ES2055887T3 - Nuevos derivados de la morfolina, su procedimiento de preparacion y las composiciones farmaceuticas que los contienen. - Google Patents
Nuevos derivados de la morfolina, su procedimiento de preparacion y las composiciones farmaceuticas que los contienen.Info
- Publication number
- ES2055887T3 ES2055887T3 ES90403123T ES90403123T ES2055887T3 ES 2055887 T3 ES2055887 T3 ES 2055887T3 ES 90403123 T ES90403123 T ES 90403123T ES 90403123 T ES90403123 T ES 90403123T ES 2055887 T3 ES2055887 T3 ES 2055887T3
- Authority
- ES
- Spain
- Prior art keywords
- morpholine
- contain
- pharmaceutical compositions
- preparation procedure
- new derivatives
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/08—Vasodilators for multiple indications
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Life Sciences & Earth Sciences (AREA)
- Neurology (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Neurosurgery (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Biomedical Technology (AREA)
- Heart & Thoracic Surgery (AREA)
- Hospice & Palliative Care (AREA)
- Cardiology (AREA)
- Psychiatry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
NUEVOS DERIVADOS DE LA MORFOLINA, UTILIZABLES COMO MEDICAMENTO Y QUE RESPONDE A LA FORMULA: EN LA QUE: X, FIJADO SOBRE EL NUCLEO AROMATICO, ES HALOGENO O TRIFLUOROMETILO, Y R'' ES HIDROGENO, (C SUB 1 TE UN DOBLE ENLACE, O ARALQUILO, EN FORMAS RACEMICAS Y ENANTIOMERO. ESTOS DERIVADOS Y SUS SALES FISIOLOGICAMENTE TOLERABLES PUEDEN UTILIZARSE EN TERAPIA, EN PARTICULAR, EN EL TRATAMIENTO DE LOS SINDROMES ISQUEMICOS Y DEL ENVEJECIMIENTO CEREBRAL.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR8914489A FR2653999A1 (fr) | 1989-11-06 | 1989-11-06 | Nouveaux derives de la morpholine, leur procede de preparation et les compositions pharmaceutiques les renfermant. |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES2055887T3 true ES2055887T3 (es) | 1994-09-01 |
Family
ID=9387096
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES90403123T Expired - Lifetime ES2055887T3 (es) | 1989-11-06 | 1990-11-06 | Nuevos derivados de la morfolina, su procedimiento de preparacion y las composiciones farmaceuticas que los contienen. |
Country Status (15)
| Country | Link |
|---|---|
| US (1) | US5026701A (es) |
| EP (1) | EP0427605B1 (es) |
| JP (1) | JPH06102660B2 (es) |
| AT (1) | ATE104976T1 (es) |
| AU (1) | AU631465B2 (es) |
| CA (1) | CA2029334A1 (es) |
| DE (1) | DE69008489T2 (es) |
| DK (1) | DK0427605T3 (es) |
| ES (1) | ES2055887T3 (es) |
| FR (1) | FR2653999A1 (es) |
| IE (1) | IE66019B1 (es) |
| NZ (1) | NZ235815A (es) |
| OA (1) | OA09467A (es) |
| PT (1) | PT95782B (es) |
| ZA (1) | ZA908883B (es) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5698007A (en) * | 1992-08-06 | 1997-12-16 | Akzo Nobel Nv | Process for agglomerating particulate material |
| BR9407469A (pt) * | 1993-09-15 | 1996-11-12 | Syntex Inc | Micofenolato mofetil anidro cristalino e formulação intravenosa do mesmo |
| US20040030131A1 (en) * | 2000-10-04 | 2004-02-12 | Martine Keenan | Pharmaceutical compounds |
| AU2005238296A1 (en) | 2004-04-30 | 2005-11-10 | Warner-Lambert Company Llc | Substituted morpholine compounds for the treatment of central nervous system disorders |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BE758766A (fr) * | 1969-11-17 | 1971-05-10 | Ici Ltd | Nouveaux derives de la morpholine et de la |
| FR2612926B1 (fr) * | 1987-03-24 | 1989-06-09 | Adir | Nouveaux derives de la morpholine, leur procede de preparation et les compositions pharmaceutiques les renfermant |
-
1989
- 1989-11-06 FR FR8914489A patent/FR2653999A1/fr active Granted
-
1990
- 1990-10-24 NZ NZ235815A patent/NZ235815A/en unknown
- 1990-10-25 US US07/603,522 patent/US5026701A/en not_active Expired - Fee Related
- 1990-11-05 PT PT95782A patent/PT95782B/pt not_active IP Right Cessation
- 1990-11-05 AU AU65771/90A patent/AU631465B2/en not_active Ceased
- 1990-11-05 CA CA002029334A patent/CA2029334A1/fr not_active Abandoned
- 1990-11-05 IE IE397290A patent/IE66019B1/en not_active IP Right Cessation
- 1990-11-06 ES ES90403123T patent/ES2055887T3/es not_active Expired - Lifetime
- 1990-11-06 DK DK90403123.4T patent/DK0427605T3/da active
- 1990-11-06 AT AT9090403123T patent/ATE104976T1/de not_active IP Right Cessation
- 1990-11-06 DE DE69008489T patent/DE69008489T2/de not_active Expired - Fee Related
- 1990-11-06 JP JP2300917A patent/JPH06102660B2/ja not_active Expired - Lifetime
- 1990-11-06 OA OA59884A patent/OA09467A/xx unknown
- 1990-11-06 ZA ZA908883A patent/ZA908883B/xx unknown
- 1990-11-06 EP EP90403123A patent/EP0427605B1/fr not_active Expired - Lifetime
Also Published As
| Publication number | Publication date |
|---|---|
| ATE104976T1 (de) | 1994-05-15 |
| CA2029334A1 (fr) | 1991-05-07 |
| DK0427605T3 (da) | 1994-07-25 |
| EP0427605B1 (fr) | 1994-04-27 |
| ZA908883B (en) | 1991-08-28 |
| NZ235815A (en) | 1992-04-28 |
| DE69008489T2 (de) | 1994-10-13 |
| OA09467A (fr) | 1992-11-15 |
| DE69008489D1 (de) | 1994-06-01 |
| AU631465B2 (en) | 1992-11-26 |
| AU6577190A (en) | 1991-07-11 |
| PT95782A (pt) | 1991-09-13 |
| JPH03184978A (ja) | 1991-08-12 |
| EP0427605A1 (fr) | 1991-05-15 |
| JPH06102660B2 (ja) | 1994-12-14 |
| FR2653999A1 (fr) | 1991-05-10 |
| FR2653999B1 (es) | 1994-04-22 |
| IE66019B1 (en) | 1995-11-29 |
| PT95782B (pt) | 1997-11-28 |
| IE903972A1 (en) | 1991-05-08 |
| US5026701A (en) | 1991-06-25 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FG2A | Definitive protection |
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