NO307968B1 - Pyrazolo- og pyrrolopyridiner og farmasøytisk blanding derav - Google Patents
Pyrazolo- og pyrrolopyridiner og farmasøytisk blanding deravInfo
- Publication number
- NO307968B1 NO307968B1 NO965378A NO965378A NO307968B1 NO 307968 B1 NO307968 B1 NO 307968B1 NO 965378 A NO965378 A NO 965378A NO 965378 A NO965378 A NO 965378A NO 307968 B1 NO307968 B1 NO 307968B1
- Authority
- NO
- Norway
- Prior art keywords
- pyrrolopyridines
- pyrazolo
- pharmaceutical mixtures
- pharmaceutical
- mixtures
- Prior art date
Links
- 239000000203 mixture Substances 0.000 title 1
- 150000005229 pyrazolopyridines Chemical class 0.000 title 1
- 150000005255 pyrrolopyridines Chemical class 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 201000010099 disease Diseases 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/04—Immunostimulants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/10—Drugs for disorders of the endocrine system of the posterior pituitary hormones, e.g. oxytocin, ADH
- A61P5/12—Drugs for disorders of the endocrine system of the posterior pituitary hormones, e.g. oxytocin, ADH for decreasing, blocking or antagonising the activity of the posterior pituitary hormones
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Diabetes (AREA)
- Immunology (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Endocrinology (AREA)
- Rheumatology (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Virology (AREA)
- Child & Adolescent Psychology (AREA)
- Anesthesiology (AREA)
- Addiction (AREA)
- Emergency Medicine (AREA)
- Hospice & Palliative Care (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Controls And Circuits For Display Device (AREA)
- Projection Apparatus (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US26005594A | 1994-06-16 | 1994-06-16 | |
| PCT/IB1995/000373 WO1995034563A1 (fr) | 1994-06-16 | 1995-05-18 | Pyrazolo et pyrrolopyridines |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| NO965378D0 NO965378D0 (no) | 1996-12-13 |
| NO965378L NO965378L (no) | 1996-12-13 |
| NO307968B1 true NO307968B1 (no) | 2000-06-26 |
Family
ID=22987613
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO965378A NO307968B1 (no) | 1994-06-16 | 1996-12-13 | Pyrazolo- og pyrrolopyridiner og farmasøytisk blanding derav |
Country Status (27)
| Country | Link |
|---|---|
| US (1) | US6248753B1 (fr) |
| EP (1) | EP0765327B1 (fr) |
| JP (1) | JP2891544B2 (fr) |
| KR (1) | KR100235277B1 (fr) |
| CN (1) | CN1056611C (fr) |
| AT (1) | ATE182332T1 (fr) |
| AU (1) | AU687196B2 (fr) |
| BR (1) | BR9502707A (fr) |
| CA (1) | CA2192820C (fr) |
| CO (1) | CO4290424A1 (fr) |
| CZ (1) | CZ287613B6 (fr) |
| DE (1) | DE69510940T2 (fr) |
| DK (1) | DK0765327T3 (fr) |
| ES (1) | ES2135062T3 (fr) |
| FI (1) | FI112659B (fr) |
| GR (1) | GR3031166T3 (fr) |
| HU (1) | HU219911B (fr) |
| IL (1) | IL114003A (fr) |
| MX (1) | MX9606504A (fr) |
| NO (1) | NO307968B1 (fr) |
| NZ (1) | NZ284846A (fr) |
| PE (1) | PE13396A1 (fr) |
| PL (1) | PL181895B1 (fr) |
| RU (1) | RU2135498C1 (fr) |
| TW (1) | TW432064B (fr) |
| WO (1) | WO1995034563A1 (fr) |
| ZA (1) | ZA954679B (fr) |
Families Citing this family (104)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6403599B1 (en) | 1995-11-08 | 2002-06-11 | Pfizer Inc | Corticotropin releasing factor antagonists |
| US7067664B1 (en) | 1995-06-06 | 2006-06-27 | Pfizer Inc. | Corticotropin releasing factor antagonists |
| AU738304B2 (en) * | 1995-10-13 | 2001-09-13 | Neurogen Corporation | Certain pyrrolopyridine derivatives; novel CRF 1 specific ligands |
| US6992188B1 (en) | 1995-12-08 | 2006-01-31 | Pfizer, Inc. | Substituted heterocyclic derivatives |
| WO1997035846A1 (fr) * | 1996-03-26 | 1997-10-02 | Dupont Pharmaceuticals Company | Pyridines et pyrimidines a fusion aryloxy et arylthio et derives de ces dernieres |
| ZA971896B (en) * | 1996-03-26 | 1998-09-07 | Du Pont Merck Pharma | Aryloxy-and arythio-fused pyridines and pyrimidines and derivatives |
| ZA972497B (en) | 1996-03-27 | 1998-09-25 | Du Pont Merck Pharma | Arylamino fused pyridines and pyrimidines |
| US6107300A (en) * | 1996-03-27 | 2000-08-22 | Dupont Pharmaceuticals | Arylamino fused pyrimidines |
| ZA973884B (en) | 1996-05-23 | 1998-11-06 | Du Pont Merck Pharma | Tetrahydropteridines and pyridylpiperazines for treatment of neurological disorders |
| US6124289A (en) | 1996-07-24 | 2000-09-26 | Dupont Pharmaceuticals Co. | Azolo triazines and pyrimidines |
| US7094782B1 (en) | 1996-07-24 | 2006-08-22 | Bristol-Myers Squibb Company | Azolo triazines and pyrimidines |
| US6191131B1 (en) | 1997-07-23 | 2001-02-20 | Dupont Pharmaceuticals Company | Azolo triazines and pyrimidines |
| US6060478A (en) * | 1996-07-24 | 2000-05-09 | Dupont Pharmaceuticals | Azolo triazines and pyrimidines |
| US6313124B1 (en) | 1997-07-23 | 2001-11-06 | Dupont Pharmaceuticals Company | Tetrazine bicyclic compounds |
| CA2262692C (fr) * | 1996-08-06 | 2002-06-11 | Pfizer Inc. | Derives 6,6- ou 6,7-bicycliques contenant pyrido ou pyrimido substitues |
| TW477787B (en) * | 1996-08-27 | 2002-03-01 | Pfizer | Pyrido six-membered nitrogen-containing cyclic ring derivatives having corticotropin releasing factor antagonist activity and pharmaceutical composition containing same |
| EP0927171B1 (fr) | 1996-09-16 | 2002-02-20 | Du Pont Pharmaceuticals Company | Pyrazinones et triazinones ainsi que leurs derives |
| JP2001511813A (ja) | 1997-02-18 | 2001-08-14 | ニューロクライン バイオサイエンシーズ,インコーポレイテッド | Crfレセプターアンタゴニストおよびそれらに関連する方法 |
| PL337888A1 (en) | 1997-07-03 | 2000-09-11 | Du Pont Pharm Co | Imidazoprimidines and imidazopyridines for use in treating neurological disorders |
| UA62972C2 (en) * | 1997-07-03 | 2004-01-15 | Application of imidazopyrimidins and imidazopyridins for the treatment of neural disorders | |
| IL134748A0 (en) | 1997-09-02 | 2001-04-30 | Du Pont Pharm Co | Heterocyclyl-substituted ring-fused pyridines and pyrimidines as corticotropin releasing hormone (crh) antagonists, useful for treating cns and stress-related disorders |
| NL1010018C2 (nl) * | 1997-09-09 | 1999-03-10 | Duphar Int Res | Chinoline en chinazoline derivaten met corticotropine releasing factor (CRF) antagonistische werking. |
| US6187777B1 (en) | 1998-02-06 | 2001-02-13 | Amgen Inc. | Compounds and methods which modulate feeding behavior and related diseases |
| US6472402B1 (en) | 1998-04-02 | 2002-10-29 | Neurogen Corporation | Aminoalkyl substituted 5,6,7,8-Tetrahydro-9H-Pyridino [2,3-B]indole derivatives |
| JP2002510686A (ja) | 1998-04-02 | 2002-04-09 | ニューロゲン コーポレイション | アミノアルキルで置換された5,6,7,8−テトラヒドロ−9H−ピリジノ[2,3−b]インドール及び5,6,7,8−テトラヒドロ−9Hピリミジノ[4,5−B]インドール誘導体:CRF1特異的配位子 |
| EP1068206A1 (fr) * | 1998-04-02 | 2001-01-17 | Neurogen Corporation | Derives aminoalkyle substitues de pyrrolo 2,3-b]pyridine et pyrrolo 2,3-d]pyrimidine: modulateurs de recepteurs de crf1 |
| US6365589B1 (en) | 1998-07-02 | 2002-04-02 | Bristol-Myers Squibb Pharma Company | Imidazo-pyridines, -pyridazines, and -triazines as corticotropin releasing factor antagonists |
| DE19837387A1 (de) * | 1998-08-18 | 2000-02-24 | Aventis Res & Tech Gmbh & Co | 3'-Desoxypentopyranosyl-Nucleinsäure, ihre Herstellung und Verwendung |
| US6174912B1 (en) | 1998-08-21 | 2001-01-16 | Dupont Pharmaceuticals Company | Nitrogen substituted imidazo[4,5-C]pyrazoles as corticotropin releasing hormone antagonists |
| US6531475B1 (en) | 1998-11-12 | 2003-03-11 | Neurocrine Biosciences, Inc. | CRF receptor antagonists and methods relating thereto |
| WO2000027850A2 (fr) | 1998-11-12 | 2000-05-18 | Neurocrine Biosciences, Inc. | Antagonistes de recepteurs du crf et methodes associees |
| US6514982B1 (en) | 1998-11-12 | 2003-02-04 | Neurocrine Biosciences, Inc. | CRF receptor antagonists and methods relating thereto |
| US6271380B1 (en) | 1998-12-30 | 2001-08-07 | Dupont Pharmaceuticals Company | 1H-imidazo[4,5-d]pyridazin-7-ones, 3H-imidazo-[4,5-c]pyridin-4-ones and corresponding thiones as corticotropin releasing factor (CRF) receptor ligands |
| EP1040831A3 (fr) * | 1999-04-02 | 2003-05-02 | Pfizer Products Inc. | Utilisation d'antagonistes du facteur de libération de la corticotropine pour la prévention de la mort subite |
| US6387894B1 (en) | 1999-06-11 | 2002-05-14 | Pfizer Inc. | Use of CRF antagonists and renin-angiotensin system inhibitors |
| US6432989B1 (en) | 1999-08-27 | 2002-08-13 | Pfizer Inc | Use of CRF antagonists to treat circadian rhythm disorders |
| ATE318267T1 (de) | 1999-09-30 | 2006-03-15 | Neurogen Corp | Einige alkylendiamin-substituierte heterocyclen |
| CO5271670A1 (es) * | 1999-10-29 | 2003-04-30 | Pfizer Prod Inc | Antagonistas del factor de liberacion de corticitropina y composiciones relacionadas |
| TWI271406B (en) | 1999-12-13 | 2007-01-21 | Eisai Co Ltd | Tricyclic condensed heterocyclic compounds, preparation method of the same and pharmaceuticals comprising the same |
| AU3264201A (en) * | 1999-12-17 | 2001-06-25 | Du Pont Pharmaceuticals Company | Imidazopyrimidinyl and imidazopyridinyl derivatives |
| EP1293213A1 (fr) * | 2000-02-14 | 2003-03-19 | Japan Tobacco Inc. | Agents prophylactiques/therapeutiques contre le stress postoperatoire |
| DE60108626T2 (de) * | 2000-04-25 | 2005-12-22 | Bristol-Myers Squibb Co. | Verwendung von 5-thio, sulfinyl- und sulfonylpyrazolo 3,4-b] pyridinen als cyclin-abhängige kinase-hemmer |
| US6630476B2 (en) | 2000-07-07 | 2003-10-07 | Bristol-Myers Squibb Pharma Company | Pyrrolo [3,4-d] pyrimidines as corticotropin releasing factor (CRF) antagonists |
| PE20020394A1 (es) | 2000-08-18 | 2002-06-21 | Agouron Pharma | Compuestos de pirazol y composiciones farmaceuticas que los contienen, que modulan y/o inhiben la actividad de erab/hadh2 |
| DE10042093A1 (de) * | 2000-08-26 | 2002-03-07 | Dresden Arzneimittel | Antikonvulsiv wirkende 6,7-Dihydro-pyrrolo[3,4-d]pyridin-5-one und Verfahren zu deren Darstellung |
| AU2002213929B2 (en) | 2000-09-22 | 2006-04-13 | Merck Sharp & Dohme B.V. | Bicyclic heteroaromatic compounds |
| DE10053275A1 (de) * | 2000-10-27 | 2002-05-02 | Dresden Arzneimittel | Neue 7-Azaindole, deren Verwendung als Inhibitoren der Phosphodiesterase 4 und Verfahren zu deren Herstellung |
| TWI312347B (en) | 2001-02-08 | 2009-07-21 | Eisai R&D Man Co Ltd | Bicyclic nitrogen-containing condensed ring compounds |
| RU2296753C2 (ru) * | 2001-02-22 | 2007-04-10 | Селлтек Р Энд Д Лимитед | Производные 3-оксо-1-циклобутена и фармацевтическая композиция на их основе |
| ES2262801T3 (es) * | 2001-02-27 | 2006-12-01 | Ortho-Mcneil Pharmaceutical, Inc. | Uso de un compuesto de carbamato para la prevencion o el tratamiento de trastorno bipolar. |
| DE10110747A1 (de) | 2001-03-07 | 2002-09-12 | Bayer Ag | Substituierte 2,6-Diamino-3,5-dicyano-4-aryl-pyridine und ihre Verwendung |
| IL158624A0 (en) | 2001-04-27 | 2004-05-12 | Eisai Co Ltd | Pyrazolo [1, 5-a] pyridines and medicines containing the same |
| GB0117396D0 (en) | 2001-07-17 | 2001-09-05 | Glaxo Group Ltd | Chemical compounds |
| CA2462806A1 (fr) * | 2001-10-08 | 2003-04-17 | F. Hoffmann-La Roche Ag | Amide d'acide 8-amino-[1,2,4]triazolo[1,5-a]pyridine-6-carboxylique |
| GB0128287D0 (en) * | 2001-11-26 | 2002-01-16 | Smithkline Beecham Plc | Novel method and compounds |
| AU2002356725B2 (en) * | 2001-12-04 | 2008-07-17 | F. Hoffmann-La Roche Ag | Ring fused pyrazole derivatives |
| AU2003214414B2 (en) * | 2002-03-28 | 2008-10-09 | Eisai R & D Management Co., Ltd. | Azaindoles as inhibitors of c-Jun N-terminal kinases |
| UA78999C2 (en) * | 2002-06-04 | 2007-05-10 | Wyeth Corp | 1-(aminoalkyl)-3-sulfonylazaindoles as ligands of 5-hydroxytryptamine-6 |
| GB0230045D0 (en) * | 2002-12-23 | 2003-01-29 | Glaxo Group Ltd | Compounds |
| RU2357967C2 (ru) * | 2002-09-16 | 2009-06-10 | Глаксо Груп Лимитед | ПРОИЗВОДНЫЕ ПИРАЗОЛО[3, 4-b]ПИРИДИНА, ФАРМАЦЕВТИЧЕСКАЯ КОМПОЗИЦИЯ (ВАРИАНТЫ), ПРИМЕНЕНИЕ (ВАРИАНТЫ), КОМПОЗИЦИЯ (ВАРИАНТЫ) |
| KR100984085B1 (ko) | 2002-10-22 | 2010-09-30 | 에자이 알앤드디 매니지먼트 가부시키가이샤 | 7-페닐 피라졸로피리딘 화합물 |
| US7176216B2 (en) | 2002-10-22 | 2007-02-13 | Eisai Co., Ltd. | 7-phenylpyrazolopyridine compounds |
| AR042667A1 (es) | 2002-12-26 | 2005-06-29 | Taisho Pharmaceutical Co Ltd | Derivados de pirrolopirimidina y pirrolopiridina sustituidos con un grupo amino ciclico |
| GB0308208D0 (en) | 2003-04-09 | 2003-05-14 | Glaxo Group Ltd | Chemical compounds |
| MY144903A (en) * | 2004-06-17 | 2011-11-30 | Novartis Ag | Pyrrolopyridine derivatives and their use as crth2 antagonists |
| RU2387654C2 (ru) * | 2004-07-27 | 2010-04-27 | Сгкс Фармасьютиклз, Инк. | Конденсированные гетероциклические модуляторы киназ |
| RU2389728C2 (ru) * | 2004-07-27 | 2010-05-20 | Сгкс Фармасьютиклз, Инк. | Модуляторы киназы на основе производных пирролопиридина |
| DE102004042607A1 (de) | 2004-09-03 | 2006-03-09 | Bayer Healthcare Ag | Substituierte Phenylaminothiazole und ihre Verwendung |
| ATE430746T1 (de) * | 2004-10-19 | 2009-05-15 | Smithkline Beecham Cork Ltd | Crf-rezeptor-antagonisten und zugehörige verfahren |
| RU2287275C1 (ru) * | 2005-06-23 | 2006-11-20 | Федеральное государственное образовательное учреждение высшего профессионального образования Кубанский государственный аграрный университет | ПРИМЕНЕНИЕ 3[(ЗАМЕЩЕННЫЙ ФЕНИЛ) КАРБОКСАМИДО]-1,4,6-ТРИМЕТИЛ-5-R ПИРАЗОЛО [4,5-b]ПИРИДИНОВ В КАЧЕСТВЕ АНТИДОТОВ 2,4-Д |
| RU2287273C1 (ru) * | 2005-06-23 | 2006-11-20 | Федеральное государственное образовательное учреждение высшего профессионального образования Кубанский государственный аграрный университет | Применение n-замещенных 3-циано-4,6-диметил-5-хлорпиридил-2-сульфониламидов в качестве антидотов гербицида 2,4-дихлорфеноксиуксусной кислоты на подсолнечнике |
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| US3925388A (en) * | 1971-08-05 | 1975-12-09 | Squibb & Sons Inc | 4-Piperazino-{8 3,4-b{9 pyridine-5-carboxylic acids and esters |
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| IT222061Z2 (it) | 1991-12-03 | 1994-12-29 | Hydro Aluminium Systems Spa | Complesso di profilati metallici per serramenti muniti di squadrette di rinforzo |
| JPH0669494B2 (ja) | 1991-12-04 | 1994-09-07 | 南雄 河野 | 医療用窓付断熱カテーテル |
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| TW370529B (en) * | 1992-12-17 | 1999-09-21 | Pfizer | Pyrazolopyrimidines |
| WO1995010506A1 (fr) | 1993-10-12 | 1995-04-20 | The Du Pont Merck Pharmaceutical Company | 1n-alkyle-n-arylpyrimidinamines et leurs derives |
-
1995
- 1995-05-18 RU RU96123712/04A patent/RU2135498C1/ru not_active IP Right Cessation
- 1995-05-18 HU HU9603469A patent/HU219911B/hu not_active IP Right Cessation
- 1995-05-18 AT AT95917436T patent/ATE182332T1/de not_active IP Right Cessation
- 1995-05-18 AU AU23505/95A patent/AU687196B2/en not_active Ceased
- 1995-05-18 KR KR1019960707183A patent/KR100235277B1/ko not_active Expired - Fee Related
- 1995-05-18 PL PL95317705A patent/PL181895B1/pl not_active IP Right Cessation
- 1995-05-18 CZ CZ19963670A patent/CZ287613B6/cs not_active IP Right Cessation
- 1995-05-18 MX MX9606504A patent/MX9606504A/es not_active IP Right Cessation
- 1995-05-18 NZ NZ284846A patent/NZ284846A/xx unknown
- 1995-05-18 CA CA002192820A patent/CA2192820C/fr not_active Expired - Fee Related
- 1995-05-18 JP JP8501868A patent/JP2891544B2/ja not_active Expired - Fee Related
- 1995-05-18 CN CN95193638A patent/CN1056611C/zh not_active Expired - Fee Related
- 1995-05-18 DE DE69510940T patent/DE69510940T2/de not_active Expired - Fee Related
- 1995-05-18 ES ES95917436T patent/ES2135062T3/es not_active Expired - Lifetime
- 1995-05-18 WO PCT/IB1995/000373 patent/WO1995034563A1/fr not_active Ceased
- 1995-05-18 DK DK95917436T patent/DK0765327T3/da active
- 1995-05-18 EP EP95917436A patent/EP0765327B1/fr not_active Expired - Lifetime
- 1995-05-25 TW TW084105306A patent/TW432064B/zh active
- 1995-06-05 IL IL11400395A patent/IL114003A/xx not_active IP Right Cessation
- 1995-06-07 BR BR9502707A patent/BR9502707A/pt not_active IP Right Cessation
- 1995-06-07 ZA ZA954679A patent/ZA954679B/xx unknown
- 1995-06-08 CO CO95024908A patent/CO4290424A1/es unknown
- 1995-06-08 PE PE1995270715A patent/PE13396A1/es not_active Application Discontinuation
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- 1996-12-13 NO NO965378A patent/NO307968B1/no not_active IP Right Cessation
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