IL100576A - Cephalosporin antibiotics - Google Patents

Cephalosporin antibiotics

Info

Publication number
IL100576A
IL100576A IL10057692A IL10057692A IL100576A IL 100576 A IL100576 A IL 100576A IL 10057692 A IL10057692 A IL 10057692A IL 10057692 A IL10057692 A IL 10057692A IL 100576 A IL100576 A IL 100576A
Authority
IL
Israel
Prior art keywords
amino
compound
group
formula
alkyl
Prior art date
Application number
IL10057692A
Other languages
English (en)
Other versions
IL100576A0 (en
Original Assignee
Eli Lilley And Company
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Eli Lilley And Company filed Critical Eli Lilley And Company
Publication of IL100576A0 publication Critical patent/IL100576A0/xx
Publication of IL100576A publication Critical patent/IL100576A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14—Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/59—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3 with hetero atoms directly attached in position 3
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cephalosporin Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Materials For Medical Uses (AREA)
  • Jellies, Jams, And Syrups (AREA)
  • Food Preservation Except Freezing, Refrigeration, And Drying (AREA)
IL10057692A 1991-01-18 1992-01-01 Cephalosporin antibiotics IL100576A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US64295991A 1991-01-18 1991-01-18

Publications (2)

Publication Number Publication Date
IL100576A0 IL100576A0 (en) 1992-09-06
IL100576A true IL100576A (en) 1995-11-27

Family

ID=24578768

Family Applications (1)

Application Number Title Priority Date Filing Date
IL10057692A IL100576A (en) 1991-01-18 1992-01-01 Cephalosporin antibiotics

Country Status (23)

Country Link
US (1) US5362722A (cs)
EP (1) EP0495584B1 (cs)
JP (1) JP3164390B2 (cs)
KR (1) KR920014818A (cs)
CN (1) CN1063286A (cs)
AT (1) ATE187729T1 (cs)
AU (1) AU642333B2 (cs)
BR (1) BR9200057A (cs)
CA (1) CA2058822C (cs)
CZ (1) CZ281684B6 (cs)
DE (1) DE69230415T2 (cs)
ES (1) ES2141096T3 (cs)
FI (1) FI920111A7 (cs)
HU (1) HUT60276A (cs)
IE (1) IE920085A1 (cs)
IL (1) IL100576A (cs)
MX (1) MX9200102A (cs)
NO (1) NO301330B1 (cs)
NZ (1) NZ241249A (cs)
PT (1) PT99983B (cs)
RU (1) RU2104280C1 (cs)
YU (1) YU2292A (cs)
ZA (1) ZA9224B (cs)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5077287A (en) * 1991-01-18 1991-12-31 Eli Lilly And Company 3-thiazolylthio carbacephem antibacterial agents
JPH05132488A (ja) * 1991-08-13 1993-05-28 Meiji Seika Kaisha Ltd 新規セフアロスポリン誘導体
JP2857532B2 (ja) * 1992-03-12 1999-02-17 明治製菓株式会社 新規セファロスポリン誘導体
US5525599A (en) * 1993-07-21 1996-06-11 Eli Lilly And Company 7-substituted-amino-3-substituted-3-cephem-4-carboxylic acids
US5496816A (en) * 1994-03-14 1996-03-05 Merck & Co., Inc. Carbapenem antibacterial compounds, compositions containing such compounds and methods of treatment
US5498777A (en) * 1994-07-20 1996-03-12 Merck & Co., Inc. 3-thioheteroaryl cephalosporin compounds, compositions and methods of use
TWI288745B (en) 2000-04-05 2007-10-21 Daiichi Seiyaku Co Ethylenediamine derivatives
US6599893B2 (en) * 2000-08-29 2003-07-29 Essential Therapeutics, Inc. Cephalosporin antibiotics and prodrugs thereof
US7365205B2 (en) 2001-06-20 2008-04-29 Daiichi Sankyo Company, Limited Diamine derivatives
RU2319699C2 (ru) 2001-06-20 2008-03-20 Дайити Санкио Компани, Лимитед Производные диаминов

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5214789A (en) * 1975-07-22 1977-02-03 Shionogi & Co Ltd Process for preparing 3-substiuted cephem compounds by ring closure
ZA766941B (en) * 1975-11-21 1978-06-28 Merck & Co Inc 3-(substituted thio)cephalosporins,derivatives and nuclear analogues thereof
EP0009008A3 (de) * 1978-09-08 1980-05-14 Ciba-Geigy Ag Cephalosporinderivate, Verfahren zu ihrer Herstellung und diese enthaltende pharmazeutische Präparate
US4500526A (en) * 1982-06-28 1985-02-19 Bristol-Myers Company Cephalosporin derivatives
GB8410992D0 (en) * 1984-04-30 1984-06-06 Glaxo Group Ltd Process
JPH0653739B2 (ja) * 1984-11-15 1994-07-20 協和醗酵工業株式会社 ３位置換カルバセフエム化合物
GB2177691A (en) * 1985-07-18 1987-01-28 Glaxo Group Ltd Cephalosporin antibiotics
US5142039A (en) * 1987-07-31 1992-08-25 Eli Lilly And Company β-lactam antibiotics
JP2568248B2 (ja) * 1988-04-22 1996-12-25 第一製薬株式会社 ３−セフェム−４−カルボン酸
DE69028285T2 (de) * 1989-12-07 1997-03-20 Meiji Seika Kaisha Cephalosporinderivate, ihre Herstellung und Anwendungen
JPH0686459B2 (ja) * 1989-12-07 1994-11-02 明治製菓株式会社 ３―置換チオ―３―セフエム化合物の製造法
IE65926B1 (en) * 1990-07-19 1995-11-29 Shionogi & Co Thioalkylthio cephalosporin derivatives
US5077287A (en) * 1991-01-18 1991-12-31 Eli Lilly And Company 3-thiazolylthio carbacephem antibacterial agents
US5247073A (en) * 1991-01-18 1993-09-21 Eli Lilly And Company 7-(Amino or protected amino)-3-thioheterobicyclic cephalosporins
JPH05132488A (ja) * 1991-08-13 1993-05-28 Meiji Seika Kaisha Ltd 新規セフアロスポリン誘導体
JPH09109037A (ja) * 1995-10-23 1997-04-28 Denso Corp スライド機能付き締付け装置

Also Published As

Publication number Publication date
ZA9224B (en) 1993-07-02
NO301330B1 (no) 1997-10-13
CZ281684B6 (cs) 1996-12-11
JPH04321691A (ja) 1992-11-11
FI920111L (fi) 1992-07-19
HU9200082D0 (en) 1992-03-30
EP0495584B1 (en) 1999-12-15
KR920014818A (ko) 1992-08-25
CS1292A3 (en) 1992-08-12
JP3164390B2 (ja) 2001-05-08
EP0495584A2 (en) 1992-07-22
IE920085A1 (en) 1992-07-29
CN1063286A (zh) 1992-08-05
PT99983A (pt) 1993-01-29
AU642333B2 (en) 1993-10-14
CA2058822C (en) 2000-06-27
FI920111A0 (fi) 1992-01-10
NZ241249A (en) 1993-04-28
AU1013492A (en) 1992-07-23
CA2058822A1 (en) 1992-07-19
MX9200102A (es) 1992-07-01
FI920111A7 (fi) 1992-07-19
DE69230415T2 (de) 2000-05-11
DE69230415D1 (de) 2000-01-20
HUT60276A (en) 1992-08-28
EP0495584A3 (en) 1992-11-04
ES2141096T3 (es) 2000-03-16
RU2104280C1 (ru) 1998-02-10
PT99983B (pt) 1999-06-30
US5362722A (en) 1994-11-08
BR9200057A (pt) 1992-09-08
ATE187729T1 (de) 2000-01-15
NO920102D0 (no) 1992-01-08
YU2292A (sh) 1994-11-15
NO920102L (no) 1992-07-20
IL100576A0 (en) 1992-09-06

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Legal Events

Date Code Title Description
FF Patent granted
RH Patent void