DK3038656T3 - Forbindelse af glycosaminoglycan, fremgangsmåde til fremstilling og anvendelse deraf - Google Patents

Forbindelse af glycosaminoglycan, fremgangsmåde til fremstilling og anvendelse deraf Download PDF

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Publication number
DK3038656T3
DK3038656T3 DK14746964.7T DK14746964T DK3038656T3 DK 3038656 T3 DK3038656 T3 DK 3038656T3 DK 14746964 T DK14746964 T DK 14746964T DK 3038656 T3 DK3038656 T3 DK 3038656T3
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glycosaminoglycan
compound
preparation
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DK14746964.7T
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English (en)
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Hua-Yang Lin
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Holy Stone Biotech Co Ltd
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/145—Amines having sulfur, e.g. thiurams (>N—C(S)—S—C(S)—N< and >N—C(S)—S—S—C(S)—N<), Sulfinylamines (—N=SO), Sulfonylamines (—N=SO2)
    • A—HUMAN NECESSITIES
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    • A61K31/16—Amides, e.g. hydroxamic acids
    • A61K31/18—Sulfonamides
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
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    • A61K31/33—Heterocyclic compounds
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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
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    • A61K31/33—Heterocyclic compounds
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    • A61K31/573—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone substituted in position 21, e.g. cortisone, dexamethasone, prednisone or aldosterone
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  • Hematology (AREA)
  • Rheumatology (AREA)
  • Diabetes (AREA)
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  • Endocrinology (AREA)
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  • Gastroenterology & Hepatology (AREA)
  • Pain & Pain Management (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Transplantation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Polysaccharides And Polysaccharide Derivatives (AREA)
DK14746964.7T 2013-08-29 2014-06-27 Forbindelse af glycosaminoglycan, fremgangsmåde til fremstilling og anvendelse deraf DK3038656T3 (da)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201361871352P 2013-08-29 2013-08-29
US14/308,972 US9572832B2 (en) 2013-08-29 2014-06-19 Compound of glycosaminoglycan and its fabrication method as well as application
PCT/EP2014/063720 WO2015028172A1 (en) 2013-08-29 2014-06-27 Compound of glycosaminoglycan, preparation method and use thereof

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Publication Number Publication Date
DK3038656T3 true DK3038656T3 (da) 2021-10-11

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DK14746964.7T DK3038656T3 (da) 2013-08-29 2014-06-27 Forbindelse af glycosaminoglycan, fremgangsmåde til fremstilling og anvendelse deraf

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Country Link
US (7) US9572832B2 (da)
EP (2) EP3038656B1 (da)
JP (2) JP6404925B2 (da)
KR (2) KR102283978B1 (da)
CN (5) CN113893354A (da)
AU (6) AU2014314536B2 (da)
BR (2) BR112016004357B1 (da)
CA (3) CA2921830C (da)
DK (1) DK3038656T3 (da)
EA (4) EA038422B1 (da)
ES (2) ES2893329T3 (da)
HU (1) HUE056434T2 (da)
LT (1) LT3038656T (da)
MY (1) MY180502A (da)
PL (1) PL3038656T3 (da)
PT (1) PT3038656T (da)
TW (2) TWI526212B (da)
WO (2) WO2015028172A1 (da)

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US9572832B2 (en) * 2013-08-29 2017-02-21 Holy Stone Healthcare Co., Ltd. Compound of glycosaminoglycan and its fabrication method as well as application
EA027663B1 (ru) * 2016-05-20 2017-08-31 Тютор С.А.С.И.Ф.И.А. Способ получения твёрдой лекарственной формы для перорального применения и твёрдая лекарственная форма для перорального применения, полученная согласно указанному способу
SG11202109152UA (en) 2019-06-03 2021-12-30 Aihol Corp Hyaluronan conjugates and uses thereof
US11458204B2 (en) 2020-06-02 2022-10-04 Aihol Corporation Method for improving substitution rate and/or substitution efficiency of hyaluronan-drug conjugates
US11643431B2 (en) 2020-06-08 2023-05-09 Aihol Corporation Uses of hyaluronan conjugate
CN117838875B (zh) * 2020-07-15 2025-01-24 上海椿安生物医药科技有限公司 用于局部递送治疗剂的药物递送系统以及其用途
CN116782906A (zh) * 2021-06-18 2023-09-19 爱禾公司 透明质酸复合物的用途
CN116726186A (zh) * 2022-03-11 2023-09-12 四川省医学科学院·四川省人民医院 药物递送系统及其在制备抗黑色素瘤药物中的应用
CN118843468A (zh) * 2022-08-05 2024-10-25 爱禾公司 透明质酸-尼美舒利复合物于治疗局部晚及或转移性肿瘤的用途
PL249385B1 (pl) * 2022-11-23 2026-04-07 Narodowy Inst Onkologii Im Marii Sklodowskiej Curie Oddzial W Gliwicach Prolek-glikokoniugat pochodny gemcytabiny, jako związek o działaniu przeciwnowotworowym, sposób otrzymywania i zastosowanie
WO2025122826A1 (en) * 2023-12-07 2025-06-12 University Of Montana Hyaluronic acid-nonsteroidal anti-inflammatory drug conjugates for treating inflammation-mediated pathologies
CN118831067A (zh) * 2024-07-18 2024-10-25 广东药科大学 一种载药纳米粒及其制备方法和应用
WO2026062560A1 (en) * 2024-09-18 2026-03-26 Didenko Kirill Methods and bioavailable highly permeable compounds for diseases treatment

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