IT1189601B - Derivati di benzimidazolo procedimento per la loro preparazione e agenti antiulcera che li contengono - Google Patents

Derivati di benzimidazolo procedimento per la loro preparazione e agenti antiulcera che li contengono

Info

Publication number
IT1189601B
IT1189601B IT67743/85A IT6774385A IT1189601B IT 1189601 B IT1189601 B IT 1189601B IT 67743/85 A IT67743/85 A IT 67743/85A IT 6774385 A IT6774385 A IT 6774385A IT 1189601 B IT1189601 B IT 1189601B
Authority
IT
Italy
Prior art keywords
benzyl
alkyl
sulphinyl
pref
effected
Prior art date
Application number
IT67743/85A
Other languages
English (en)
Other versions
IT8567743A0 (it
Inventor
Okabe Susumu
Satoh Masaru
Yamakawa Tomio
Nomura Yutaka
Hayashi Masatoshi
Original Assignee
Nippon Chemiphar Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from JP59182400A external-priority patent/JPS6160660A/ja
Priority claimed from JP60061195A external-priority patent/JPH0764826B2/ja
Priority claimed from JP60061194A external-priority patent/JPH068283B2/ja
Application filed by Nippon Chemiphar Co filed Critical Nippon Chemiphar Co
Publication of IT8567743A0 publication Critical patent/IT8567743A0/it
Application granted granted Critical
Publication of IT1189601B publication Critical patent/IT1189601B/it

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/24—Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • C07D235/28—Sulfur atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/24—Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • C07D235/26—Oxygen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
IT67743/85A 1984-08-31 1985-08-30 Derivati di benzimidazolo procedimento per la loro preparazione e agenti antiulcera che li contengono IT1189601B (it)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP59182400A JPS6160660A (ja) 1984-08-31 1984-08-31 ベンズイミダゾ−ル誘導体およびその製造法ならびにこれを含有する抗潰瘍剤
JP60061195A JPH0764826B2 (ja) 1985-03-26 1985-03-26 ベンズイミダゾール誘導体
JP60061194A JPH068283B2 (ja) 1985-03-26 1985-03-26 ベンズイミダゾ−ル誘導体およびその製造法ならびにこれを含有する抗潰瘍剤

Publications (2)

Publication Number Publication Date
IT8567743A0 IT8567743A0 (it) 1985-08-30
IT1189601B true IT1189601B (it) 1988-02-04

Family

ID=27297422

Family Applications (1)

Application Number Title Priority Date Filing Date
IT67743/85A IT1189601B (it) 1984-08-31 1985-08-30 Derivati di benzimidazolo procedimento per la loro preparazione e agenti antiulcera che li contengono

Country Status (14)

Country Link
KR (1) KR920004936B1 (it)
AR (1) AR242195A1 (it)
AU (3) AU4640985A (it)
BE (1) BE903128A (it)
BR (1) BR8504252A (it)
CH (1) CH665417A5 (it)
DE (1) DE3531487C2 (it)
ES (1) ES8703142A1 (it)
FR (1) FR2569691B1 (it)
GB (1) GB2163747B (it)
IT (1) IT1189601B (it)
MX (1) MX159807A (it)
NL (1) NL8502384A (it)
SE (1) SE500669C2 (it)

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US6380222B2 (en) 1996-10-11 2002-04-30 Astrazeneca Ab Use of an H+, K+-atpase inhibitor in the treatment of nasal polyps
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JP4988088B2 (ja) 1998-08-12 2012-08-01 ニコメッド ゲゼルシャフト ミット ベシュレンクテル ハフツング ピリジン−２−イルメチルスルフィニル−１ｈ−ベンズイミダゾール、もしくはピリジン−２−イルメチルスルフィニル−１ｈ−ベンズイミダゾールの骨格を有する化合物、またはその薬学的に許容される塩の経口投与形組成物を固定的に組み合わせた組成物
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US6544556B1 (en) 2000-09-11 2003-04-08 Andrx Corporation Pharmaceutical formulations containing a non-steroidal antiinflammatory drug and a proton pump inhibitor
SE0101379D0 (sv) 2001-04-18 2001-04-18 Diabact Ab Komposition som hämmar utsöndring av magsyra
US8206741B2 (en) 2001-06-01 2012-06-26 Pozen Inc. Pharmaceutical compositions for the coordinated delivery of NSAIDs
SE0102993D0 (sv) 2001-09-07 2001-09-07 Astrazeneca Ab New self emulsifying drug delivery system
US8101209B2 (en) 2001-10-09 2012-01-24 Flamel Technologies Microparticulate oral galenical form for the delayed and controlled release of pharmaceutical active principles
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SE0203065D0 (sv) 2002-10-16 2002-10-16 Diabact Ab Gastric acid secretion inhibiting composition
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KR20060092255A (ko) 2003-09-26 2006-08-22 알자 코포레이션 고도의 약물적재를 제공하는 약물코팅제 및 그의 제조방법
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US10624858B2 (en) 2004-08-23 2020-04-21 Intellipharmaceutics Corp Controlled release composition using transition coating, and method of preparing same
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TR201910825T4 (tr) 2006-12-22 2019-08-21 Ironwood Pharmaceuticals Inc Yemek borusu rahatsizliklarini tedavi̇ etmek i̇çi̇n yöntemler ve bi̇leşi̇mler
BRPI0918492A2 (pt) 2008-09-09 2015-12-01 Astrazeneca Ab uso de naproxen, ou sal farmaceuticamente aceitável do mesmo, e esomeprazol, ou sal farmaceuticamente aceitável do mesmo
EP2445499A4 (en) 2009-06-25 2013-02-27 Astrazeneca Ab METHOD FOR TREATING A PATIENT WITH RISK OF DEVELOPING A NSAID-ASSOCIATED SPURGE
WO2011080500A2 (en) 2009-12-29 2011-07-07 Orexo Ab New pharmaceutical dosage form for the treatment of gastric acid-related disorders
WO2011080501A2 (en) 2009-12-29 2011-07-07 Orexo Ab New pharmaceutical dosage form for the treatment of gastric acid-related disorders
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US20130156720A1 (en) 2010-08-27 2013-06-20 Ironwood Pharmaceuticals, Inc. Compositions and methods for treating or preventing metabolic syndrome and related diseases and disorders
EP2601947A1 (en) 2011-12-05 2013-06-12 Abo Bakr Mohammed Ali Al-Mehdar Fixed-dose combination for treatment of helicobacter pylori associated diseases
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US4359465A (en) * 1980-07-28 1982-11-16 The Upjohn Company Methods for treating gastrointestinal inflammation
EP0174717B1 (en) * 1984-07-06 1992-01-22 FISONS plc Benzimidazoles, and their production formulation and use as gastric acid secretion inhibitors

Also Published As

Publication number Publication date
FR2569691A1 (fr) 1986-03-07
IT8567743A0 (it) 1985-08-30
SE8504048D0 (sv) 1985-08-30
GB8521493D0 (en) 1985-10-02
DE3531487C2 (de) 1995-08-17
KR860001793A (ko) 1986-03-22
SE500669C2 (sv) 1994-08-08
FR2569691B1 (fr) 1989-08-04
GB2163747B (en) 1989-02-08
GB2163747A (en) 1986-03-05
AU4127189A (en) 1989-12-21
NL8502384A (nl) 1986-03-17
ES546445A0 (es) 1986-11-16
AR242195A1 (es) 1993-03-31
BE903128A (fr) 1985-12-16
BR8504252A (pt) 1986-06-17
MX159807A (es) 1989-08-31
AU2975092A (en) 1993-01-28
KR920004936B1 (ko) 1992-06-22
ES8703142A1 (es) 1986-11-16
SE8504048L (sv) 1986-03-01
AU647978B2 (en) 1994-03-31
AU4640985A (en) 1986-03-06
CH665417A5 (fr) 1988-05-13
DE3531487A1 (de) 1986-03-13

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