NO20062370L - Amidderivater - Google Patents

Amidderivater

Info

Publication number
NO20062370L
NO20062370L NO20062370A NO20062370A NO20062370L NO 20062370 L NO20062370 L NO 20062370L NO 20062370 A NO20062370 A NO 20062370A NO 20062370 A NO20062370 A NO 20062370A NO 20062370 L NO20062370 L NO 20062370L
Authority
NO
Norway
Prior art keywords
trifluoromethyl
halogen
alkyl
amide derivatives
heterocyclyloxy
Prior art date
Application number
NO20062370A
Other languages
English (en)
Inventor
Dearg Sutherland Brown
Ian Alun Nash
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=29595715&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20062370(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of NO20062370L publication Critical patent/NO20062370L/no

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    • C04B—LIME, MAGNESIA; SLAG; CEMENTS; COMPOSITIONS THEREOF, e.g. MORTARS, CONCRETE OR LIKE BUILDING MATERIALS; ARTIFICIAL STONE; CERAMICS; REFRACTORIES; TREATMENT OF NATURAL STONE
    • C04B35/00—Shaped ceramic products characterised by their composition; Ceramics compositions; Processing powders of inorganic compounds preparatory to the manufacturing of ceramic products
    • C04B35/622—Forming processes; Processing powders of inorganic compounds preparatory to the manufacturing of ceramic products
    • C04B35/626—Preparing or treating the powders individually or as batches ; preparing or treating macroscopic reinforcing agents for ceramic products, e.g. fibres; mechanical aspects section B
    • C04B35/63—Preparing or treating the powders individually or as batches ; preparing or treating macroscopic reinforcing agents for ceramic products, e.g. fibres; mechanical aspects section B using additives specially adapted for forming the products, e.g.. binder binders
    • C04B35/632—Organic additives
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/517—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
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    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72—Quinazolines; Hydrogenated quinazolines
    • C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
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    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
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    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D487/08—Bridged systems

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  • Chemical & Material Sciences (AREA)
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Abstract

Det beskrives en forbindelse med formel I der m er 0-2 og hver R1 er en gruppe som hydroksy, halogeno, trifluormetyl, hetero-syklyl og heterosyklyloksy; R2 er halogen, trifluormetyl eller (Ci-6)alkyl; R3 er hydrogen, halogen eller (Ci^)alkyl; og R4 er (C3-6)sykloalkyl; eller farmasøytisk akseptable salter derav. Videre beskrives prosesser for deres fremstilling, farmasøytiske preparater inneholdende forbindelsene og deres anvendelse ved behandling av sykdommer eller medisinske tilstander som medieres av cytokiner.
NO20062370A 2003-10-24 2006-05-24 Amidderivater NO20062370L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0324790.5A GB0324790D0 (en) 2003-10-24 2003-10-24 Amide derivatives
PCT/GB2004/004474 WO2005042502A1 (en) 2003-10-24 2004-10-22 Amide derivatives

Publications (1)

Publication Number Publication Date
NO20062370L true NO20062370L (no) 2006-07-18

Family

ID=29595715

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20062370A NO20062370L (no) 2003-10-24 2006-05-24 Amidderivater

Country Status (27)

Country Link
US (1) US7750154B2 (no)
EP (1) EP1682520B1 (no)
JP (1) JP4987478B2 (no)
KR (1) KR101127697B1 (no)
CN (2) CN1898216A (no)
AR (1) AR046308A1 (no)
AT (1) ATE499347T1 (no)
AU (1) AU2004285749B2 (no)
BR (1) BRPI0415746A (no)
CA (1) CA2543351C (no)
DE (1) DE602004031543D1 (no)
ES (1) ES2359409T3 (no)
GB (1) GB0324790D0 (no)
IL (1) IL175065A (no)
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