NO324621B1 - Farmasoytiske blandinger for forlenget peptidfrigjoring - Google Patents

Farmasoytiske blandinger for forlenget peptidfrigjoring Download PDF

Info

Publication number: NO324621B1
Authority: NO; Norway
Prior art keywords: peptide; mixture according; pharmaceutical mixture; hormone; factor
Prior art date: 1998-03-25

Application number

NO20004741A

Other languages

English (en)

Norwegian (no)

Other versions

NO20004741L (no

NO20004741D0 (no

Inventor

Marc Pellet

Frederic Bismuth

Original Assignee

Sod Conseils Rech Applic

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1998-03-25

Filing date

2000-09-22

Publication date

2007-11-26

2000-09-22 Application filed by Sod Conseils Rech Applic filed Critical Sod Conseils Rech Applic

2000-09-22 Publication of NO20004741D0 publication Critical patent/NO20004741D0/no

2000-11-22 Publication of NO20004741L publication Critical patent/NO20004741L/no

2007-11-26 Publication of NO324621B1 publication Critical patent/NO324621B1/no

Links

108090000765 processed proteins & peptides Proteins 0.000 title claims abstract description 76
239000008194 pharmaceutical composition Substances 0.000 title abstract 2
239000000203 mixture Substances 0.000 claims abstract description 78
150000003839 salts Chemical class 0.000 claims abstract description 54
239000007787 solid Substances 0.000 claims abstract description 20
XLYOFNOQVPJJNP-UHFFFAOYSA-N water Substances O XLYOFNOQVPJJNP-UHFFFAOYSA-N 0.000 claims abstract description 20
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RUGAHXUZHWYHNG-NLGNTGLNSA-N acetic acid;(4r,7s,10s,13r,16s,19r)-10-(4-aminobutyl)-n-[(2s,3r)-1-amino-3-hydroxy-1-oxobutan-2-yl]-19-[[(2r)-2-amino-3-naphthalen-2-ylpropanoyl]amino]-16-[(4-hydroxyphenyl)methyl]-13-(1h-indol-3-ylmethyl)-6,9,12,15,18-pentaoxo-7-propan-2-yl-1,2-dithia-5, Chemical compound CC(O)=O.CC(O)=O.CC(O)=O.CC(O)=O.CC(O)=O.C([C@H]1C(=O)N[C@H](CC=2C3=CC=CC=C3NC=2)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(N[C@@H](CSSC[C@@H](C(=O)N1)NC(=O)[C@H](N)CC=1C=C2C=CC=CC2=CC=1)C(=O)N[C@@H]([C@@H](C)O)C(N)=O)=O)C(C)C)C1=CC=C(O)C=C1.C([C@H]1C(=O)N[C@H](CC=2C3=CC=CC=C3NC=2)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(N[C@@H](CSSC[C@@H](C(=O)N1)NC(=O)[C@H](N)CC=1C=C2C=CC=CC2=CC=1)C(=O)N[C@@H]([C@@H](C)O)C(N)=O)=O)C(C)C)C1=CC=C(O)C=C1 RUGAHXUZHWYHNG-NLGNTGLNSA-N 0.000 claims description 21
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Classifications

- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
- A61K9/0024—Solid, semi-solid or solidifying implants, which are implanted or injected in body tissue
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
- A61K38/08—Peptides having 5 to 11 amino acids
- A61K38/09—Luteinising hormone-releasing hormone [LHRH], i.e. Gonadotropin-releasing hormone [GnRH]; Related peptides
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/19—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles lyophilised, i.e. freeze-dried, solutions or dispersions

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Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Epidemiology (AREA)
Veterinary Medicine (AREA)
Chemical & Material Sciences (AREA)
Engineering & Computer Science (AREA)
Public Health (AREA)
Medicinal Chemistry (AREA)
General Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Bioinformatics & Cheminformatics (AREA)
Immunology (AREA)
Proteomics, Peptides & Aminoacids (AREA)
Endocrinology (AREA)
Gastroenterology & Hepatology (AREA)
Reproductive Health (AREA)
Biomedical Technology (AREA)
Neurosurgery (AREA)
Dermatology (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Medicinal Preparation (AREA)
Peptides Or Proteins (AREA)

NO20004741A 1998-03-25 2000-09-22 Farmasoytiske blandinger for forlenget peptidfrigjoring NO324621B1 (no)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
FR9803667A FR2776520B1 (fr)	1998-03-25	1998-03-25	Nouvelles compositions pharmaceutiques destinees a la liberation prolongee de peptides et leur procede de preparation
PCT/FR1999/000667 WO1999048517A1 (fr)	1998-03-25	1999-03-22	Compositions pharmaceutiques destinees a la liberation prolongee de peptides et leur procede de preparation

Publications (3)

Publication Number	Publication Date
NO20004741D0 NO20004741D0 (no)	2000-09-22
NO20004741L NO20004741L (no)	2000-11-22
NO324621B1 true NO324621B1 (no)	2007-11-26

Family

ID=9524472

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO20004741A NO324621B1 (no)	1998-03-25	2000-09-22	Farmasoytiske blandinger for forlenget peptidfrigjoring

Country Status (19)

Country	Link
US (1)	US6503534B1 (pl)
EP (1)	EP1066049B1 (pl)
JP (1)	JP4162381B2 (pl)
AR (1)	AR020062A1 (pl)
AT (1)	ATE241377T1 (pl)
AU (1)	AU756148B2 (pl)
CA (1)	CA2324901C (pl)
CZ (1)	CZ298941B6 (pl)
DE (1)	DE69908326T2 (pl)
DK (1)	DK1066049T3 (pl)
ES (1)	ES2200507T3 (pl)
FR (1)	FR2776520B1 (pl)
HU (1)	HU228903B1 (pl)
IL (2)	IL138533A0 (pl)
NO (1)	NO324621B1 (pl)
PL (1)	PL197775B1 (pl)
PT (1)	PT1066049E (pl)
RU (1)	RU2224538C2 (pl)
WO (1)	WO1999048517A1 (pl)

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BR122013009981B1 (pt)	2009-04-23	2020-02-11	United-Ah Ii, Llc	Composição para sincronizar o tempo de inseminação
TWI508734B (zh)	2009-05-01	2015-11-21	Ferring Int Ct Sa	用於前列腺癌之治療的組成物
TW201043221A (en) *	2009-05-06	2010-12-16	Ferring Int Ct Sa	Kit and method for preparation of a Degarelix solution
US20110039787A1 (en) *	2009-07-06	2011-02-17	Ferring International Center S.A.	Compositions, kits and methods for treating benign prostate hyperplasia
JP5801807B2 (ja) *	2009-08-14	2015-10-28	フェーズバイオファーマシューティカルズ，インコーポレイテッド	修飾された血管作動性腸管ペプチド
BR112012017435A2 (pt) *	2010-01-13	2020-08-25	Ipsen Pharma S.A.S	processo para a preparação de composições farmacêuticas para a liberação sustentada de análogos de somatostatina
ES2617336T3 (es)	2010-10-27	2017-06-16	Ferring B.V.	Procedimiento para la fabricación de degarelix y sus productos intermedios
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JO3755B1 (ar)	2011-01-26	2021-01-31	Ferring Bv	تركيبات تستوستيرون
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CN113398243A (zh)	2012-11-28	2021-09-17	联合动物健康第二有限责任公司	用于同步小母猪的授精时间的方法
EP2823808A1 (en)	2013-07-09	2015-01-14	Ipsen Pharma S.A.S.	Pharmaceutical composition for a sustained release of lanreotide
TW201605488A (zh)	2013-10-15	2016-02-16	大塚製藥股份有限公司	用以預防及／或治療多囊腎病之藥物
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1998
- 1998-03-25 FR FR9803667A patent/FR2776520B1/fr not_active Expired - Lifetime
1999
- 1999-03-22 DE DE69908326T patent/DE69908326T2/de not_active Expired - Lifetime
- 1999-03-22 JP JP2000537564A patent/JP4162381B2/ja not_active Expired - Lifetime
- 1999-03-22 CZ CZ20003432A patent/CZ298941B6/cs not_active IP Right Cessation
- 1999-03-22 EP EP99910418A patent/EP1066049B1/fr not_active Expired - Lifetime
- 1999-03-22 DK DK99910418T patent/DK1066049T3/da active
- 1999-03-22 US US09/646,519 patent/US6503534B1/en not_active Expired - Lifetime
- 1999-03-22 RU RU2000126755/15A patent/RU2224538C2/ru active
- 1999-03-22 HU HU0101545A patent/HU228903B1/hu unknown
- 1999-03-22 WO PCT/FR1999/000667 patent/WO1999048517A1/fr not_active Ceased
- 1999-03-22 PL PL343005A patent/PL197775B1/pl unknown
- 1999-03-22 IL IL13853399A patent/IL138533A0/xx active IP Right Grant
- 1999-03-22 PT PT99910418T patent/PT1066049E/pt unknown
- 1999-03-22 ES ES99910418T patent/ES2200507T3/es not_active Expired - Lifetime
- 1999-03-22 CA CA2324901A patent/CA2324901C/fr not_active Expired - Lifetime
- 1999-03-22 AU AU29384/99A patent/AU756148B2/en not_active Expired
- 1999-03-22 AT AT99910418T patent/ATE241377T1/de active
- 1999-03-23 AR ARP990101275A patent/AR020062A1/es not_active Application Discontinuation
2000
- 2000-09-18 IL IL138533A patent/IL138533A/en not_active IP Right Cessation
- 2000-09-22 NO NO20004741A patent/NO324621B1/no not_active IP Right Cessation

Also Published As

Publication number	Publication date
JP2002507578A (ja)	2002-03-12
EP1066049B1 (fr)	2003-05-28
NO20004741L (no)	2000-11-22
CA2324901C (fr)	2012-01-24
RU2224538C2 (ru)	2004-02-27
HUP0101545A1 (hu)	2001-11-28
IL138533A0 (en)	2001-10-31
AR020062A1 (es)	2002-04-10
PL343005A1 (en)	2001-07-30
PL197775B1 (pl)	2008-04-30
PT1066049E (pt)	2003-10-31
FR2776520B1 (fr)	2000-05-05
WO1999048517A1 (fr)	1999-09-30
ATE241377T1 (de)	2003-06-15
AU756148B2 (en)	2003-01-02
NO20004741D0 (no)	2000-09-22
CZ20003432A3 (cs)	2001-02-14
HUP0101545A3 (en)	2001-12-28
CA2324901A1 (fr)	1999-09-30
DE69908326D1 (de)	2003-07-03
DK1066049T3 (da)	2003-09-29
IL138533A (en)	2006-12-31
EP1066049A1 (fr)	2001-01-10
CZ298941B6 (cs)	2008-03-19
AU2938499A (en)	1999-10-18
ES2200507T3 (es)	2004-03-01
JP4162381B2 (ja)	2008-10-08
DE69908326T2 (de)	2004-03-25
US6503534B1 (en)	2003-01-07
HU228903B1 (en)	2013-06-28
FR2776520A1 (fr)	1999-10-01

Legal Events

Date	Code	Title	Description
2019-04-08	MK1K	Patent expired

Publication	Publication Date	Title
US6503534B1 (en)	2003-01-07	Pharmaceutical compositions for prolonged peptide release and preparation method
JP4489186B2 (ja)	2010-06-23	薬用組成物からのペプチドの持続的放出
KR101466933B1 (ko)	2014-12-01	펩타이드의 지속 방출 전달을 위한 의약 조성물
RU2198678C2 (ru)	2003-02-20	Композиции пролонгированного высвобождения и способ их получения
RU2453329C2 (ru)	2012-06-20	Препараты с задержкой высвобождения, содержащие полимеры с очень низкой молекулярной массой
AU2012268987B2 (en)	2016-09-08	Freeze-dried formulations of FGF-18
NO323296B1 (no)	2007-03-05	Stabil vandig formulering av en peptidbeslektet forbindelse, fremgangsmate for fremstilling av denne og anvendelse derav for fremstillingen av medikamenter.
KR20080089643A (ko)	2008-10-07	안정성이 강화된 약학 조성물
JP2010043105A (ja)	2010-02-25	非水性プロトン性ペプチド配合物
JPH0797334A (ja)	1995-04-11	徐放性製剤
SK283926B6 (sk)	2004-05-04	Implantovateľné zariadenie na dodávanie liečiva, spôsob jeho prípravy a použitie formulácie peptidovej zlúčeniny
JP2019073564A (ja)	2019-05-16	ランレオチドの持続放出用の医薬組成物
JP2006505538A (ja)	2006-02-16	徐放性を有する薬剤学的に活性なペプチドのための投与形及びそれらの製造方法
JP2005510544A (ja)	2005-04-21	Ｌｈｒｈアンタゴニストの注入溶液
HK1144067A (en)	2011-01-28	Sustained release of peptides from pharmaceutical compositions