ID16520A - Pirimido (1,2-a)indol baru - Google Patents

Pirimido (1,2-a)indol baru

Info

Publication number
ID16520A
ID16520A IDP971112A ID971112A ID16520A ID 16520 A ID16520 A ID 16520A ID P971112 A IDP971112 A ID P971112A ID 971112 A ID971112 A ID 971112A ID 16520 A ID16520 A ID 16520A
Authority
ID
Indonesia
Prior art keywords
pirimido
new indol
indol
new
Prior art date
Application number
IDP971112A
Other languages
English (en)
Indonesian (id)
Inventor
D Ulrich Muller
Peter Dr Eckenberg
Rudi Dr Grutzmann
Hilmar Dr Bischoff
Dirk Dr Denzer
Stefan Dr Lohmer
Ulrich Dr Nielsch
Peter Dr Kolkhof
Stefan Dr Wohlfeil
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ag filed Critical Bayer Ag
Publication of ID16520A publication Critical patent/ID16520A/id

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
IDP971112A 1996-04-04 1997-04-02 Pirimido (1,2-a)indol baru ID16520A (id)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19613550A DE19613550A1 (de) 1996-04-04 1996-04-04 Neue Pyrimido[1,2-a]indole

Publications (1)

Publication Number Publication Date
ID16520A true ID16520A (id) 1997-10-09

Family

ID=7790502

Family Applications (1)

Application Number Title Priority Date Filing Date
IDP971112A ID16520A (id) 1996-04-04 1997-04-02 Pirimido (1,2-a)indol baru

Country Status (33)

Country Link
US (1) US6114341A (fr)
EP (1) EP0799828A3 (fr)
JP (1) JPH1059972A (fr)
KR (1) KR970070008A (fr)
CN (2) CN1067393C (fr)
AR (1) AR006497A1 (fr)
AU (1) AU725786B2 (fr)
BG (1) BG62934B1 (fr)
BR (1) BR9701675A (fr)
CA (1) CA2201434A1 (fr)
CO (1) CO4520306A1 (fr)
CZ (1) CZ102297A3 (fr)
DE (1) DE19613550A1 (fr)
DZ (1) DZ2201A1 (fr)
EE (1) EE9700078A (fr)
HN (1) HN1997000045A (fr)
HR (1) HRP970154A2 (fr)
HU (1) HUP9700708A3 (fr)
ID (1) ID16520A (fr)
IL (3) IL120590A (fr)
MA (1) MA24131A1 (fr)
MY (1) MY126362A (fr)
NO (1) NO309092B1 (fr)
NZ (1) NZ314497A (fr)
PE (1) PE42398A1 (fr)
PL (1) PL319249A1 (fr)
SG (1) SG63698A1 (fr)
SK (1) SK42797A3 (fr)
SV (1) SV1997000025A (fr)
TN (1) TNSN97061A1 (fr)
TR (1) TR199700261A2 (fr)
YU (1) YU12397A (fr)
ZA (1) ZA972829B (fr)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE19826469A1 (de) * 1998-06-13 2000-05-25 Bayer Ag Verfahren zur Herstellung von 2,4-Dimethylcarbolin und 2,4-Dimethylpyrimido[1,2-a]indol
AU2001244635A1 (en) * 2000-03-30 2001-10-15 Yamanouchi Pharmaceutical Co..Ltd. Hydrazide derivatives
DE10030375A1 (de) * 2000-06-21 2002-01-03 Bayer Ag Verwendung von MTP-Inhibitoren zur Senkung von ppTRL
JP4254093B2 (ja) * 2001-10-17 2009-04-15 宇部興産株式会社 5−ハロゲノインドールの製法
DE10349175A1 (de) * 2003-10-22 2005-05-19 Bayer Healthcare Ag Mittel zur Gewichtsreduktion
PT1725234E (pt) 2004-03-05 2013-03-04 Univ Pennsylvania Métodos com efeitos secundários reduzidos para tratamento de patologias ou doenças associadas a hiperlipidemia e hipercolesterolemia
EP1737460A2 (fr) * 2004-04-09 2007-01-03 Janssen Pharmaceutica N.V. Mode d'administration intermittent pour le traitement de l'obésité avec des inhibiteurs de mtp
MX2007013932A (es) 2005-05-12 2008-01-28 Bard Inc C R Filtro de coagulo de sangre removible.
WO2006129193A2 (fr) * 2005-05-27 2006-12-07 Pfizer Products Inc. Polytherapie pour le traitement de l'obesite ou le maintien du poids apres une perte ponderale
US8062327B2 (en) 2005-08-09 2011-11-22 C. R. Bard, Inc. Embolus blood clot filter and delivery system
EP1951220A2 (fr) * 2005-10-18 2008-08-06 Aegerion Pharmaceuticals Compositions destinees a l'abbaissement du cholesterol serique et/ou des triglycerides
WO2007133366A2 (fr) 2006-05-02 2007-11-22 C. R. Bard, Inc. Filtre à veine cave formé à partir d'une feuille
JP2010513534A (ja) * 2006-12-21 2010-04-30 エージェリオン ファーマシューティカルズ, インコーポレイテッド Mtpインヒビターおよびコレステロール吸収インヒビターを含む組み合わせを用いて肥満症を処置する方法
BR112023000808A2 (pt) 2020-07-29 2023-02-07 Amryt Pharmaceuticals Inc Lomitapida para uso em métodos para tratar hiperlipidemia e hipercolesterolemia em pacientes pediátricos

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2200584A1 (de) * 1971-01-11 1972-07-27 Wyeth John & Brother Ltd Heterocyclische Verbindungen,Verfahren zu ihrer Herstellung und ihre Verwendung in pharmazeutischen Zubereitungen
ZA718536B (en) * 1971-01-11 1972-09-27 Wyeth John & Brother Ltd Heterocyclic compounds
GB8614246D0 (en) * 1986-06-11 1986-07-16 Wyeth John & Brother Ltd Substituted pyrimidoindoles
DE4112533A1 (de) * 1991-04-17 1992-10-22 Bayer Ag Verfahren zur herstellung von enantiomerenreinen substituierten (chinolin-2-yl-methoxy)phenyl-essigsaeuren
DE4200954A1 (de) * 1991-04-26 1992-10-29 Bayer Ag Heterocyclisch substituierte phenylessigsaeurederivate
DE4208051A1 (de) * 1992-03-13 1993-09-16 Bayer Ag Substituierte phenylessigsaeureamide
DE4309968A1 (de) * 1993-03-26 1994-09-29 Bayer Ag Phenylglycinamide von heterocyclisch substituierten Phenylessigsäurederivaten
US5576342A (en) * 1992-03-13 1996-11-19 Bayer Aktiengesellschaft Phenylglycinamides of heterocyclically substitued phenylacetic acid derivatives
DE4208052A1 (de) * 1992-03-13 1993-09-16 Bayer Ag Imidazolyl substituierte phenylessigsaeureamide
US5705498A (en) * 1992-11-05 1998-01-06 Smithkline Beecham Plc. Piperidine derivatives as 5-HT4 receptor antagonists
DE4302956A1 (de) * 1993-02-03 1994-08-04 Bayer Ag Substituierte Imidazo(4,5-b)pyridine und Benzimidazole

Also Published As

Publication number Publication date
MA24131A1 (fr) 1997-10-01
AR006497A1 (es) 1999-08-25
EE9700078A (et) 1997-10-15
CZ102297A3 (en) 1997-10-15
MX9702445A (es) 1997-10-31
TNSN97061A1 (fr) 2005-03-15
ZA972829B (en) 1997-10-31
EP0799828A2 (fr) 1997-10-08
IL131645A0 (en) 2001-01-28
NZ314497A (en) 1999-10-28
AU1660397A (en) 1997-10-09
PL319249A1 (en) 1997-10-13
IL120590A (en) 2000-02-17
CO4520306A1 (es) 1997-10-15
PE42398A1 (es) 1998-10-12
HUP9700708A3 (en) 2000-01-28
CN1312246A (zh) 2001-09-12
MY126362A (en) 2006-09-29
NO971512L (no) 1997-10-06
CN1067393C (zh) 2001-06-20
NO971512D0 (no) 1997-04-03
SG63698A1 (en) 1999-03-30
HN1997000045A (es) 1997-06-26
NO309092B1 (no) 2000-12-11
CA2201434A1 (fr) 1997-10-04
HU9700708D0 (en) 1997-05-28
HUP9700708A2 (hu) 1998-10-28
TR199700261A2 (xx) 1997-10-21
EP0799828A3 (fr) 1998-04-08
US6114341A (en) 2000-09-05
AU725786B2 (en) 2000-10-19
KR970070008A (ko) 1997-11-07
YU12397A (en) 1999-11-22
CN1176965A (zh) 1998-03-25
DZ2201A1 (fr) 2002-12-03
IL131645A (en) 2000-12-06
DE19613550A1 (de) 1997-10-09
SV1997000025A (es) 1997-10-23
JPH1059972A (ja) 1998-03-03
BG62934B1 (bg) 2000-11-30
HRP970154A2 (en) 1998-04-30
IL120590A0 (en) 1997-08-14
BR9701675A (pt) 1998-11-03
BG101379A (en) 1997-11-28
SK42797A3 (en) 1997-11-05

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