NO20064017L - Fremgangsmate for fremstilling av enantiomert rene 1-substituerte -3-aminoalkoholer - Google Patents

Fremgangsmate for fremstilling av enantiomert rene 1-substituerte -3-aminoalkoholer

Info

Publication number: NO20064017L
Authority: NO; Norway
Prior art keywords: amino alcohols; substituted; amino; preparation; enantiomerically pure
Prior art date: 2004-02-19

Application number

NO20064017A

Other languages

English (en)

Norwegian (no)

Inventor

Hans-Peter Mettler

Dominique Michel

John Mcgarrity

Original Assignee

Lonza Ag Lonza Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2004-02-19

Filing date

2006-09-06

Publication date

2006-09-15

2004-02-19 Priority claimed from EP04003809A external-priority patent/EP1566383A1/fr

2006-09-06 Application filed by Lonza Ag Lonza Ltd filed Critical Lonza Ag Lonza Ltd

2006-09-15 Publication of NO20064017L publication Critical patent/NO20064017L/no

Links

238000000034 method Methods 0.000 title abstract 2
XSQUKJJJFZCRTK-UHFFFAOYSA-N Urea Chemical compound NC(N)=O XSQUKJJJFZCRTK-UHFFFAOYSA-N 0.000 abstract 3
150000003839 salts Chemical class 0.000 abstract 3
125000003545 alkoxy group Chemical group 0.000 abstract 2
125000000217 alkyl group Chemical group 0.000 abstract 2
150000001414 amino alcohols Chemical class 0.000 abstract 2
238000009876 asymmetric hydrogenation reaction Methods 0.000 abstract 2
125000005843 halogen group Chemical group 0.000 abstract 2
125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 2
125000002941 2-furyl group Chemical group O1C([*])=C([H])C([H])=C1[H] 0.000 abstract 1
125000000175 2-thienyl group Chemical group S1C([*])=C([H])C([H])=C1[H] 0.000 abstract 1
150000001732 carboxylic acid derivatives Chemical class 0.000 abstract 1
150000001735 carboxylic acids Chemical class 0.000 abstract 1
230000007062 hydrolysis Effects 0.000 abstract 1
238000006460 hydrolysis reaction Methods 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
- C07D333/14—Radicals substituted by singly bound hetero atoms other than halogen
- C07D333/20—Radicals substituted by singly bound hetero atoms other than halogen by nitrogen atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C213/00—Preparation of compounds containing amino and hydroxy, amino and etherified hydroxy or amino and esterified hydroxy groups bound to the same carbon skeleton
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
- C07D307/04—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
- C07D307/18—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D307/22—Nitrogen atoms not forming part of a nitro radical
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
- C07D333/22—Radicals substituted by doubly bound hetero atoms, or by two hetero atoms other than halogen singly bound to the same carbon atom
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/07—Optical isomers

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Heterocyclic Compounds Containing Sulfur Atoms (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Furan Compounds (AREA)

NO20064017A 2004-02-19 2006-09-06 Fremgangsmate for fremstilling av enantiomert rene 1-substituerte -3-aminoalkoholer NO20064017L (no)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
EP04003809A EP1566383A1 (fr)	2004-02-19	2004-02-19	Procédé de préparation des enantiomers pures des dérivés de 3-aminoalcools substitués
EP04010043		2004-04-28
PCT/EP2005/001781 WO2005080370A1 (fr)	2004-02-19	2005-02-21	Procede de preparation de 3-aminoalcools 1-substitues enantiomeriquement purs

Publications (1)

Publication Number	Publication Date
NO20064017L true NO20064017L (no)	2006-09-15

Family

ID=34889010

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO20064017A NO20064017L (no)	2004-02-19	2006-09-06	Fremgangsmate for fremstilling av enantiomert rene 1-substituerte -3-aminoalkoholer

Country Status (20)

Country	Link
US (3)	US7973182B2 (fr)
EP (1)	EP1720852B1 (fr)
JP (2)	JP2007523124A (fr)
KR (1)	KR101160502B1 (fr)
CN (1)	CN102627572A (fr)
AU (1)	AU2005215906C1 (fr)
BR (1)	BRPI0506796A (fr)
CA (1)	CA2556891C (fr)
CY (1)	CY1113261T1 (fr)
DK (1)	DK1720852T3 (fr)
EA (1)	EA200601513A1 (fr)
ES (1)	ES2391399T3 (fr)
IL (1)	IL177561A (fr)
NO (1)	NO20064017L (fr)
NZ (1)	NZ549381A (fr)
PL (1)	PL1720852T3 (fr)
PT (1)	PT1720852E (fr)
SG (1)	SG135196A1 (fr)
SI (1)	SI1720852T1 (fr)
WO (1)	WO2005080370A1 (fr)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
CA2556891C (fr)	2004-02-19	2012-12-18	Lonza Ag	Procede de preparation de 3-aminoalcools 1-substitues enantiomeriquement purs
EA200701613A1 (ru) *	2005-02-21	2008-02-28	Лонца Аг	Способ получения энантиомерно чистых 1-замещенных 3-аминоспиртов
EP2044049A2 (fr)	2006-07-03	2009-04-08	Ranbaxy Laboratories Limited	Procédé de préparation de sels énantiomöriquement purs de n-méthyl-3-(1-naphtalènoxy)-3-(2-thiényl) propanamine
EP2329013B1 (fr)	2008-08-27	2015-10-28	Codexis, Inc.	Polypeptides de kétoréductase servant à préparer une 3-aryl-3-hydroxypropanamine à partir d'une 3-aryl-3-kétopropanamine
WO2010025287A2 (fr)	2008-08-27	2010-03-04	Codexis, Inc.	Polypeptides cétoréductases pour la production de 3-aryl-3-hydroxypropanamine à partir de a 3-aryl-3-cétopropanamine
WO2011128370A1 (fr)	2010-04-13	2011-10-20	Krka, D.D., Novo Mesto	Synthèse de duloxétine et/ou de ses sels pharmaceutiquement acceptables de celle-ci
CN104056663B (zh) *	2013-03-22	2016-12-28	上海交通大学	一种面手性双反应中心钌催化剂及其合成与应用
CN110054563A (zh) *	2019-06-10	2019-07-26	江西隆莱生物制药有限公司	丁内酯类化合物的制备方法及其中间体
CN111793056A (zh) *	2020-07-27	2020-10-20	广州康瑞泰药业有限公司	一种度洛西汀中间体的制备方法

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DE3031248A1 (de) *	1980-08-19	1982-04-01	Ruhrchemie Ag, 4200 Oberhausen	Verfahren zur herstellung von 3-dimethylamino-2,2-dimethylpropanal
US5362866A (en)	1983-09-02	1994-11-08	Molecular Biosystems, Inc.	Oligonucleotide polymeric support system with an oxidation cleavable link
KR880007433A (ko) *	1986-12-22	1988-08-27	메리 앤 터커	3-아릴옥시-3-치환된 프로판아민
US4948813A (en) *	1987-11-30	1990-08-14	E. I. Du Pont De Nemours And Company	Benzylketone phospholipase A2 inhibitors
CA2042346A1 (fr)	1990-05-17	1991-11-18	Michael Alexander Staszak	Synthese chirale de 1-aryl-3-aminopropan-1-ols
JPH0570412A (ja) *	1991-09-13	1993-03-23	Fuji Yakuhin Kogyo Kk	光学活性なβ−アミノアルコールの製造方法
US5491234A (en) *	1992-03-30	1996-02-13	Pfizer Inc.	Pyrimidine derivatives for enhancing antitumor activity
DK0647648T3 (da)	1993-10-08	1999-09-27	Hoffmann La Roche	Optisk aktive phosphorforbindelser
US5362886A (en)	1993-10-12	1994-11-08	Eli Lilly And Company	Asymmetric synthesis
IT1270082B (it) *	1994-07-12	1997-04-28	Univ Degli Studi Milano	Difosfine eteroaromatiche come leganti chirali, complessi tra dette difosfine e metalli di transizione ed impiego di detti complessi come catalizzatori chirali
TW514634B (en) *	1997-10-14	2002-12-21	Lilly Co Eli	Process to make chiral compounds
US6008412A (en) *	1997-10-14	1999-12-28	Eli Lilly And Company	Process to make chiral compounds
US6162929A (en)	1997-12-23	2000-12-19	Hoffmann-La Roche Inc.	Process for the manufacture of bisphosphine oxide and bisphosphonate compounds
JP3549390B2 (ja)	1998-03-23	2004-08-04	高砂香料工業株式会社	ルテニウム−ホスフィン錯体及びその製造方法
DE69933904T2 (de)	1998-05-08	2007-09-06	Takasago International Corp.	Ruthenium-iodo optisch aktiver Phosphinkomplex
FR2816946B1 (fr)	2000-11-17	2004-04-02	Ppg Sipsy	Diphosphines chirales dissymetriques, leurs utilisations pour la preparation de complexes diphosphino-metalliques, et les complexes diphosphino-metalliques ainsi obtenus
DE10207586A1 (de) *	2002-02-22	2003-09-11	Degussa	Herstellung von N-Methyl-3-hydroxy-3-(2-thienyl)propanamin über neue carbamatgruppenhaltige Thiophenderivate als Zwischenprodukte
FR2841899A1 (fr)	2002-07-05	2004-01-09	Ppg Sipsy	Procede de resolution asymetrique d'un racemique faisant intervenir l'acide diprogulique et utilisation dudit acide comme agent de resolution asymetrique
WO2004005307A1 (fr) *	2002-07-09	2004-01-15	Lonza Ag	Procede de preparation de 3-n-methylamino-1-(2-thienyl)-1-propanol optiquement actif
DK1539673T3 (da)	2002-07-09	2008-01-21	Lonza Ag	Fremgangsmåde til fremstilling af N-monosubstituerede beta-aminoalkoholer
CA2556891C (fr)	2004-02-19	2012-12-18	Lonza Ag	Procede de preparation de 3-aminoalcools 1-substitues enantiomeriquement purs

2005
- 2005-02-21 CA CA2556891A patent/CA2556891C/fr not_active Expired - Fee Related
- 2005-02-21 EP EP05715425A patent/EP1720852B1/fr not_active Expired - Lifetime
- 2005-02-21 BR BRPI0506796-0A patent/BRPI0506796A/pt not_active IP Right Cessation
- 2005-02-21 NZ NZ549381A patent/NZ549381A/en not_active IP Right Cessation
- 2005-02-21 DK DK05715425.4T patent/DK1720852T3/da active
- 2005-02-21 PT PT05715425T patent/PT1720852E/pt unknown
- 2005-02-21 CN CN2012100464149A patent/CN102627572A/zh active Pending
- 2005-02-21 ES ES05715425T patent/ES2391399T3/es not_active Expired - Lifetime
- 2005-02-21 SI SI200531602T patent/SI1720852T1/sl unknown
- 2005-02-21 EA EA200601513A patent/EA200601513A1/ru unknown
- 2005-02-21 JP JP2006553562A patent/JP2007523124A/ja active Pending
- 2005-02-21 PL PL05715425T patent/PL1720852T3/pl unknown
- 2005-02-21 SG SG200706103-9A patent/SG135196A1/en unknown
- 2005-02-21 KR KR1020067018840A patent/KR101160502B1/ko not_active Expired - Fee Related
- 2005-02-21 AU AU2005215906A patent/AU2005215906C1/en not_active Ceased
- 2005-02-21 WO PCT/EP2005/001781 patent/WO2005080370A1/fr not_active Ceased
- 2005-02-21 US US10/590,140 patent/US7973182B2/en not_active Expired - Fee Related
2006
- 2006-08-17 IL IL177561A patent/IL177561A/en not_active IP Right Cessation
- 2006-09-06 NO NO20064017A patent/NO20064017L/no not_active Application Discontinuation
2011
- 2011-03-08 US US13/064,146 patent/US8198468B2/en not_active Expired - Fee Related
- 2011-03-08 US US13/064,147 patent/US8193380B2/en not_active Expired - Fee Related
2012
- 2012-06-14 JP JP2012134968A patent/JP2012229223A/ja not_active Withdrawn
- 2012-10-10 CY CY20121100937T patent/CY1113261T1/el unknown

Also Published As

Publication number	Publication date
CA2556891C (fr)	2012-12-18
AU2005215906B2 (en)	2011-08-18
US7973182B2 (en)	2011-07-05
AU2005215906C1 (en)	2012-03-01
PL1720852T3 (pl)	2012-12-31
CY1113261T1 (el)	2016-04-13
EA200601513A1 (ru)	2007-02-27
US20080154047A1 (en)	2008-06-26
IL177561A0 (en)	2006-12-10
CN102627572A (zh)	2012-08-08
US20110207946A1 (en)	2011-08-25
AU2005215906A1 (en)	2005-09-01
EP1720852B1 (fr)	2012-07-11
US20110207945A1 (en)	2011-08-25
SI1720852T1 (sl)	2012-11-30
CA2556891A1 (fr)	2005-09-01
IL177561A (en)	2011-12-29
DK1720852T3 (da)	2012-10-22
WO2005080370A1 (fr)	2005-09-01
KR20070009587A (ko)	2007-01-18
JP2007523124A (ja)	2007-08-16
ES2391399T3 (es)	2012-11-26
JP2012229223A (ja)	2012-11-22
US8193380B2 (en)	2012-06-05
PT1720852E (pt)	2012-10-22
NZ549381A (en)	2010-05-28
US8198468B2 (en)	2012-06-12
BRPI0506796A (pt)	2007-05-22
EP1720852A1 (fr)	2006-11-15
SG135196A1 (en)	2007-09-28
KR101160502B1 (ko)	2012-06-28

Legal Events

Date	Code	Title	Description
2014-09-22	FC2A	Withdrawal, rejection or dismissal of laid open patent application

Publication	Publication Date	Title
NO20064017L (no)	2006-09-15	Fremgangsmate for fremstilling av enantiomert rene 1-substituerte -3-aminoalkoholer
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