ES2290754T3 - Derivados de triazolopirimidina como inhibidores de la glucogeno sintasa cinasa 3. - Google Patents

Derivados de triazolopirimidina como inhibidores de la glucogeno sintasa cinasa 3. Download PDF

Info

Publication number: ES2290754T3
Authority: ES; Spain
Prior art keywords: alkyloxy; alkyl; carboxyl; cyano; hydroxyl
Prior art date: 2003-07-16
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Expired - Lifetime

Application number

ES04766189T

Other languages

English (en)

Spanish (es)

Inventor

Eddy Jean Edgard Janssen Pharmaceutica NV FREYNE

Christopher John Janssen Pharmaceutica N.V. LOVE

Ludwig Paul Janssen Pharmaceutica N.V. COOYMANS

Nele c/o Janssen Pharmaceutica N.V. VANDERMAESEN

Peter J.J.A Janssen Pharmaceutica N.V BUIJNSTERS

Marc c/o Janssen Pharmaceutica N.V. WILLEMS

Werner C.J. Janssen Pharmaceutica N.V. EMBRECHTS

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Janssen Pharmaceutica NV

Original Assignee

Janssen Pharmaceutica NV

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2003-07-16

Filing date

2004-07-12

Publication date

2008-02-16

2004-07-12 Application filed by Janssen Pharmaceutica NV filed Critical Janssen Pharmaceutica NV

2008-02-16 Application granted granted Critical

2008-02-16 Publication of ES2290754T3 publication Critical patent/ES2290754T3/es

2024-07-12 Anticipated expiration legal-status Critical

Status Expired - Lifetime legal-status Critical Current

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Classifications

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- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
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- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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ES04766189T 2003-07-16 2004-07-12 Derivados de triazolopirimidina como inhibidores de la glucogeno sintasa cinasa 3. Expired - Lifetime ES2290754T3 (es)

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WOPCT/EP03/50310		2003-07-16
EP0350310		2003-07-16

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ES2290754T3 true ES2290754T3 (es)	2008-02-16

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ES04766189T Expired - Lifetime ES2290754T3 (es)	2003-07-16	2004-07-12	Derivados de triazolopirimidina como inhibidores de la glucogeno sintasa cinasa 3.

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US (2)	US7560458B2 (pt)
EP (1)	EP1658292B1 (pt)
JP (1)	JP2009514782A (pt)
KR (1)	KR20060120393A (pt)
CN (1)	CN100404536C (pt)
AP (1)	AP2006003486A0 (pt)
AR (1)	AR045698A1 (pt)
AT (1)	ATE370142T1 (pt)
AU (1)	AU2004260738B2 (pt)
BR (1)	BRPI0412596A (pt)
CA (1)	CA2531333A1 (pt)
DE (1)	DE602004008303T2 (pt)
DK (1)	DK1658292T3 (pt)
EA (1)	EA010109B1 (pt)
ES (1)	ES2290754T3 (pt)
IL (1)	IL173139A (pt)
JO (1)	JO2460B1 (pt)
MX (1)	MXPA06000540A (pt)
NO (1)	NO20060678L (pt)
NZ (1)	NZ545058A (pt)
PA (1)	PA8607001A1 (pt)
PL (1)	PL1658292T3 (pt)
PT (1)	PT1658292E (pt)
TW (1)	TW200524935A (pt)
WO (1)	WO2005012307A1 (pt)
ZA (1)	ZA200600385B (pt)

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2004
- 2004-07-12 DK DK04766189T patent/DK1658292T3/da active
- 2004-07-12 PL PL04766189T patent/PL1658292T3/pl unknown
- 2004-07-12 CA CA002531333A patent/CA2531333A1/en not_active Abandoned
- 2004-07-12 CN CNB2004800201486A patent/CN100404536C/zh not_active Expired - Fee Related
- 2004-07-12 ES ES04766189T patent/ES2290754T3/es not_active Expired - Lifetime
- 2004-07-12 AP AP2006003486A patent/AP2006003486A0/xx unknown
- 2004-07-12 NZ NZ545058A patent/NZ545058A/en not_active IP Right Cessation
- 2004-07-12 MX MXPA06000540A patent/MXPA06000540A/es active IP Right Grant
- 2004-07-12 JO JO200496A patent/JO2460B1/en active
- 2004-07-12 EA EA200600258A patent/EA010109B1/ru not_active IP Right Cessation
- 2004-07-12 WO PCT/EP2004/051455 patent/WO2005012307A1/en not_active Ceased
- 2004-07-12 JP JP2006519926A patent/JP2009514782A/ja not_active Withdrawn
- 2004-07-12 KR KR1020057024541A patent/KR20060120393A/ko not_active Ceased
- 2004-07-12 EP EP04766189A patent/EP1658292B1/en not_active Expired - Lifetime
- 2004-07-12 BR BRPI0412596-7A patent/BRPI0412596A/pt not_active IP Right Cessation
- 2004-07-12 PT PT04766189T patent/PT1658292E/pt unknown
- 2004-07-12 DE DE602004008303T patent/DE602004008303T2/de not_active Expired - Lifetime
- 2004-07-12 AT AT04766189T patent/ATE370142T1/de active
- 2004-07-12 US US10/564,844 patent/US7560458B2/en not_active Expired - Fee Related
- 2004-07-12 AU AU2004260738A patent/AU2004260738B2/en not_active Ceased
- 2004-07-15 TW TW093121066A patent/TW200524935A/zh unknown
- 2004-07-15 PA PA20048607001A patent/PA8607001A1/es unknown
- 2004-07-15 AR ARP040102496A patent/AR045698A1/es not_active Application Discontinuation
2006
- 2006-01-12 IL IL173139A patent/IL173139A/en not_active IP Right Cessation
- 2006-01-13 ZA ZA200600385A patent/ZA200600385B/en unknown
- 2006-02-10 NO NO20060678A patent/NO20060678L/no not_active Application Discontinuation
2008
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Publication number	Publication date
US20060205721A1 (en)	2006-09-14
ZA200600385B (en)	2007-05-30
BRPI0412596A (pt)	2006-09-19
MXPA06000540A (es)	2006-03-30
EA010109B1 (ru)	2008-06-30
TW200524935A (en)	2005-08-01
CA2531333A1 (en)	2005-02-10
PA8607001A1 (es)	2005-05-10
AU2004260738A1 (en)	2005-02-10
EA200600258A1 (ru)	2006-06-30
AP2006003486A0 (en)	2006-02-28
DE602004008303T2 (de)	2008-05-08
DK1658292T3 (da)	2007-11-12
US20090036471A1 (en)	2009-02-05
US7560458B2 (en)	2009-07-14
PT1658292E (pt)	2007-10-25
NZ545058A (en)	2008-05-30
EP1658292A1 (en)	2006-05-24
KR20060120393A (ko)	2006-11-27
DE602004008303D1 (de)	2007-09-27
AR045698A1 (es)	2005-11-09
WO2005012307A1 (en)	2005-02-10
CN1823068A (zh)	2006-08-23
IL173139A (en)	2010-04-29
AU2004260738B2 (en)	2009-07-16
JP2009514782A (ja)	2009-04-09
EP1658292B1 (en)	2007-08-15
IL173139A0 (en)	2006-06-11
ATE370142T1 (de)	2007-09-15
JO2460B1 (en)	2009-01-20
CN100404536C (zh)	2008-07-23
PL1658292T3 (pl)	2008-01-31
NO20060678L (no)	2006-02-10

Publication	Publication Date	Title
ES2290754T3 (es)	2008-02-16	Derivados de triazolopirimidina como inhibidores de la glucogeno sintasa cinasa 3.
ES2317031T3 (es)	2009-04-16	Derivados de triazolopirimidina como inhibidores de la glucogeno-sintasa-quinasa 3.
ES2588238T3 (es)	2016-10-31	Derivados de pirazolopirimidin-4,6-diona y su uso como producto farmacéutico
JP6473133B2 (ja)	2019-02-20	Ｋｒａｓｇ１２ｃの共有結合性阻害剤
CN101970444A (zh)	2011-02-09	有机化合物
BRPI0910690B1 (pt)	2020-10-20	derivados de 1-heterociclil-1,5-di-hidro-pirazolo[3,4-d]pirimidin-4-ona
AU2014400628A1 (en)	2017-01-19	Aminopyridazinone compounds as protein kinase inhibitors
EP4061817A1 (en)	2022-09-28	Adenosine receptor antagonist compounds
CN119403803A (zh)	2025-02-07	Parg抑制剂
CN105916858B (zh)	2018-09-14	稠合咪唑基衍生物、其制备和作为药物的用途
US20100160349A1 (en)	2010-06-24	Triazolopyrimidine derivatives as glycogen synthase kinase 3 inhibitors
AU2004260739B2 (en)	2010-02-11	Triazolopyrimidine derivatives as glycogen synthase kinase 3 inhibitors
HK1155905A (en)	2012-06-01	Organic compounds