LU92636I2 - Zolpidem et ses sels pharmaceutiquement acceptables - Google Patents

Zolpidem et ses sels pharmaceutiquement acceptables Download PDF

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Publication number
LU92636I2
LU92636I2 LU92636C LU92636C LU92636I2 LU 92636 I2 LU92636 I2 LU 92636I2 LU 92636 C LU92636 C LU 92636C LU 92636 C LU92636 C LU 92636C LU 92636 I2 LU92636 I2 LU 92636I2
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LU
Luxembourg
Prior art keywords
zolpidem
pharmaceutically acceptable
acceptable salts
microparticles
bioadhesion
Prior art date
Application number
LU92636C
Other languages
English (en)
Original Assignee
Orexo Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=20412702&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=LU92636(I2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Orexo Ab filed Critical Orexo Ab
Publication of LU92636I2 publication Critical patent/LU92636I2/fr

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/006—Oral mucosa, e.g. mucoadhesive forms, sublingual droplets; Buccal patches or films; Buccal sprays
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/136—Amines having aromatic rings, e.g. ketamine, nortriptyline having the amino group directly attached to the aromatic ring, e.g. benzeneamine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19—Carboxylic acids, e.g. valproic acid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19—Carboxylic acids, e.g. valproic acid
    • A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/196—Carboxylic acids, e.g. valproic acid having an amino group the amino group being directly attached to a ring, e.g. anthranilic acid, mefenamic acid, diclofenac, chlorambucil
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/34—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
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    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/34—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
    • A61K31/341—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide not condensed with another ring, e.g. ranitidine, furosemide, bufetolol, muscarine
    • A—HUMAN NECESSITIES
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    • A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/5415—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with carbocyclic ring systems, e.g. phenothiazine, chlorpromazine, piroxicam
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    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
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  • Proteomics, Peptides & Aminoacids (AREA)
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LU92636C 1998-09-24 2015-01-20 Zolpidem et ses sels pharmaceutiquement acceptables LU92636I2 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
SE9803240A SE9803240D0 (sv) 1998-09-24 1998-09-24 A pharmaceutical composition having a rapid action

Publications (1)

Publication Number Publication Date
LU92636I2 true LU92636I2 (fr) 2015-03-20

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ID=20412702

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Application Number Title Priority Date Filing Date
LU92636C LU92636I2 (fr) 1998-09-24 2015-01-20 Zolpidem et ses sels pharmaceutiquement acceptables

Country Status (29)

Country Link
US (8) US6761910B1 (fr)
EP (5) EP1652518B1 (fr)
JP (1) JP3381220B2 (fr)
KR (1) KR100760536B1 (fr)
CN (1) CN1173694C (fr)
AT (1) ATE365540T1 (fr)
AU (1) AU764346B2 (fr)
BG (1) BG65502B1 (fr)
BR (1) BRPI9913945B8 (fr)
CA (3) CA2820588C (fr)
CY (5) CY1107711T1 (fr)
CZ (2) CZ2008315A3 (fr)
DE (1) DE69936393T2 (fr)
DK (5) DK1115383T3 (fr)
EE (3) EE05555B1 (fr)
ES (5) ES2507579T3 (fr)
HU (2) HU230468B1 (fr)
IL (1) IL142135A0 (fr)
LU (1) LU92636I2 (fr)
MX (1) MXPA01003068A (fr)
NO (1) NO332226B1 (fr)
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US7910132B2 (en) 2011-03-22
PT2236132E (pt) 2014-07-31
EP2236133A1 (fr) 2010-10-06
IL142135A0 (en) 2002-03-10
TR200100855T2 (tr) 2001-10-22
PT2236133E (pt) 2014-07-16
CY1107711T1 (el) 2013-04-18
EP2805716A1 (fr) 2014-11-26
HU0800435D0 (en) 2008-09-29
CA2629988C (fr) 2014-01-07
CN1326340A (zh) 2001-12-12
EE05555B1 (et) 2012-08-15
CA2345121C (fr) 2008-06-10
AU6492799A (en) 2000-04-10
HUP0103856A2 (hu) 2002-02-28
JP3381220B2 (ja) 2003-02-24
EE200800028A (et) 2008-08-15
RU2193879C1 (ru) 2002-12-10
ES2289829T3 (es) 2008-02-01
NO20011473L (no) 2001-05-23
US20080286368A1 (en) 2008-11-20
ES2507579T3 (es) 2014-10-15
EE04927B1 (et) 2007-12-17
EP2236132A1 (fr) 2010-10-06
HUP0103856A3 (en) 2003-11-28
EP1115383A1 (fr) 2001-07-18
HK1148457A1 (en) 2011-09-09
KR20010075315A (ko) 2001-08-09
CA2345121A1 (fr) 2000-03-30
CY1114620T1 (el) 2016-10-05
EP1652518B1 (fr) 2013-08-07
CY1115688T1 (el) 2017-01-25
EE200700030A (et) 2007-08-15
SK4022001A3 (en) 2001-11-06
DK2236132T3 (da) 2014-08-04
HU230342B1 (hu) 2016-02-29
US20140030336A1 (en) 2014-01-30
US20040213855A1 (en) 2004-10-28
DE69936393D1 (de) 2007-08-09

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