ECSP034567A - Inhibidores de espiropirimidin-2,4,6-triona metaloproteinasas - Google Patents

Inhibidores de espiropirimidin-2,4,6-triona metaloproteinasas

Info

Publication number: ECSP034567A
Authority: EC; Ecuador
Prior art keywords: spiropirimidin; triona; inhibitors; metaloproteinase inhibitors; metaloproteinase
Prior art date: 2000-10-26

Application number

EC2003004567A

Other languages

English (en)

Spanish (es)

Inventor

Mark Carl Noe

Martin James Wythes

Brian S Bronk

Original Assignee

Pfizer Prod Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-10-26

Filing date

2003-04-25

Publication date

2003-06-25

2003-04-25 Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc

2003-06-25 Publication of ECSP034567A publication Critical patent/ECSP034567A/es

Links

239000003112 inhibitor Substances 0.000 title abstract 2
125000003341 7 membered heterocyclic group Chemical group 0.000 abstract 1
206010061218 Inflammation Diseases 0.000 abstract 1
102000005741 Metalloproteases Human genes 0.000 abstract 1
108010006035 Metalloproteases Proteins 0.000 abstract 1
206010028980 Neoplasm Diseases 0.000 abstract 1
201000011510 cancer Diseases 0.000 abstract 1
230000004054 inflammatory process Effects 0.000 abstract 1
239000008194 pharmaceutical composition Substances 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
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- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/10—Spiro-condensed systems
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Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Physical Education & Sports Medicine (AREA)
Immunology (AREA)
Reproductive Health (AREA)
Endocrinology (AREA)
Oncology (AREA)
Rheumatology (AREA)
Pain & Pain Management (AREA)
Orthopedic Medicine & Surgery (AREA)
Dermatology (AREA)
Communicable Diseases (AREA)
Gynecology & Obstetrics (AREA)
Diabetes (AREA)
Pulmonology (AREA)
Ophthalmology & Optometry (AREA)
Heart & Thoracic Surgery (AREA)
Pregnancy & Childbirth (AREA)
Hematology (AREA)
Tropical Medicine & Parasitology (AREA)
Cardiology (AREA)
Virology (AREA)
Obesity (AREA)
Psychology (AREA)

EC2003004567A 2000-10-26 2003-04-25 Inhibidores de espiropirimidin-2,4,6-triona metaloproteinasas ECSP034567A (es)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US24338900P	2000-10-26	2000-10-26

Publications (1)

Publication Number	Publication Date
ECSP034567A true ECSP034567A (es)	2003-06-25

Family

ID=22918584

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
EC2003004567A ECSP034567A (es)	2000-10-26	2003-04-25	Inhibidores de espiropirimidin-2,4,6-triona metaloproteinasas

Country Status (32)

Country	Link
EP (1)	EP1332146A2 (bg)
JP (1)	JP2004518635A (bg)
KR (1)	KR20040004412A (bg)
CN (1)	CN1501937A (bg)
AP (1)	AP2001002318A0 (bg)
AR (1)	AR035069A1 (bg)
AU (1)	AU2002210813A1 (bg)
BG (1)	BG107653A (bg)
BR (1)	BR0114913A (bg)
CA (1)	CA2425283A1 (bg)
CZ (1)	CZ20031083A3 (bg)
EA (1)	EA005762B1 (bg)
EC (1)	ECSP034567A (bg)
EE (1)	EE200300196A (bg)
GT (1)	GT200100213A (bg)
HN (1)	HN2001000244A (bg)
HR (1)	HRP20030332A2 (bg)
HU (1)	HUP0301577A3 (bg)
IL (1)	IL154948A0 (bg)
IS (1)	IS6762A (bg)
MA (1)	MA26957A1 (bg)
MX (1)	MXPA03003735A (bg)
NO (1)	NO20031853L (bg)
OA (1)	OA12529A (bg)
PA (1)	PA8531401A1 (bg)
PE (1)	PE20020589A1 (bg)
PL (1)	PL366201A1 (bg)
SK (1)	SK4972003A3 (bg)
SV (1)	SV2003000705A (bg)
TN (1)	TNSN01149A1 (bg)
WO (1)	WO2002034753A2 (bg)
ZA (1)	ZA200302190B (bg)

Families Citing this family (39)

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EP1368323B1 (en)	2001-02-14	2010-06-30	Warner-Lambert Company LLC	Pyrimidine matrix metalloproteinase inhibitors
DOP2002000333A (es)	2001-02-14	2002-09-30	Warner Lambert Co	Derivados de acido isoftalico como inhibidores de metaloproteinasas de la matriz
MXPA03005870A (es)	2001-02-14	2005-02-14	Warner Lambert Co	Inhibirores de benzotiadiazina de metaloproteinasas de la matriz.
PA8539501A1 (es)	2001-02-14	2002-09-30	Warner Lambert Co	Compuestos triazolo como inhibidores de mmp
DOP2002000332A (es)	2001-02-14	2002-08-30	Warner Lambert Co	Inhibidores de piridina de metaloproteinasas de la matriz
US6924276B2 (en)	2001-09-10	2005-08-02	Warner-Lambert Company	Diacid-substituted heteroaryl derivatives as matrix metalloproteinase inhibitors
EP1434585A1 (en)	2001-10-12	2004-07-07	Warner-Lambert Company LLC	Alkyne matrix metalloproteinase inhibitors
US6962922B2 (en)	2001-10-12	2005-11-08	Warner-Lambert Company Llc	Alkynylated quinazoline compounds
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2001
- 2001-10-23 BR BR0114913-0A patent/BR0114913A/pt not_active IP Right Cessation
- 2001-10-23 HU HU0301577A patent/HUP0301577A3/hu unknown
- 2001-10-23 EP EP01978721A patent/EP1332146A2/en not_active Withdrawn
- 2001-10-23 JP JP2002537743A patent/JP2004518635A/ja not_active Withdrawn
- 2001-10-23 HR HR20030332A patent/HRP20030332A2/hr not_active Application Discontinuation
- 2001-10-23 SK SK497-2003A patent/SK4972003A3/sk unknown
- 2001-10-23 CA CA002425283A patent/CA2425283A1/en not_active Abandoned
- 2001-10-23 PL PL01366201A patent/PL366201A1/xx not_active Application Discontinuation
- 2001-10-23 WO PCT/IB2001/001986 patent/WO2002034753A2/en not_active Ceased
- 2001-10-23 KR KR10-2003-7005753A patent/KR20040004412A/ko not_active Ceased
- 2001-10-23 OA OA1200300123A patent/OA12529A/en unknown
- 2001-10-23 EE EEP200300196A patent/EE200300196A/xx unknown
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- 2001-10-23 AU AU2002210813A patent/AU2002210813A1/en not_active Abandoned
- 2001-10-23 MX MXPA03003735A patent/MXPA03003735A/es unknown
- 2001-10-23 AP APAP/P/2001/002318A patent/AP2001002318A0/en unknown
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- 2001-10-23 EA EA200300306A patent/EA005762B1/ru not_active IP Right Cessation
- 2001-10-23 CN CNA018179231A patent/CN1501937A/zh active Pending
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- 2001-10-25 PE PE2001001060A patent/PE20020589A1/es not_active Application Discontinuation
- 2001-10-25 SV SV2001000705A patent/SV2003000705A/es unknown
- 2001-10-25 TN TNTNSN01149A patent/TNSN01149A1/fr unknown
- 2001-10-25 GT GT200100213A patent/GT200100213A/es unknown
- 2001-10-26 PA PA20018531401A patent/PA8531401A1/es unknown
2003
- 2003-03-19 ZA ZA200302190A patent/ZA200302190B/en unknown
- 2003-03-20 BG BG107653A patent/BG107653A/bg unknown
- 2003-03-27 IS IS6762A patent/IS6762A/is unknown
- 2003-04-22 MA MA27117A patent/MA26957A1/fr unknown
- 2003-04-24 NO NO20031853A patent/NO20031853L/no not_active Application Discontinuation
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Also Published As

Publication number	Publication date
AU2002210813A1 (en)	2002-05-06
EP1332146A2 (en)	2003-08-06
HN2001000244A (es)	2003-11-07
JP2004518635A (ja)	2004-06-24
EA005762B1 (ru)	2005-06-30
SK4972003A3 (en)	2004-05-04
NO20031853D0 (no)	2003-04-24
BR0114913A (pt)	2003-07-01
MXPA03003735A (es)	2003-07-28
OA12529A (en)	2006-06-02
EE200300196A (et)	2003-10-15
KR20040004412A (ko)	2004-01-13
GT200100213A (es)	2002-07-03
TNSN01149A1 (fr)	2005-11-10
WO2002034753A2 (en)	2002-05-02
BG107653A (bg)	2003-12-31
IL154948A0 (en)	2003-10-31
IS6762A (is)	2003-03-27
PA8531401A1 (es)	2003-06-30
WO2002034753A3 (en)	2002-08-15
CA2425283A1 (en)	2002-05-02
EA200300306A1 (ru)	2003-08-28
HUP0301577A2 (hu)	2003-11-28
HRP20030332A2 (en)	2003-06-30
AP2001002318A0 (en)	2001-12-31
HUP0301577A3 (en)	2006-02-28
SV2003000705A (es)	2003-01-13
PE20020589A1 (es)	2002-07-06
MA26957A1 (fr)	2004-12-20
ZA200302190B (en)	2004-04-28
CN1501937A (zh)	2004-06-02
AR035069A1 (es)	2004-04-14
NO20031853L (no)	2003-06-23
PL366201A1 (en)	2005-01-24
CZ20031083A3 (cs)	2004-03-17

Publication	Publication Date	Title
ECSP034567A (es)	2003-06-25	Inhibidores de espiropirimidin-2,4,6-triona metaloproteinasas
UY27777A1 (es)	2003-11-28	Inhibidores de metaloproteinasa de heteroariloxi-aril-espiro-pirimidina-2,4,6-triona n-sustituida
ECSP034568A (es)	2003-06-25	Inhibidores de metaloproteinasa del tipo pirimidin 2,4,6-triona
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BR0316680A (pt)	2005-10-18	Pirimidinas inibidoras de chk, pdk e akt, sua produção e uso como agentes farmacêuticos
PA8572101A1 (es)	2003-12-10	Inhibidores de metaloproteinasa de aril-heteroariloxi-ariloxi-pirimidina-2,4,6-triona
BRPI0413452A (pt)	2006-10-17	composto, composição farmacêutica, kit, artigo de fabricação, e, métodos de inibir dpp-iv, terapêutico e de tratar um estado de doença, cáncer, distúrbios autoimunes, uma condição einfecção por hiv
HN2000000137A (es)	2001-02-02	Pirimidina-2,4,6-trionas inhibidores de metaloproteinasas
SE0001899D0 (sv)	2000-05-22	New compounds
ECSP066314A (es)	2006-07-28	Derivados piridilo y su uso como agentes terapéuticos
ATE437872T1 (de)	2009-08-15	Proteinkinaseinhibitoren
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BR0315580A (pt)	2005-08-30	Derivados de metileno uréia
SE0401342D0 (sv)	2004-05-25	Therapeutic compounds
AR047529A1 (es)	2006-01-25	Compuestos de quinolina sustituidos
UY27872A1 (es)	2003-12-31	Inhibidores de caspasa y usos de los mismos.
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ATE275143T1 (de)	2004-09-15	Verbindungen
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