NO314405B1 - Farmasöytisk aktive forbindelser og liposomer og anvendelse derav - Google Patents

Farmasöytisk aktive forbindelser og liposomer og anvendelse derav Download PDF

Info

Publication number: NO314405B1
Authority: NO; Norway
Prior art keywords: group; carbons; alkyl; formula; chain
Prior art date: 1994-02-02

Application number

NO19963224A

Other languages

English (en)

Norwegian (no)

Other versions

NO963224L (no

NO963224D0 (no

Inventor

Yong-Wei Pei

Eric Mayhew

Imran Ahmad

Andrew Stuart Janoff

Original Assignee

Liposome Co Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1994-02-02

Filing date

1996-08-01

Publication date

2003-03-17

1996-08-01 Application filed by Liposome Co Inc filed Critical Liposome Co Inc

1996-08-01 Publication of NO963224D0 publication Critical patent/NO963224D0/no

1996-09-27 Publication of NO963224L publication Critical patent/NO963224L/no

2003-03-17 Publication of NO314405B1 publication Critical patent/NO314405B1/no

Links

150000001875 compounds Chemical class 0.000 title claims abstract description 61
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125000000217 alkyl group Chemical group 0.000 claims abstract description 74
125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 claims abstract description 40
230000002401 inhibitory effect Effects 0.000 claims abstract description 31
125000004432 carbon atom Chemical group C* 0.000 claims abstract description 20
125000003342 alkenyl group Chemical group 0.000 claims abstract description 18
125000000304 alkynyl group Chemical group 0.000 claims abstract description 18
125000001931 aliphatic group Chemical group 0.000 claims abstract description 12
125000002924 primary amino group Chemical group [H]N([H])* 0.000 claims abstract description 12
150000002632 lipids Chemical class 0.000 claims description 41
125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 claims description 34
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239000012867 bioactive agent Substances 0.000 claims description 18
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Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/10—Dispersions; Emulsions
- A61K9/127—Synthetic bilayered vehicles, e.g. liposomes or liposomes with cholesterol as the only non-phosphatidyl surfactant
- A61K9/1271—Non-conventional liposomes, e.g. PEGylated liposomes or liposomes coated or grafted with polymers
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
- C07F7/02—Silicon compounds
- C07F7/08—Compounds having one or more C—Si linkages
- C07F7/18—Compounds having one or more C—Si linkages as well as one or more C—O—Si linkages
- C07F7/1804—Compounds having Si-O-C linkages
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
- Y10T—TECHNICAL SUBJECTS COVERED BY FORMER US CLASSIFICATION
- Y10T428/00—Stock material or miscellaneous articles
- Y10T428/29—Coated or structually defined flake, particle, cell, strand, strand portion, rod, filament, macroscopic fiber or mass thereof
- Y10T428/2982—Particulate matter [e.g., sphere, flake, etc.]
- Y10T428/2984—Microcapsule with fluid core [includes liposome]

Landscapes

Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Veterinary Medicine (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Epidemiology (AREA)
Dispersion Chemistry (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Medicinal Preparation (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Steroid Compounds (AREA)
Manufacturing Of Micro-Capsules (AREA)

NO19963224A 1994-02-02 1996-08-01 Farmasöytisk aktive forbindelser og liposomer og anvendelse derav NO314405B1 (no)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US19029594A	1994-02-02	1994-02-02
PCT/US1995/001490 WO1995021175A1 (en)	1994-02-02	1995-02-02	Pharmaceutically active compounds and liposomes, and methods of use therof

Publications (3)

Publication Number	Publication Date
NO963224D0 NO963224D0 (no)	1996-08-01
NO963224L NO963224L (no)	1996-09-27
NO314405B1 true NO314405B1 (no)	2003-03-17

Family

ID=22700754

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO19963224A NO314405B1 (no)	1994-02-02	1996-08-01	Farmasöytisk aktive forbindelser og liposomer og anvendelse derav

Country Status (14)

Country	Link
US (3)	US5631394A (de)
EP (2)	EP0742789B1 (de)
JP (1)	JPH09508900A (de)
AT (1)	ATE195944T1 (de)
AU (1)	AU691886B2 (de)
CA (1)	CA2182485A1 (de)
DE (1)	DE69518627T2 (de)
DK (1)	DK0742789T3 (de)
ES (1)	ES2149350T3 (de)
FI (1)	FI116620B (de)
GR (1)	GR3034521T3 (de)
NO (1)	NO314405B1 (de)
PT (1)	PT742789E (de)
WO (1)	WO1995021175A1 (de)

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1995
- 1995-02-02 ES ES95910923T patent/ES2149350T3/es not_active Expired - Lifetime
- 1995-02-02 CA CA002182485A patent/CA2182485A1/en not_active Abandoned
- 1995-02-02 US US08/383,291 patent/US5631394A/en not_active Expired - Fee Related
- 1995-02-02 EP EP95910923A patent/EP0742789B1/de not_active Expired - Lifetime
- 1995-02-02 EP EP00102434A patent/EP1008342A3/de not_active Withdrawn
- 1995-02-02 AT AT95910923T patent/ATE195944T1/de not_active IP Right Cessation
- 1995-02-02 PT PT95910923T patent/PT742789E/pt unknown
- 1995-02-02 AU AU18712/95A patent/AU691886B2/en not_active Ceased
- 1995-02-02 JP JP7520799A patent/JPH09508900A/ja not_active Ceased
- 1995-02-02 DK DK95910923T patent/DK0742789T3/da active
- 1995-02-02 DE DE69518627T patent/DE69518627T2/de not_active Expired - Fee Related
- 1995-02-02 WO PCT/US1995/001490 patent/WO1995021175A1/en not_active Ceased
- 1995-10-19 US US08/545,164 patent/US5681589A/en not_active Expired - Lifetime
- 1995-10-19 US US08/547,688 patent/US5677337A/en not_active Expired - Lifetime
1996
- 1996-08-01 NO NO19963224A patent/NO314405B1/no unknown
- 1996-08-01 FI FI963045A patent/FI116620B/fi not_active IP Right Cessation
2000
- 2000-09-29 GR GR20000402211T patent/GR3034521T3/el not_active IP Right Cessation

Also Published As

Publication number	Publication date
US5631394A (en)	1997-05-20
ATE195944T1 (de)	2000-09-15
JPH09508900A (ja)	1997-09-09
EP1008342A3 (de)	2004-12-29
US5681589A (en)	1997-10-28
FI963045L (fi)	1996-08-01
FI116620B (fi)	2006-01-13
EP0742789B1 (de)	2000-08-30
FI963045A0 (fi)	1996-08-01
DE69518627D1 (de)	2000-10-05
WO1995021175A1 (en)	1995-08-10
EP0742789A1 (de)	1996-11-20
DK0742789T3 (da)	2000-11-13
CA2182485A1 (en)	1995-08-10
AU1871295A (en)	1995-08-21
GR3034521T3 (en)	2000-12-29
US5677337A (en)	1997-10-14
ES2149350T3 (es)	2000-11-01
PT742789E (pt)	2000-12-29
DE69518627T2 (de)	2001-01-11
EP1008342A2 (de)	2000-06-14
NO963224L (no)	1996-09-27
NO963224D0 (no)	1996-08-01
AU691886B2 (en)	1998-05-28

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