JO3408B1 - مركبات بترين سلفون اميد ثيازول و أوكسازول - Google Patents

مركبات بترين سلفون اميد ثيازول و أوكسازول

Info

Publication number
JO3408B1
JO3408B1 JOP/2009/0162A JOP20090162A JO3408B1 JO 3408 B1 JO3408 B1 JO 3408B1 JO P20090162 A JOP20090162 A JO P20090162A JO 3408 B1 JO3408 B1 JO 3408B1
Authority
JO
Jordan
Prior art keywords
benzene sulfonamide
oxazole compounds
thiazole
sulfonamide thiazole
oxazole
Prior art date
Application number
JOP/2009/0162A
Other languages
English (en)
Inventor
W Johnson Neil
Howard Dickerson Scott
Wilson Brian
Leroy Adams Jerry
Stellwagen John
Petrov Kimberly
Schaaf Gregory
Edward Uehling David
Gregory Waterson Alex
M Ralph Jeffrey
Tian Xinrong
Renae Rheault Tara
Kuntz Kevin
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=41265326&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=JO3408(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Application granted granted Critical
Publication of JO3408B1 publication Critical patent/JO3408B1/ar

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A61K31/427—Thiazoles not condensed and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/04—Antineoplastic agents specific for metastasis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Epidemiology (AREA)
  • Oncology (AREA)
  • Hematology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

Abstract

يتعلق الاختراع الحالي بتوفير مركبات ثيازول سلفوناميد و أوكسازول سلفوناميد، وتركيبات تحتوي على ثيازول سلفوناميد و أوكسازول سلفوناميد. كما يتعلق الاختراع الحالي بعمليات لتحضيرها وطرق لاستخدامها كعوامل صيدلانية.
JOP/2009/0162A 2008-05-06 2009-05-04 مركبات بترين سلفون اميد ثيازول و أوكسازول JO3408B1 (ar)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US5074408P 2008-05-06 2008-05-06

Publications (1)

Publication Number Publication Date
JO3408B1 true JO3408B1 (ar) 2019-10-20

Family

ID=41265326

Family Applications (1)

Application Number Title Priority Date Filing Date
JOP/2009/0162A JO3408B1 (ar) 2008-05-06 2009-05-04 مركبات بترين سلفون اميد ثيازول و أوكسازول

Country Status (34)

Country Link
US (6) US7994185B2 (ar)
EP (2) EP2282636B1 (ar)
JP (1) JP5426664B2 (ar)
KR (1) KR101628746B1 (ar)
CN (1) CN102083312B (ar)
AR (1) AR071617A1 (ar)
AU (1) AU2009244491B2 (ar)
BR (1) BRPI0912541B8 (ar)
CA (1) CA2723396C (ar)
CL (1) CL2009001065A1 (ar)
CO (1) CO6321189A2 (ar)
CY (1) CY1117615T1 (ar)
DK (1) DK2282636T3 (ar)
DO (1) DOP2010000326A (ar)
EA (1) EA019349B1 (ar)
ES (1) ES2576684T3 (ar)
HR (1) HRP20160447T1 (ar)
HU (1) HUE028820T2 (ar)
IL (1) IL209018A (ar)
JO (1) JO3408B1 (ar)
MA (1) MA32369B1 (ar)
MX (1) MX2010012074A (ar)
MY (1) MY155317A (ar)
NZ (1) NZ588970A (ar)
PE (1) PE20091952A1 (ar)
PL (1) PL2282636T3 (ar)
RS (1) RS54725B1 (ar)
SG (1) SG190624A1 (ar)
SI (1) SI2282636T1 (ar)
TW (1) TWI432430B (ar)
UA (1) UA103319C2 (ar)
UY (1) UY31806A (ar)
WO (1) WO2009137391A2 (ar)
ZA (1) ZA201007960B (ar)

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