NO320495B1 - Intrakonazolininneholdende partikler og farmasoytiske doseringsformer inneholdende disse samt fremgamsmater for fremstilling av det samme - Google Patents

Intrakonazolininneholdende partikler og farmasoytiske doseringsformer inneholdende disse samt fremgamsmater for fremstilling av det samme Download PDF

Info

Publication number: NO320495B1
Authority: NO; Norway
Prior art keywords: dosage form; itraconazole; particles; mixture; weight
Prior art date: 1996-05-20

Application number

NO19982599A

Other languages

English (en)

Norwegian (no)

Other versions

NO982599L (no

NO982599D0 (no

Inventor

Daniel Joseph Christiaan Thone

Lieven Elvire Colette Baert

Geert Verreck

Original Assignee

Janssen Pharmaceutica Nv

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1996-05-20

Filing date

1998-06-05

Publication date

2005-12-12

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=26142825&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO320495(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

1998-06-05 Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv

1998-06-05 Publication of NO982599D0 publication Critical patent/NO982599D0/no

1998-11-19 Publication of NO982599L publication Critical patent/NO982599L/no

2005-12-12 Publication of NO320495B1 publication Critical patent/NO320495B1/no

Links

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Classifications

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- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A—HUMAN NECESSITIES
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- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/141—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
- A61K9/146—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic macromolecular compounds
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1629—Organic macromolecular compounds
- A61K9/1652—Polysaccharides, e.g. alginate, cellulose derivatives; Cyclodextrin
- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
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- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/2027—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
- A61K9/2077—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2806—Coating materials
- A61K9/2833—Organic macromolecular compounds
- A61K9/286—Polysaccharides, e.g. gums; Cyclodextrin
- A61K9/2866—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/10—Antimycotics

Landscapes

Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Chemical & Material Sciences (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Medicinal Chemistry (AREA)
General Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Pharmacology & Pharmacy (AREA)
Epidemiology (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Organic Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Oncology (AREA)
Communicable Diseases (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Medicinal Preparation (AREA)
Agricultural Chemicals And Associated Chemicals (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

NO19982599A 1996-05-20 1998-06-05 Intrakonazolininneholdende partikler og farmasoytiske doseringsformer inneholdende disse samt fremgamsmater for fremstilling av det samme NO320495B1 (no)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
EP96201430		1996-05-20
EP97200698		1997-03-07
PCT/EP1997/002507 WO1997044014A1 (en)	1996-05-20	1997-05-12	Antifungal compositions with improved bioavailability

Publications (3)

Publication Number	Publication Date
NO982599D0 NO982599D0 (no)	1998-06-05
NO982599L NO982599L (no)	1998-11-19
NO320495B1 true NO320495B1 (no)	2005-12-12

Family

ID=26142825

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO19982599A NO320495B1 (no)	1996-05-20	1998-06-05	Intrakonazolininneholdende partikler og farmasoytiske doseringsformer inneholdende disse samt fremgamsmater for fremstilling av det samme

Country Status (33)

Country	Link
US (4)	US6509038B2 (pl)
EP (1)	EP0904060B1 (pl)
JP (1)	JP3391801B2 (pl)
KR (1)	KR19990044257A (pl)
CN (1)	CN1165291C (pl)
AR (1)	AR007195A1 (pl)
AT (1)	ATE255883T1 (pl)
AU (1)	AU722101B2 (pl)
BG (1)	BG64368B1 (pl)
BR (1)	BR9706897B1 (pl)
CA (1)	CA2240161C (pl)
CY (1)	CY2434B1 (pl)
CZ (1)	CZ293841B6 (pl)
DE (1)	DE69726729T2 (pl)
DK (1)	DK0904060T3 (pl)
EA (1)	EA001219B1 (pl)
EE (1)	EE03902B1 (pl)
ES (1)	ES2212810T3 (pl)
HR (1)	HRP970270B1 (pl)
HU (1)	HU227745B1 (pl)
ID (1)	ID16926A (pl)
IL (1)	IL124935A (pl)
MX (1)	MX9805418A (pl)
MY (1)	MY123827A (pl)
NO (1)	NO320495B1 (pl)
NZ (1)	NZ330739A (pl)
PL (1)	PL188566B1 (pl)
PT (1)	PT904060E (pl)
SI (1)	SI0904060T1 (pl)
SK (1)	SK284145B6 (pl)
TR (1)	TR199801225T2 (pl)
TW (1)	TW460282B (pl)
WO (1)	WO1997044014A1 (pl)

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KR19990001564A (ko) *	1997-06-16	1999-01-15	유충식	용해도를 개선한 아졸계 항진균제 및 이를 함유하는 제제
KR100514330B1 (ko) *	1997-12-31	2006-02-17	주식회사 중외제약	난용성 약물을 함유하는 코팅정
KR100288890B1 (ko) *	1997-12-31	2001-05-02	최현식	이트라코나졸 경구용 제제 및 그의 제조방법
CA2317106C (en) *	1997-12-31	2004-11-23	Choongwae Pharma Corporation	Method and composition of an oral preparation of itraconazole
AU736555B2 (en)	1998-01-07	2001-08-02	Meiji Seika Pharma Co., Ltd.	A composition comprising a crystallographically stable, amphorous cephalosporin and processes for the preparation thereof
ES2157731B1 (es) *	1998-07-21	2002-05-01	Liconsa Liberacion Controlada	Preparacion farmaceutica oral de un compuesto de actividad antifungica y procedimiento para su preparacion.
ES2251985T3 (es) *	1999-03-24	2006-05-16	R.P. Scherer Technologies, Inc.	Particula granulada para mejorar la solubilidad acuosa de farmacos, y su procedimiento de preparacion.
KR100331529B1 (ko) *	1999-06-16	2002-04-06	민경윤	난용성 항진균제의 경구투여용 조성물 및 그의 제조 방법
CA2359945C (en)	1999-11-12	2011-04-26	Abbott Laboratories	Inhibitors of crystallization in a solid dispersion
EP2415462A1 (en)	1999-12-23	2012-02-08	Mayne Pharma International Pty Ltd.	Improved pharmaceutical compositions for poorly soluble drugs
FR2803748A1 (fr) *	2000-01-14	2001-07-20	Ethypharm Lab Prod Ethiques	Composition d'itraconazole et procede de preparation
DE10026698A1 (de)	2000-05-30	2001-12-06	Basf Ag	Selbstemulgierende Wirkstoffformulierung und Verwendung dieser Formulierung
NZ540748A (en) *	2000-06-22	2007-04-27	Novartis Ag	An oral solid pharmaceutical composition comprising valsartan and a filler in a weight ratio from 2:1 to 1:1
DE10038571A1 (de) *	2000-08-03	2002-02-14	Knoll Ag	Zusammensetzungen und Dosierungsformen zur Anwendung in der Mundhöhle bei der Bhandlung von Mykosen
US20050048126A1 (en) *	2000-12-22	2005-03-03	Barrett Rabinow	Formulation to render an antimicrobial drug potent against organisms normally considered to be resistant to the drug
US6869617B2 (en)	2000-12-22	2005-03-22	Baxter International Inc.	Microprecipitation method for preparing submicron suspensions
US8067032B2 (en)	2000-12-22	2011-11-29	Baxter International Inc.	Method for preparing submicron particles of antineoplastic agents
US9700866B2 (en)	2000-12-22	2017-07-11	Baxter International Inc.	Surfactant systems for delivery of organic compounds
US6951656B2 (en)	2000-12-22	2005-10-04	Baxter International Inc.	Microprecipitation method for preparing submicron suspensions
US6884436B2 (en) *	2000-12-22	2005-04-26	Baxter International Inc.	Method for preparing submicron particle suspensions
US6977085B2 (en)	2000-12-22	2005-12-20	Baxter International Inc.	Method for preparing submicron suspensions with polymorph control
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- 1998-06-05 NO NO19982599A patent/NO320495B1/no not_active IP Right Cessation
- 1998-06-11 BG BG102532A patent/BG64368B1/bg unknown
- 1998-07-02 MX MX9805418A patent/MX9805418A/es active IP Right Grant
2002
- 2002-08-14 US US10/218,851 patent/US7081255B2/en not_active Expired - Fee Related
2004
- 2004-03-29 CY CY0400023A patent/CY2434B1/xx unknown
2006
- 2006-06-01 US US11/445,849 patent/US8591948B2/en not_active Expired - Fee Related
2013
- 2013-11-01 US US14/069,842 patent/US9642806B2/en not_active Expired - Fee Related

Also Published As

Publication number	Publication date
AU722101B2 (en)	2000-07-20
JP3391801B2 (ja)	2003-03-31
EE9800304A (et)	1999-02-15
TR199801225T2 (xx)	1998-11-23
NO982599L (no)	1998-11-19
MY123827A (en)	2006-06-30
HRP970270A2 (en)	1998-04-30
SK284145B6 (sk)	2004-10-05
US20010007678A1 (en)	2001-07-12
US20030082239A1 (en)	2003-05-01
ATE255883T1 (de)	2003-12-15
IL124935A (en)	2001-06-14
US7081255B2 (en)	2006-07-25
WO1997044014A1 (en)	1997-11-27
EA199800571A1 (ru)	1998-12-24
PL188566B1 (pl)	2005-02-28
PT904060E (pt)	2004-04-30
CZ293841B6 (cs)	2004-08-18
NZ330739A (en)	1999-06-29
DE69726729D1 (de)	2004-01-22
US20060263436A1 (en)	2006-11-23
DK0904060T3 (da)	2004-04-13
SI0904060T1 (en)	2004-04-30
HUP9901620A3 (en)	2000-03-28
US8591948B2 (en)	2013-11-26
BG102532A (en)	1999-02-26
CN1209740A (zh)	1999-03-03
CY2434B1 (en)	2004-11-12
HU227745B1 (en)	2012-02-28
PL330931A1 (en)	1999-06-07
AR007195A1 (es)	1999-10-13
IL124935A0 (en)	1999-01-26
EE03902B1 (et)	2002-12-16
CA2240161A1 (en)	1997-11-27
ID16926A (id)	1997-11-20
CA2240161C (en)	2005-05-24
BR9706897B1 (pt)	2010-09-21
BG64368B1 (bg)	2004-12-30
KR19990044257A (ko)	1999-06-25
HRP970270B1 (en)	2005-02-28
EA001219B1 (ru)	2000-12-25
TW460282B (en)	2001-10-21
ES2212810T3 (es)	2004-08-01
MX9805418A (es)	1998-10-31
EP0904060A1 (en)	1999-03-31
NO982599D0 (no)	1998-06-05
US20140134244A1 (en)	2014-05-15
CN1165291C (zh)	2004-09-08
CZ188598A3 (cs)	1998-11-11
DE69726729T2 (de)	2004-12-02
SK84898A3 (en)	1999-03-12
HUP9901620A2 (hu)	1999-10-28
JPH11509238A (ja)	1999-08-17
AU2956297A (en)	1997-12-09
BR9706897A (pt)	1999-08-31
US6509038B2 (en)	2003-01-21
EP0904060B1 (en)	2003-12-10
HK1018002A1 (en)	1999-12-10
US9642806B2 (en)	2017-05-09

Legal Events

Date	Code	Title	Description
2017-05-22	MK1K	Patent expired

Publication	Publication Date	Title
NO320495B1 (no)	2005-12-12	Intrakonazolininneholdende partikler og farmasoytiske doseringsformer inneholdende disse samt fremgamsmater for fremstilling av det samme
EP0969821B1 (en)	2003-06-04	Pellets having a core coated with an antifungal and a polymer
EP0872233A1 (en)	1998-10-21	Antiretroviral compositions with improved bioavailability
AU766041B2 (en)	2003-10-09	Pellets having a core coated with an antifungal and a polymer
JP5763735B2 (ja)	2015-08-12	改善された生物学的利用能をもつイトラコナゾール組成物
EP1028730B1 (en)	2002-04-17	Compositions of lipid lowering agents
EP2696857A1 (en)	2014-02-19	Pharmaceutical composition comprising bosentan
HK1018002B (en)	2004-04-16	Antifungal compositions with improved bioavailability
UA72424C2 (en)	2005-03-15	Particles, solid dispersion and dosage form of itraconazole, method for their manufacture (variants) and pharmaceutical package
HK1022840B (en)	2003-09-05	Pellets having a core coated with an antifungal and a polymer