MA31338B1 - Agent thérapeutique pour une affection abdominale inflammatoire qui comprend un dérivé de 2-amino-1,3-propanediol en tant qu'ingrédient actif et procédé pour le traitement d'une affection abdominale inflammatoire - Google Patents

Agent thérapeutique pour une affection abdominale inflammatoire qui comprend un dérivé de 2-amino-1,3-propanediol en tant qu'ingrédient actif et procédé pour le traitement d'une affection abdominale inflammatoire

Info

Publication number
MA31338B1
MA31338B1 MA31196A MA31196A MA31338B1 MA 31338 B1 MA31338 B1 MA 31338B1 MA 31196 A MA31196 A MA 31196A MA 31196 A MA31196 A MA 31196A MA 31338 B1 MA31338 B1 MA 31338B1
Authority
MA
Morocco
Prior art keywords
inflammatory bowel
bowel disease
amino
disease
derivative
Prior art date
Application number
MA31196A
Other languages
Arabic (ar)
English (en)
Inventor
Ryotaro Kojima
Koichi Nakamaru
Tokutarou Yasue
Original Assignee
Kyorin Seiyaku Kk
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=38345101&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MA31338(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Kyorin Seiyaku Kk filed Critical Kyorin Seiyaku Kk
Publication of MA31338B1 publication Critical patent/MA31338B1/fr

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/137—Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Emergency Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

L'invention concerne un dérivé de 2-amino-1,3-propanediol représenté par la formule (1) (par exemple le chlorhydrate de 2-amino-2-[4-(3-benzyloxyphénylthio)-2-chlorophényl]éthyl-1,3-propanediol), qui est un agoniste du récepteur de la sphingosine-1-phosphate, ou un sel ou solvate acceptable du point de vue pharmaceutique de celui-ci. Il apparaît que le dérivé, le sel ou le solvate est utile en tant qu'agent thérapeutique ou agent prophylactique pour une affection abdominale inflammatoire telle que la maladie de crohn, la maladie de crohn du gros intestin, la maladie de behcet intestinale, la rectocolite hémorragique, l'ulcère rectal hémorragique ou la pochite.
MA31196A 2006-02-06 2008-08-26 Agent thérapeutique pour une affection abdominale inflammatoire qui comprend un dérivé de 2-amino-1,3-propanediol en tant qu'ingrédient actif et procédé pour le traitement d'une affection abdominale inflammatoire MA31338B1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2006027883 2006-02-06
PCT/JP2007/051887 WO2007091501A1 (fr) 2006-02-06 2007-02-05 Agent thérapeutique pour une affection abdominale inflammatoire qui comprend un dérivé de 2-amino-1,3-propanediol en tant qu'ingrédient actif et procédé pour le traitement d'une affection abdominale inflammatoire

Publications (1)

Publication Number Publication Date
MA31338B1 true MA31338B1 (fr) 2010-05-03

Family

ID=38345101

Family Applications (1)

Application Number Title Priority Date Filing Date
MA31196A MA31338B1 (fr) 2006-02-06 2008-08-26 Agent thérapeutique pour une affection abdominale inflammatoire qui comprend un dérivé de 2-amino-1,3-propanediol en tant qu'ingrédient actif et procédé pour le traitement d'une affection abdominale inflammatoire

Country Status (29)

Country Link
US (1) US8318811B2 (fr)
EP (2) EP2520291A1 (fr)
JP (1) JP5042042B2 (fr)
KR (1) KR101334153B1 (fr)
CN (1) CN101378743B (fr)
AU (1) AU2007213194B9 (fr)
BR (1) BRPI0706971A2 (fr)
CA (1) CA2641546C (fr)
CY (1) CY1116112T1 (fr)
DK (1) DK1982708T3 (fr)
EC (1) ECSP088662A (fr)
ES (1) ES2524056T3 (fr)
GT (1) GT200800148A (fr)
HR (1) HRP20080421B1 (fr)
IL (1) IL192150A (fr)
MA (1) MA31338B1 (fr)
MX (1) MX2008008872A (fr)
MY (1) MY151193A (fr)
NO (1) NO20082708L (fr)
NZ (1) NZ568907A (fr)
PL (1) PL1982708T3 (fr)
PT (1) PT1982708E (fr)
RU (1) RU2428976C2 (fr)
SG (1) SG169370A1 (fr)
SI (1) SI1982708T1 (fr)
TN (1) TNSN08246A1 (fr)
TW (1) TWI389683B (fr)
WO (1) WO2007091501A1 (fr)
ZA (1) ZA200806199B (fr)

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TWI389683B (zh) 2006-02-06 2013-03-21 Kyorin Seiyaku Kk A therapeutic agent for an inflammatory bowel disease or an inflammatory bowel disease treatment using a 2-amino-1,3-propanediol derivative as an active ingredient
JP5140593B2 (ja) 2006-08-08 2013-02-06 杏林製薬株式会社 アミノアルコール誘導体及びそれらを有効成分とする免疫抑制剤
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TW200946105A (en) 2008-02-07 2009-11-16 Kyorin Seiyaku Kk Therapeutic agent or preventive agent for inflammatory bowel disease containing amino alcohol derivative as active ingredient
EP2305305A4 (fr) * 2008-05-20 2013-02-13 Kyorin Seiyaku Kk Agent d'induction/d'entretien de rémission
HRP20161133T1 (hr) 2008-07-23 2016-12-02 Arena Pharmaceuticals, Inc. DERIVATI SUSPSTITUIRANE 1,2,3,4-TETRAHIDROCIKLOPENTA[b]INDOL-3-IL-OCTENE KISELINE KORISNI U LIJEČENJU AUTOIMUNIH I UPALNIH POREMEĆAJA
CN105816453B (zh) 2008-08-27 2021-03-05 艾尼纳制药公司 用于治疗自身免疫性病症和炎性病症的作为s1p1受体激动剂的经取代的三环酸衍生物
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KR101787543B1 (ko) 2014-08-22 2017-10-19 샘표식품 주식회사 발효배양 산삼을 포함하는 항염증 조성물
AU2016205361C1 (en) 2015-01-06 2021-04-08 Arena Pharmaceuticals, Inc. Methods of treating conditions related to the S1P1 receptor
PL3310760T3 (pl) 2015-06-22 2023-03-06 Arena Pharmaceuticals, Inc. Krystaliczna sól L-argininy kwasu (R)-2-(7-(4-cyklopentylo-3-(trifluorometylo)benzyloksy)- 1,2,3,4-tetrahydrocyklo-penta[b]indol-3-ilo)octowego do zastosowania w zaburzeniach związanych z receptorem S1P1
JP2020507610A (ja) 2017-02-16 2020-03-12 アリーナ ファーマシューティカルズ， インコーポレイテッド 腸管外症状を伴う炎症性腸疾患の治療のための化合物および方法
KR20190116416A (ko) 2017-02-16 2019-10-14 아레나 파마슈티칼스, 인크. 원발 담즙성 담관염을 치료하기 위한 화합물 및 방법
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CN112512516A (zh) 2018-07-27 2021-03-16 普瑞奥治疗有限公司 用于在已经经历造血干细胞移植的患者中抑制血液恶性肿瘤复发的活性剂
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TWI389683B (zh) 2013-03-21
NO20082708L (no) 2008-09-02
IL192150A (en) 2015-04-30
PT1982708E (pt) 2014-12-23
AU2007213194A1 (en) 2007-08-16
DK1982708T3 (en) 2014-12-01
AU2007213194B9 (en) 2013-05-16
ECSP088662A (es) 2008-09-29
CN101378743B (zh) 2014-05-28
MY151193A (en) 2014-04-30
HK1126119A1 (en) 2009-08-28
JP5042042B2 (ja) 2012-10-03
HRP20080421B1 (hr) 2015-07-17
EP1982708B1 (fr) 2014-11-05
US20090137685A1 (en) 2009-05-28
SI1982708T1 (sl) 2015-01-30
EP2520291A1 (fr) 2012-11-07
HRP20080421A2 (en) 2008-12-31
MX2008008872A (es) 2008-10-23
WO2007091501A1 (fr) 2007-08-16
CY1116112T1 (el) 2017-02-08
GT200800148A (es) 2008-10-29
KR101334153B1 (ko) 2013-11-28
TW200806281A (en) 2008-02-01
BRPI0706971A2 (pt) 2011-09-27
EP1982708A4 (fr) 2010-03-17
AU2007213194B2 (en) 2013-03-14
EP1982708A1 (fr) 2008-10-22
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NZ568907A (en) 2011-08-26
IL192150A0 (en) 2008-12-29
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JPWO2007091501A1 (ja) 2009-07-02
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CA2641546A1 (fr) 2007-08-16
RU2008135264A (ru) 2010-03-20
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US8318811B2 (en) 2012-11-27
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PL1982708T3 (pl) 2015-03-31
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