IS5053A - 6-Fenýlpýridýl-2-amín afleiður nytsamlegar sem nituroxíð sýntasa tálmar - Google Patents

6-Fenýlpýridýl-2-amín afleiður nytsamlegar sem nituroxíð sýntasa tálmar

Info

Publication number: IS5053A
Authority: IS; Iceland
Prior art keywords: phenylpyridyl; nitric oxide; oxide synthase; amine derivatives; synthase inhibitors
Prior art date: 1996-12-06

Application number

IS5053A

Other languages

English (en)

Inventor

Adams Lowe John Iii

Original Assignee

Pfizer Inc.

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1996-12-06

Filing date

1999-05-18

Publication date

1999-05-18

1999-05-18 Application filed by Pfizer Inc. filed Critical Pfizer Inc.

1999-05-18 Publication of IS5053A publication Critical patent/IS5053A/is

Links

239000000236 nitric oxide synthase inhibitor Substances 0.000 title 1
CSYSULGPHGCBQD-UHFFFAOYSA-N s-ethylisothiouronium diethylphosphate Chemical compound CCSC(N)=N.CCOP(O)(=O)OCC CSYSULGPHGCBQD-UHFFFAOYSA-N 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/72—Nitrogen atoms
- C07D213/73—Unsubstituted amino or imino radicals
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- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/10—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing aromatic rings
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

Landscapes

Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Life Sciences & Earth Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Chemical Kinetics & Catalysis (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Pain & Pain Management (AREA)
Diabetes (AREA)
Ophthalmology & Optometry (AREA)
Pulmonology (AREA)
Psychiatry (AREA)
Hematology (AREA)
Psychology (AREA)
Rheumatology (AREA)
Immunology (AREA)
Orthopedic Medicine & Surgery (AREA)
Emergency Medicine (AREA)
Heart & Thoracic Surgery (AREA)
Obesity (AREA)
Hospice & Palliative Care (AREA)
Addiction (AREA)
Endocrinology (AREA)
Physical Education & Sports Medicine (AREA)
Cardiology (AREA)
Urology & Nephrology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Pyridine Compounds (AREA)
Plural Heterocyclic Compounds (AREA)

IS5053A 1996-12-06 1999-05-18 6-Fenýlpýridýl-2-amín afleiður nytsamlegar sem nituroxíð sýntasa tálmar IS5053A (is)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US3279396P	1996-12-06	1996-12-06
PCT/IB1997/001446 WO1998024766A1 (en)	1996-12-06	1997-11-17	6-phenylpyridyl-2-amine derivatives useful as nos inhibitors

Publications (1)

Publication Number	Publication Date
IS5053A true IS5053A (is)	1999-05-18

Family

ID=21866837

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
IS5053A IS5053A (is)	1996-12-06	1999-05-18	6-Fenýlpýridýl-2-amín afleiður nytsamlegar sem nituroxíð sýntasa tálmar

Country Status (42)

Country	Link
US (3)	US6235750B1 (is)
EP (1)	EP0946512B1 (is)
JP (2)	JP3604399B2 (is)
KR (1)	KR100360633B1 (is)
CN (1)	CN1117077C (is)
AP (1)	AP848A (is)
AR (1)	AR010331A1 (is)
AT (1)	ATE251612T1 (is)
AU (2)	AU4791797A (is)
BG (1)	BG103540A (is)
BR (1)	BR9714381A (is)
CA (1)	CA2273479C (is)
CZ (1)	CZ293863B6 (is)
DE (1)	DE69725465T2 (is)
DK (1)	DK0946512T3 (is)
DZ (1)	DZ2361A1 (is)
EA (1)	EA002907B1 (is)
ES (1)	ES2206691T3 (is)
HN (2)	HN1997000027A (is)
HR (1)	HRP970664A2 (is)
HU (1)	HUP0001848A3 (is)
ID (1)	ID19056A (is)
IL (1)	IL130111A0 (is)
IS (1)	IS5053A (is)
MA (1)	MA26453A1 (is)
NO (1)	NO313517B1 (is)
NZ (1)	NZ335733A (is)
OA (1)	OA11123A (is)
PA (1)	PA8442201A1 (is)
PE (1)	PE46499A1 (is)
PL (1)	PL333918A1 (is)
PT (1)	PT946512E (is)
SI (1)	SI0946512T1 (is)
SK (1)	SK70899A3 (is)
TN (1)	TNSN97198A1 (is)
TR (1)	TR199901259T2 (is)
TW (1)	TW491840B (is)
UA (1)	UA59379C2 (is)
UY (1)	UY24799A1 (is)
WO (1)	WO1998024766A1 (is)
YU (1)	YU25399A (is)
ZA (1)	ZA9710906B (is)

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PT891332E (pt) *	1996-03-29	2004-07-30	Pfizer	Derivados de 6-fenilpiridil-2-amina
US20010049379A1 (en)	1997-08-27	2001-12-06	Lowe John Adams	2-aminopyridines containing fused ring substituents
HN1998000118A (es)	1997-08-27	1999-02-09	Pfizer Prod Inc	2 - aminopiridinas que contienen sustituyentes de anillos condensados.
HN1998000125A (es)	1997-08-28	1999-02-09	Pfizer Prod Inc	2-aminopiridinas con sustituyentes alcoxi ramificados
CA2334012C (en)	1998-06-03	2006-05-02	Pfizer Products Inc.	2-aminopyridines containing fused ring substituents as nitric oxide synthase inhibitors
FR2780971B1 (fr) *	1998-07-08	2001-09-28	Sod Conseils Rech Applic	Nouveaux derives de 2-aminopyridines, leur application en tant que medicaments et compositions pharmaceutiques les contenant
AR019190A1 (es) *	1998-07-08	2001-12-26	Sod Conseils Rech Applic	Derivados de 2-aminopiridinas, productos intermedios para su preparacion, medicamentos y composiciones farmaceuticas que los contienen y su uso para preparar medicamentos
FR2791674A1 (fr) *	1999-04-02	2000-10-06	Sod Conseils Rech Applic	Nouveaux derives de 2-aminopyridines, leur utilisation en tant que medicaments et compositions pharmaceutiques les contenant
SK1702001A3 (en) *	1998-08-11	2003-02-04	Pfizer Prod Inc	New pharmaceutical uses for NOS inhibitors
US7115557B2 (en)	1998-09-25	2006-10-03	Sciaticon Ab	Use of certain drugs for treating nerve root injury
SE9803710L (sv)	1998-09-25	2000-03-26	A & Science Invest Ab	Användning av vissa substanser för behandling av nervrotsskador
CN1341099A (zh)	1999-02-25	2002-03-20	辉瑞产品公司	含有稠合环取代基的2－氨基吡啶
MXPA01013452A (es) *	1999-07-23	2002-07-02	Shionogi & Co	Inhibodores de diferenciacion th2.
FR2804429B1 (fr) *	2000-01-31	2003-05-09	Adir	Nouveaux derives de 4-sulfonamides piperidine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
WO2002080853A2 (en) *	2001-04-09	2002-10-17	Bristol-Myers Squibb Company	Fused heterocyclic inhibitors of factor xa
US20030045449A1 (en) *	2001-08-15	2003-03-06	Pfizer, Inc.	Pharmaceutical combinations for the treatment of neurodegenerative diseases
MXPA05011070A (es) *	2003-04-14	2005-12-12	Pfizer Prod Inc	Derivados de 3-azabiciclo [3.2.1] octano.
CN1295216C (zh) *	2003-07-04	2007-01-17	中国人民解放军军事医学科学院毒物药物研究所	吲哚酮类衍生物及其用于制备抗肿瘤药物的用途
CA2598484A1 (en) *	2005-02-21	2006-08-24	Proximagen Ltd.	Inhibition or treatment of dyskinesia
WO2006105795A1 (en) *	2005-04-08	2006-10-12	Leo Pharma A/S	Novel indolinone derivatives
CN101522614B (zh)	2006-08-09	2014-06-25	史密丝克莱恩比彻姆公司	作为阿片样物质受体的拮抗剂或反向激动剂的化合物
EP2152271B1 (en)	2007-06-08	2015-10-21	Janssen Pharmaceutica, N.V.	Piperidine/piperazine derivatives
AU2008258487B2 (en)	2007-06-08	2012-11-15	Janssen Pharmaceutica N.V.	Piperidine/piperazine derivatives
CA2687918C (en)	2007-06-08	2016-11-08	Janssen Pharmaceutica N.V.	Piperidine/piperazine derivatives
JO2972B1 (en)	2007-06-08	2016-03-15	جانسين فارماسوتيكا ان. في	Piperidine / piperazine derivatives
JP5579170B2 (ja)	2008-06-05	2014-08-27	ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ	Ｄｇａｔ阻害剤とｐｐａｒ作動薬を含有する薬剤組み合わせ物
UA105182C2 (ru)	2008-07-03	2014-04-25	Ньюрексон, Інк.	Бензоксазины, бензотиазины и родственные соединения, которые имеют ингибирующую nos активность
US8889674B2 (en) *	2009-03-05	2014-11-18	Shionogi & Co., Ltd.	Piperidine and pyrrolidine derivatives having NPY Y5 receptor antagonism
US11013844B2 (en) *	2014-11-20	2021-05-25	City Of Hope	Treatment device for plasma virus inactivation
CA3032586A1 (en)	2016-08-12	2018-02-15	Athenex, Inc.	Biaryl compounds and use thereof for modulating a kinase cascade
BR112020005489A2 (pt)	2017-09-22	2020-09-24	Jubilant Epipad Llc,	composto da fórmula (i), composto de fórmula (ii), composto de fórmula (iii), processo de preparação de compostos de fórmula (i), processo de preparação de compostos de fórmula (ii), processo de preparação de compostos de fórmula (iii), composição farmacêutica, método para inibir uma ou mais famílias pad em uma célula, método para tratar uma afeção mediada por um ou mais pads, utilização do composto, método para o tratamento e/ou prevenção de uma afeção mediada por um ou mais distúrbios da família pad, método para o tratamento de artrite reumatoide e método de tratamento de câncer
CN111225915B (zh)	2017-10-18	2023-03-07	朱比兰特埃皮帕德有限公司	作为pad抑制剂的咪唑并吡啶化合物
EP3707135A1 (en)	2017-11-06	2020-09-16	Jubilant Prodel LLC	Pyrimidine derivatives as inhibitors of pd1/pd-l1 activation
IL274762B2 (en)	2017-11-24	2023-10-01	Jubilant Episcribe Llc	Novel heterocyclic compounds as prmt5 inhibitors
EP3765453A1 (en)	2018-03-13	2021-01-20	Jubilant Prodel LLC	Bicyclic compounds as inhibitors of pd1/pd-l1 interaction/activation
US20220267269A1 (en) *	2019-06-14	2022-08-25	Srx Cardio, Llc	Compounds for the modulation of proprotein convertase subtilisin/kexin type 9 (pcsk9)
US12115154B2 (en) *	2020-12-16	2024-10-15	Srx Cardio, Llc	Compounds for the modulation of proprotein convertase subtilisin/kexin type 9 (PCSK9)

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WO1992014780A1 (en)	1991-02-19	1992-09-03	Akzo N.V.	Stabilized carbon monoxide-olefin copolymers
JPH08504798A (ja) *	1992-12-18	1996-05-21	ザウエルカムファウンデーションリミテッド	酵素阻害薬としての，ピリミジン，ピリジン，プテリジノンおよびインダゾール誘導体
US5621004A (en)	1994-06-03	1997-04-15	Robert W. Dunn	Method for treating emesis
WO1996018616A1 (en) *	1994-12-12	1996-06-20	Merck & Co., Inc.	Substituted 2-aminopyridines as inhibitors of nitric oxide synthase
PT891332E (pt) *	1996-03-29	2004-07-30	Pfizer	Derivados de 6-fenilpiridil-2-amina
US6093743A (en)	1998-06-23	2000-07-25	Medinox Inc.	Therapeutic methods employing disulfide derivatives of dithiocarbamates and compositions useful therefor

1997
- 1997-02-18 HN HN1997000027A patent/HN1997000027A/es unknown
- 1997-11-17 SK SK708-99A patent/SK70899A3/sk unknown
- 1997-11-17 UA UA99063103A patent/UA59379C2/uk unknown
- 1997-11-17 CZ CZ19992017A patent/CZ293863B6/cs not_active IP Right Cessation
- 1997-11-17 BR BR9714381-2A patent/BR9714381A/pt not_active Application Discontinuation
- 1997-11-17 WO PCT/IB1997/001446 patent/WO1998024766A1/en not_active Ceased
- 1997-11-17 CA CA002273479A patent/CA2273479C/en not_active Expired - Fee Related
- 1997-11-17 TR TR1999/01259T patent/TR199901259T2/xx unknown
- 1997-11-17 DK DK97910587T patent/DK0946512T3/da active
- 1997-11-17 EP EP97910587A patent/EP0946512B1/en not_active Expired - Lifetime
- 1997-11-17 DE DE69725465T patent/DE69725465T2/de not_active Expired - Fee Related
- 1997-11-17 ES ES97910587T patent/ES2206691T3/es not_active Expired - Lifetime
- 1997-11-17 CN CN97180350A patent/CN1117077C/zh not_active Expired - Fee Related
- 1997-11-17 PT PT97910587T patent/PT946512E/pt unknown
- 1997-11-17 IL IL13011197A patent/IL130111A0/xx unknown
- 1997-11-17 EA EA199900448A patent/EA002907B1/ru not_active IP Right Cessation
- 1997-11-17 AT AT97910587T patent/ATE251612T1/de not_active IP Right Cessation
- 1997-11-17 HU HU0001848A patent/HUP0001848A3/hu unknown
- 1997-11-17 YU YU25399A patent/YU25399A/sh unknown
- 1997-11-17 NZ NZ335733A patent/NZ335733A/xx unknown
- 1997-11-17 PL PL97333918A patent/PL333918A1/xx unknown
- 1997-11-17 JP JP52539798A patent/JP3604399B2/ja not_active Expired - Fee Related
- 1997-11-17 SI SI9730597T patent/SI0946512T1/xx unknown
- 1997-11-17 KR KR1019997004981A patent/KR100360633B1/ko not_active Expired - Fee Related
- 1997-11-17 AU AU47917/97A patent/AU4791797A/en not_active Abandoned
- 1997-11-18 HN HN1997000149A patent/HN1997000149A/es unknown
- 1997-11-22 TW TW086117501A patent/TW491840B/zh active
- 1997-12-01 PE PE1997001080A patent/PE46499A1/es not_active Application Discontinuation
- 1997-12-03 MA MA24884A patent/MA26453A1/fr unknown
- 1997-12-03 TN TNTNSN97198A patent/TNSN97198A1/fr unknown
- 1997-12-03 DZ DZ970211A patent/DZ2361A1/xx active
- 1997-12-03 UY UY24799A patent/UY24799A1/es unknown
- 1997-12-04 PA PA19978442201A patent/PA8442201A1/es unknown
- 1997-12-04 HR HR60/032,793A patent/HRP970664A2/hr not_active Application Discontinuation
- 1997-12-04 AR ARP970105713A patent/AR010331A1/es not_active Application Discontinuation
- 1997-12-04 AP APAP/P/1997/001156A patent/AP848A/en active
- 1997-12-04 ZA ZA9710906A patent/ZA9710906B/xx unknown
- 1997-12-05 ID IDP973838A patent/ID19056A/id unknown
1999
- 1999-05-18 IS IS5053A patent/IS5053A/is unknown
- 1999-06-01 OA OA9900115A patent/OA11123A/en unknown
- 1999-06-03 US US09/325,480 patent/US6235750B1/en not_active Expired - Fee Related
- 1999-06-04 NO NO19992725A patent/NO313517B1/no unknown
- 1999-06-30 BG BG103540A patent/BG103540A/bg unknown
2001
- 2001-03-08 US US09/802,086 patent/US20020032191A1/en not_active Abandoned
- 2001-09-13 AU AU72050/01A patent/AU766080B2/en not_active Ceased
- 2001-09-27 US US09/965,564 patent/US20020103227A1/en not_active Abandoned
2004
- 2004-06-24 JP JP2004186311A patent/JP2005170924A/ja active Pending

Also Published As

Publication number	Publication date
DE69725465D1 (de)	2003-11-13
AP9701156A0 (en)	1998-01-31
AU7205001A (en)	2001-11-15
UY24799A1 (es)	2001-08-27
YU25399A (sh)	2001-07-10
AP848A (en)	2000-06-09
TR199901259T2 (xx)	1999-08-23
AU766080B2 (en)	2003-10-09
DE69725465T2 (de)	2004-05-06
SI0946512T1 (en)	2004-04-30
PT946512E (pt)	2004-01-30
CA2273479C (en)	2006-02-07
OA11123A (en)	2003-04-07
PE46499A1 (es)	1999-05-12
NO992725L (no)	1999-06-04
HN1997000149A (es)	1997-12-26
ID19056A (id)	1998-06-11
US6235750B1 (en)	2001-05-22
EA002907B1 (ru)	2002-10-31
BR9714381A (pt)	2000-05-02
HRP970664A2 (en)	1998-10-31
PA8442201A1 (es)	2000-05-24
SK70899A3 (en)	2002-04-04
PL333918A1 (en)	2000-01-31
KR20000057413A (ko)	2000-09-15
CA2273479A1 (en)	1998-06-11
CZ293863B6 (cs)	2004-08-18
EP0946512A1 (en)	1999-10-06
WO1998024766A1 (en)	1998-06-11
EA199900448A1 (ru)	2000-02-28
AR010331A1 (es)	2000-06-07
IL130111A0 (en)	2000-06-01
JP2005170924A (ja)	2005-06-30
DZ2361A1 (fr)	2002-12-28
JP3604399B2 (ja)	2004-12-22
TNSN97198A1 (fr)	2005-03-15
DK0946512T3 (da)	2004-01-12
MA26453A1 (fr)	2004-12-20
HN1997000027A (es)	1997-06-05
NO992725D0 (no)	1999-06-04
HUP0001848A2 (hu)	2001-04-28
US20020032191A1 (en)	2002-03-14
NO313517B1 (no)	2002-10-14
CZ201799A3 (cs)	2000-07-12
HUP0001848A3 (en)	2002-03-28
NZ335733A (en)	2001-01-26
BG103540A (bg)	2000-12-29
ZA9710906B (en)	1999-06-09
ES2206691T3 (es)	2004-05-16
KR100360633B1 (ko)	2002-11-13
CN1117077C (zh)	2003-08-06
CN1239952A (zh)	1999-12-29
US20020103227A1 (en)	2002-08-01
ATE251612T1 (de)	2003-10-15
TW491840B (en)	2002-06-21
EP0946512B1 (en)	2003-10-08
UA59379C2 (uk)	2003-09-15
JP2000505814A (ja)	2000-05-16
AU4791797A (en)	1998-06-29

Publication	Publication Date	Title
IS5053A (is)	1999-05-18	6-Fenýlpýridýl-2-amín afleiður nytsamlegar sem nituroxíð sýntasa tálmar
EE200000716A (et)	2002-04-15	Lämmastikoksiidi süntaasi inhibiitorid
EE04013B1 (et)	2003-04-15	Lämmastikoksiidi süntaasi inhibiitorid
AU4149696A (en)	1996-06-06	Substituted heterocycles as inhibitors of nitric oxide synthase
SI1686119T1 (sl)	2009-12-31	Derivati pirimidin-5-ona kot inhibitorji ldl-pla2
GB0031179D0 (en)	2001-01-31	Nitric oxide synthase inhibitors
IL154841A0 (en)	2003-10-31	2-amino-2-alkyl-5- heptenoic and heptynoic acid derivatives useful as nitric oxide synthase inhibitors
AU4515896A (en)	1996-07-03	Substituted 2-acylamino-pyridines as inhibitors of nitric oxide synthase
EE200000519A (et)	2002-02-15	Lämmastikoksiidi süntaasi inhibiitoritena toimivad halogeenitud amidinoaminohappederivaadid
IS2312B (is)	2007-11-15	Afleiður ísósorbíð einnítrats og notkun þeirra sem æðavíkkarar með lága þolmyndun
IL125738A0 (en)	1999-04-11	Hydroxyamidino derivatives useful as nitric oxide synthase inhibitors
ATE252547T1 (de)	2003-11-15	Matrixmetalloproteinaseinhibitoren
EE9900474A (et)	2000-06-15	Amidiini derivaadid lämmastikoksiidi süntaasi inhibiitoritena
MA24854A1 (fr)	1999-12-31	Inhibiteurs d'oxyde nitrique synthase
ZA971944B (en)	1998-03-06	Hydroxyamidino derivatives useful as nitric oxide synthase inhibitors.
HRP980381B1 (en)	2002-02-28	Nitric oxide synthase inhibitors
SI1084104T1 (en)	2003-12-31	Nitric oxide synthase inhibitors
SI0958277T1 (en)	2002-06-30	Nitric oxide synthase inhibitors
GB9605700D0 (en)	1996-05-22	Hexahydro-5-imino,4-heteroazepine derivatives as inhibitors of nitric oxide synthases
GB9605162D0 (en)	1996-05-15	Hexahydro-5-imino-1,4-heteroazepine derivatives as inhibitors of nitric oxide synthases
GB9604090D0 (en)	1996-05-01	Substituted saturated aza heterocycles as inhibitors of nitric oxide synthase
GB0031177D0 (en)	2001-01-31	Nitric oxide synthase inhibitors
SE9802118D0 (sv)	1998-06-15	Mycobacterial inhibitors