MA38385A1 - Nouvelle composition pour la stéatose hépatique non alcoolique (nafld) - Google Patents
Nouvelle composition pour la stéatose hépatique non alcoolique (nafld)Info
- Publication number
- MA38385A1 MA38385A1 MA38385A MA38385A MA38385A1 MA 38385 A1 MA38385 A1 MA 38385A1 MA 38385 A MA38385 A MA 38385A MA 38385 A MA38385 A MA 38385A MA 38385 A1 MA38385 A1 MA 38385A1
- Authority
- MA
- Morocco
- Prior art keywords
- nafld
- liver disease
- fatty liver
- alcoholic fatty
- new composition
- Prior art date
Links
- 208000008338 non-alcoholic fatty liver disease Diseases 0.000 title abstract 3
- 150000001875 compounds Chemical class 0.000 abstract 3
- 210000004185 liver Anatomy 0.000 abstract 2
- 206010016654 Fibrosis Diseases 0.000 abstract 1
- 230000007882 cirrhosis Effects 0.000 abstract 1
- 208000019425 cirrhosis of liver Diseases 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 208000035475 disorder Diseases 0.000 abstract 1
- 206010053219 non-alcoholic steatohepatitis Diseases 0.000 abstract 1
- 230000037390 scarring Effects 0.000 abstract 1
- 230000007863 steatosis Effects 0.000 abstract 1
- 231100000240 steatosis hepatitis Toxicity 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Gastroenterology & Hepatology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicinal Preparation (AREA)
Abstract
La présente invention concerne un composé de formule (i) ou un produit pharmaceutique acceptable correspondant, où 'r' est décrit dans la description. De plus, l'invention concerne une composition comprenant une quantité thérapeutique efficace du composé de formule (i) et des procédés d'utilisation des composés pour traiter ou prévenir des troubles tels que la stéatose hépatique non alcoolique (nafld) comprenant le foie stéatosique (stéatose), la stéatohépatite non alcoolique (nash) et la cirrhose (cicatrisation avancée du foie).
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IN1468MU2013 IN2013MU01468A (fr) | 2013-04-22 | 2013-06-25 | |
| PCT/IN2013/000391 WO2014174524A1 (fr) | 2013-04-22 | 2013-06-25 | Nouvelle composition pour la stéatose hépatique non alcoolique (nafld) |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MA38385A1 true MA38385A1 (fr) | 2017-09-29 |
Family
ID=49253372
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MA38385A MA38385A1 (fr) | 2013-04-22 | 2013-06-25 | Nouvelle composition pour la stéatose hépatique non alcoolique (nafld) |
Country Status (21)
| Country | Link |
|---|---|
| US (3) | US20160166539A1 (fr) |
| EP (1) | EP2988736A1 (fr) |
| JP (1) | JP6246895B2 (fr) |
| KR (1) | KR101617812B1 (fr) |
| CN (1) | CN105377246B (fr) |
| AP (1) | AP2015008674A0 (fr) |
| AU (1) | AU2013387996B2 (fr) |
| BR (1) | BR112015020600A2 (fr) |
| CA (1) | CA2900435C (fr) |
| EA (1) | EA201592020A1 (fr) |
| GE (1) | GEP201706663B (fr) |
| HK (1) | HK1214968A1 (fr) |
| IL (2) | IL240183A (fr) |
| IN (1) | IN2013MU01468A (fr) |
| MA (1) | MA38385A1 (fr) |
| MX (1) | MX346943B (fr) |
| MY (1) | MY180160A (fr) |
| PH (1) | PH12015501795A1 (fr) |
| SG (1) | SG11201506218UA (fr) |
| UA (1) | UA114360C2 (fr) |
| WO (1) | WO2014174524A1 (fr) |
Families Citing this family (20)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR101633720B1 (ko) | 2011-01-31 | 2016-06-27 | 카딜라 핼쓰캐어 리미티드 | 지방이상증의 치료 |
| US20130158077A1 (en) | 2011-12-19 | 2013-06-20 | Ares Trading S.A. | Pharmaceutical compositions |
| UA114360C2 (uk) | 2013-04-22 | 2017-05-25 | Каділа Хелткере Лімітед | Спосіб лікування та/або зменшення інтенсивності неалкогольної жирової хвороби печінки (нжхп) |
| US20160107989A1 (en) | 2013-05-30 | 2016-04-21 | Cadila Healthcare Limited | A process for preparation of pyrroles having hypolipidemic hypocholesteremic activities |
| TW201513857A (zh) | 2013-07-05 | 2015-04-16 | Cadila Healthcare Ltd | 協同性組成物 |
| IN2013MU02470A (fr) * | 2013-07-25 | 2015-06-26 | Cadila Healthcare Ltd | |
| IN2013MU02905A (fr) | 2013-09-06 | 2015-07-03 | Cadila Healthcare Ltd | |
| US10385017B2 (en) | 2015-10-14 | 2019-08-20 | Cadila Healthcare Limited | Pyrrole compound, compositions and process for preparation thereof |
| CN117137917A (zh) * | 2016-04-22 | 2023-12-01 | 景凯生物科技股份有限公司 | 纳美芬、纳曲酮或其衍生物在治疗(非)酒精性脂肪肝炎或非酒精性脂肪性肝病的应用 |
| MX382765B (es) * | 2016-12-09 | 2025-03-13 | Zydus Lifesciences Ltd | Tratamiento para la colangitis biliar primaria. |
| SI4122464T1 (sl) | 2017-03-28 | 2024-07-31 | Gilead Sciences, Inc. | Terapevtske kombinacije za zdravljenje bolezni jeter |
| GB201710229D0 (en) | 2017-06-27 | 2017-08-09 | Tdeltas Ltd | Compounds for new use |
| US10980810B2 (en) * | 2017-10-06 | 2021-04-20 | Gilead Sciences, Inc. | Combination therapy comprising an ACC inhibitor |
| CN109675016A (zh) * | 2017-10-18 | 2019-04-26 | 上海贺普药业股份有限公司 | 非酒精性脂肪性肝病的治疗药物 |
| CN110934866B (zh) * | 2018-09-25 | 2023-12-01 | 深圳微芯生物科技股份有限公司 | 西格列羧及其相关化合物的应用 |
| US12201609B2 (en) * | 2018-12-18 | 2025-01-21 | Zydus Lifesciences Limited | Saroglitazar for the treatment of hepatocellular carcinoma |
| EP3923932A4 (fr) * | 2019-02-13 | 2022-11-16 | Cadila Healthcare Limited | Traitement du syndrome des ovaires polykystiques (pcos) |
| WO2022128870A1 (fr) * | 2020-12-18 | 2022-06-23 | Société des Produits Nestlé S.A. | Compositions et procédés utilisant au moins une glycine ou un dérivé de celle-ci et/ou au moins une n-acétylcystéine ou un dérivé de celle-ci, et au moins un thymol et/ou du carvacrol |
| WO2022246243A1 (fr) * | 2021-05-21 | 2022-11-24 | HepQuant, LLC | Procédés de définition d'un changement fonctionnel et de ralentissement de la progression dans une maladie hépatique chronique |
| WO2025238663A1 (fr) * | 2024-05-16 | 2025-11-20 | Zydus Lifesciences Limited | Saroglitazar pour le traitement de maladies hépatiques alcooliques |
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| US4444784A (en) | 1980-08-05 | 1984-04-24 | Merck & Co., Inc. | Antihypercholesterolemic compounds |
| DK149080C (da) | 1980-06-06 | 1986-07-28 | Sankyo Co | Fremgangsmaade til fremstilling af derivater af ml-236b-carboxylsyre |
| US5354772A (en) | 1982-11-22 | 1994-10-11 | Sandoz Pharm. Corp. | Indole analogs of mevalonolactone and derivatives thereof |
| FI94339C (fi) | 1989-07-21 | 1995-08-25 | Warner Lambert Co | Menetelmä farmaseuttisesti käyttökelpoisen /R-(R*,R*)/-2-(4-fluorifenyyli)- , -dihydroksi-5-(1-metyylietyyli)-3-fenyyli-4-/(fenyyliamino)karbonyyli/-1H-pyrroli-1-heptaanihapon ja sen farmaseuttisesti hyväksyttävien suolojen valmistamiseksi |
| US5089514A (en) | 1990-06-14 | 1992-02-18 | Pfizer Inc. | 3-coxazolyl [phenyl, chromanyl or benzofuranyl]-2-hydroxypropionic acid derivatives and analogs as hypoglycemic agents |
| CZ1095A3 (en) | 1992-07-03 | 1995-10-18 | Smithkline Beecham Plc | Heterocyclic compounds, process of their preparation, their use for the preparation of a pharmaceutical preparation and the pharmaceutical composition containing thereof |
| GB9225386D0 (en) | 1992-12-04 | 1993-01-27 | Smithkline Beecham Plc | Novel compounds |
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| EP1123269A1 (fr) | 1998-10-21 | 2001-08-16 | Novo Nordisk A/S | Nouveaux composes, leur preparation et leur utilisation |
| WO2000023451A1 (fr) | 1998-10-21 | 2000-04-27 | Novo Nordisk A/S | Nouveaux composes, leur preparation et leur utilisation |
| EP1123292A1 (fr) | 1998-10-21 | 2001-08-16 | Novo Nordisk A/S | Nouveaux composes, leur preparation et leur utilisation |
| CO5150173A1 (es) | 1998-12-10 | 2002-04-29 | Novartis Ag | Compuestos n-(glicilo sustituido)-2-cianopirrolidinas inhibidores de peptidasa de dipeptidilo-iv (dpp-iv) los cuales son efectivos en el tratamiento de condiciones mediadas por la inhibicion de dpp-iv |
| ES2449194T3 (es) | 2000-01-19 | 2014-03-18 | Cadila Healthcare Limited | Compuestos que tienen actividades hipolipidémica e hipocolesterolémica, procedimiento para su preparación y composiciones farmacéuticas que los contienen |
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| WO2002024625A2 (fr) | 2000-09-22 | 2002-03-28 | Dr. Reddy's Research Foundation | Procede ameliore pour la preparation de derives d'acide 3-aryl-2-hydroxy propanoique |
| UA74912C2 (en) | 2001-07-06 | 2006-02-15 | Merck & Co Inc | Beta-aminotetrahydroimidazo-(1,2-a)-pyrazines and tetratriazolo-(4,3-a)-pyrazines as inhibitors of dipeptylpeptidase for the treatment or prevention of diabetes |
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| US7407955B2 (en) | 2002-08-21 | 2008-08-05 | Boehringer Ingelheim Pharma Gmbh & Co., Kg | 8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions |
| US20070051626A1 (en) | 2003-09-26 | 2007-03-08 | Chiho Itou | Cataphoresis apparatus cataphoresis method, and detection method for organism-related material using the apparatus and the method |
| UA85871C2 (uk) | 2004-03-15 | 2009-03-10 | Такеда Фармасьютікал Компані Лімітед | Інгібітори дипептидилпептидази |
| CA2623762A1 (fr) * | 2005-09-19 | 2007-03-29 | Johnson & Johnson Pharmaceutical Research & Development, L.L.C. | Modulation de l'expression du recepteur du glucagon |
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| JP2008184429A (ja) * | 2007-01-30 | 2008-08-14 | Japan Health Science Foundation | 肝臓トリグリセリド濃度低下剤 |
| LT2641596T (lt) | 2009-11-26 | 2018-08-10 | Genfit | 1,3-difenilprop-2-en-1-ono darinių panaudojimas kepenų sutrikimų gydymui |
| EP2627323A4 (fr) | 2010-10-12 | 2014-03-12 | Univ Johns Hopkins | Compositions antitussives comprenant de la mémantine |
| KR101633720B1 (ko) * | 2011-01-31 | 2016-06-27 | 카딜라 핼쓰캐어 리미티드 | 지방이상증의 치료 |
| UA114360C2 (uk) | 2013-04-22 | 2017-05-25 | Каділа Хелткере Лімітед | Спосіб лікування та/або зменшення інтенсивності неалкогольної жирової хвороби печінки (нжхп) |
| US20160107989A1 (en) | 2013-05-30 | 2016-04-21 | Cadila Healthcare Limited | A process for preparation of pyrroles having hypolipidemic hypocholesteremic activities |
| TW201513857A (zh) | 2013-07-05 | 2015-04-16 | Cadila Healthcare Ltd | 協同性組成物 |
| IN2013MU02470A (fr) | 2013-07-25 | 2015-06-26 | Cadila Healthcare Ltd | |
| US9951009B2 (en) | 2013-08-29 | 2018-04-24 | Cadila Healthcare Limited | Polymorphic form of pyrrole derivative and intermediate thereof |
| IN2013MU02905A (fr) | 2013-09-06 | 2015-07-03 | Cadila Healthcare Ltd |
-
2013
- 2013-06-25 UA UAA201509744A patent/UA114360C2/uk unknown
- 2013-06-25 EP EP13767126.9A patent/EP2988736A1/fr not_active Withdrawn
- 2013-06-25 JP JP2016505927A patent/JP6246895B2/ja active Active
- 2013-06-25 KR KR1020157024370A patent/KR101617812B1/ko active Active
- 2013-06-25 GE GEAP201313941A patent/GEP201706663B/en unknown
- 2013-06-25 MX MX2015010769A patent/MX346943B/es active IP Right Grant
- 2013-06-25 MY MYPI2015002026A patent/MY180160A/en unknown
- 2013-06-25 IN IN1468MU2013 patent/IN2013MU01468A/en unknown
- 2013-06-25 WO PCT/IN2013/000391 patent/WO2014174524A1/fr not_active Ceased
- 2013-06-25 US US14/782,609 patent/US20160166539A1/en not_active Abandoned
- 2013-06-25 MA MA38385A patent/MA38385A1/fr unknown
- 2013-06-25 EA EA201592020A patent/EA201592020A1/ru unknown
- 2013-06-25 BR BR112015020600A patent/BR112015020600A2/pt not_active IP Right Cessation
- 2013-06-25 CA CA2900435A patent/CA2900435C/fr not_active Expired - Fee Related
- 2013-06-25 AP AP2015008674A patent/AP2015008674A0/xx unknown
- 2013-06-25 SG SG11201506218UA patent/SG11201506218UA/en unknown
- 2013-06-25 AU AU2013387996A patent/AU2013387996B2/en not_active Ceased
- 2013-06-25 CN CN201380075905.9A patent/CN105377246B/zh active Active
- 2013-06-25 HK HK16103017.5A patent/HK1214968A1/zh unknown
-
2015
- 2015-07-28 IL IL240183A patent/IL240183A/en not_active IP Right Cessation
- 2015-08-14 PH PH12015501795A patent/PH12015501795A1/en unknown
-
2016
- 2016-08-11 IL IL247231A patent/IL247231A/en not_active IP Right Cessation
- 2016-11-04 US US15/343,859 patent/US9814697B2/en active Active
-
2017
- 2017-11-02 US US15/801,738 patent/US20180185330A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| IL240183A0 (en) | 2015-09-24 |
| US20160166539A1 (en) | 2016-06-16 |
| CA2900435C (fr) | 2017-02-14 |
| MY180160A (en) | 2020-11-23 |
| AU2013387996A1 (en) | 2015-09-24 |
| UA114360C2 (uk) | 2017-05-25 |
| IL247231A (en) | 2017-03-30 |
| CN105377246A (zh) | 2016-03-02 |
| JP2016515608A (ja) | 2016-05-30 |
| IL240183A (en) | 2016-08-31 |
| PH12015501795A1 (en) | 2015-11-09 |
| MX346943B (es) | 2017-04-06 |
| MX2015010769A (es) | 2015-11-26 |
| US20180185330A1 (en) | 2018-07-05 |
| CN105377246B (zh) | 2018-03-20 |
| BR112015020600A2 (pt) | 2017-07-18 |
| KR20150118990A (ko) | 2015-10-23 |
| WO2014174524A8 (fr) | 2015-10-01 |
| CA2900435A1 (fr) | 2014-10-30 |
| US9814697B2 (en) | 2017-11-14 |
| GEP201706663B (en) | 2017-05-10 |
| KR101617812B1 (ko) | 2016-05-03 |
| JP6246895B2 (ja) | 2017-12-13 |
| WO2014174524A1 (fr) | 2014-10-30 |
| IN2013MU01468A (fr) | 2015-04-17 |
| EA201592020A1 (ru) | 2016-05-31 |
| US20170087127A1 (en) | 2017-03-30 |
| AP2015008674A0 (en) | 2015-08-31 |
| EP2988736A1 (fr) | 2016-03-02 |
| SG11201506218UA (en) | 2015-09-29 |
| HK1214968A1 (zh) | 2016-08-12 |
| AU2013387996B2 (en) | 2015-12-10 |
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