ES2916998T3 - Análogos del EGF(A) con sustituyentes de ácidos grasos - Google Patents

Análogos del EGF(A) con sustituyentes de ácidos grasos Download PDF

Info

Publication number: ES2916998T3
Authority: ES; Spain
Prior art keywords: ethoxy; peptide; egf; amino; acetyl
Prior art date: 2016-01-13
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Active

Application number

ES17701078T

Other languages

English (en)

Spanish (es)

Inventor

Jianhe Chen

Jesper F Lau

János Tibor Kodra

Birgit Wieczorek

Lars Linderoth

Henning Thøgersen

Salka Elbøl Rasmussen

Patrick William Garibay

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Novo Nordisk AS

Original Assignee

Novo Nordisk AS

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2016-01-13

Filing date

2017-01-13

Publication date

2022-07-06

2017-01-13 Application filed by Novo Nordisk AS filed Critical Novo Nordisk AS

2022-07-06 Application granted granted Critical

2022-07-06 Publication of ES2916998T3 publication Critical patent/ES2916998T3/es

Status Active legal-status Critical Current

2037-01-13 Anticipated expiration legal-status Critical

Links

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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- A61K38/177—Receptors; Cell surface antigens; Cell surface determinants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/475—Growth factors; Growth regulators
- C07K14/485—Epidermal growth factor [EGF], i.e. urogastrone
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/705—Receptors; Cell surface antigens; Cell surface determinants

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ES17701078T 2016-01-13 2017-01-13 Análogos del EGF(A) con sustituyentes de ácidos grasos Active ES2916998T3 (es)

Applications Claiming Priority (4)

Application Number	Priority Date	Filing Date	Title
CN2016070791		2016-01-13
CN2016076580		2016-03-17
EP16195965		2016-10-27
PCT/EP2017/050668 WO2017121850A1 (en)	2016-01-13	2017-01-13	Egf(a) analogues with fatty acid substituents

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ES17701078T Active ES2916998T3 (es)	2016-01-13	2017-01-13	Análogos del EGF(A) con sustituyentes de ácidos grasos

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JP (2)	JP6797926B2 (2)
KR (1)	KR102417487B1 (2)
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AU (1)	AU2017207862B2 (2)
BR (1)	BR112018013820A2 (2)
CA (1)	CA3010756A1 (2)
CL (1)	CL2018001868A1 (2)
CO (1)	CO2018007440A2 (2)
DK (1)	DK3402811T3 (2)
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HU (1)	HUE058647T2 (2)
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SI3402811T1 (sl)	2016-01-13	2022-06-30	Novo Nordisk A/S	Analogi EGF(A) z maščobnokislinskimi substituenti
CA3068956A1 (en)	2017-07-19	2019-01-24	Novo Nordisk A/S	Bifunctional compounds
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2017
- 2017-01-13 SI SI201731149T patent/SI3402811T1/sl unknown
- 2017-01-13 US US16/069,932 patent/US10822385B2/en active Active
- 2017-01-13 RS RS20220538A patent/RS63298B1/sr unknown
- 2017-01-13 PE PE2018001257A patent/PE20181376A1/es unknown
- 2017-01-13 CA CA3010756A patent/CA3010756A1/en not_active Withdrawn
- 2017-01-13 PL PL17701078T patent/PL3402811T3/pl unknown
- 2017-01-13 LT LTEPPCT/EP2017/050668T patent/LT3402811T/lt unknown
- 2017-01-13 BR BR112018013820-7A patent/BR112018013820A2/pt not_active Application Discontinuation
- 2017-01-13 JP JP2018536444A patent/JP6797926B2/ja active Active
- 2017-01-13 DK DK17701078.2T patent/DK3402811T3/da active
- 2017-01-13 RU RU2018127882A patent/RU2747877C2/ru active
- 2017-01-13 MY MYPI2018702319A patent/MY195199A/en unknown
- 2017-01-13 HU HUE17701078A patent/HUE058647T2/hu unknown
- 2017-01-13 WO PCT/EP2017/050668 patent/WO2017121850A1/en not_active Ceased
- 2017-01-13 ES ES17701078T patent/ES2916998T3/es active Active
- 2017-01-13 MX MX2018008681A patent/MX2018008681A/es unknown
- 2017-01-13 KR KR1020187022105A patent/KR102417487B1/ko not_active Expired - Fee Related
- 2017-01-13 HR HRP20220720TT patent/HRP20220720T1/hr unknown
- 2017-01-13 EP EP17701078.2A patent/EP3402811B1/en active Active
- 2017-01-13 CN CN201780006783.6A patent/CN108473550B/zh active Active
- 2017-01-13 AU AU2017207862A patent/AU2017207862B2/en not_active Ceased
2018
- 2018-06-14 IL IL260043A patent/IL260043A/en unknown
- 2018-07-09 CL CL2018001868A patent/CL2018001868A1/es unknown
- 2018-07-10 SA SA518391996A patent/SA518391996B1/ar unknown
- 2018-07-12 PH PH12018501502A patent/PH12018501502A1/en unknown
- 2018-07-16 CO CONC2018/0007440A patent/CO2018007440A2/es unknown
2020
- 2020-09-17 US US17/024,264 patent/US20200407409A1/en not_active Abandoned
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Also Published As

Publication number	Publication date
CN108473550A (zh)	2018-08-31
AU2017207862A1 (en)	2018-07-05
DK3402811T3 (da)	2022-06-13
US20200407409A1 (en)	2020-12-31
JP6797926B2 (ja)	2020-12-09
PE20181376A1 (es)	2018-09-05
WO2017121850A1 (en)	2017-07-20
PL3402811T3 (pl)	2022-07-11
EP3402811A1 (en)	2018-11-21
JP2019505521A (ja)	2019-02-28
EP3402811B1 (en)	2022-03-30
KR20180100177A (ko)	2018-09-07
RS63298B1 (sr)	2022-07-29
CN108473550B (zh)	2022-11-22
PH12018501502A1 (en)	2019-03-25
US10822385B2 (en)	2020-11-03
US20190016768A1 (en)	2019-01-17
MY195199A (en)	2023-01-11
KR102417487B1 (ko)	2022-07-06
CO2018007440A2 (es)	2018-09-28
RU2018127882A3 (2)	2020-06-19
IL260043A (en)	2018-07-31
RU2018127882A (ru)	2020-02-13
MX2018008681A (es)	2018-09-17
SI3402811T1 (sl)	2022-06-30
SA518391996B1 (ar)	2021-07-14
HRP20220720T1 (hr)	2022-09-30
LT3402811T (lt)	2022-06-10
HUE058647T2 (hu)	2022-09-28
CA3010756A1 (en)	2017-07-20
BR112018013820A2 (pt)	2018-12-11
RU2747877C2 (ru)	2021-05-17
CL2018001868A1 (es)	2018-08-31
AU2017207862B2 (en)	2020-12-17
JP2021035989A (ja)	2021-03-04

Publication	Publication Date	Title
ES2916998T3 (es)	2022-07-06	Análogos del EGF(A) con sustituyentes de ácidos grasos
ES2625735T3 (es)	2017-07-20	Análogos y derivados de GLP-1
ES2674946T3 (es)	2018-07-05	Análogos de glucagón que muestran actividad de receptor de GIP
EA020326B1 (ru)	2014-10-30	Агонисты смешанного действия на основе глюкозозависимого инсулинотропного пептида для лечения нарушений обмена веществ и ожирения
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TW202028229A (zh)	2020-08-01	包含胰島素肽及ｅｇｆ（ａ）肽之雙功能化合物
CA2792663A1 (en)	2011-09-29	Novel glucagon analogues
CN104411322B (zh)	2017-05-24	双酰化glp‑1衍生物
EA019203B1 (ru)	2014-01-30	Коагонисты глюкагонового рецептора/glp-1-рецептора
KR20230104118A (ko)	2023-07-07	Glp-1 전구약물 및 이의 용도
JP2018505146A (ja)	2018-02-22	Ｆｇｆ２１誘導体及びその使用
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US20200165313A1 (en)	2020-05-28	Egf(a) analogues, preparation, formulations and uses thereof
KR20210126088A (ko)	2021-10-19	지속성 glp-2 유사체
HK1262866B (en)	2022-07-22	Egf(a) analogues with fatty acid substituents
CA3195872A1 (en)	2022-05-12	Glp-1 prodrugs and uses hereof
JP2026031900A (ja)	2026-02-25	Ｆｃ－アシル化ポリペプチドコンジュゲート