BRPI0514833A - fenilaminotiazóis substituìdos e seu uso - Google Patents

fenilaminotiazóis substituìdos e seu uso

Info

Publication number
BRPI0514833A
BRPI0514833A BRPI0514833-2A BRPI0514833A BRPI0514833A BR PI0514833 A BRPI0514833 A BR PI0514833A BR PI0514833 A BRPI0514833 A BR PI0514833A BR PI0514833 A BRPI0514833 A BR PI0514833A
Authority
BR
Brazil
Prior art keywords
phenylaminothiazoles
substituted
treatment
diseases
prophylaxis
Prior art date
Application number
BRPI0514833-2A
Other languages
English (en)
Inventor
Jens-Kerim Ergueden
Gunter Karig
Ulrich Rosentreter
Barbara Albrecht
Kerstin Henninger
Joachim Huetter
Nicole Diedrichs
Peter Nell
Sabine Arndt
Walter Huebsch
Andreas Knorr
Karl-Heinz Schlemmer
Dirk Brohm
Original Assignee
Bayer Healthcare Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Healthcare Ag filed Critical Bayer Healthcare Ag
Publication of BRPI0514833A publication Critical patent/BRPI0514833A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

FENILAMINOTIAZóIS SUBSTITUìDOS E SEU USO. Refere-se aos novos derivados de fenilaminotiazol, processos para sua produção, seu uso para o tratamento e/ou profilaxia de doenças, bem como seu uso para a produção de medicamentos para o tratamento e/ou profilaxia de doenças, preferentemente para o tratamento e/ou prevenção de hipertonia e de outras doenças cardiovasculares.
BRPI0514833-2A 2004-09-03 2005-08-30 fenilaminotiazóis substituìdos e seu uso BRPI0514833A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE102004042607A DE102004042607A1 (de) 2004-09-03 2004-09-03 Substituierte Phenylaminothiazole und ihre Verwendung
PCT/EP2005/009316 WO2006027142A1 (de) 2004-09-03 2005-08-30 Substituierte phenylaminothiazole und ihre verwendung

Publications (1)

Publication Number Publication Date
BRPI0514833A true BRPI0514833A (pt) 2008-06-24

Family

ID=35852458

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0514833-2A BRPI0514833A (pt) 2004-09-03 2005-08-30 fenilaminotiazóis substituìdos e seu uso

Country Status (24)

Country Link
US (1) US8691850B2 (pt)
EP (1) EP1812430B1 (pt)
JP (1) JP4999691B2 (pt)
KR (1) KR20070057235A (pt)
CN (1) CN101056875A (pt)
AR (1) AR050551A1 (pt)
AT (1) ATE428710T1 (pt)
AU (1) AU2005281941A1 (pt)
BR (1) BRPI0514833A (pt)
CA (1) CA2578596C (pt)
DE (2) DE102004042607A1 (pt)
EC (1) ECSP077296A (pt)
ES (1) ES2324049T3 (pt)
GT (1) GT200500238A (pt)
IL (1) IL181670A0 (pt)
MA (1) MA28869B1 (pt)
MX (1) MX2007002470A (pt)
NO (1) NO20071343L (pt)
PE (1) PE20060589A1 (pt)
SV (1) SV2006002218A (pt)
TW (1) TW200621765A (pt)
UY (1) UY29099A1 (pt)
WO (1) WO2006027142A1 (pt)
ZA (1) ZA200701820B (pt)

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DE102006056740A1 (de) 2006-12-01 2008-06-05 Bayer Healthcare Ag Cyclisch substituierte 3,5-Dicyano-2-thiopyridine und ihre Verwendung
DE102007035367A1 (de) 2007-07-27 2009-01-29 Bayer Healthcare Ag Substituierte Aryloxazole und ihre Verwendung
DE102007036076A1 (de) 2007-08-01 2009-02-05 Bayer Healthcare Aktiengesellschaft Dipeptoid-Produgs und ihre Verwendung
DE102007061764A1 (de) 2007-12-20 2009-06-25 Bayer Healthcare Ag Anellierte Cyanopyridine und ihre Verwendung
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DE102010030688A1 (de) 2010-06-30 2012-01-05 Bayer Schering Pharma Aktiengesellschaft Substituierte Dicyanopyridine und ihre Verwendung
AU2014305843B2 (en) 2013-08-09 2019-08-29 Ardelyx, Inc. Compounds and methods for inhibiting phosphate transport
WO2018153900A1 (de) 2017-02-22 2018-08-30 Bayer Aktiengesellschaft Selektive partielle adenosin a1 rezeptor-agonisten in kombination mit sglt-2-hemmern
WO2018153897A1 (de) 2017-02-22 2018-08-30 Bayer Pharma Aktiengesellschaft Selektive partielle adenosin a1 rezeptor-agonisten in kombination mit hcn-kanal-hemmern
WO2018153895A1 (de) 2017-02-22 2018-08-30 Bayer Pharma Aktiengesellschaft Selektive partielle adenosin a1 rezeptor-agonisten in kombination mit einem inhibitor der neutralen endopeptidase und/oder einem angiotensin ii rezeptor-antagonisten
WO2018153899A1 (de) 2017-02-22 2018-08-30 Bayer Pharma Aktiengesellschaft Selektive partielle adenosin a1 rezeptor-agonisten in kombination mit stimulatoren und/oder aktivatoren der löslichen guanylatcyclase (sgc)
WO2018153898A1 (de) 2017-02-22 2018-08-30 Bayer Pharma Aktiengesellschaft Selektive partielle adenosin a1 rezeptor-agonisten in kombination mit mineralocorticoid-rezeptor-antagonisten
JP7323913B2 (ja) * 2019-04-12 2023-08-09 国立大学法人 筑波大学 睡眠誘導剤である複素環化合物

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Also Published As

Publication number Publication date
MX2007002470A (es) 2009-02-12
PE20060589A1 (es) 2006-08-12
GT200500238A (es) 2006-04-10
WO2006027142A1 (de) 2006-03-16
IL181670A0 (en) 2007-07-04
DE102004042607A1 (de) 2006-03-09
ES2324049T3 (es) 2009-07-29
MA28869B1 (fr) 2007-09-03
KR20070057235A (ko) 2007-06-04
ZA200701820B (en) 2008-08-27
NO20071343L (no) 2007-05-30
EP1812430A1 (de) 2007-08-01
AU2005281941A1 (en) 2006-03-16
CN101056875A (zh) 2007-10-17
ECSP077296A (es) 2007-04-26
CA2578596A1 (en) 2006-03-16
SV2006002218A (es) 2006-10-04
JP4999691B2 (ja) 2012-08-15
AR050551A1 (es) 2006-11-01
JP2008511614A (ja) 2008-04-17
UY29099A1 (es) 2006-04-28
EP1812430B1 (de) 2009-04-15
TW200621765A (en) 2006-07-01
CA2578596C (en) 2012-10-23
DE502005007106D1 (de) 2009-05-28
US8691850B2 (en) 2014-04-08
US20080269300A1 (en) 2008-10-30
ATE428710T1 (de) 2009-05-15

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Legal Events

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B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE AS 5A E 6A ANUIDADES.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2160 DE 29/05/2012.