ITMI20022076A1 - Sali di intermedi del cefdinir. - Google Patents

Sali di intermedi del cefdinir.

Info

Publication number
ITMI20022076A1
ITMI20022076A1 IT002076A ITMI20022076A ITMI20022076A1 IT MI20022076 A1 ITMI20022076 A1 IT MI20022076A1 IT 002076 A IT002076 A IT 002076A IT MI20022076 A ITMI20022076 A IT MI20022076A IT MI20022076 A1 ITMI20022076 A1 IT MI20022076A1
Authority
IT
Italy
Prior art keywords
cefdinir
salts
sub
disclosed
general formula
Prior art date
Application number
IT002076A
Other languages
English (en)
Inventor
Marco Alpegiani
Walter Cabri
Gomez Patricio Martin
Giovanni Pozzi
Original Assignee
Antibioticos Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Antibioticos Spa filed Critical Antibioticos Spa
Priority to IT002076A priority Critical patent/ITMI20022076A1/it
Priority to JP2004544046A priority patent/JP2006501305A/ja
Priority to AT03788921T priority patent/ATE332304T1/de
Priority to AU2003293585A priority patent/AU2003293585A1/en
Priority to DE60306667T priority patent/DE60306667D1/de
Priority to ES03788921T priority patent/ES2268467T3/es
Priority to CA002500791A priority patent/CA2500791A1/en
Priority to EP03788921A priority patent/EP1546155B1/en
Priority to PCT/EP2003/010718 priority patent/WO2004035800A2/en
Priority to US10/529,649 priority patent/US7405294B2/en
Publication of ITMI20022076A1 publication Critical patent/ITMI20022076A1/it
Priority to US12/181,438 priority patent/US20090036672A1/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Cephalosporin Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
IT002076A 2002-10-01 2002-10-01 Sali di intermedi del cefdinir. ITMI20022076A1 (it)

Priority Applications (11)

Application Number Priority Date Filing Date Title
IT002076A ITMI20022076A1 (it) 2002-10-01 2002-10-01 Sali di intermedi del cefdinir.
ES03788921T ES2268467T3 (es) 2002-10-01 2003-09-26 Sales de intermediario de cefdinir.
AT03788921T ATE332304T1 (de) 2002-10-01 2003-09-26 Cefdinir salze als zwischenprodukte
AU2003293585A AU2003293585A1 (en) 2002-10-01 2003-09-26 Intermediate cefdinir salts
DE60306667T DE60306667D1 (de) 2002-10-01 2003-09-26 Cefdinir salze als zwischenprodukte
JP2004544046A JP2006501305A (ja) 2002-10-01 2003-09-26 セフジニル中間体塩
CA002500791A CA2500791A1 (en) 2002-10-01 2003-09-26 Intermediate cefdinir salts
EP03788921A EP1546155B1 (en) 2002-10-01 2003-09-26 Intermediate cefdinir salts
PCT/EP2003/010718 WO2004035800A2 (en) 2002-10-01 2003-09-26 Intermediate cefdinir salts
US10/529,649 US7405294B2 (en) 2002-10-01 2003-09-26 Intermediate cefdinir salts
US12/181,438 US20090036672A1 (en) 2002-10-01 2008-07-29 Intermediate cefdinir salts

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT002076A ITMI20022076A1 (it) 2002-10-01 2002-10-01 Sali di intermedi del cefdinir.

Publications (1)

Publication Number Publication Date
ITMI20022076A1 true ITMI20022076A1 (it) 2004-04-02

Family

ID=32104767

Family Applications (1)

Application Number Title Priority Date Filing Date
IT002076A ITMI20022076A1 (it) 2002-10-01 2002-10-01 Sali di intermedi del cefdinir.

Country Status (10)

Country Link
US (1) US7405294B2 (it)
EP (1) EP1546155B1 (it)
JP (1) JP2006501305A (it)
AT (1) ATE332304T1 (it)
AU (1) AU2003293585A1 (it)
CA (1) CA2500791A1 (it)
DE (1) DE60306667D1 (it)
ES (1) ES2268467T3 (it)
IT (1) ITMI20022076A1 (it)
WO (1) WO2004035800A2 (it)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN115612473A (zh) * 2022-10-11 2023-01-17 中国科学院兰州化学物理研究所 一种耐高温酸化缓蚀剂及其制备方法和应用、缓蚀酸化压裂液

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ITMI20020913A0 (it) * 2002-04-29 2002-04-29 Acs Dobfar Spa Nuova forma cristallina del cefdinir
AU2003255424A1 (en) * 2002-08-13 2004-03-03 Sandoz Ag A cefdinir intermediate
US7244842B2 (en) * 2002-11-15 2007-07-17 Orchid Chemicals & Pharmaceuticals Ltd. Amorphous hydrate of a cephalosporin antibiotic
MXPA05010205A (es) * 2003-03-24 2005-11-08 Acs Dobfar Spa Nuevo cristal del acido 7-[2-(2- aminotiazol- 4-il)-2- hidroxiiminoacetamido] -3-vinil-3- cefem-4 -carboxilico (isomero syn) y metodo para la preparacion del mismo.
US20050209211A1 (en) * 2004-03-16 2005-09-22 Devalina Law Trihemihydrate, anhydrate and novel hydrate forms of Cefdinir
US20050245738A1 (en) * 2004-05-03 2005-11-03 Lupin Ltd Stable bioavailable crystalline form or cefdinir and a process for the preparation thereof
JP4856795B2 (ja) * 2004-07-05 2012-01-18 オーキッド ケミカルズ アンド ファーマシューティカルズ リミテッド セファロスポリン抗生物質の製造における新規な塩
ITMI20042231A1 (it) * 2004-11-19 2005-02-19 Antibioticos Spa Cefdinir sale d'ammonio in forma cristallina
MX2007006018A (es) 2004-11-30 2007-06-07 Astellas Pharma Inc Suspension farmaceutica oral novedosa de cristal de cefdinir.
EP1848724A2 (en) * 2005-10-31 2007-10-31 Teva Pharmaceutical Industries Ltd Process for the preparation of cefdinir
US20070128268A1 (en) * 2005-12-07 2007-06-07 Herwig Jennewein Pharmaceutical compositions comprising an antibiotic
ITMI20071628A1 (it) * 2007-08-06 2007-11-05 Acs Dobfar Spa Sintesi di 3-alchenilcefalosporine e nuovi intermedi utili ad esse correlati
US8290559B2 (en) * 2007-12-17 2012-10-16 Dexcom, Inc. Systems and methods for processing sensor data
KR101058135B1 (ko) * 2008-04-04 2011-08-24 대웅바이오 주식회사 세프디니르 합성에 유용한 중간체 및 이를 이용하여세프디니르를 제조하는 방법
CN101481383B (zh) * 2008-12-31 2012-01-11 杭州奥默医药技术有限公司 头孢地尼酸式复盐化合物及制备方法
TR200909784A1 (tr) 2009-12-25 2011-07-21 Bi̇lgi̇ç Mahmut Yeni sefdinir tuzları
CN102020664B (zh) * 2010-11-30 2012-12-12 浙江工业大学 一种头孢地尼的合成方法
CN102617506B (zh) * 2011-01-31 2015-04-01 石药集团中奇制药技术(石家庄)有限公司 一种头孢地尼及其中间体的制备方法
CN102617601A (zh) * 2011-01-31 2012-08-01 石药集团中奇制药技术(石家庄)有限公司 一种头孢地尼的制备方法

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ZA806977B (en) * 1979-11-19 1981-10-28 Fujisawa Pharmaceutical Co 7-acylamino-3-vinylcephalosporanic acid derivatives and processes for the preparation thereof
US5114958A (en) * 1991-05-09 1992-05-19 Warner-Lambert Company 1,2,4-oxadiazole and 1,2,4-thiadiazole derivatives of fenamates as antiinflammatory agents
PT874853E (pt) * 1995-12-27 2002-09-30 Hanmi Pharmaceutical Co Ltd Processo de preparacao de cefdinir
TW538045B (en) * 1997-01-16 2003-06-21 Biochemie Gmbh Process for purifying cefixime
AT405283B (de) * 1997-04-04 1999-06-25 Biochemie Gmbh Neues kristallines 7-(z)-(2-(2-aminothiazol-4-yl) -2-hydroxyiminoacetamido)-3-vinyl-3-cephem-4- carbonsäure dicyclohexylammoniumsalz und verfahren zu dessen herstellung
US6319955B1 (en) * 1998-01-06 2001-11-20 The General Hospital Corporation Use of MEK1 inhibitors as protective agents against damage due to ischemia
WO2000017206A1 (en) * 1998-09-18 2000-03-30 Cubist Pharmaceuticals, Inc. Tetracyclic heterocycles as antimicrobial agents
US6346583B1 (en) * 1999-08-25 2002-02-12 General Electric Company Polar solvent compatible polyethersiloxane elastomers
BR0017026A (pt) * 1999-12-15 2003-01-07 Cubist Pharm Inc Lipeptìdeos como agentes antibacterianos
JP4544692B2 (ja) * 2000-04-13 2010-09-15 大塚化学株式会社 3−ビニル−セフェム化合物の製造方法
KR100451672B1 (ko) 2001-06-05 2004-10-08 한미약품 주식회사 결정성 세프디니르 산부가염, 이의 제조방법 및 이를이용한 세프디니르의 제조방법
CA2379375A1 (en) * 2002-03-28 2003-09-28 Apotex Inc. Sulfonamide derivatives of 3-substituted imidazol[1,2-d]-1,2,4-thiadiazoles and 3-substituted-[1,2,4] thiadiazolo[4,5-a] benzimidazole as inhibitors of fibrin cross-linking and transglutaminases
US6960654B2 (en) * 2002-06-11 2005-11-01 The Board Of Trustees Of The University Of Illinois Method of forming glycosidic bonds from thioglycosides using an N,N-dialkylsulfinamide
US7244842B2 (en) * 2002-11-15 2007-07-17 Orchid Chemicals & Pharmaceuticals Ltd. Amorphous hydrate of a cephalosporin antibiotic
ITMI20022724A1 (it) * 2002-12-20 2004-06-21 Antibioticos Spa Sali cristallini del cefdinir.
US20050119244A1 (en) * 2003-12-02 2005-06-02 Acs Dobfar S.P.A. Process for preparing cephalosporins with salified intermediate
US20050245738A1 (en) * 2004-05-03 2005-11-03 Lupin Ltd Stable bioavailable crystalline form or cefdinir and a process for the preparation thereof
JP4856795B2 (ja) * 2004-07-05 2012-01-18 オーキッド ケミカルズ アンド ファーマシューティカルズ リミテッド セファロスポリン抗生物質の製造における新規な塩
ITMI20042231A1 (it) * 2004-11-19 2005-02-19 Antibioticos Spa Cefdinir sale d'ammonio in forma cristallina

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN115612473A (zh) * 2022-10-11 2023-01-17 中国科学院兰州化学物理研究所 一种耐高温酸化缓蚀剂及其制备方法和应用、缓蚀酸化压裂液

Also Published As

Publication number Publication date
WO2004035800A3 (en) 2004-08-26
US7405294B2 (en) 2008-07-29
ATE332304T1 (de) 2006-07-15
CA2500791A1 (en) 2004-04-29
ES2268467T3 (es) 2007-03-16
DE60306667D1 (de) 2006-08-17
EP1546155B1 (en) 2006-07-05
AU2003293585A8 (en) 2004-05-04
JP2006501305A (ja) 2006-01-12
EP1546155A2 (en) 2005-06-29
US20060111566A1 (en) 2006-05-25
WO2004035800A2 (en) 2004-04-29
AU2003293585A1 (en) 2004-05-04

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