NO20045054L - 4-substituerte imidazol-2-tioner og imidazol-2-oner som agonister av alfa-2B og alfa-2C adrenerge reseptorer - Google Patents

4-substituerte imidazol-2-tioner og imidazol-2-oner som agonister av alfa-2B og alfa-2C adrenerge reseptorer

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Publication number
NO20045054L
NO20045054L NO20045054A NO20045054A NO20045054L NO 20045054 L NO20045054 L NO 20045054L NO 20045054 A NO20045054 A NO 20045054A NO 20045054 A NO20045054 A NO 20045054A NO 20045054 L NO20045054 L NO 20045054L
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NO
Norway
Prior art keywords
alpha
imidazol
agonists
ions
ones
Prior art date
Application number
NO20045054A
Other languages
English (en)
Other versions
NO330692B1 (no
Inventor
Michael E Garst
Ken Chow
Daniel W Gil
Larry A Wheeler
Phong X Nguyen
Todd Heidelbaugh
Dario Gomez
Original Assignee
Allergan Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Allergan Inc filed Critical Allergan Inc
Publication of NO20045054L publication Critical patent/NO20045054L/no
Publication of NO330692B1 publication Critical patent/NO330692B1/no

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    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/70—One oxygen atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
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    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/84—Sulfur atoms
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    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
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    • C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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    • C07D—HETEROCYCLIC COMPOUNDS
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    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/08—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing alicyclic rings

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  • Orthopedic Medicine & Surgery (AREA)
  • Ophthalmology & Optometry (AREA)
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  • Urology & Nephrology (AREA)
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  • Transplantation (AREA)
  • Otolaryngology (AREA)
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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
NO20045054A 2002-05-21 2004-11-19 4-substituerte imidazol-2-tioner og imidazol-2-oner for behandling av sykdom samt anvendelse av disse for fremstilling av medikament for behandling av sykdom NO330692B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US15332802A 2002-05-21 2002-05-21
PCT/US2003/015441 WO2003099795A1 (en) 2002-05-21 2003-05-16 4-substituted imidazole-2-thiones and imidazol-2-ones as agonists of the alpha-2b and alpha-2c adrenergic receptors

Publications (2)

Publication Number Publication Date
NO20045054L true NO20045054L (no) 2005-02-10
NO330692B1 NO330692B1 (no) 2011-06-14

Family

ID=29582081

Family Applications (1)

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NO20045054A NO330692B1 (no) 2002-05-21 2004-11-19 4-substituerte imidazol-2-tioner og imidazol-2-oner for behandling av sykdom samt anvendelse av disse for fremstilling av medikament for behandling av sykdom

Country Status (17)

Country Link
US (5) US7091232B2 (no)
EP (1) EP1507767A1 (no)
JP (2) JP2005531581A (no)
KR (1) KR101016151B1 (no)
CN (1) CN1332952C (no)
AU (2) AU2003245286A1 (no)
BR (1) BR0311326A (no)
CA (1) CA2486537C (no)
CO (1) CO5621366A2 (no)
IL (1) IL165280A (no)
MX (1) MXPA04011546A (no)
NO (1) NO330692B1 (no)
NZ (1) NZ536626A (no)
PL (1) PL213028B1 (no)
RU (1) RU2318816C2 (no)
WO (1) WO2003099795A1 (no)
ZA (1) ZA200409333B (no)

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