JPH01311095A - ４―デメトキシ―４′―デオキシ―４′―ヨードアントラサイクリングリコシド - Google Patents

４―デメトキシ―４′―デオキシ―４′―ヨードアントラサイクリングリコシド

Info

Publication number
JPH01311095A
JPH01311095A JP1101521A JP10152189A JPH01311095A JP H01311095 A JPH01311095 A JP H01311095A JP 1101521 A JP1101521 A JP 1101521A JP 10152189 A JP10152189 A JP 10152189A JP H01311095 A JPH01311095 A JP H01311095A
Authority
JP
Japan
Prior art keywords
demethoxy
formula
deoxy
pharmaceutically acceptable
acid addition
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP1101521A
Other languages
English (en)
Japanese (ja)
Inventor
Antonino Suarato
アントニノ・スアラト
Michele Caruso
ミケル・カルソ
Sergio Penco
セルジオ・ペンコ
Fernando Giuliani
フエルナンド・ジユリアニ
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Italia SRL
Original Assignee
Farmitalia Carlo Erba SRL
Carlo Erba SpA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Farmitalia Carlo Erba SRL, Carlo Erba SpA filed Critical Farmitalia Carlo Erba SRL
Publication of JPH01311095A publication Critical patent/JPH01311095A/ja
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D309/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings
    • C07D309/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • C07D309/08—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D309/14—Nitrogen atoms not forming part of a nitro radical
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
JP1101521A 1988-04-22 1989-04-20 ４―デメトキシ―４′―デオキシ―４′―ヨードアントラサイクリングリコシド Pending JPH01311095A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB8809615A GB2218087B (en) 1988-04-22 1988-04-22 4-demethoxy-4'-deoxy-4'iodo anthracycline glycosides
GB8809615.1 1988-04-22

Publications (1)

Publication Number Publication Date
JPH01311095A true JPH01311095A (ja) 1989-12-15

Family

ID=10635701

Family Applications (1)

Application Number Title Priority Date Filing Date
JP1101521A Pending JPH01311095A (ja) 1988-04-22 1989-04-20 ４―デメトキシ―４′―デオキシ―４′―ヨードアントラサイクリングリコシド

Country Status (4)

Country Link
JP (1) JPH01311095A (it)
DE (1) DE3912867A1 (it)
GB (1) GB2218087B (it)
IT (1) IT1230065B (it)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9418260D0 (en) * 1994-09-09 1994-10-26 Erba Carlo Spa Anthracycline derivatives

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3803124A (en) * 1968-04-12 1974-04-09 Farmaceutici It Soc Process for the preparation of adriamycin and adriamycinone and adriamycin derivatives
US4438105A (en) * 1982-04-19 1984-03-20 Farmaitalia Carlo Erba S.P.A 4'-Iododerivatives of anthracycline glycosides
GB8321676D0 (en) * 1983-08-11 1983-09-14 Erba Farmitalia 4'-haloanthrocycline glycosides
GB2169286A (en) * 1985-01-05 1986-07-09 Erba Farmitalia 4'-Deoxy-4'-halodoxorubicin-14-esters

Also Published As

Publication number Publication date
DE3912867A1 (de) 1989-11-02
IT8920197A0 (it) 1989-04-19
GB2218087B (en) 1991-01-30
GB8809615D0 (en) 1988-05-25
IT1230065B (it) 1991-09-27
GB2218087A (en) 1989-11-08

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