DK34793A - Vandoploeseligt, farmaceutisk acceptabelt salt af et monoacylderivat af rapamycin, fremgangsmaade til dets fremstilling og injicerbart, farmaceutisk praeparat indeholdende det - Google Patents

Vandoploeseligt, farmaceutisk acceptabelt salt af et monoacylderivat af rapamycin, fremgangsmaade til dets fremstilling og injicerbart, farmaceutisk praeparat indeholdende det

Info

Publication number
DK34793A
DK34793A DK034793A DK34793A DK34793A DK 34793 A DK34793 A DK 34793A DK 034793 A DK034793 A DK 034793A DK 34793 A DK34793 A DK 34793A DK 34793 A DK34793 A DK 34793A
Authority
DK
Denmark
Prior art keywords
sub
pharmaceutical
preparation
water soluble
injectable
Prior art date
Application number
DK034793A
Other languages
English (en)
Other versions
DK170750B1 (da
DK34793D0 (da
Inventor
Valentino John Stella
Paul Edwin Kennedy
Original Assignee
Univ Kansas
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Univ Kansas filed Critical Univ Kansas
Publication of DK34793D0 publication Critical patent/DK34793D0/da
Publication of DK34793A publication Critical patent/DK34793A/da
Application granted granted Critical
Publication of DK170750B1 publication Critical patent/DK170750B1/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H1/00—Processes for the preparation of sugar derivatives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D498/18—Bridged systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
DK034793A 1985-12-06 1993-03-25 Vandopløselige, farmaceutisk acceptable salte af i 43-stillingen monosubstitueret rapamycin, fremgangsmåde til fremstilling heraf og injicerbare, farmaceutiske præparater indeholdende et sådant salt. DK170750B1 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US80615285 1985-12-06
US06/806,152 US4650803A (en) 1985-12-06 1985-12-06 Prodrugs of rapamycin

Publications (3)

Publication Number Publication Date
DK34793D0 DK34793D0 (da) 1993-03-25
DK34793A true DK34793A (da) 1993-03-25
DK170750B1 DK170750B1 (da) 1996-01-08

Family

ID=25193443

Family Applications (2)

Application Number Title Priority Date Filing Date
DK584886A DK169409B1 (da) 1985-12-06 1986-12-05 Vanduopløselige, farmaceutisk acceptable salte af substituerede derivater af rapamycin og farmaceutisk præparat indeholdende et sådant salt
DK034793A DK170750B1 (da) 1985-12-06 1993-03-25 Vandopløselige, farmaceutisk acceptable salte af i 43-stillingen monosubstitueret rapamycin, fremgangsmåde til fremstilling heraf og injicerbare, farmaceutiske præparater indeholdende et sådant salt.

Family Applications Before (1)

Application Number Title Priority Date Filing Date
DK584886A DK169409B1 (da) 1985-12-06 1986-12-05 Vanduopløselige, farmaceutisk acceptable salte af substituerede derivater af rapamycin og farmaceutisk præparat indeholdende et sådant salt

Country Status (16)

Country Link
US (1) US4650803A (da)
EP (1) EP0227355B1 (da)
JP (2) JPH0670066B2 (da)
KR (2) KR940004072B1 (da)
AT (1) ATE74134T1 (da)
AU (1) AU583439B2 (da)
CA (2) CA1273920A (da)
DE (1) DE3684574D1 (da)
DK (2) DK169409B1 (da)
ES (1) ES2032750T3 (da)
GB (1) GB2183647A (da)
GR (1) GR3004530T3 (da)
HU (1) HU198054B (da)
IE (1) IE64506B1 (da)
PT (1) PT83843B (da)
ZA (1) ZA869181B (da)

Cited By (2)

* Cited by examiner, † Cited by third party
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US2420367A (en) * 1943-11-09 1947-05-13 Celanese Corp Fluffing up artificial staple fibers
US4748768A (en) * 1982-11-23 1988-06-07 Jacobsen Poul E B Method for the production of a mattress

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US4650803A (en) 1987-03-17
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GB2183647B (da) 1989-10-18
AU583439B2 (en) 1989-04-27
EP0227355B1 (en) 1992-03-25
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AU6608086A (en) 1987-06-11
KR870006072A (ko) 1987-07-09
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KR940004072B1 (ko) 1994-05-11
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JPS62215592A (ja) 1987-09-22
DE3684574D1 (de) 1992-04-30
GR3004530T3 (da) 1993-04-28
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GB2183647A (en) 1987-06-10
ATE74134T1 (de) 1992-04-15
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