
- 2001-05-10 CN CNB018093302A patent/CN1174979C/zh not_active Expired - Fee Related
- 2001-05-10 SK SK1587-2002A patent/SK286778B6/sk not_active IP Right Cessation
- 2001-05-10 DE DE60101386T patent/DE60101386T2/de not_active Expired - Lifetime
- 2001-05-10 MX MXPA02011084A patent/MXPA02011084A/es active IP Right Grant
- 2001-05-10 HU HU0302016A patent/HUP0302016A2/hu unknown
- 2001-05-10 NZ NZ522116A patent/NZ522116A/en not_active IP Right Cessation
- 2001-05-10 CZ CZ20023721A patent/CZ301464B6/cs not_active IP Right Cessation
- 2001-05-10 WO PCT/EP2001/005320 patent/WO2001085725A1/en not_active Ceased
- 2001-05-10 DK DK01938214T patent/DK1283838T3/da active
- 2001-05-10 EP EP01938214A patent/EP1283838B1/en not_active Expired - Lifetime
- 2001-05-10 US US10/257,677 patent/US6911448B2/en not_active Expired - Fee Related
- 2001-05-10 DZ DZ013370A patent/DZ3370A1/xx active
- 2001-05-10 AT AT01938214T patent/ATE255578T1/de active
- 2001-05-10 CA CA2405971A patent/CA2405971C/en not_active Expired - Fee Related
- 2001-05-10 JP JP2001582326A patent/JP2003532729A/ja not_active Ceased
- 2001-05-10 RU RU2002133458/04A patent/RU2261250C2/ru not_active IP Right Cessation
- 2001-05-11 AR ARP010102239A patent/AR028443A1/es active IP Right Grant
- 2001-10-05 UA UA2002129990A patent/UA72337C2/uk unknown
2002
- 2002-10-08 IL IL152177A patent/IL152177A/en not_active IP Right Cessation
- 2002-10-22 ZA ZA200208537A patent/ZA200208537B/en unknown
- 2002-11-08 NO NO20025365A patent/NO323778B1/no not_active IP Right Cessation
2005
- 2005-05-16 US US11/129,465 patent/US7297699B2/en not_active Expired - Lifetime

Also Published As

Publication number	Publication date
DZ3370A1 (fr)	2001-11-15
CZ301464B6 (cs)	2010-03-10
NO323778B1 (no)	2007-07-02
JP2003532729A (ja)	2003-11-05
NZ522116A (en)	2004-04-30
CN1174979C (zh)	2004-11-10
ATE255578T1 (de)	2003-12-15
AU2001263927B2 (en)	2004-09-30
CN1429226A (zh)	2003-07-09
DE60101386T2 (de)	2004-05-27
US7297699B2 (en)	2007-11-20
US6911448B2 (en)	2005-06-28
US20030119849A1 (en)	2003-06-26
CZ20023721A3 (cs)	2003-02-12
WO2001085725A1 (en)	2001-11-15
NO20025365L (no)	2002-11-08
BR0110592A (pt)	2003-04-01
AU6392701A (en)	2001-11-20
US20060089366A1 (en)	2006-04-27
CA2405971A1 (en)	2001-11-15
IL152177A (en)	2009-08-03
MXPA02011084A (es)	2003-03-10
RU2261250C2 (ru)	2005-09-27
PT1283838E (pt)	2004-04-30
PL358201A1 (en)	2004-08-09
ES2211809T3 (es)	2004-07-16
SK286778B6 (sk)	2009-05-07
EP1283838A1 (en)	2003-02-19
CA2405971C (en)	2010-03-30
TR200302294T4 (tr)	2004-02-23
IL152177A0 (en)	2003-05-29
UA72337C2 (uk)	2005-02-15
SK15872002A3 (sk)	2003-04-01
EP1283838B1 (en)	2003-12-03
PL198857B1 (pl)	2008-07-31
HK1055952A1 (en)	2004-01-30
NO20025365D0 (no)	2002-11-08
ZA200208537B (en)	2004-01-22
DE60101386D1 (de)	2004-01-15
HUP0302016A2 (hu)	2003-09-29
AR028443A1 (es)	2003-05-07

Publication	Publication Date	Title
NO20023787D0 (no)	2002-08-09	Piperazin- og piperidinderivater
DK1325008T3 (da)	2006-02-13	Piperazinderivater
ATE397595T1 (de)	2008-06-15	Piperazin-derivate
DZ3306A1 (fr)	2001-10-04	Derives de piperazine
AR028343A1 (es)	2003-05-07	Derivados de pirrolidina y piperidina
DE60103472D1 (de)	2004-07-01	Rohrschneider
DE50105915D1 (de)	2005-05-19	Schutzhülle
NO20032585L (no)	2003-07-21	ABCA-1 forhoyende forbindelser
NO20026125L (no)	2003-02-04	Tetrahydropyridin- eller piperidin-heterocykliske derivater
DE60101386D1 (de)	2004-01-15	Piperazin- und piperidinverbindungen
NO20043079L (no)	2004-09-21	Piperazinderivat
DK1131308T3 (da)	2004-06-28	Piperazin- og piperidinderivater
NO20031572L (no)	2003-06-10	Brodannete piperazinderivater
NO20023954D0 (no)	2002-08-20	Substituerte piperasinforbindelser
DE50113112D1 (de)	2007-11-22	Schaltungsanordnung
DE60109953D1 (de)	2005-05-12	Kapazitiver wandler
ATE268757T1 (de)	2004-06-15	Piperidinalkohole
DE60139781D1 (de)	2009-10-15	4-substituierte piperidinverbindung
PT1131308E (pt)	2004-10-29	Novos compostos de piperazina e piperidina
DE50115426D1 (de)	2010-05-20	Schaltungsanordnung
FR2814381B1 (fr)	2004-06-04	Dechiqueteur
FI20001114L (fi)	2001-11-11	Kulmasuoja
DK1037892T3 (da)	2005-02-07	Piperidinderivater
ITMI20000805A0 (it)	2000-04-12	Lettino termale-estetico
SE0003782D0 (sv)	2000-10-14	Inbrottsskydd