ID21755A - Antijamur azol yang mengandung ester asam amino - Google Patents

Antijamur azol yang mengandung ester asam amino

Info

Publication number: ID21755A
Authority: ID; Indonesia
Prior art keywords: amino acid; antijamur; azol; acid esters; contains amino
Prior art date: 1997-02-11

Application number

IDW990505A

Other languages

English (en)

Inventor

Lieven Meerpoel

Jan Heeres

Robert Josef Maria B Hendrickx

Original Assignee

Janssen Pharmaceutica Nv

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1997-02-11

Filing date

1998-02-03

Publication date

1999-07-22

1998-02-03 Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv

1999-07-22 Publication of ID21755A publication Critical patent/ID21755A/id

Links

PLIKAWJENQZMHA-UHFFFAOYSA-N 4-aminophenol Chemical compound NC1=CC=C(O)C=C1 PLIKAWJENQZMHA-UHFFFAOYSA-N 0.000 title 1
-1 AMINO ACID ESTERS Chemical class 0.000 title 1
KAESVJOAVNADME-UHFFFAOYSA-N Pyrrole Chemical compound C=1C=CNC=1 KAESVJOAVNADME-UHFFFAOYSA-N 0.000 abstract 2
WNXJIVFYUVYPPR-UHFFFAOYSA-N 1,3-dioxolane Chemical class C1COCO1 WNXJIVFYUVYPPR-UHFFFAOYSA-N 0.000 abstract 1
125000000815 N-oxide group Chemical group 0.000 abstract 1
125000002252 acyl group Chemical group 0.000 abstract 1
150000001413 amino acids Chemical class 0.000 abstract 1
229940121375 antifungal agent Drugs 0.000 abstract 1
150000001875 compounds Chemical class 0.000 abstract 1
239000003814 drug Substances 0.000 abstract 1
239000000203 mixture Substances 0.000 abstract 1
150000003839 salts Chemical class 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/10—Antimycotics
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Public Health (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Oncology (AREA)
Communicable Diseases (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Dermatology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Agricultural Chemicals And Associated Chemicals (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

IDW990505A 1997-02-11 1998-02-03 Antijamur azol yang mengandung ester asam amino ID21755A (id)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
EP97200374		1997-02-11
EP97203228		1997-10-15

Publications (1)

Publication Number	Publication Date
ID21755A true ID21755A (id)	1999-07-22

Family

ID=26146124

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
IDW990505A ID21755A (id)	1997-02-11	1998-02-03	Antijamur azol yang mengandung ester asam amino

Country Status (31)

Country	Link
US (3)	US6262052B1 (id)
EP (1)	EP0958289B1 (id)
JP (1)	JP4347911B2 (id)
KR (1)	KR100509171B1 (id)
CN (1)	CN1238353C (id)
AT (1)	ATE270290T1 (id)
AU (1)	AU725302C (id)
BG (1)	BG63872B1 (id)
BR (1)	BR9809744A (id)
CA (1)	CA2262791C (id)
CZ (1)	CZ297197B6 (id)
DE (1)	DE69824834T2 (id)
DK (1)	DK0958289T3 (id)
EE (1)	EE03876B1 (id)
ES (1)	ES2224364T3 (id)
HU (1)	HU227744B1 (id)
ID (1)	ID21755A (id)
IL (2)	IL128513A (id)
MY (1)	MY129537A (id)
NO (1)	NO316668B1 (id)
NZ (1)	NZ334477A (id)
PL (1)	PL191152B1 (id)
PT (1)	PT958289E (id)
RU (1)	RU2197489C2 (id)
SI (1)	SI0958289T1 (id)
SK (1)	SK284910B6 (id)
TR (1)	TR199900584T2 (id)
TW (1)	TW495508B (id)
UA (1)	UA61919C2 (id)
WO (1)	WO1998034934A1 (id)
ZA (1)	ZA981079B (id)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
EP0957101A1 (en)	1998-05-14	1999-11-17	Janssen Pharmaceutica N.V.	Water soluble azoles as broad-spectrum antifungals
AU1915500A (en)	1998-11-20	2000-06-13	Bristol-Myers Squibb Company	Water soluble prodrugs of azole compounds
ES2194723T3 (es)	1999-05-04	2003-12-01	Janssen Pharmaceutica Nv	Eteres antifungicos.
WO2003052117A2 (en) *	2001-09-19	2003-06-26	Massachusetts Institute Of Technology	Methods and products related to non-viral transfection
ITMI20032020A1 (it)	2003-10-17	2005-04-18	Italfarmaco Spa	Nuovi agenti antifungini azolici con diminuita interazione con i citocromi metabolici
EP2571871B1 (en) *	2010-05-19	2017-06-21	Sandoz AG	Process for the preparation of chiral triazolones
US20170290333A1 (en)	2014-12-30	2017-10-12	Dow Agrosciences Llc	Picolinamide compounds with fungicidal activity
BR102019004480B1 (pt) *	2018-03-08	2023-03-28	Dow Agrosciences Llc	Picolinamidas como fungicidas
CN111138421A (zh) *	2019-12-26	2020-05-12	上海英诺富成生物科技有限公司	抗真菌水溶性化合物及其制备方法与应用

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4267179A (en)	1978-06-23	1981-05-12	Janssen Pharmaceutica, N.V.	Heterocyclic derivatives of (4-phenylpiperazin-1-yl-aryloxymethyl-1,3-dioxolan-2-yl)methyl-1H-imidazoles and 1H-1,2,4-triazoles
US4791111A (en) *	1985-12-23	1988-12-13	Janssen Pharmaceutica, N.V.	[[4-[4-(4-phenyl-1-piperazinyl)phenoxymethyl]-1,3-dioxolan-2-yl]methyl]-1H-imidazoles and 1H-1,2,4-triazoles having anti-microbial properties
US4916134A (en)	1987-03-25	1990-04-10	Janssen Pharmacuetica N.V.	4-[4-[4-[4-[[2-(2,4-difluorophenyl)-2-(1H-azolylmethyl)-1,3-dioxolan-4-yl]me]phenyl]-1-piperazinyl]phenyl]triazolones
CA1331757C (en)	1988-02-29	1994-08-30	Janssen Pharmaceutica Naamloze Vennootschap	5-lipoxygenase inhibiting 4-(4-phenyl-1-piperazinyl)phenols
NZ233502A (en) *	1989-06-09	1991-11-26	Janssen Pharmaceutica Nv	4-(1,2,4-triazole- or imidazole-phenyl-substituted) -1-(1,3-dioxolan-4-ylmethoxyphenyl) piperazine derivatives; preparatory processes: fungicidal and antiviral compositions
HU221189B1 (en)	1992-03-18	2002-08-28	Janssen Pharmaceutica Nv	Itraconazole and saperconazole stereoisomers, their cyclodextrin complexes and pharmaceutical compositions containing them and process for producing them
PL181193B1 (pl)	1993-12-21	2001-06-29	Schering Corp	Nowe pochodne tetrahydrofuranowe o działaniu przeciwgrzybicznym, kompozycja farmaceutyczna do leczenia infekcji grzybiczych oraz sposób wytwarzania tych związków
NZ278882A (en) *	1994-01-24	1997-06-24	Janssen Pharmaceutica Nv	Piperazine-containing azole antifungal compounds
SK27097A3 (en) *	1995-06-02	1997-09-10	Schering Corp	Tetrahydrofuran antifungals
CA2224707A1 (en) *	1995-06-19	1997-01-03	Schering Corporation	Tetrahydrofuran antifungals

1998
- 1998-02-03 AU AU66207/98A patent/AU725302C/en not_active Expired
- 1998-02-03 SK SK1059-99A patent/SK284910B6/sk not_active IP Right Cessation
- 1998-02-03 NZ NZ334477A patent/NZ334477A/en not_active IP Right Cessation
- 1998-02-03 DK DK98908064T patent/DK0958289T3/da active
- 1998-02-03 DE DE69824834T patent/DE69824834T2/de not_active Expired - Lifetime
- 1998-02-03 JP JP53376398A patent/JP4347911B2/ja not_active Expired - Lifetime
- 1998-02-03 PT PT98908064T patent/PT958289E/pt unknown
- 1998-02-03 CN CNB988011352A patent/CN1238353C/zh not_active Expired - Lifetime
- 1998-02-03 EP EP98908064A patent/EP0958289B1/en not_active Expired - Lifetime
- 1998-02-03 SI SI9830687T patent/SI0958289T1/xx unknown
- 1998-02-03 HU HU0001050A patent/HU227744B1/hu unknown
- 1998-02-03 US US09/355,369 patent/US6262052B1/en not_active Expired - Lifetime
- 1998-02-03 ES ES98908064T patent/ES2224364T3/es not_active Expired - Lifetime
- 1998-02-03 BR BR9809744-0A patent/BR9809744A/pt not_active Application Discontinuation
- 1998-02-03 ID IDW990505A patent/ID21755A/id unknown
- 1998-02-03 WO PCT/EP1998/000646 patent/WO1998034934A1/en not_active Ceased
- 1998-02-03 IL IL12851398A patent/IL128513A/en not_active IP Right Cessation
- 1998-02-03 RU RU99106585/04A patent/RU2197489C2/ru active
- 1998-02-03 PL PL332008A patent/PL191152B1/pl unknown
- 1998-02-03 KR KR10-1999-7001983A patent/KR100509171B1/ko not_active Expired - Lifetime
- 1998-02-03 TR TR1999/00584T patent/TR199900584T2/xx unknown
- 1998-02-03 CZ CZ0283599A patent/CZ297197B6/cs not_active IP Right Cessation
- 1998-02-03 CA CA002262791A patent/CA2262791C/en not_active Expired - Lifetime
- 1998-02-03 EE EEP199900100A patent/EE03876B1/xx unknown
- 1998-02-03 AT AT98908064T patent/ATE270290T1/de active
- 1998-02-09 MY MYPI98000513A patent/MY129537A/en unknown
- 1998-02-09 TW TW087101662A patent/TW495508B/zh not_active IP Right Cessation
- 1998-02-10 ZA ZA9801079A patent/ZA981079B/xx unknown
- 1998-03-02 UA UA99020835A patent/UA61919C2/uk unknown
1999
- 1999-02-02 NO NO19990484A patent/NO316668B1/no not_active IP Right Cessation
- 1999-02-11 BG BG103171A patent/BG63872B1/bg unknown
2001
- 2001-05-04 US US09/848,989 patent/US6512116B2/en not_active Expired - Lifetime
2002
- 2002-04-23 IL IL149285A patent/IL149285A/en not_active IP Right Cessation
- 2002-11-15 US US10/298,038 patent/US6703506B2/en not_active Expired - Lifetime

Also Published As

Publication number	Publication date
US20030158210A1 (en)	2003-08-21
PL191152B1 (pl)	2006-03-31
AU725302B2 (en)	2000-10-12
IL149285A0 (en)	2002-11-10
BG103171A (en)	1999-09-30
PL332008A1 (en)	1999-08-16
IL149285A (en)	2007-08-19
US6703506B2 (en)	2004-03-09
ES2224364T3 (es)	2005-03-01
CA2262791A1 (en)	1998-08-13
BR9809744A (pt)	2000-06-20
US20010039281A1 (en)	2001-11-08
UA61919C2 (uk)	2003-12-15
JP4347911B2 (ja)	2009-10-21
SK105999A3 (en)	2000-06-12
HUP0001050A2 (hu)	2001-04-28
CN1236366A (zh)	1999-11-24
RU2197489C2 (ru)	2003-01-27
DK0958289T3 (da)	2004-11-01
EP0958289A1 (en)	1999-11-24
TW495508B (en)	2002-07-21
CZ283599A3 (cs)	2000-02-16
SK284910B6 (sk)	2006-02-02
DE69824834D1 (de)	2004-08-05
US6262052B1 (en)	2001-07-17
NO316668B1 (no)	2004-03-29
ZA981079B (en)	1999-08-10
DE69824834T2 (de)	2005-07-21
NZ334477A (en)	2001-05-25
AU6620798A (en)	1998-08-26
CN1238353C (zh)	2006-01-25
NO990484L (no)	1999-10-11
BG63872B1 (bg)	2003-04-30
IL128513A0 (en)	2000-01-31
KR20000068526A (ko)	2000-11-25
CA2262791C (en)	2008-10-28
HU227744B1 (en)	2012-02-28
CZ297197B6 (cs)	2006-09-13
JP2001508080A (ja)	2001-06-19
NO990484D0 (no)	1999-02-02
MY129537A (en)	2007-04-30
PT958289E (pt)	2004-11-30
EP0958289B1 (en)	2004-06-30
IL128513A (en)	2002-11-10
EE9900100A (et)	1999-10-15
SI0958289T1 (en)	2004-12-31
EE03876B1 (et)	2002-10-15
TR199900584T2 (xx)	1999-10-21
WO1998034934A1 (en)	1998-08-13
HUP0001050A3 (en)	2001-07-30
AU725302C (en)	2001-08-23
US6512116B2 (en)	2003-01-28
ATE270290T1 (de)	2004-07-15
KR100509171B1 (ko)	2005-08-22

Publication	Publication Date	Title
BG60102B2 (bg)	1993-10-29	Метод за получаване на 5-флуор-2(((4-циклопропил- метокси-2-пиридинил)метил)тионил)-1н-бензимидазол
RU95108387A (ru)	1996-12-10	Дикетопиперазин, способ его получения, фармацевтическая композиция, применение дикетопиперазина
RU95101048A (ru)	1996-10-27	Производные пролинамида, фармкомпозиция на их основе
PT948527E (pt)	2002-11-29	Novos derivados de ciclosporina sua preparacao e composicoes farmaceuticas que os contem
ATE260658T1 (de)	2004-03-15	Pharmazeutische zubereitungen zur verminderung von atmungsdepressionen
AU8985391A (en)	1992-07-02	Trifluoromethylketone derivatives, processes for preparation thereof and use thereof
SE0102055D0 (sv)	2001-06-08	New Compounds
PT958289E (pt)	2004-11-30	Ester de amino acidos contendo antifungicos de azol
AU5879798A (en)	1998-09-08	Agents inhibiting progress of pterygium and postoperative recurrence of the same
NZ332655A (en)	2000-04-28	Pharmaceutical compositions containing diclofenac and alkali metal bicarbonates
DE69330601D1 (de)	2001-09-20	Serotoninergische ergolin derivate
RU95113437A (ru)	1997-02-20	(h±)-сложный этиловый эфир транс-2-диметиламино-1-фенил-3-циклогексентранс-1-карбоновой кислоты в виде первичного ортофосфата и твердая фармацевтическая композиция с обезболивающей активностью
AR002264A1 (es)	1998-03-11	6-[triazolil[3(trifluormetil)fenil]metil]-2-quinolinonas y quinolintionas, un procedimiento para su preparacion, una composicion que las comprende, unprocedimiento para su preparacion, el uso de las mismas para la preparacion de un medicamento y un intermediario.
RU94040865A (ru)	1996-08-10	Производные пептида и их терапевтически приемлемые соли, способ их получения, фармацевтическая и косметическая композиция с антивирусной активностью
ES2094608T3 (es)	1997-01-16	Mezclas fungicidas.
IL111138A (en)	1997-04-15	Pharmaceutical compositions comprising penciclovir and/or its bioprecursor and/or its derivatives for the treatment and prophylaxis of post-herpetic neuralgia
ATE268768T1 (de)	2004-06-15	Antithrombosemittel
ES8104271A1 (es)	1981-04-16	Procedimiento para la preparacion de 5-(2-((3-(1,3-benzodio-sol-5-il)-1-metilpropil)amino)-1-hidroxietil-2-metoxibenza- mida y de sus sales e isomeros opticos farmaceuticamente aceptables
YU47871B (sh)	1996-02-19	Derivati aminokiselina
NO931091L (no)	1993-03-24	Analoger av sykloinopeptid a og anvendelse derav