DK2508521T4 - Dimaleat af en aminocrotonylforbindelse og fremgangsmåde til fremstilling deraf - Google Patents

Dimaleat af en aminocrotonylforbindelse og fremgangsmåde til fremstilling deraf Download PDF

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Publication number
DK2508521T4
DK2508521T4 DK12155662.5T DK12155662T DK2508521T4 DK 2508521 T4 DK2508521 T4 DK 2508521T4 DK 12155662 T DK12155662 T DK 12155662T DK 2508521 T4 DK2508521 T4 DK 2508521T4
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Prior art keywords
aminocrotonyl
dimaleate
compound
preparation
aminocrotonyl compound
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DK12155662.5T
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English (en)
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DK2508521T3 (da
Inventor
Werner Rall
Christian Kulinna
Juergen Schnaubelt
Peter Sieger
Rainer Soyka
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Boehringer Ingelheim Int
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Pulmonology (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pyrrole Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
DK12155662.5T 2003-10-17 2004-10-12 Dimaleat af en aminocrotonylforbindelse og fremgangsmåde til fremstilling deraf DK2508521T4 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10349113A DE10349113A1 (de) 2003-10-17 2003-10-17 Verfahren zur Herstellung von Aminocrotonylverbindungen
EP04765927.1A EP1678165B1 (de) 2003-10-17 2004-10-12 Verfahren zur herstellung von aminocrotonylverbindungen

Publications (2)

Publication Number Publication Date
DK2508521T3 DK2508521T3 (da) 2016-03-29
DK2508521T4 true DK2508521T4 (da) 2022-10-03

Family

ID=34428508

Family Applications (2)

Application Number Title Priority Date Filing Date
DK12155662.5T DK2508521T4 (da) 2003-10-17 2004-10-12 Dimaleat af en aminocrotonylforbindelse og fremgangsmåde til fremstilling deraf
DK04765927.1T DK1678165T3 (da) 2003-10-17 2004-10-12 Fremgangsmåde til fremstilling af aminocrotonylforbindelser

Family Applications After (1)

Application Number Title Priority Date Filing Date
DK04765927.1T DK1678165T3 (da) 2003-10-17 2004-10-12 Fremgangsmåde til fremstilling af aminocrotonylforbindelser

Country Status (34)

Country Link
US (2) US20050085495A1 (da)
EP (2) EP2508521B2 (da)
JP (2) JP4594317B2 (da)
KR (2) KR101282812B1 (da)
CN (2) CN1867564B (da)
AR (1) AR046118A1 (da)
AU (2) AU2004281938B2 (da)
BR (2) BR122013033343B8 (da)
CA (2) CA2541928C (da)
CY (2) CY1114866T1 (da)
DE (1) DE10349113A1 (da)
DK (2) DK2508521T4 (da)
EA (1) EA016624B1 (da)
EC (1) ECSP066509A (da)
ES (2) ES2440466T3 (da)
HR (2) HRP20160246T4 (da)
HU (1) HUE028254T2 (da)
IL (2) IL174951A (da)
ME (1) ME00341B (da)
MX (2) MX338920B (da)
MY (2) MY149921A (da)
NO (2) NO333971B1 (da)
NZ (2) NZ583049A (da)
PE (2) PE20050965A1 (da)
PL (2) PL1678165T3 (da)
PT (2) PT1678165E (da)
RS (3) RS60563B1 (da)
SG (1) SG139743A1 (da)
SI (2) SI2508521T2 (da)
TW (2) TWI348468B (da)
UA (2) UA91006C2 (da)
UY (2) UY28559A1 (da)
WO (1) WO2005037824A2 (da)
ZA (1) ZA200602234B (da)

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