NO166860C - Analogifremgangsmaate for fremstilling av terapeutisk aktive monosulfaktamer. - Google Patents

Analogifremgangsmaate for fremstilling av terapeutisk aktive monosulfaktamer.

Info

Publication number: NO166860C
Authority: NO; Norway
Prior art keywords: sub; monosulfactures; preparation; therapeutically active; analogy procedure
Prior art date: 1986-01-06

Application number

NO870031A

Other languages

English (en)

Norwegian (no)

Other versions

NO870031L (no

NO870031D0 (no

NO166860B (no

Inventor

Joseph Edward Sundeen

Original Assignee

Squibb & Sons Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1986-01-06

Filing date

1987-01-05

Publication date

1991-09-11

1987-01-05 Application filed by Squibb & Sons Inc filed Critical Squibb & Sons Inc

1987-01-05 Publication of NO870031D0 publication Critical patent/NO870031D0/no

1987-07-07 Publication of NO870031L publication Critical patent/NO870031L/no

1990-12-13 Priority to NO905385A priority Critical patent/NO905385D0/no

1991-06-03 Publication of NO166860B publication Critical patent/NO166860B/no

1991-09-11 Publication of NO166860C publication Critical patent/NO166860C/no

Links

UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 1
230000003213 activating effect Effects 0.000 abstract 1
125000004442 acylamino group Chemical group 0.000 abstract 1
125000000217 alkyl group Chemical group 0.000 abstract 1
230000000844 anti-bacterial effect Effects 0.000 abstract 1
239000003782 beta lactam antibiotic agent Substances 0.000 abstract 1
229910052739 hydrogen Inorganic materials 0.000 abstract 1
239000001257 hydrogen Substances 0.000 abstract 1
125000002950 monocyclic group Chemical group 0.000 abstract 1
239000002132 β-lactam antibiotic Substances 0.000 abstract 1
229940124586 β-lactam antibiotics Drugs 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Oncology (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Communicable Diseases (AREA)
Public Health (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Agricultural Chemicals And Associated Chemicals (AREA)
Plural Heterocyclic Compounds (AREA)
Thiazole And Isothizaole Compounds (AREA)
Cephalosporin Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Medicines Containing Material From Animals Or Micro-Organisms (AREA)
Saccharide Compounds (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

NO870031A 1986-01-06 1987-01-05 Analogifremgangsmaate for fremstilling av terapeutisk aktive monosulfaktamer. NO166860C (no)

Priority Applications (1)

Application Number	Priority Date	Filing Date	Title
NO905385A NO905385D0 (no)	1986-01-06	1990-12-13	Tiazolderivater egnet som mellomprodukter ved fremstilling av terapeutisk aktive monosulfaktamer.

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US06/816,475 US4684722A (en)	1986-01-06	1986-01-06	Monosulfactams

Publications (4)

Publication Number	Publication Date
NO870031D0 NO870031D0 (no)	1987-01-05
NO870031L NO870031L (no)	1987-07-07
NO166860B NO166860B (no)	1991-06-03
NO166860C true NO166860C (no)	1991-09-11

Family

ID=25220721

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO870031A NO166860C (no)	1986-01-06	1987-01-05	Analogifremgangsmaate for fremstilling av terapeutisk aktive monosulfaktamer.

Country Status (21)

Country	Link
US (1)	US4684722A (da)
EP (1)	EP0229012B1 (da)
JP (1)	JPS62158278A (da)
KR (1)	KR900002244B1 (da)
AT (1)	ATE64393T1 (da)
AU (3)	AU602133B2 (da)
CA (1)	CA1308107C (da)
DD (3)	DD256700A5 (da)
DE (1)	DE3770644D1 (da)
DK (1)	DK3087A (da)
ES (1)	ES2038127T3 (da)
FI (1)	FI870030L (da)
GR (1)	GR3002312T3 (da)
HU (2)	HU198700B (da)
IL (1)	IL81153A (da)
NO (1)	NO166860C (da)
NZ (1)	NZ218682A (da)
PH (1)	PH23052A (da)
SU (1)	SU1517762A3 (da)
YU (2)	YU227886A (da)
ZA (1)	ZA8771B (da)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
JPS6452767A (en) *	1986-03-19	1989-02-28	Banyu Pharma Co Ltd	2-(2-aminothiazol-4-yl)-2-(1-carboxy-1-vinyloxyimino)acetic acid derivative and production thereof
JPS6393796A (ja) *	1986-10-09	1988-04-25	Shin Etsu Chem Co Ltd	ペプチド合成の脱保護基用薬剤
US5143913A (en) *	1988-04-04	1992-09-01	E. R. Squibb & Sons, Inc.	[3S(Z)]-3-[[(2-amino-4-thiazolyl)[[2-(hydroxyamino)-2-oxoethoxy]imino]acetyl]amino]-2,2-dimethyl-4-oxo-1-azetidinyl sulfate
JPH07165740A (ja) *	1994-11-07	1995-06-27	Banyu Pharmaceut Co Ltd	２−（２−アミノチアゾリル）−２−（１−カルボキシ−１−ビニルオキシイミノ）酢酸及びその製法
WO1997026250A1 (en) *	1996-01-16	1997-07-24	Merck & Co., Inc.	Integrin receptor antagonists
US5952306A (en) *	1996-01-16	1999-09-14	Merck & Co., Inc.	Integrin receptor antagonists
US9120796B2 (en)	2013-10-02	2015-09-01	Cubist Pharmaceuticals, Inc.	B-lactamase inhibitor picoline salt
MA44083A (fr)	2015-12-15	2021-06-02	Merck Sharp & Dohme	Composés de biarylmonobactame pour le traitement d'infections bactériennes
WO2017155765A1 (en)	2016-03-07	2017-09-14	Merck Sharp & Dohme Corp.	Bicyclic aryl monobactam compounds and methods of use thereof for the treatment of bacterial infections
US10002721B1 (en) *	2017-02-27	2018-06-19	Carling Technologies, Inc.	Multiple contact circuit breaker
EA202090604A1 (ru)	2017-10-02	2020-10-15	Мерк Шарп энд Доум Корп.	Хроманмонобактамовые соединения для лечения бактериальных инфекций
CN113754651B (zh)	2020-06-02	2023-04-18	中国医学科学院医药生物技术研究所	一种β-内酰胺化合物、其用途及其制备方法
CN118255695B (zh) *	2024-02-26	2025-03-14	广州艾奇西医药科技有限公司	一种β-内酰胺类化合物的中间体的纯化方法和制备方法

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
AU526540B2 (en) *	1976-04-12	1983-01-20	Fujisawa Pharmaceutical Co., Ltd.	Oximes of substituted phenyl, thiazolyl - glyoxylic acids
DE2716677C2 (de) *	1977-04-15	1985-10-10	Hoechst Ag, 6230 Frankfurt	Cephemderivate und Verfahren zu ihrer Herstellung
GB1602725A (en) *	1977-04-27	1981-11-18	Glaxo Operations Ltd	7-(a-oxyiminoacetamido)-ceph-3-em-4-carboxylic acid derivatives
US4409214A (en) *	1979-11-19	1983-10-11	Fujisawa Pharmaceutical, Co., Ltd.	7-Acylamino-3-vinylcephalosporanic acid derivatives and processes for the preparation thereof
US4533660A (en) *	1980-10-31	1985-08-06	E. R. Squibb & Sons, Inc.	Antibacterial O-sulfated β-lactam hydroxamic acids
JPS58113174A (ja) *	1981-12-26	1983-07-05	Toyama Chem Co Ltd	新規なアゼチジン誘導体またはその塩類を含有する抗菌剤
US4443374A (en) *	1982-02-01	1984-04-17	E. R. Squibb & Sons, Inc.	Process for preparing (3S)-3-[[(2-amino-4-thiazolyl)[(1-carboxy-1-methylethoxy)imino]-acetyl]amino]-2-oxo-1-azetidinesulfonic acid, and 4-substituted derivatives
AU564150B2 (en) *	1982-04-30	1987-08-06	Takeda Chemical Industries Ltd.	1-sulfo-2-azetidinone derivatives
JPS58206589A (ja) *	1982-05-26	1983-12-01	Yamanouchi Pharmaceut Co Ltd	２−アゼチジノン誘導体
KR900005112B1 (ko) *	1982-05-31	1990-07-19	반유세이야꾸 가부시끼가이샤	2-옥소-1-아제티딘술폰산 유도체의 제조방법
JPS58210060A (ja) *	1982-05-31	1983-12-07	Takeda Chem Ind Ltd	２−オキソアゼチジン誘導体、その製造法および用途
EP0096296B1 (de) *	1982-06-03	1987-07-29	F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft	1-Sulfo-2-oxoazetidinderivate
EP0096297B1 (de) *	1982-06-03	1988-06-15	F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft	Verfahren zur Herstellung von 1-Sulfo-2-oxoazetidinderivaten
US4704457A (en) *	1982-06-21	1987-11-03	E. R. Squibb & Sons, Inc.	Process for the preparation of (3S)-3-[[[2-(protected amino)-4-thiazolyl]-oxoacetyl]amino]-2-oxo-1-azetidinesulfonic acid and 4-substituted derivatives thereof
GB8413152D0 (en) *	1983-06-03	1984-06-27	Ici Pharma	Cephalosporin derivatives
DE3342929A1 (de) *	1983-11-26	1985-06-05	Bayer Ag, 5090 Leverkusen	Ss-lactamantibiotika, verfahren zu deren herstellung sowie ihre verwendung als arzneimittel

1986
- 1986-01-06 US US06/816,475 patent/US4684722A/en not_active Expired - Fee Related
- 1986-12-08 CA CA000524775A patent/CA1308107C/en not_active Expired - Lifetime
- 1986-12-17 NZ NZ218682A patent/NZ218682A/xx unknown
- 1986-12-19 PH PH34627A patent/PH23052A/en unknown
- 1986-12-19 AU AU66808/86A patent/AU602133B2/en not_active Ceased
- 1986-12-26 JP JP61315973A patent/JPS62158278A/ja active Pending
- 1986-12-30 YU YU02278/86A patent/YU227886A/xx unknown
1987
- 1987-01-04 IL IL81153A patent/IL81153A/xx unknown
- 1987-01-05 ES ES198787100056T patent/ES2038127T3/es not_active Expired - Lifetime
- 1987-01-05 KR KR1019870000006A patent/KR900002244B1/ko not_active Expired
- 1987-01-05 AT AT87100056T patent/ATE64393T1/de not_active IP Right Cessation
- 1987-01-05 DK DK003087A patent/DK3087A/da not_active Application Discontinuation
- 1987-01-05 EP EP87100056A patent/EP0229012B1/en not_active Expired - Lifetime
- 1987-01-05 NO NO870031A patent/NO166860C/no unknown
- 1987-01-05 HU HU875581A patent/HU198700B/hu not_active IP Right Cessation
- 1987-01-05 DD DD87299092A patent/DD256700A5/de unknown
- 1987-01-05 HU HU8722A patent/HU198926B/hu not_active IP Right Cessation
- 1987-01-05 DE DE8787100056T patent/DE3770644D1/de not_active Expired - Fee Related
- 1987-01-05 FI FI870030A patent/FI870030L/fi not_active Application Discontinuation
- 1987-01-05 SU SU874028791A patent/SU1517762A3/ru active
- 1987-01-06 ZA ZA8771A patent/ZA8771B/xx unknown
- 1987-07-08 YU YU01278/87A patent/YU127887A/xx unknown
1988
- 1988-01-05 DD DD88312099A patent/DD267039A5/de unknown
- 1988-01-05 DD DD88312098A patent/DD267035A5/de not_active IP Right Cessation
1990
- 1990-07-10 AU AU58851/90A patent/AU617059B2/en not_active Expired - Fee Related
- 1990-07-10 AU AU58850/90A patent/AU5885090A/en not_active Abandoned
1991
- 1991-07-15 GR GR91401016T patent/GR3002312T3/el unknown

Also Published As

Publication number	Publication date
IL81153A (en)	1991-06-10
FI870030A7 (fi)	1987-07-07
DD256700A5 (de)	1988-05-18
YU227886A (en)	1988-02-29
IL81153A0 (en)	1987-08-31
HUT48876A (en)	1989-07-28
ES2038127T3 (es)	1993-07-16
NO870031L (no)	1987-07-07
SU1517762A3 (ru)	1989-10-23
DK3087A (da)	1987-07-07
DK3087D0 (da)	1987-01-05
FI870030L (fi)	1987-07-07
AU602133B2 (en)	1990-10-04
AU5885190A (en)	1990-10-25
ZA8771B (en)	1987-08-26
NO870031D0 (no)	1987-01-05
KR870007164A (ko)	1987-08-17
US4684722A (en)	1987-08-04
DE3770644D1 (de)	1991-07-18
DD267035A5 (de)	1989-04-19
AU617059B2 (en)	1991-11-14
DD267039A5 (de)	1989-04-19
NZ218682A (en)	1990-05-28
HUT44540A (en)	1988-03-28
ATE64393T1 (de)	1991-06-15
AU6680886A (en)	1987-07-09
HU198926B (en)	1989-12-28
HU198700B (en)	1989-11-28
NO166860B (no)	1991-06-03
AU5885090A (en)	1990-11-15
YU127887A (en)	1988-04-30
FI870030A0 (fi)	1987-01-05
KR900002244B1 (ko)	1990-04-07
EP0229012A1 (en)	1987-07-15
CA1308107C (en)	1992-09-29
PH23052A (en)	1989-03-10
JPS62158278A (ja)	1987-07-14
GR3002312T3 (en)	1992-12-30
EP0229012B1 (en)	1991-06-12

Publication	Publication Date	Title
AU5860386A (en)	1986-11-18	Nitrogen-containing heterocycles
NO166860C (no)	1991-09-11	Analogifremgangsmaate for fremstilling av terapeutisk aktive monosulfaktamer.
GR880100248A (el)	1989-01-31	Ουσιες για την προφυλαξη και θεραπεια ρετροιογενην φλεγμωνων.
FI875218A0 (fi)	1987-11-26	Ns. aktiivisesta panssarista tehty panssariseinä
AU7998687A (en)	1988-06-23	Additives enhancing topical actions of therapeutic agents
IT8847884A0 (it)	1988-04-22	Elettrodo enzimatico e modulo di elettrodo nonche' relativo metodo di impiego
NO176275C (no)	1995-03-08	Analogifremgangsmåte for fremstilling av terapeutisk aktive pyridazinonderivater
EP0350012A3 (en)	1990-09-05	Antiviral composition
NO168362C (no)	1992-02-12	Analogifremgangsmaate for fremstilling av terapeutisk aktive peptidforbindelser
JO1704B1 (en)	1992-12-15	New potent compounds
CA2053359A1 (en)	1992-05-06	Heteroaroyl derivatives of monocyclic beta-lactam antibiotics
NO172849C (no)	1993-09-15	Analogifremgangsmaate for fremstilling av terapeutisk aktive tiazol- og oksazol-derivater
AU4059485A (en)	1985-10-03	Substituted benzopyrans
EG17752A (en)	1990-10-30	Benzoylurea derivatives
ES8701161A1 (es)	1986-11-16	Un procedimiento para preparar derivados de piridiloxi
CA1270247C (en)	1990-06-12	3-ACYLAMINO-2-OXO-1-AZETIDINESULFONIC ACIDS
AU585279B2 (en)	1989-06-15	Pesticidal biphenylyloxy and biphenylylalkoxy aryl acyl urea compounds
GR3007423T3 (da)	1993-07-30
CA1271750C (en)	1990-07-17	3-ACYLAMINO-2-OXO-1-AZETIDINESULFONIC ACIDS
FI841240A0 (fi)	1984-03-28	Foerbaettringar i makrolidantibiotika.
SU1271155A1 (ru)	1996-04-20	Способ создания лазерноактивных центров окраски tl°va*99+ в кристаллах kcl-tl
SU1203863A1 (ru)	2000-02-20	6-циклогексил-2-окса-6-азаспиро (3,3) гептан, подавляющий рост сульфатвосстанавливающих бактерий
SE9000857D0 (sv)	1990-03-09	Novel use of theraeutically active compound
SU1116706A1 (ru)	1996-05-20	Производные 2,3,4,5-тетрагидро-1н-1,5-бензодиазепинона-2, проявляющие противовоспалительную активность
GB8629579D0 (en)	1987-01-21	Stabilisation of yeast enzymes