LTC2552902I2 - Nenukleozidinės reversinės transkriptazės inhibitoriai - Google Patents

Nenukleozidinės reversinės transkriptazės inhibitoriai

Info

Publication number
LTC2552902I2
LTC2552902I2 LTPA2019506C LTC2552902I2 LT C2552902 I2 LTC2552902 I2 LT C2552902I2 LT PA2019506 C LTPA2019506 C LT PA2019506C LT C2552902 I2 LTC2552902 I2 LT C2552902I2
Authority
LT
Lithuania
Prior art keywords
reverse transcriptase
transcriptase inhibitors
nucleoside reverse
nucleoside
inhibitors
Prior art date
Application number
Other languages
English (en)
Original Assignee
Merck Canada Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=44710363&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=LTC2552902(I2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Merck Canada Inc filed Critical Merck Canada Inc
Publication of LTPA2019506I1 publication Critical patent/LTPA2019506I1/lt
Publication of LTC2552902I2 publication Critical patent/LTC2552902I2/lt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Communicable Diseases (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Virology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Molecular Biology (AREA)
  • AIDS & HIV (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
LTPA2019506 2010-03-30 2019-04-11 Nenukleozidinės reversinės transkriptazės inhibitoriai LTC2552902I2 (lt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US31882410P 2010-03-30 2010-03-30
US32157310P 2010-04-07 2010-04-07
PCT/CA2011/000320 WO2011120133A1 (en) 2010-03-30 2011-03-28 Non-nucleoside reverse transcriptase inhibitors

Publications (2)

Publication Number Publication Date
LTPA2019506I1 LTPA2019506I1 (lt) 2019-04-25
LTC2552902I2 true LTC2552902I2 (lt) 2019-12-10

Family

ID=44710363

Family Applications (3)

Application Number Title Priority Date Filing Date
LTEP15157348.2T LT2924034T (lt) 2010-03-30 2011-03-28 Farmacinė kompozicija, apimanti nenukleozidinį atvirkštinės transkriptazės inhibitorių
LTPA2019507C LTC2924034I2 (lt) 2010-03-30 2019-04-11 Farmacinė kompozicija, apimanti nenukleozidinį atvirkštinės transkriptazės inhibitorių
LTPA2019506 LTC2552902I2 (lt) 2010-03-30 2019-04-11 Nenukleozidinės reversinės transkriptazės inhibitoriai

Family Applications Before (2)

Application Number Title Priority Date Filing Date
LTEP15157348.2T LT2924034T (lt) 2010-03-30 2011-03-28 Farmacinė kompozicija, apimanti nenukleozidinį atvirkštinės transkriptazės inhibitorių
LTPA2019507C LTC2924034I2 (lt) 2010-03-30 2019-04-11 Farmacinė kompozicija, apimanti nenukleozidinį atvirkštinės transkriptazės inhibitorių

Country Status (44)

Country Link
US (2) US8486975B2 (lt)
EP (2) EP2924034B1 (lt)
JP (2) JP5281718B2 (lt)
KR (1) KR101421861B1 (lt)
CN (1) CN102971308B (lt)
AR (1) AR080859A1 (lt)
AU (1) AU2011235568B2 (lt)
BR (1) BR112012024691B1 (lt)
CA (1) CA2794377C (lt)
CL (1) CL2012002744A1 (lt)
CO (1) CO6630126A2 (lt)
CR (1) CR20120503A (lt)
CY (3) CY1118774T1 (lt)
DK (2) DK2924034T3 (lt)
DO (1) DOP2012000256A (lt)
EA (1) EA024804B1 (lt)
EC (1) ECSP12012201A (lt)
ES (2) ES2609636T3 (lt)
FI (1) FIC20190021I1 (lt)
GE (1) GEP20156368B (lt)
HN (1) HN2012002039A (lt)
HR (2) HRP20150427T1 (lt)
HU (4) HUE025336T2 (lt)
IL (2) IL222030A (lt)
LT (3) LT2924034T (lt)
LU (2) LUC00114I2 (lt)
MA (1) MA34170B1 (lt)
ME (2) ME02570B (lt)
MX (1) MX2012011379A (lt)
MY (1) MY163979A (lt)
NI (1) NI201200146A (lt)
NL (1) NL300980I2 (lt)
NO (2) NO2019019I1 (lt)
NZ (1) NZ602670A (lt)
PE (1) PE20130158A1 (lt)
PH (1) PH12012501923A1 (lt)
PL (2) PL2924034T3 (lt)
PT (2) PT2924034T (lt)
RS (2) RS55505B1 (lt)
SG (1) SG184347A1 (lt)
SI (2) SI2924034T1 (lt)
TN (1) TN2012000455A1 (lt)
TW (1) TWI458719B (lt)
WO (1) WO2011120133A1 (lt)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MX2012011379A (es) * 2010-03-30 2012-11-30 Merck Canada Inc Inhibidores no nucleosidicos de la transcriptasa inversa.
WO2012048113A2 (en) 2010-10-07 2012-04-12 The General Hospital Corporation Biomarkers of cancer
EP2900240B1 (en) * 2012-09-26 2020-01-08 Merck Sharp & Dohme Corp. Crystalline form of a reverse transcriptase inhibitor
JO3470B1 (ar) 2012-10-08 2020-07-05 Merck Sharp & Dohme مشتقات 5- فينوكسي-3h-بيريميدين-4-أون واستخدامها كمثبطات ناسخ عكسي ل hiv
CN104994855B (zh) * 2012-12-05 2018-06-05 默沙东公司 制备逆转录酶抑制剂的方法
EP3071037A4 (en) * 2013-11-22 2017-08-02 Merck Sharp & Dohme Corp. Composition of a non-nucleoside reverse transcriptase inhibitor
KR101803671B1 (ko) * 2013-12-04 2017-11-30 머크 샤프 앤드 돔 코포레이션 역전사효소 억제제의 제조 방법
SI3125894T1 (sl) 2014-04-01 2020-12-31 Merck Sharp & Dohme Corp. Predzdravila inhibitorjev reverzne transkriptaze HIV
EP3161159B1 (en) 2014-06-25 2020-08-05 The General Hospital Corporation Targeting human satellite ii (hsatii)
RU2736941C2 (ru) 2015-12-02 2020-11-23 Мерк Шарп энд Доум Корп. Фармацевтические композиции, содержащие доравирин, тенофовира дизопроксила фумарат и ламивудин
WO2018175271A1 (en) * 2017-03-24 2018-09-27 Merck Sharp & Dohme Corp. Formulation for parenteral administration
RU2019136678A (ru) 2017-04-18 2021-05-18 Сипла Лимитед Комбинированная терапия для применения в лечении ретровирусных инфекций
EP4317972A3 (en) 2018-02-06 2024-03-13 The General Hospital Corporation Repeat rna as biomarkers of tumor immune response
WO2020018352A1 (en) 2018-07-17 2020-01-23 Merck Sharp & Dohme Corp. Hiv drug combination for increasing barrier against resistance
MX2021007382A (es) 2018-12-18 2021-07-15 Merck Sharp & Dohme Llc Derivados de pirimidona como agentes citotoxicos selectivos contra celulas infectadas por vih.
CN110801455B (zh) * 2019-11-12 2020-06-02 河北医科大学第二医院 用于治疗mrsa的药物组合物及其应用
CN114163309B (zh) * 2021-12-27 2023-04-25 甘肃皓天医药科技有限责任公司 一种多拉韦林中间体的制备方法
CN114349690B (zh) * 2022-02-15 2023-04-25 甘肃皓天医药科技有限责任公司 一种多拉韦林中间体合成方法
CN116903590A (zh) * 2023-06-06 2023-10-20 延边大学 一种含杂环结构的吡啶酮类化合物及其制备方法和用途
CN120157613A (zh) * 2023-12-15 2025-06-17 山东诚创蓝海医药科技有限公司 多拉韦林中间体及其应用和合成方法

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE9904045D0 (sv) 1999-11-09 1999-11-09 Astra Ab Compounds
TW200423930A (en) * 2003-02-18 2004-11-16 Hoffmann La Roche Non-nucleoside reverse transcriptase inhibitors
TW200505441A (en) * 2003-03-24 2005-02-16 Hoffmann La Roche Non-nucleoside reverse transcriptase inhibitorsⅠ
WO2004085406A1 (en) 2003-03-24 2004-10-07 F. Hoffmann-La Roche Ag Benzyl-pyridazinons as reverse transcriptase inhibitors
US7166738B2 (en) 2004-04-23 2007-01-23 Roche Palo Alto Llc Non-nucleoside reverse transcriptase inhibitors
AU2005235692B2 (en) 2004-04-23 2011-11-10 F. Hoffmann-La Roche Ag Non-nucleoside reverse transcriptase inhibitors
JP2008525419A (ja) 2004-12-22 2008-07-17 ファイザー・リミテッド Hiv−1逆転写酵素の非ヌクレオシド阻害剤
AR057455A1 (es) 2005-07-22 2007-12-05 Merck & Co Inc Inhibidores de la transcriptasa reversa de vih y composicion farmaceutica
ES2320042T3 (es) 2005-10-19 2009-05-18 F. Hoffmann-La Roche Ag Inhibidores de transcriptasa reversa con nucleosidos de n-fenil fenilacetamida.
EP1940781A1 (en) 2005-10-19 2008-07-09 F.Hoffmann-La Roche Ag Phenyl-acetamide nnrt inhibitors
TW200831085A (en) 2006-12-13 2008-08-01 Merck & Co Inc Non-nucleoside reverse transcriptase inhibitors
CN101952274A (zh) 2007-11-20 2011-01-19 默沙东公司 非核苷逆转录酶抑制剂
MX2012011379A (es) * 2010-03-30 2012-11-30 Merck Canada Inc Inhibidores no nucleosidicos de la transcriptasa inversa.

Also Published As

Publication number Publication date
EA024804B1 (ru) 2016-10-31
LUC00113I9 (lt) 2024-06-07
EP2552902A1 (en) 2013-02-06
AR080859A1 (es) 2012-05-16
CY2019026I1 (el) 2020-05-29
CR20120503A (es) 2013-01-09
KR20120128703A (ko) 2012-11-27
NL300980I2 (nl) 2021-06-17
CY2019025I2 (el) 2019-11-27
IL222030A (en) 2014-07-31
US20110245296A1 (en) 2011-10-06
HUS1900022I1 (hu) 2019-05-28
KR101421861B1 (ko) 2014-07-22
CY2019025I1 (el) 2019-11-27
EA201290976A1 (ru) 2013-03-29
IL233334A (en) 2015-09-24
CO6630126A2 (es) 2013-03-01
EP2552902B1 (en) 2015-03-11
TN2012000455A1 (en) 2014-01-30
EP2924034A1 (en) 2015-09-30
NO2019018I1 (no) 2019-04-24
BR112012024691B1 (pt) 2020-11-17
GEP20156368B (en) 2015-09-25
PL2552902T3 (pl) 2015-10-30
PT2924034T (pt) 2017-01-06
LT2924034T (lt) 2016-12-27
PT2552902E (pt) 2015-06-02
HK1175471A1 (en) 2013-07-05
JP2013209405A (ja) 2013-10-10
DK2924034T3 (en) 2017-02-06
ECSP12012201A (es) 2012-10-30
HRP20161680T1 (hr) 2017-01-27
HN2012002039A (es) 2015-08-24
SI2924034T1 (sl) 2017-05-31
SI2552902T1 (sl) 2015-10-30
CN102971308B (zh) 2015-02-04
MX2012011379A (es) 2012-11-30
AU2011235568A1 (en) 2012-11-01
SG184347A1 (en) 2012-11-29
NO2019019I1 (no) 2019-04-24
JP2013510800A (ja) 2013-03-28
HUE025336T2 (en) 2016-03-29
AU2011235568B2 (en) 2013-09-12
ES2536295T3 (es) 2015-05-22
MY163979A (en) 2017-11-15
CN102971308A (zh) 2013-03-13
LTC2924034I2 (lt) 2020-10-12
TWI458719B (zh) 2014-11-01
TW201139409A (en) 2011-11-16
PH12012501923A1 (en) 2013-02-04
BR112012024691A2 (pt) 2019-07-02
CA2794377A1 (en) 2011-10-06
HUS1900021I1 (hu) 2019-05-28
LTPA2019506I1 (lt) 2019-04-25
EP2924034B1 (en) 2016-11-02
HUE031785T2 (en) 2017-08-28
HK1209121A1 (en) 2016-03-24
CA2794377C (en) 2015-06-16
PL2924034T3 (pl) 2017-07-31
LTPA2019507I1 (lt) 2019-04-25
US8486975B2 (en) 2013-07-16
JP5886790B2 (ja) 2016-03-16
NL300980I1 (nl) 2019-04-24
ME02181B (me) 2015-10-20
HRP20150427T1 (hr) 2015-07-03
RS55505B1 (sr) 2017-05-31
ES2609636T3 (es) 2017-04-21
CY1118774T1 (el) 2017-07-12
LUC00114I1 (lt) 2019-04-17
EP2552902A4 (en) 2013-09-04
ME02570B (me) 2017-06-20
DOP2012000256A (es) 2012-12-15
NZ602670A (en) 2014-09-26
FIC20190021I1 (fi) 2019-04-17
LUC00113I2 (lt) 2024-05-22
LUC00114I2 (lt) 2020-07-10
CY2019026I2 (el) 2020-05-29
PE20130158A1 (es) 2013-02-28
JP5281718B2 (ja) 2013-09-04
WO2011120133A1 (en) 2011-10-06
IL233334A0 (en) 2014-09-01
CL2012002744A1 (es) 2012-12-14
DK2552902T3 (en) 2015-06-15
MA34170B1 (fr) 2013-04-03
NI201200146A (es) 2013-03-18
RS54017B1 (sr) 2015-10-30
US20130296382A1 (en) 2013-11-07

Similar Documents

Publication Publication Date Title
LTPA2019506I1 (lt) Nenukleozidinės reversinės transkriptazės inhibitoriai
FR25C1006I2 (fr) Inhibiteurs de pyrazolyl-quinoxaline kinase
EP2604688A4 (en) VARIANTE REVERSE TRANSKRIPTASE
SMT201500271B (it) Inibitori di neprilisina
HRP20181786T1 (hr) Inhibitori aktivacije t-stanica
IL237582A0 (en) Cdk inhibitors
DK2371923T3 (da) Aflejringshæmmer
DK2448938T3 (da) Pyrimidinoner som pi3k-inhibitorer
DK2710007T3 (da) Kinasehæmmere
LT2841428T (lt) Dnr-pk inhibitoriai
DK3196202T3 (da) Heterocyclylaminer som pi3k-inhibitorer
EP2554796A4 (en) TURBINE
DK2920149T3 (da) 3-aminocycloalkyl-forbindelser som ror-gamma-t-inhibitorer og anvendelser deraf
DK2421825T3 (da) Azetidinyldiamider som monoacylglycerollipase-inhibitorer
EP4300014C0 (en) FRIDGE
EP2540987A4 (en) TURBINE
BR112013025761A2 (pt) inibidores de hsp90
EP2563127A4 (en) PROLYLCARBOXYPEPTIDASE INHIBITORS
EP2549107A4 (en) Freezing machine
BR112012019494A2 (pt) dispositivo elétrico
EP2663574A4 (en) RETRO VIRUS REPLICATION INHIBITORS
BR112013005966A2 (pt) refrigerador
RU2016124545A (ru) Композиция ненуклеозидного ингибитора обратной транскриптазы
DK2564056T3 (da) Turbine
BR112013012958A2 (pt) inibidores integrin ligado com quinase