NO308663B1 - AnalogifremgangsmÕte ved fremstilling av biologisk aktive forbindelser - Google Patents

AnalogifremgangsmÕte ved fremstilling av biologisk aktive forbindelser Download PDF

Info

Publication number: NO308663B1
Authority: NO; Norway
Prior art keywords: formula; compounds; boc; compound; mineral
Prior art date: 1990-05-15

Application number

NO911880A

Other languages

English (en)

Norwegian (no)

Other versions

NO911880L (no

NO911880D0 (no

Inventor

Jacques Chauveau

Michel Delaage

Anne Morel

Louis Segu

Original Assignee

Immunotech Sa

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1990-05-15

Filing date

1991-05-14

Publication date

2000-10-09

1990-05-15 Priority claimed from FR9006292A external-priority patent/FR2662082B1/fr

1991-01-30 Priority claimed from FR9101292A external-priority patent/FR2671971B1/fr

1991-05-14 Application filed by Immunotech Sa filed Critical Immunotech Sa

1991-05-14 Publication of NO911880D0 publication Critical patent/NO911880D0/no

1991-11-18 Publication of NO911880L publication Critical patent/NO911880L/no

2000-10-09 Publication of NO308663B1 publication Critical patent/NO308663B1/no

Links

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GETQZCLCWQTVFV-UHFFFAOYSA-N trimethylamine Chemical compound CN(C)C GETQZCLCWQTVFV-UHFFFAOYSA-N 0.000 description 1
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Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
- C07C229/02—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton
- C07C229/34—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton containing six-membered aromatic rings
- C07C229/36—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton containing six-membered aromatic rings with at least one amino group and one carboxyl group bound to the same carbon atom of the carbon skeleton
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
- C07D209/14—Radicals substituted by nitrogen atoms, not forming part of a nitro radical
- C07D209/16—Tryptamines
- G—PHYSICS
- G01—MEASURING; TESTING
- G01N—INVESTIGATING OR ANALYSING MATERIALS BY DETERMINING THEIR CHEMICAL OR PHYSICAL PROPERTIES
- G01N33/00—Investigating or analysing materials by specific methods not covered by groups G01N1/00 - G01N31/00
- G01N33/48—Biological material, e.g. blood, urine; Haemocytometers
- G01N33/50—Chemical analysis of biological material, e.g. blood, urine; Testing involving biospecific ligand binding methods; Immunological testing
- G01N33/74—Chemical analysis of biological material, e.g. blood, urine; Testing involving biospecific ligand binding methods; Immunological testing involving hormones or other non-cytokine intercellular protein regulatory factors such as growth factors, including receptors to hormones and growth factors
- G01N33/78—Thyroid gland hormones, e.g. T3, T4, TBH, TBG or their receptors

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Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Organic Chemistry (AREA)
Molecular Biology (AREA)
Engineering & Computer Science (AREA)
Urology & Nephrology (AREA)
Endocrinology (AREA)
Biomedical Technology (AREA)
Hematology (AREA)
Immunology (AREA)
Analytical Chemistry (AREA)
Food Science & Technology (AREA)
Medicinal Chemistry (AREA)
Physics & Mathematics (AREA)
Cell Biology (AREA)
Biochemistry (AREA)
General Health & Medical Sciences (AREA)
General Physics & Mathematics (AREA)
Pathology (AREA)
Biotechnology (AREA)
Microbiology (AREA)
Peptides Or Proteins (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Indole Compounds (AREA)
Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
Steroid Compounds (AREA)
Investigating Or Analysing Biological Materials (AREA)
Measuring Or Testing Involving Enzymes Or Micro-Organisms (AREA)
Medicinal Preparation (AREA)

NO911880A 1990-05-15 1991-05-14 AnalogifremgangsmÕte ved fremstilling av biologisk aktive forbindelser NO308663B1 (no)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
FR9006292A FR2662082B1 (fr)	1990-05-15	1990-05-15	Nouveaux derives de mediateurs endogenes, leurs sels, procede de preparation et applications.
FR9101292A FR2671971B1 (fr)	1991-01-30	1991-01-30	Nouveaux derives de la serotonine, application a titre de medicament et compositions les renfermant.

Publications (3)

Publication Number	Publication Date
NO911880D0 NO911880D0 (no)	1991-05-14
NO911880L NO911880L (no)	1991-11-18
NO308663B1 true NO308663B1 (no)	2000-10-09

Family

ID=26228029

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NO911880A NO308663B1 (no)	1990-05-15	1991-05-14	AnalogifremgangsmÕte ved fremstilling av biologisk aktive forbindelser

Country Status (12)

Country	Link
US (1)	US5298491A (da)
EP (1)	EP0457701B1 (da)
JP (1)	JP2968623B2 (da)
KR (1)	KR0138750B1 (da)
AT (1)	ATE118758T1 (da)
AU (1)	AU650265B2 (da)
CA (1)	CA2042295A1 (da)
DE (1)	DE69107512T2 (da)
DK (1)	DK0457701T3 (da)
ES (1)	ES2039313T3 (da)
IE (1)	IE67888B1 (da)
NO (1)	NO308663B1 (da)

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TW288010B (da) *	1992-03-05	1996-10-11	Pfizer
NZ251047A (en) *	1992-04-10	1996-09-25	Pfizer	Acylaminoindole derivatives and medicaments
TW251284B (da) *	1992-11-02	1995-07-11	Pfizer
FR2699918B1 (fr) *	1992-12-30	1995-03-17	Pf Medicament	Ligands sélectifs des récepteurs 5HY1D-5HT1B dérivés d'indole-pipérazine utiles comme médicaments.
DK0703923T3 (da) *	1993-06-18	1999-06-21	Nycomed Imaging As	Faktor VII afledte peptider
AU729415B2 (en)	1996-07-12	2001-02-01	Millennium Pharmaceuticals, Inc.	Chemokine receptor antagonists and methods of use therefor
FR2773489B1 (fr) *	1998-01-15	2001-03-23	Immunotech Sa	Nouvelle composition destinee a la voie oromuqueuse notamment pernasale
KR100596641B1 (ko) *	1998-12-11	2006-10-04	이승진	진단용 공중합성 미셀 및 그의 제조방법
US7163918B2 (en)	2000-08-22	2007-01-16	New River Pharmaceuticals Inc.	Iodothyronine compositions
US8394813B2 (en)	2000-11-14	2013-03-12	Shire Llc	Active agent delivery systems and methods for protecting and administering active agents
US20060014697A1 (en) *	2001-08-22	2006-01-19	Travis Mickle	Pharmaceutical compositions for prevention of overdose or abuse
DK1523486T3 (da)	2002-06-21	2008-03-03	Suven Life Sciences Ltd	Tetracykliske arylsulfonylindoler med serotoninreceptor-affinitet
DE60329607D1 (de)	2002-06-21	2009-11-19	Suven Life Sciences Ltd	Sich als therapeutische mittel eignende arylalkylindole mit affinität für den serotoninrezeptor, verfahren zu deren herstellung und pharmazeutische zusammensetzungen, die diese enthalten
JP4559230B2 (ja) *	2002-11-28	2010-10-06	スベンライフサイエンシズリミティド	セロトニン受容体に対する親和性を有する新規ｎ−アリールスルホニル−３−置換されたインドール、その調製方法、それを含有する医薬組成物
MXPA05005700A (es)	2002-11-28	2005-08-16	Suven Life Sciences Ltd	N-arilsulfonil-3-aminoalcoxiindoles.
EA009367B1 (ru)	2002-12-18	2007-12-28	Сувен Лайф Сайенсиз Лимитед	ПРОИЗВОДНЫЕ 5-ТИА-5-ДИОКСО-4b-АЗАИНДЕНО[2,1-a]ИНДЕНА, ОБЛАДАЮЩИЕ АФФИННОСТЬЮ К РЕЦЕПТОРУ СЕРОТОНИНА

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US2703325A (en) *	1951-12-06	1955-03-01	Upjohn Co	Preparation of 5-benzyloxytryptamines
US3182071A (en) *	1961-06-27	1965-05-04	Warner Lambert Pharmaceutical	Acylated indole derivatives
US3686213A (en) *	1970-08-28	1972-08-22	American Cyanamid Co	Substituted aminoethyl indoles
US4046636A (en) *	1974-06-20	1977-09-06	Syva Company	Diazepam enzyme conjugates
US3878187A (en) *	1972-09-11	1975-04-15	Syva Co	Polypeptide derivatives of amphetamine and analogs for immunoassays
US4040907A (en) *	1974-06-20	1977-08-09	Syva Company	Iodothyronine enzyme conjugates
DE2737802A1 (de) *	1977-08-22	1979-03-08	Henning Berlin Gmbh	Arzneimittel oder diagnostikum zur behandlung oder feststellung von schilddruesenfunktionsstoerungen und verfahren zu dessen herstellung
FR2437398A1 (fr) *	1978-06-20	1980-04-25	Commissariat Energie Atomique	Compose iode utilisable comme traceur en radio-immunologie
ZA795239B (en) *	1978-10-12	1980-11-26	Glaxo Group Ltd	Heterocyclic compounds
ZW19381A1 (en) *	1980-08-12	1983-03-09	Glaxo Group Ltd	Heterocyclic compounds
US4426453A (en) *	1980-09-18	1984-01-17	Amersham International Limited	Derivatives of iodothyronine compounds and their use in an assay for the free iodothyronine compounds
EP0099707B1 (en) *	1982-07-16	1986-12-10	Beecham Group Plc	2-aminoethyl ether derivatives, processes for their preparation and pharmaceutical compositions containing them
JPS60132935A (ja) *	1983-12-20	1985-07-16	Sumitomo Chem Co Ltd	フエニルセリン誘導体及びその製造方法
FR2562671B1 (fr) *	1984-04-10	1986-07-25	Immunotech Sa	Procede pour le dosage immunologique des monoamines
US4833153A (en) *	1985-11-08	1989-05-23	Glaxo Group Limited	Indole derivatives
GB8530507D0 (en) *	1985-12-11	1986-01-22	Glaxo Group Plc	Chemical compounds
US4910193A (en) *	1985-12-16	1990-03-20	Sandoz Ltd.	Treatment of gastrointestinal disorders
DE3628795A1 (de) *	1986-08-25	1988-03-03	Hoechst Ag	Neue thyroninderivate
US5019586A (en) *	1987-04-14	1991-05-28	Glaxo Group Limited	Ketone derivatives
GB8801306D0 (en) *	1988-01-21	1988-02-17	Ici Plc	Chemical compounds
GB8802127D0 (en) *	1988-02-01	1988-03-02	Glaxo Group Ltd	Chemical compounds
US4933324A (en) *	1988-02-26	1990-06-12	Shashoua Victor E	Fatty acid-neuroactive drug conjugate as a prodrug
FR2671971B1 (fr) *	1991-01-30	1994-01-28	Immunotech	Nouveaux derives de la serotonine, application a titre de medicament et compositions les renfermant.
FR2662082B1 (fr) *	1990-05-15	1994-12-23	Immunotech Sa	Nouveaux derives de mediateurs endogenes, leurs sels, procede de preparation et applications.

1991
- 1991-05-10 CA CA002042295A patent/CA2042295A1/fr not_active Abandoned
- 1991-05-13 EP EP91430009A patent/EP0457701B1/fr not_active Expired - Lifetime
- 1991-05-13 US US07/699,027 patent/US5298491A/en not_active Expired - Lifetime
- 1991-05-13 ES ES91430009T patent/ES2039313T3/es not_active Expired - Lifetime
- 1991-05-13 DE DE69107512T patent/DE69107512T2/de not_active Expired - Lifetime
- 1991-05-13 DK DK91430009.0T patent/DK0457701T3/da active
- 1991-05-13 AT AT91430009T patent/ATE118758T1/de not_active IP Right Cessation
- 1991-05-14 AU AU77045/91A patent/AU650265B2/en not_active Ceased
- 1991-05-14 NO NO911880A patent/NO308663B1/no unknown
- 1991-05-14 KR KR1019910007750A patent/KR0138750B1/ko not_active Expired - Fee Related
- 1991-05-14 IE IE164991A patent/IE67888B1/en unknown
- 1991-05-15 JP JP3205013A patent/JP2968623B2/ja not_active Expired - Fee Related

Also Published As

Publication number	Publication date
AU650265B2 (en)	1994-06-16
KR910020034A (ko)	1991-12-19
JP2968623B2 (ja)	1999-10-25
JPH04288044A (ja)	1992-10-13
IE67888B1 (en)	1996-05-01
KR0138750B1 (ko)	1998-05-01
DE69107512D1 (de)	1995-03-30
CA2042295A1 (fr)	1991-11-16
IE911649A1 (en)	1991-11-20
NO911880L (no)	1991-11-18
US5298491A (en)	1994-03-29
EP0457701A1 (fr)	1991-11-21
DE69107512T2 (de)	1995-06-29
ES2039313T1 (es)	1993-10-01
EP0457701B1 (fr)	1995-02-22
ATE118758T1 (de)	1995-03-15
ES2039313T3 (es)	1995-04-16
AU7704591A (en)	1991-11-21
NO911880D0 (no)	1991-05-14
DK0457701T3 (da)	1996-02-05

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