NO312679B1 - N6 heterocykliske substituerte adenosinderivater, farmasöytisk sammensetning inneholdende samme, og anvendelse avsamme for fremstilling av preparat - Google Patents

N6 heterocykliske substituerte adenosinderivater, farmasöytisk sammensetning inneholdende samme, og anvendelse avsamme for fremstilling av preparat Download PDF

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Publication number
NO312679B1
NO312679B1 NO19990787A NO990787A NO312679B1 NO 312679 B1 NO312679 B1 NO 312679B1 NO 19990787 A NO19990787 A NO 19990787A NO 990787 A NO990787 A NO 990787A NO 312679 B1 NO312679 B1 NO 312679B1
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NO
Norway
Prior art keywords
preparation
pharmaceutical composition
compound
same
receptor
Prior art date
Application number
NO19990787A
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English (en)
Norwegian (no)
Other versions
NO990787L (no
NO990787D0 (no
Inventor
Robert T Lum
Jurg Roland Pfister
Steven R Schow
Michael M Wick
Marek G Nelson
George F Schreiner
Original Assignee
Cv Therapeutics Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Cv Therapeutics Inc filed Critical Cv Therapeutics Inc
Publication of NO990787L publication Critical patent/NO990787L/no
Publication of NO990787D0 publication Critical patent/NO990787D0/no
Priority to NO20020758A priority Critical patent/NO322459B1/no
Priority to NO20020759A priority patent/NO20020759D0/no
Publication of NO312679B1 publication Critical patent/NO312679B1/no

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/16—Purine radicals
    • C07H19/167—Purine radicals with ribosyl as the saccharide radical
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/16—Purine radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/06—Antiarrhythmics

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Cardiology (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
NO19990787A 1996-08-27 1999-02-19 N6 heterocykliske substituerte adenosinderivater, farmasöytisk sammensetning inneholdende samme, og anvendelse avsamme for fremstilling av preparat NO312679B1 (no)

Priority Applications (2)

Application Number Priority Date Filing Date Title
NO20020758A NO322459B1 (no) 1996-08-27 2002-02-15 N6 heterocykliske substituerte adenosinderivater, farmasoytiske sammensetninger omfattende samme, og anvendelse av samme for fremstilling av medikament.
NO20020759A NO20020759D0 (no) 1996-08-27 2002-02-15 N<o>6</o> heterocykliske substituerte adenosinderivater

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US08702234 US5789416B1 (en) 1996-08-27 1996-08-27 N6 mono heterocyclic substituted adenosine derivatives
PCT/US1997/014724 WO1998008855A2 (en) 1996-08-27 1997-08-20 N6 heterocyclic substituted adenosine derivatives

Publications (3)

Publication Number Publication Date
NO990787L NO990787L (no) 1999-02-19
NO990787D0 NO990787D0 (no) 1999-02-19
NO312679B1 true NO312679B1 (no) 2002-06-17

Family

ID=24820367

Family Applications (3)

Application Number Title Priority Date Filing Date
NO19990787A NO312679B1 (no) 1996-08-27 1999-02-19 N6 heterocykliske substituerte adenosinderivater, farmasöytisk sammensetning inneholdende samme, og anvendelse avsamme for fremstilling av preparat
NO20020758A NO322459B1 (no) 1996-08-27 2002-02-15 N6 heterocykliske substituerte adenosinderivater, farmasoytiske sammensetninger omfattende samme, og anvendelse av samme for fremstilling av medikament.
NO20020759A NO20020759D0 (no) 1996-08-27 2002-02-15 N<o>6</o> heterocykliske substituerte adenosinderivater

Family Applications After (2)

Application Number Title Priority Date Filing Date
NO20020758A NO322459B1 (no) 1996-08-27 2002-02-15 N6 heterocykliske substituerte adenosinderivater, farmasoytiske sammensetninger omfattende samme, og anvendelse av samme for fremstilling av medikament.
NO20020759A NO20020759D0 (no) 1996-08-27 2002-02-15 N<o>6</o> heterocykliske substituerte adenosinderivater

Country Status (24)

Country Link
US (1) US5789416B1 (de)
EP (3) EP0920438B1 (de)
JP (1) JP3157842B2 (de)
KR (1) KR100331775B1 (de)
CN (1) CN100363377C (de)
AT (2) ATE234323T1 (de)
AU (1) AU726597B2 (de)
BR (1) BR9711444A (de)
CA (1) CA2264155C (de)
CZ (1) CZ296855B6 (de)
DE (2) DE69719816T2 (de)
DK (2) DK0992510T3 (de)
ES (2) ES2189330T3 (de)
GE (1) GEP20012419B (de)
GR (1) GR3036332T3 (de)
HU (1) HU226057B1 (de)
IL (2) IL128652A0 (de)
NO (3) NO312679B1 (de)
NZ (3) NZ334095A (de)
PL (1) PL187635B1 (de)
PT (1) PT920438E (de)
TR (2) TR199900377T2 (de)
UA (1) UA62936C2 (de)
WO (1) WO1998008855A2 (de)

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Also Published As

Publication number Publication date
NO990787L (no) 1999-02-19
KR20000035867A (ko) 2000-06-26
ATE202361T1 (de) 2001-07-15
IL128652A (en) 2008-06-05
EP0920438B1 (de) 2001-06-20
NO20020759L (no) 1999-02-19
EP0920438A2 (de) 1999-06-09
DK0920438T3 (da) 2001-09-10
NO20020758D0 (no) 2002-02-15
HK1020967A1 (en) 2000-05-26
CZ61499A3 (cs) 1999-10-13
US5789416A (en) 1998-08-04
CA2264155C (en) 2003-11-18
TR200202287T2 (tr) 2003-01-21
ATE234323T1 (de) 2003-03-15
NO20020759D0 (no) 2002-02-15
US5789416B1 (en) 1999-10-05
DE69705312T2 (de) 2001-10-11
DE69705312D1 (de) 2001-07-26
CA2264155A1 (en) 1998-03-05
CN1234803A (zh) 1999-11-10
EP1081155A2 (de) 2001-03-07
BR9711444A (pt) 2000-01-18
JP3157842B2 (ja) 2001-04-16
NZ505428A (en) 2005-03-24
PL187635B1 (pl) 2004-08-31
HUP0001640A2 (hu) 2001-05-28
AU726597B2 (en) 2000-11-16
CZ296855B6 (cs) 2006-07-12
NO990787D0 (no) 1999-02-19
DE69719816D1 (de) 2003-04-17
GEP20012419B (en) 2001-04-25
EP1081155A3 (de) 2003-05-02
DK0992510T3 (da) 2003-07-07
DE69719816T2 (de) 2003-12-18
ES2157593T3 (es) 2001-08-16
NZ334095A (en) 2000-10-27
IL128652A0 (en) 2000-01-31
EP0992510A1 (de) 2000-04-12
WO1998008855A3 (en) 1998-09-03
EP0992510B1 (de) 2003-03-12
ES2189330T3 (es) 2003-07-01
KR100331775B1 (ko) 2002-04-09
CN100363377C (zh) 2008-01-23
NO322459B1 (no) 2006-10-09
GR3036332T3 (en) 2001-11-30
NO20020758L (no) 1999-02-19
UA62936C2 (en) 2004-01-15
AU4080997A (en) 1998-03-19
WO1998008855A2 (en) 1998-03-05
JP2000501426A (ja) 2000-02-08
HU226057B1 (en) 2008-04-28
NZ512242A (en) 2004-01-30
PL331853A1 (en) 1999-08-16
PT920438E (pt) 2001-10-30
TR199900377T2 (xx) 1999-05-21
HUP0001640A3 (en) 2002-04-29

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