IS7382A - Píperidínafleiður - Google Patents
PíperidínafleiðurInfo
- Publication number
- IS7382A IS7382A IS7382A IS7382A IS7382A IS 7382 A IS7382 A IS 7382A IS 7382 A IS7382 A IS 7382A IS 7382 A IS7382 A IS 7382A IS 7382 A IS7382 A IS 7382A
- Authority
- IS
- Iceland
- Prior art keywords
- piperidine
- Prior art date
Links
- NQRYJNQNLNOLGT-UHFFFAOYSA-N Piperidine Chemical compound C1CCNCC1 NQRYJNQNLNOLGT-UHFFFAOYSA-N 0.000 title 2
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/04—Ortho-condensed systems
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Pain & Pain Management (AREA)
- Psychiatry (AREA)
- Epidemiology (AREA)
- Hospice & Palliative Care (AREA)
- Immunology (AREA)
- Anesthesiology (AREA)
- Rheumatology (AREA)
- Addiction (AREA)
- Pulmonology (AREA)
- Otolaryngology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB0203020.3A GB0203020D0 (en) | 2002-02-08 | 2002-02-08 | Chemical compounds |
| PCT/EP2003/001308 WO2003066635A1 (en) | 2002-02-08 | 2003-02-10 | Piperidine derivatives |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| IS7382A true IS7382A (is) | 2004-08-04 |
| IS2402B IS2402B (is) | 2008-09-15 |
Family
ID=9930717
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IS7382A IS2402B (is) | 2002-02-08 | 2004-08-04 | Píperidínafleiður |
Country Status (26)
| Country | Link |
|---|---|
| US (3) | US7189713B2 (is) |
| EP (2) | EP1666465B1 (is) |
| JP (1) | JP4488743B2 (is) |
| KR (1) | KR101011316B1 (is) |
| CN (1) | CN1319973C (is) |
| AR (1) | AR038818A1 (is) |
| AT (2) | ATE308543T1 (is) |
| AU (1) | AU2003205753B9 (is) |
| BR (1) | BRPI0307123B8 (is) |
| CA (1) | CA2475619C (is) |
| CO (1) | CO5611152A2 (is) |
| DE (2) | DE60320865D1 (is) |
| DK (1) | DK1472256T3 (is) |
| ES (2) | ES2250870T3 (is) |
| GB (1) | GB0203020D0 (is) |
| IL (2) | IL162765A0 (is) |
| IS (1) | IS2402B (is) |
| MX (1) | MXPA04006791A (is) |
| MY (1) | MY130411A (is) |
| NO (1) | NO329379B1 (is) |
| NZ (1) | NZ533785A (is) |
| PL (1) | PL211082B1 (is) |
| RU (1) | RU2336276C2 (is) |
| TW (1) | TWI291466B (is) |
| WO (1) | WO2003066635A1 (is) |
| ZA (1) | ZA200404842B (is) |
Families Citing this family (26)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB0203020D0 (en) * | 2002-02-08 | 2002-03-27 | Glaxo Group Ltd | Chemical compounds |
| TWI283241B (en) | 2002-05-29 | 2007-07-01 | Tanabe Seiyaku Co | Novel piperidine compound |
| EP1594574A2 (en) * | 2003-01-27 | 2005-11-16 | Glaxo Group Limited | Nk1 receptor antagonists for the treatment of functional dyspepsia |
| GB0308968D0 (en) * | 2003-04-17 | 2003-05-28 | Glaxo Group Ltd | Medicaments |
| US20060030600A1 (en) * | 2004-08-06 | 2006-02-09 | Patrick Schnider | Dual NK1/NK3 receptor antagonists for the treatment of schizophrenia |
| WO2006094948A1 (en) * | 2005-03-08 | 2006-09-14 | Janssen Pharmaceutica N.V. | Diaza-spiro-[4.4]-nonane derivatives as neurokinin (nk1) antagonists |
| HRP20110457T1 (hr) * | 2005-09-09 | 2011-07-31 | Glaxosmithkline Llc | Derivati piridina i njihova upotreba u liječenju psihotičnih poremećaja |
| AR057828A1 (es) | 2005-09-29 | 2007-12-19 | Astrazeneca Ab | Compuestos derivados de azetidina, su preparacion y composicion farmaceuutica |
| EP1976527A4 (en) * | 2006-01-11 | 2009-04-22 | Merck & Co Inc | CONDENSED TRIAZOL TACHYKININE RECEPTOR ANTAGONISTS |
| US7872022B2 (en) * | 2006-04-03 | 2011-01-18 | Hoffmann-La Roche Inc. | Serotonin transporter (SERT) inhibitors for the treatment of depression and anxiety |
| GB0621229D0 (en) * | 2006-10-20 | 2006-12-06 | Glaxo Group Ltd | Novel use |
| JP2010516734A (ja) | 2007-01-24 | 2010-05-20 | グラクソ グループ リミテッド | ３，５−ジアミノ−６−（２，３−ジクロロフェニル）−１，２，４−トリアジンまたはｒ（−）−２，４−ジアミノ−５−（２，３−ジクロロフェニル）−６−フルオロメチルピリミジンを含む医薬組成物 |
| WO2009002770A1 (en) * | 2007-06-22 | 2008-12-31 | Merck & Co., Inc. | 6.5-pyrrolopiperidine tachykinin receptor antagonists |
| GB0806652D0 (en) * | 2008-04-11 | 2008-05-14 | Glaxo Group Ltd | Anhydrous crystal form of orvepitant maleate |
| GB0812849D0 (en) * | 2008-07-14 | 2008-08-20 | Glaxo Wellcome Mfg Pte Ltd | Novel compounds |
| GB0814340D0 (en) | 2008-08-05 | 2008-09-10 | Smithkline Beecham Corp | Anhydrous crystol form fo a pyridine derivative |
| DK2729147T3 (en) | 2011-07-04 | 2017-12-18 | Irbm - Science Park S P A | NK-1 RECEPTOR ANTAGONISTS FOR TREATMENT OF CORNOVA |
| AU2013224181A1 (en) * | 2012-02-22 | 2014-10-02 | Leo Pharma A/S | Novel neurokinin 1 receptor antagonist compounds |
| HUE046508T2 (hu) | 2012-10-11 | 2020-03-30 | Nerre Therapeutics Ltd | Orvepitant krónikus viszketés kezelésére |
| WO2015024203A1 (en) * | 2013-08-20 | 2015-02-26 | Leo Pharma A/S | Novel neurokinin 1 receptor antagonist compounds ii |
| CN105579456A (zh) * | 2013-08-20 | 2016-05-11 | 利奥制药有限公司 | 新型神经激肽1受体拮抗剂化合物ii |
| SI3377064T1 (sl) * | 2016-01-08 | 2019-11-29 | Nerre Therapeutics Ltd | Orvepitant za zdravljenje kroničnega kašlja |
| IL312486B2 (en) | 2017-04-10 | 2025-05-01 | Chase Therapeutics Corp | NK1 antagonist combination and method for treating synucleinopathies |
| JP7158425B2 (ja) | 2017-06-30 | 2022-10-21 | チェイス セラピューティクス コーポレイション | Ｎｋ－１アンタゴニスト組成物およびうつ病の処置における使用法 |
| KR20220165251A (ko) | 2020-04-03 | 2022-12-14 | 네르 쎄라퓨틱스 리미티드 | 패혈증, 패혈성 쇼크, 급성 호흡 곤란 증후군 (ards) 또는 다발성 기관 기능장애 증후군 (mods)으로부터 선택된 질환을 치료하기 위한 nk-1 수용체 길항제 |
| MX2022014901A (es) | 2020-06-02 | 2023-01-18 | Nerre Therapeutics Ltd | Antagonistas del receptor de neuroquinina (nk)-1 para su uso en el tratamiento de condiciones de fibrosis pulmonar promovidas por lesion mecanica a los pulmones. |
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| AUPO735997A0 (en) | 1997-06-17 | 1997-07-10 | Fujisawa Pharmaceutical Co., Ltd. | Piperazine derivatives |
| CA2301770A1 (en) | 1997-08-27 | 1999-03-04 | Merck & Co., Inc. | Inhibitors of prenyl-protein transferase |
| EP1034164B1 (en) | 1997-11-24 | 2004-05-19 | Merck & Co., Inc. | Substituted beta-alanine derivatives as cell adhesion inhibitors |
| WO1999037304A1 (en) | 1998-01-27 | 1999-07-29 | Aventis Pharmaceuticals Products Inc. | SUBSTITUTED OXOAZAHETEROCYCLYL FACTOR Xa INHIBITORS |
| GB9923748D0 (en) | 1999-10-07 | 1999-12-08 | Glaxo Group Ltd | Chemical compounds |
| WO2002000631A2 (en) * | 2000-06-29 | 2002-01-03 | Fujisawa Pharmaceutical Co., Ltd. | Benzhydryl derivatives |
| AUPR237301A0 (en) * | 2001-01-02 | 2001-01-25 | Fujisawa Pharmaceutical Co., Ltd. | Benzhydryl derivatives |
| EP2301565A1 (de) | 2000-10-12 | 2011-03-30 | ViroLogik GmbH | Verwendung von Proteasome Hemmern zur Behandlung von Virus-Infektionen |
| GB0025354D0 (en) * | 2000-10-17 | 2000-11-29 | Glaxo Group Ltd | Chemical compounds |
| US20030022891A1 (en) | 2000-12-01 | 2003-01-30 | Anandan Palani | MCH antagonists and their use in the treatment of obesity |
| GB0203020D0 (en) * | 2002-02-08 | 2002-03-27 | Glaxo Group Ltd | Chemical compounds |
| US20040029865A1 (en) | 2002-05-23 | 2004-02-12 | Acker Brad A. | Bis-arylsulfones |
| MY141736A (en) | 2002-10-08 | 2010-06-15 | Elanco Animal Health Ireland | Substituted 1,4-di-piperidin-4-yi-piperazine derivatives and their use as neurokinin antagonists |
| GB0308968D0 (en) | 2003-04-17 | 2003-05-28 | Glaxo Group Ltd | Medicaments |
-
2002
- 2002-02-08 GB GBGB0203020.3A patent/GB0203020D0/en not_active Ceased
-
2003
- 2003-02-06 TW TW092102350A patent/TWI291466B/zh not_active IP Right Cessation
- 2003-02-06 MY MYPI20030409A patent/MY130411A/en unknown
- 2003-02-06 AR ARP030100377A patent/AR038818A1/es active IP Right Grant
- 2003-02-10 EP EP05077500A patent/EP1666465B1/en not_active Expired - Lifetime
- 2003-02-10 MX MXPA04006791A patent/MXPA04006791A/es active IP Right Grant
- 2003-02-10 ES ES03702621T patent/ES2250870T3/es not_active Expired - Lifetime
- 2003-02-10 IL IL16276503A patent/IL162765A0/xx unknown
- 2003-02-10 AT AT03702621T patent/ATE308543T1/de active
- 2003-02-10 CN CNB03803431XA patent/CN1319973C/zh not_active Expired - Lifetime
- 2003-02-10 KR KR1020047012190A patent/KR101011316B1/ko not_active Expired - Lifetime
- 2003-02-10 ES ES05077500T patent/ES2304660T3/es not_active Expired - Lifetime
- 2003-02-10 RU RU2004126957/04A patent/RU2336276C2/ru active
- 2003-02-10 AU AU2003205753A patent/AU2003205753B9/en not_active Expired
- 2003-02-10 BR BRPI0307123A patent/BRPI0307123B8/pt not_active IP Right Cessation
- 2003-02-10 WO PCT/EP2003/001308 patent/WO2003066635A1/en not_active Ceased
- 2003-02-10 DK DK03702621T patent/DK1472256T3/da active
- 2003-02-10 PL PL373532A patent/PL211082B1/pl unknown
- 2003-02-10 DE DE60320865T patent/DE60320865D1/de not_active Expired - Lifetime
- 2003-02-10 CA CA2475619A patent/CA2475619C/en not_active Expired - Lifetime
- 2003-02-10 NZ NZ533785A patent/NZ533785A/en not_active IP Right Cessation
- 2003-02-10 EP EP03702621A patent/EP1472256B1/en not_active Expired - Lifetime
- 2003-02-10 US US10/502,255 patent/US7189713B2/en not_active Expired - Lifetime
- 2003-02-10 DE DE60302137T patent/DE60302137T2/de not_active Expired - Lifetime
- 2003-02-10 AT AT05077500T patent/ATE394375T1/de not_active IP Right Cessation
- 2003-02-10 JP JP2003566008A patent/JP4488743B2/ja not_active Expired - Lifetime
-
2004
- 2004-06-18 ZA ZA2004/04842A patent/ZA200404842B/en unknown
- 2004-06-28 IL IL162765A patent/IL162765A/en active IP Right Grant
- 2004-08-02 NO NO20043239A patent/NO329379B1/no not_active IP Right Cessation
- 2004-08-04 IS IS7382A patent/IS2402B/is unknown
- 2004-08-06 CO CO04076757A patent/CO5611152A2/es active IP Right Grant
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2006
- 2006-12-11 US US11/608,853 patent/US7652012B2/en not_active Expired - Lifetime
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2009
- 2009-12-08 US US12/633,265 patent/US20100152446A1/en not_active Abandoned
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