NO20062258L - Nye metoder - Google Patents

Nye metoder

Info

Publication number: NO20062258L
Authority: NO; Norway
Prior art keywords: mandelic acid; alkyl; acid derivatives; cleaved; new methods
Prior art date: 2003-11-28

Application number

NO20062258A

Other languages

English (en)

Norwegian (no)

Inventor

Hans Jorgen Blixt

Bo Lars Gustaf Bosson

Roberto Giuseppe Gatti

Michael William Senior

Simone Zaramella

Kurt Vogtli

Andrea Zistler

Original Assignee

Astrazeneca Ab

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2003-11-28

Filing date

2006-05-19

Publication date

2006-08-23

2006-05-19 Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab

2006-08-23 Publication of NO20062258L publication Critical patent/NO20062258L/no

Links

238000000034 method Methods 0.000 title abstract 2
QBYIENPQHBMVBV-HFEGYEGKSA-N (2R)-2-hydroxy-2-phenylacetic acid Chemical class O[C@@H](C(O)=O)c1ccccc1.O[C@@H](C(O)=O)c1ccccc1 QBYIENPQHBMVBV-HFEGYEGKSA-N 0.000 abstract 3
125000000217 alkyl group Chemical group 0.000 abstract 3
IWYDHOAUDWTVEP-UHFFFAOYSA-N mandelic acid Chemical class OC(=O)C(O)C1=CC=CC=C1 IWYDHOAUDWTVEP-UHFFFAOYSA-N 0.000 abstract 2
-1 mandelic acid cyclic amide salts Chemical class 0.000 abstract 2
DASQIKOOFDJYKA-UHFFFAOYSA-N CCIF Chemical compound CCIF DASQIKOOFDJYKA-UHFFFAOYSA-N 0.000 abstract 1
230000015572 biosynthetic process Effects 0.000 abstract 1
238000003776 cleavage reaction Methods 0.000 abstract 1
150000001875 compounds Chemical class 0.000 abstract 1
150000003950 cyclic amides Chemical class 0.000 abstract 1
229910052736 halogen Inorganic materials 0.000 abstract 1
150000002367 halogens Chemical class 0.000 abstract 1
239000000543 intermediate Substances 0.000 abstract 1
229960002510 mandelic acid Drugs 0.000 abstract 1
239000002184 metal Substances 0.000 abstract 1
239000000203 mixture Substances 0.000 abstract 1
150000003839 salts Chemical class 0.000 abstract 1
230000007017 scission Effects 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C51/00—Preparation of carboxylic acids or their salts, halides or anhydrides
- C07C51/42—Separation; Purification; Stabilisation; Use of additives
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C231/00—Preparation of carboxylic acid amides
- C07C231/16—Preparation of optical isomers
- C07C231/20—Preparation of optical isomers by separation of optical isomers
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C237/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups
- C07C237/24—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atom of at least one of the carboxamide groups bound to a carbon atom of a ring other than a six-membered aromatic ring of the carbon skeleton
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C51/00—Preparation of carboxylic acids or their salts, halides or anhydrides
- C07C51/42—Separation; Purification; Stabilisation; Use of additives
- C07C51/487—Separation; Purification; Stabilisation; Use of additives by treatment giving rise to chemical modification
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C59/00—Compounds having carboxyl groups bound to acyclic carbon atoms and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups
- C07C59/40—Unsaturated compounds
- C07C59/58—Unsaturated compounds containing ether groups, groups, groups, or groups
- C07C59/64—Unsaturated compounds containing ether groups, groups, groups, or groups containing six-membered aromatic rings

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Engineering & Computer Science (AREA)
Oil, Petroleum & Natural Gas (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Analytical Chemistry (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Pyrrole Compounds (AREA)

NO20062258A 2003-11-28 2006-05-19 Nye metoder NO20062258L (no)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
SE0303220A SE0303220D0 (sv)	2003-11-28	2003-11-28	New process
PCT/GB2004/004964 WO2005054168A2 (en)	2003-11-28	2004-11-25	A process for resolving, optionally substituted, mandelic acids by salt formation with a chiral base cyclic amide

Publications (1)

Publication Number	Publication Date
NO20062258L true NO20062258L (no)	2006-08-23

Family

ID=29729226

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO20062258A NO20062258L (no)	2003-11-28	2006-05-19	Nye metoder

Country Status (15)

Country	Link
US (1)	US7960582B2 (pt)
EP (1)	EP1692089A2 (pt)
JP (1)	JP4906511B2 (pt)
KR (1)	KR101134767B1 (pt)
CN (2)	CN100448834C (pt)
AU (2)	AU2004295152B2 (pt)
BR (1)	BRPI0416931A (pt)
CA (1)	CA2546694A1 (pt)
IL (1)	IL175488A (pt)
NO (1)	NO20062258L (pt)
NZ (1)	NZ547354A (pt)
SE (1)	SE0303220D0 (pt)
SG (2)	SG148212A1 (pt)
WO (1)	WO2005054168A2 (pt)
ZA (1)	ZA200604192B (pt)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
AR035216A1 (es)	2000-12-01	2004-05-05	Astrazeneca Ab	Derivados de acido mandelico ,derivados farmaceuticamente aceptables, uso de estos derivados para la fabricacion de medicamentos, metodos de tratamiento ,procesos para la preparacion de estos derivados, y compuestos intermediarios
AR034517A1 (es)	2001-06-21	2004-02-25	Astrazeneca Ab	Formulacion farmaceutica
SE0201661D0 (sv) *	2002-05-31	2002-05-31	Astrazeneca Ab	New salts
US7781424B2 (en) *	2003-05-27	2010-08-24	Astrazeneca Ab	Modified release pharmaceutical formulation
SE0303220D0 (sv)	2003-11-28	2003-11-28	Astrazeneca Ab	New process
GB0510546D0 (en) *	2005-05-24	2005-06-29	Astrazeneca Ab	New process
TW200827336A (en)	2006-12-06	2008-07-01	Astrazeneca Ab	New crystalline forms
TW200900033A (en) *	2007-06-21	2009-01-01	Wen-Qing Li	Automatic brewing machine
US20090061000A1 (en) *	2007-08-31	2009-03-05	Astrazeneca Ab	Pharmaceutical formulation use 030
CN103450008B (zh) *	2013-09-02	2015-02-25	江苏宝众宝达药业有限公司	一种从废水中回收扁桃酸的方法
CN104447294A (zh) *	2014-11-24	2015-03-25	苏州乔纳森新材料科技有限公司	一种3-环己烯-1-甲酸的手性拆分方法

Family Cites Families (19)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US1867274A (en) *	1929-11-20	1932-07-12	Lilly Co Eli	Resolution of ephedrine and its homologues and of mandelic acid, and certain intermediates
JPS581105B2 (ja) *	1977-03-24	1983-01-10	日本化薬株式会社	光学活性アミノ酸−マンデル酸複合体及びその製造法
JPS5416442A (en) *	1977-07-08	1979-02-07	Sumitomo Chem Co Ltd	Optical resolution of 3-pheoxymandelic acid
US4239912A (en) *	1978-12-08	1980-12-16	American Cyanamid Company	Process for resolving DL-Mandelic acid with novel 2-benzylamino-1-butanols
US4259521A (en) *	1979-10-09	1981-03-31	American Cyanamid Company	Process for resolving DL-mandelic acid
US4260815A (en) *	1979-10-09	1981-04-07	American Cyanamid Company	Process for preparing a solution of DL-mandelic acid
JPH01221345A (ja) *	1988-02-27	1989-09-04	Ajinomoto Co Inc	マンデル酸誘導体の光学分割方法
DE4137663A1 (de) *	1991-11-12	1993-05-13	Degussa	Verfahren zur herstellung optisch aktiver 1,3-imidazolidin-4-one und deren verwendung
JPH11228546A (ja) *	1998-02-09	1999-08-24	Koei Chem Co Ltd	光学活性２−（Ｎ−ｔｅｒｔ−ブチルカルバモイル）ピペラジンの製造法
JP2001002641A (ja) *	1999-06-24	2001-01-09	Daito Chemix Corp	光学活性３−アミノピロリジン−２−オン誘導体の製造法
JP2001072644A (ja) *	1999-09-06	2001-03-21	Yamakawa Yakuhin Kogyo Kk	光学活性な２−クロロマンデル酸の製造方法および製造の中間体
WO2001040168A1 (en)	1999-11-29	2001-06-07	Mitsubishi Rayon Co., Ltd.	Acetalsulfonate derivative, process for producing the same, and process for producing styrene oxide derivative
EP1341762A1 (en) *	2000-11-20	2003-09-10	Eli Lilly And Company	Process for resolving racemic mixtures of piperidine derivatives
US7129233B2 (en) *	2000-12-01	2006-10-31	Astrazeneca Ab	Mandelic acid derivatives and their use as thrombin inhibitors
AR035216A1 (es) *	2000-12-01	2004-05-05	Astrazeneca Ab	Derivados de acido mandelico ,derivados farmaceuticamente aceptables, uso de estos derivados para la fabricacion de medicamentos, metodos de tratamiento ,procesos para la preparacion de estos derivados, y compuestos intermediarios
AR034517A1 (es) *	2001-06-21	2004-02-25	Astrazeneca Ab	Formulacion farmaceutica
SE0303220D0 (sv)	2003-11-28	2003-11-28	Astrazeneca Ab	New process
GB0503672D0 (en) *	2005-02-23	2005-03-30	Astrazeneca Ab	New process
GB0510546D0 (en)	2005-05-24	2005-06-29	Astrazeneca Ab	New process

2003
- 2003-11-28 SE SE0303220A patent/SE0303220D0/xx unknown
2004
- 2004-11-25 CN CNB2004800349394A patent/CN100448834C/zh not_active Expired - Fee Related
- 2004-11-25 KR KR1020067012985A patent/KR101134767B1/ko not_active Expired - Fee Related
- 2004-11-25 JP JP2006540610A patent/JP4906511B2/ja not_active Expired - Fee Related
- 2004-11-25 EP EP04819714A patent/EP1692089A2/en not_active Withdrawn
- 2004-11-25 SG SG200808873-4A patent/SG148212A1/en unknown
- 2004-11-25 US US10/579,854 patent/US7960582B2/en not_active Expired - Fee Related
- 2004-11-25 CA CA002546694A patent/CA2546694A1/en not_active Abandoned
- 2004-11-25 NZ NZ547354A patent/NZ547354A/en unknown
- 2004-11-25 CN CNA2008101754369A patent/CN101407453A/zh active Pending
- 2004-11-25 AU AU2004295152A patent/AU2004295152B2/en not_active Ceased
- 2004-11-25 WO PCT/GB2004/004964 patent/WO2005054168A2/en not_active Ceased
- 2004-11-25 SG SG200808874-2A patent/SG148213A1/en unknown
- 2004-11-25 BR BRPI0416931-0A patent/BRPI0416931A/pt active Search and Examination
2006
- 2006-05-08 IL IL175488A patent/IL175488A/en not_active IP Right Cessation
- 2006-05-19 NO NO20062258A patent/NO20062258L/no not_active Application Discontinuation
- 2006-05-24 ZA ZA200604192A patent/ZA200604192B/en unknown
2009
- 2009-08-11 AU AU2009208107A patent/AU2009208107A1/en not_active Ceased

Also Published As

Publication number	Publication date
SE0303220D0 (sv)	2003-11-28
CN1886359A (zh)	2006-12-27
BRPI0416931A (pt)	2007-01-16
SG148213A1 (en)	2008-12-31
AU2009208107A1 (en)	2009-09-03
SG148212A1 (en)	2008-12-31
IL175488A0 (en)	2006-09-05
JP2007513885A (ja)	2007-05-31
ZA200604192B (en)	2007-11-28
JP4906511B2 (ja)	2012-03-28
CN100448834C (zh)	2009-01-07
KR101134767B1 (ko)	2012-04-13
AU2004295152A1 (en)	2005-06-16
KR20060109965A (ko)	2006-10-23
NZ547354A (en)	2010-02-26
WO2005054168A2 (en)	2005-06-16
CA2546694A1 (en)	2005-06-16
IL175488A (en)	2012-02-29
AU2004295152B2 (en)	2009-07-02
WO2005054168A3 (en)	2005-10-27
US20080312457A1 (en)	2008-12-18
CN101407453A (zh)	2009-04-15
US7960582B2 (en)	2011-06-14
EP1692089A2 (en)	2006-08-23

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Legal Events

Date	Code	Title	Description
2012-06-25	FC2A	Withdrawal, rejection or dismissal of laid open patent application