JPH06506443A - アザ二環式およびアザ三環式誘導体、その製法および中間体ならびに該化合物含有の医薬組成物 - Google Patents

アザ二環式およびアザ三環式誘導体、その製法および中間体ならびに該化合物含有の医薬組成物

Info

Publication number
JPH06506443A
JPH06506443A JP4502573A JP50257392A JPH06506443A JP H06506443 A JPH06506443 A JP H06506443A JP 4502573 A JP4502573 A JP 4502573A JP 50257392 A JP50257392 A JP 50257392A JP H06506443 A JPH06506443 A JP H06506443A
Authority
JP
Japan
Prior art keywords
hydrogen
alkyl
formula
compound
tables
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP4502573A
Other languages
English (en)
Japanese (ja)
Inventor
キング，フランシス・デイビッド
Original Assignee
スミスクライン・ビーチャム・パブリック・リミテッド・カンパニー
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB919100370A external-priority patent/GB9100370D0/en
Priority claimed from GB919100580A external-priority patent/GB9100580D0/en
Application filed by スミスクライン・ビーチャム・パブリック・リミテッド・カンパニー filed Critical スミスクライン・ビーチャム・パブリック・リミテッド・カンパニー
Publication of JPH06506443A publication Critical patent/JPH06506443A/ja
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
    • C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
JP4502573A 1991-01-09 1992-01-09 アザ二環式およびアザ三環式誘導体、その製法および中間体ならびに該化合物含有の医薬組成物 Pending JPH06506443A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
GB919100370A GB9100370D0 (en) 1991-01-09 1991-01-09 Pharmaceuticals
GB9100370.7 1991-01-09
GB919100580A GB9100580D0 (en) 1991-01-10 1991-01-10 Pharmaceuticals
GB9100580.1 1991-01-10
PCT/GB1992/000050 WO1992012149A1 (fr) 1991-01-09 1992-01-09 Derives azabicydiques et azatricydiques, leurs procedes et intermediaires de preparation et compositions pharmaceutiques les contenant

Publications (1)

Publication Number Publication Date
JPH06506443A true JPH06506443A (ja) 1994-07-21

Family

ID=26298233

Family Applications (1)

Application Number Title Priority Date Filing Date
JP4502573A Pending JPH06506443A (ja) 1991-01-09 1992-01-09 アザ二環式およびアザ三環式誘導体、その製法および中間体ならびに該化合物含有の医薬組成物

Country Status (4)

Country Link
EP (1) EP0566609A1 (fr)
JP (1) JPH06506443A (fr)
AU (1) AU1161292A (fr)
WO (1) WO1992012149A1 (fr)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2008044701A1 (fr) 2006-10-11 2008-04-17 Nippon Soda Co., Ltd. Procédé de production d'un dérivé de pipéridine-4-one

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9214184D0 (en) * 1992-07-03 1992-08-12 Smithkline Beecham Plc Pharmaceuticals
JP3235913B2 (ja) * 1993-07-30 2001-12-04 エーザイ株式会社 アミノ安息香酸誘導体
GB9721139D0 (en) 1997-10-07 1997-12-03 Glaxo Group Ltd Medicaments
IT1303123B1 (it) * 1998-10-13 2000-10-30 Rotta Research Lab Derivati basici di benz(e)isoindol-1-oni e pirrolo(3,4-c)chinolin-1-oni ad attivita' 5ht3 antagonista, loro preparazione ed
TW200306189A (en) 2002-03-21 2003-11-16 Merz Pharma Gmbh & Co Kgaa Azabicyclic, azatricyclic and azaspirocyclic derivatives of aminocyclohexane NMDA, 5HT3, and neuronal nicotinic receptor antagonists
ES2405594T3 (es) 2002-09-25 2013-05-31 Memory Pharmaceuticals Corporation Idazoles, benzotiazoles y benzisotiazoles, y preparación y usos de los mismos
US6984652B2 (en) 2003-09-05 2006-01-10 Warner-Lambert Company Llc Gyrase inhibitors
WO2005063767A2 (fr) 2003-12-22 2005-07-14 Memory Pharmaceuticals Corporation Indoles, 1h-indazoles, 1,2-benzisoxazoles, et 1,2-benzisothiazoles, et leur preparation et utilisation
RU2417225C2 (ru) 2004-03-25 2011-04-27 Мемори Фармасьютиклз Корпорейшн Индазолы, бензотиазолы, бензоизотиазолы, бензизоксазолы и их получение и применение
CA2567977A1 (fr) 2004-04-22 2006-01-05 Memory Pharmaceutical Corporation Indoles, 1h-indazoles, 1,2-benzisoxazoles, 1,2-benzoisothiazoles, leur preparation et leurs utilisations
JP2007538011A (ja) 2004-05-07 2007-12-27 メモリー・ファーマシューティカルズ・コーポレイション １ｈ−インダゾール、ベンゾチアゾール、１，２−ベンゾイソキサゾール、１，２−ベンゾイソチアゾール、およびクロモン、ならびにそれらの調製および使用
BRPI0512046A (pt) 2004-06-15 2008-02-06 Pfizer derivados de ácido benzimidazolona carboxìlico
US7737163B2 (en) 2004-06-15 2010-06-15 Pfizer Inc. Benzimidazolone carboxylic acid derivatives
JP2008525464A (ja) 2004-12-22 2008-07-17 メモリー・ファーマシューティカルズ・コーポレイション α−７ニコチン性受容体リガンド並びにその製造及び使用
EA012615B1 (ru) 2005-02-22 2009-10-30 Пфайзер Инк. Производные оксииндола в качестве агонистов 5-htрецептора
US8106066B2 (en) 2005-09-23 2012-01-31 Memory Pharmaceuticals Corporation Indazoles, benzothiazoles, benzoisothiazoles, benzisoxazoles, pyrazolopyridines, isothiazolopyridines, and preparation and uses thereof
WO2022175402A1 (fr) 2021-02-18 2022-08-25 Aprea Therapeutics Ab Dérivés de quinuclidine-3-one

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL59004A0 (en) * 1978-12-30 1980-03-31 Beecham Group Ltd Substituted benzamides their preparation and pharmaceutical compositions containing them

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2008044701A1 (fr) 2006-10-11 2008-04-17 Nippon Soda Co., Ltd. Procédé de production d'un dérivé de pipéridine-4-one

Also Published As

Publication number Publication date
WO1992012149A1 (fr) 1992-07-23
EP0566609A1 (fr) 1993-10-27
AU1161292A (en) 1992-08-17

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