DK362889A - Thiazolderivater - Google Patents

Thiazolderivater Download PDF

Info

Publication number: DK362889A
Authority: DK; Denmark
Prior art keywords: substituted; group; hydrogen atom; acyl group; thiazole
Prior art date: 1988-07-22

Application number

DK362889A

Other languages

Danish (da)

English (en)

Other versions

DK362889D0 (da

Inventor

Tetsuya Aono

Masahiro Suno

Go Kito

Original Assignee

Takeda Chemical Industries Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1988-07-22

Filing date

1989-07-21

Publication date

1990-01-23

1989-07-21 Application filed by Takeda Chemical Industries Ltd filed Critical Takeda Chemical Industries Ltd

1989-07-21 Publication of DK362889D0 publication Critical patent/DK362889D0/da

1990-01-23 Publication of DK362889A publication Critical patent/DK362889A/da

Links

FZWLAAWBMGSTSO-UHFFFAOYSA-N Thiazole Chemical compound C1=CSC=N1 FZWLAAWBMGSTSO-UHFFFAOYSA-N 0.000 title 1
125000001931 aliphatic group Chemical group 0.000 abstract 2
125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 2
WRDQLFOQEXCULO-UHFFFAOYSA-N 2h-[1,3]thiazolo[5,4-b]azepine Chemical class C1=CC=CC2=NCSC2=N1 WRDQLFOQEXCULO-UHFFFAOYSA-N 0.000 abstract 1
125000002252 acyl group Chemical group 0.000 abstract 1
125000003118 aryl group Chemical group 0.000 abstract 1
230000015572 biosynthetic process Effects 0.000 abstract 1
125000001589 carboacyl group Chemical group 0.000 abstract 1
230000002401 inhibitory effect Effects 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Veterinary Medicine (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Public Health (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Cardiology (AREA)
Heart & Thoracic Surgery (AREA)
Urology & Nephrology (AREA)
Biomedical Technology (AREA)
Immunology (AREA)
Hematology (AREA)
Obesity (AREA)
Pulmonology (AREA)
Vascular Medicine (AREA)
Diabetes (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Pain & Pain Management (AREA)
Rheumatology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Plural Heterocyclic Compounds (AREA)

DK362889A 1988-07-22 1989-07-21 Thiazolderivater DK362889A (da)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
JP18422088		1988-07-22
JP8653689		1989-04-05

Publications (2)

Publication Number	Publication Date
DK362889D0 DK362889D0 (da)	1989-07-21
DK362889A true DK362889A (da)	1990-01-23

Family

ID=26427638

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK362889A DK362889A (da)	1988-07-22	1989-07-21	Thiazolderivater

Country Status (11)

Country	Link
US (3)	US4956360A (fr)
EP (1)	EP0351856B1 (fr)
JP (1)	JP3054738B2 (fr)
KR (1)	KR970011396B1 (fr)
AT (1)	ATE184610T1 (fr)
AU (1)	AU610739B2 (fr)
CA (1)	CA1336431C (fr)
DE (1)	DE68929074T2 (fr)
DK (1)	DK362889A (fr)
IL (1)	IL91063A (fr)
NZ (1)	NZ230042A (fr)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
IL89351A0 (en) *	1988-03-14	1989-09-10	Lundbeck & Co As H	4,5,6,7-tetrahydroisothiazolo(4,5-c)pyridines,process for their preparation and pharmaceutical compositions containing them
DE3820775A1 (de) *	1988-06-20	1989-12-21	Thomae Gmbh Dr K	Neue 4,5,7,8-tetrahydro-6h-thiazolo(5,4,-d)azepine, ihre herstellung und ihre verwendung als arzneimittel
DE4134467A1 (de) *	1991-10-18	1993-04-22	Thomae Gmbh Dr K	Heterobiarylderivate, diese verbindungen enthaltende arzneimittel und verfahren zu ihrer herstellung
IL97249A (en) *	1990-02-23	1995-01-24	Takeda Chemical Industries Ltd	Compounds of 7,6,5,4-tetrahydrothiazole] B-5,4 [pyridine and compounds of 5,6-dihydro-H4-pyrrolo] D-3,2 [thiazole, their manufacture, and pharmaceutical compositions including or
RU2124503C1 (ru) *	1992-05-18	1999-01-10	И.Р.Сквибб энд Санз, Инк.	Гетероциклические азотсодержащие производные карбоновой кислоты, способ их получения и фармацевтическая композиция
GB9219779D0 (en) *	1992-09-18	1992-10-28	Rhone Poulenc Agriculture	Compositions of new matter
DE4324580A1 (de) *	1993-07-22	1995-01-26	Thomae Gmbh Dr K	Bicyclische Heterocyclen, diese Verbindungen enthaltende Arzneimittel und Verfahren zu ihrer Herstellung
EP0743064A1 (fr) *	1995-05-17	1996-11-20	Eli Lilly And Company	Antagonistes des leucotriènes pour utilisation dans le traitement ou dans la prévention de la maladie d'Alzheimer
US5891460A (en) *	1995-06-07	1999-04-06	University Of Southern California University Park Campus	Method for reducing or preventing post-surgical adhesion formation using ketotifen and analogs thereof
GB2312621B (en) *	1996-05-02	1998-03-11	Pharma Nord Uk Limited	Anti-oxidant medicament
US6433935B2 (en)	1996-07-02	2002-08-13	Three-Five Systems, Inc.	Display illumination system
AU5886500A (en) *	1999-06-23	2001-01-09	Sepracor, Inc.	Indolyl-benzimidazole antibacterials, and methods of use thereof
US6649318B1 (en)	2000-04-20	2003-11-18	Eastman Kodak Company	Self-contained imaging media comprising microencapsulated color formers and a resilient layer
RU2188824C1 (ru) *	2000-12-18	2002-09-10	Военно-медицинская академия	2-амино-4-ацетилтиазоло[5,4-b]индол, защищающий организм от воздействия гипоксии и токсического отека легкого
US7148248B2 (en)	2002-11-29	2006-12-12	Masako Nozaki	Method of treating or inhibiting the development of brain inflammation and sepsis
EP1424101A3 (fr) *	2002-11-29	2004-08-18	NOZAKI, Masako	Utilisation d'un antagoniste du leucotriène c4/d4 pour la préparation d'un médicament pour le traitement ou la prévention d'une inflammation ou septicémie du cerveau
DK1691814T3 (da) *	2003-12-01	2012-10-29	Cambridge Entpr Ltd	Antiinflammatoriske midler
RU2281950C2 (ru) *	2004-09-21	2006-08-20	Военно-медицинская академия им. С.М. Кирова	4-АЦЕТИЛТИАЗОЛО[5,4-b]ИНДОЛ-2-СУКЦИНИМИД, ЗАЩИЩАЮЩИЙ ОРГАНИЗМ ОТ ГИПОКСИИ И ОБЛАДАЮЩИЙ ПРОФИЛАКТИЧЕСКИМ ДЕЙСТВИЕМ В ОТНОШЕНИИ ТОКСИЧЕСКОГО ОТЕКА ЛЕГКОГО
EP1896036B1 (fr)	2005-06-15	2013-01-23	Cambridge Enterprise Limited	Agents anti-inflammatoires
GB201009603D0 (en) *	2010-06-08	2010-07-21	Cambridge Entpr Ltd	Anti-inflammatory agent

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
BG17785A3 (bg) *	1970-08-14	1973-12-25	Dr. Karl Thomae Gmbh	Метод за получаване на нови азетинови производни
JPS53121781A (en) *	1977-03-30	1978-10-24	Torii Yakuhin Kk	Caprolactum derivatives
AU554388B2 (en) *	1981-06-15	1986-08-21	American Home Products Corporation	Alpha-phenyl-2-(aza)benzothiazolylthioglycolic acid derivatives
JPS5837097A (ja) *	1981-08-28	1983-03-04	味の素株式会社	界面活性剤
JPS63283591A (ja) *	1986-12-17	1988-11-21	Toray Ind Inc	Ｌ−α−アミノ−ε−カプロラクタムの製造法

1989
- 1989-07-19 JP JP01187790A patent/JP3054738B2/ja not_active Expired - Lifetime
- 1989-07-20 EP EP89113362A patent/EP0351856B1/fr not_active Expired - Lifetime
- 1989-07-20 DE DE68929074T patent/DE68929074T2/de not_active Expired - Fee Related
- 1989-07-20 AT AT89113362T patent/ATE184610T1/de not_active IP Right Cessation
- 1989-07-21 CA CA000606328A patent/CA1336431C/fr not_active Expired - Fee Related
- 1989-07-21 NZ NZ230042A patent/NZ230042A/en unknown
- 1989-07-21 DK DK362889A patent/DK362889A/da not_active Application Discontinuation
- 1989-07-21 IL IL9106389A patent/IL91063A/en not_active IP Right Cessation
- 1989-07-21 AU AU38862/89A patent/AU610739B2/en not_active Ceased
- 1989-07-21 US US07/383,071 patent/US4956360A/en not_active Expired - Lifetime
- 1989-07-22 KR KR1019890010423A patent/KR970011396B1/ko not_active Expired - Lifetime
1990
- 1990-07-27 US US07/558,507 patent/US5118806A/en not_active Expired - Fee Related
1992
- 1992-03-17 US US07/852,657 patent/US5300639A/en not_active Expired - Fee Related

Also Published As

Publication number	Publication date
US4956360A (en)	1990-09-11
JPH0347188A (ja)	1991-02-28
AU3886289A (en)	1990-01-25
ATE184610T1 (de)	1999-10-15
DE68929074D1 (de)	1999-10-21
KR910002873A (ko)	1991-02-26
US5118806A (en)	1992-06-02
JP3054738B2 (ja)	2000-06-19
IL91063A0 (en)	1990-02-09
NZ230042A (en)	1990-10-26
DK362889D0 (da)	1989-07-21
CA1336431C (fr)	1995-07-25
IL91063A (en)	1994-12-29
EP0351856A2 (fr)	1990-01-24
EP0351856B1 (fr)	1999-09-15
US5300639A (en)	1994-04-05
EP0351856A3 (fr)	1991-08-07
DE68929074T2 (de)	2000-01-05
KR970011396B1 (ko)	1997-07-10
AU610739B2 (en)	1991-05-23

Legal Events

Date	Code	Title	Description
1989-07-21	A0	Application filed
1996-03-25	AHB	Application shelved due to non-payment

Publication	Publication Date	Title
DK362889A (da)	1990-01-23	Thiazolderivater
NO904377L (no)	1991-04-12	Tricykliske karbapenemforbindelser.
ATE93849T1 (de)	1993-09-15	Imidoaromatische percarbonsaeure.
IT1215739B (it)	1990-02-22	Perossiacidi immido aromatici come agenti sbiancanti.
FI982436A0 (fi)	1998-11-10	Kondensoituneet heterosykliset yhdisteet
ID17851A (id)	1998-01-29	Persenyawaan heterosiklis, produksi dan pemakaiannya
NO893453L (no)	1990-03-01	Antibakterielle spiro-forbindelser og fremgangsmaate for deres fremstilling.
ATE123778T1 (de)	1995-06-15	Beta-lactam-derivate.
TW198022B (fr)	1993-01-11
FI911080A0 (fi)	1991-03-04	Menetelmä 1,5-bentsotiatsepiinijohdannaisten valmistamiseksi
AU7819187A (en)	1988-03-17	New phenyl, pyrrolidin-2-yl substituted 5-ring heterocycles having antiphycsotic properties
DE3884499D1 (de)	1993-11-04	Heterozyklische peroxycarbonsaeure.
ATE148699T1 (de)	1997-02-15	Herstellung von 2-(2-thienyl)äthylamin und synthese von thieno(3,2-c)pyridinderivaten daraus
IT1219690B (it)	1990-05-24	Perossiacidi eterociclici azotati monopersolfati
ATE119909T1 (de)	1995-04-15	3-deoxymycaminosyltylonolidderivate.
DE69317920D1 (de)	1998-05-20	Thiazolderivate von Alcoxyacrylaten mit fungizider Wirkung