NO924076L - Antihypertensive midler - Google Patents

Antihypertensive midler

Info

Publication number: NO924076L
Authority: NO; Norway
Prior art keywords: lower alkyl; aryl; halogen; optionally substituted; antihypertensive agents
Prior art date: 1991-02-27

Application number

NO92924076A

Other languages

English (en)

Norwegian (no)

Other versions

NO924076D0 (no

Inventor

Jose Repolles Moliner

Francisco Pubill Coy

Lydia Cabeza Llorente

Carlos Malet Falco

Original Assignee

Lacer Sa

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1991-02-27

Filing date

1992-10-21

Publication date

1992-12-21

1992-10-21 Application filed by Lacer Sa filed Critical Lacer Sa

1992-10-21 Publication of NO924076D0 publication Critical patent/NO924076D0/no

1992-12-21 Publication of NO924076L publication Critical patent/NO924076L/no

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/08—Tripeptides
- C07K5/0821—Tripeptides with the first amino acid being heterocyclic, e.g. His, Pro, Trp
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/02—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
- C07K5/0202—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -NH-X-X-C(=0)-, X being an optionally substituted carbon atom or a heteroatom, e.g. beta-amino acids
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/02—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
- C07K5/0205—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -NH-(X)3-C(=0)-, e.g. statine or derivatives thereof
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/08—Tripeptides
- C07K5/0827—Tripeptides containing heteroatoms different from O, S, or N
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Biochemistry (AREA)
Biophysics (AREA)
Genetics & Genomics (AREA)
Molecular Biology (AREA)
Proteomics, Peptides & Aminoacids (AREA)
Crystallography & Structural Chemistry (AREA)
Engineering & Computer Science (AREA)
Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Bioinformatics & Cheminformatics (AREA)
Animal Behavior & Ethology (AREA)
Heart & Thoracic Surgery (AREA)
Cardiology (AREA)
Peptides Or Proteins (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Pyridine Compounds (AREA)

NO92924076A 1991-02-27 1992-10-21 Antihypertensive midler NO924076L (no)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
EP91102950A EP0500989B1 (de)	1991-02-27	1991-02-27	Antihypertensive N-(alpha-substituiertes Pyridyl)-carbonyldipeptide
PCT/EP1992/000400 WO1992015608A1 (en)	1991-02-27	1992-02-26	N-(α-SUBSTITUTED-PYRIDINYL)CARBONYL DIPEPTIDE ANTIHYPERTENSIVE AGENTS

Publications (2)

Publication Number	Publication Date
NO924076D0 NO924076D0 (no)	1992-10-21
NO924076L true NO924076L (no)	1992-12-21

Family

ID=8206465

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO92924076A NO924076L (no)	1991-02-27	1992-10-21	Antihypertensive midler

Country Status (18)

Country	Link
US (1)	US5432159A (de)
EP (1)	EP0500989B1 (de)
JP (1)	JPH05507295A (de)
AT (1)	ATE174343T1 (de)
AU (1)	AU650954B2 (de)
BR (1)	BR9204779A (de)
CA (1)	CA2081471A1 (de)
CZ (1)	CZ280952B6 (de)
DE (1)	DE69130605T2 (de)
ES (1)	ES2037613B1 (de)
FI (1)	FI924850L (de)
HU (1)	HUT62313A (de)
NO (1)	NO924076L (de)
PL (1)	PL167915B1 (de)
PT (1)	PT100148B (de)
RO (1)	RO111369B1 (de)
RU (1)	RU2098424C1 (de)
WO (1)	WO1992015608A1 (de)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
WO1995014033A1 (en) *	1993-11-19	1995-05-26	Aktiebolaget Astra	Novel dipeptide derivatives
AU738037B2 (en) *	1997-04-04	2001-09-06	Pfizer Products Inc.	Nicotinamide derivatives
CN1200946C (zh) *	1998-09-22	2005-05-11	钟渊化学工业株式会社	制备n2－(1(s)－羧基－3－苯基丙基)－l－赖氨酰－l－脯氨酸的方法
JP2004520386A (ja)	2001-01-31	2004-07-08	ファイザー・プロダクツ・インク	Ｐｄｅ４アイソザイムの阻害剤として有用なニコチンアミドビアリール誘導体
US7250518B2 (en)	2001-01-31	2007-07-31	Pfizer Inc.	Nicotinamide acids, amides, and their mimetics active as inhibitors of PDE4 isozymes
DE60113731T2 (de)	2001-01-31	2006-06-29	Pfizer Products Inc., Groton	Als inhibitoren von pde4-isozymen geeignete etherderivate
WO2002060898A1 (en)	2001-01-31	2002-08-08	Pfizer Products Inc.	Thiazolyl-, oxazolyl-, pyrrolyl-, and imidazolyl-acid amide derivatives useful as inhibitors of pde4 isozymes
WO2003033471A1 (en) *	2001-10-17	2003-04-24	Tobishi Pharmaceutical Co.,Ltd	Novel pyridone derivative and remedial agent for circulatory disease containing the same
KR20040094677A (ko) *	2002-01-29	2004-11-10	와이어쓰	코넥신 헤미채널 조절을 위한 조성물 및 방법
SI21507A (sl) *	2003-05-16	2004-12-31	LEK farmacevtska dru�ba d.d.	Postopek za pripravo spojin z ace inhibitornim delovanjem
CN101155798A (zh) *	2005-04-14	2008-04-02	默克公司	Vla-4拮抗剂

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
AU537592B2 (en) *	1979-04-02	1984-07-05	E.R. Squibb & Sons, Inc.	Mercaptoacyldipeptides
NZ202232A (en) *	1981-11-06	1985-08-16	Smithkline Beckman Corp	N-carboxyalkylproline-containing tripeptides and pharmaceutical compositions
DE3332633A1 (de) *	1983-09-09	1985-04-04	Luitpold-Werk Chemisch-pharmazeutische Fabrik GmbH & Co, 8000 München	Substituierte carbonsaeurederivate, verfahren zu ihrer herstellung, und arzneimittel

1991
- 1991-02-27 AT AT91102950T patent/ATE174343T1/de not_active IP Right Cessation
- 1991-02-27 EP EP91102950A patent/EP0500989B1/de not_active Expired - Lifetime
- 1991-02-27 DE DE69130605T patent/DE69130605T2/de not_active Expired - Fee Related
- 1991-12-16 ES ES9102792A patent/ES2037613B1/es not_active Expired - Fee Related
1992
- 1992-02-21 PT PT100148A patent/PT100148B/pt not_active IP Right Cessation
- 1992-02-26 RU RU9292016314A patent/RU2098424C1/ru active
- 1992-02-26 AU AU12783/92A patent/AU650954B2/en not_active Ceased
- 1992-02-26 WO PCT/EP1992/000400 patent/WO1992015608A1/en not_active Ceased
- 1992-02-26 JP JP92504931A patent/JPH05507295A/ja active Pending
- 1992-02-26 PL PL92296625A patent/PL167915B1/pl unknown
- 1992-02-26 FI FI924850A patent/FI924850L/fi unknown
- 1992-02-26 CA CA002081471A patent/CA2081471A1/en not_active Abandoned
- 1992-02-26 CZ CS923220A patent/CZ280952B6/cs unknown
- 1992-02-26 US US07/938,248 patent/US5432159A/en not_active Expired - Lifetime
- 1992-02-26 BR BR9204779A patent/BR9204779A/pt not_active Application Discontinuation
- 1992-02-26 RO RO92-01349A patent/RO111369B1/ro unknown
- 1992-02-26 HU HU9203324A patent/HUT62313A/hu unknown
- 1992-10-21 NO NO92924076A patent/NO924076L/no unknown

Also Published As

Publication number	Publication date
HU9203324D0 (en)	1993-01-28
BR9204779A (pt)	1993-08-17
EP0500989A1 (de)	1992-09-02
WO1992015608A1 (en)	1992-09-17
DE69130605T2 (de)	1999-05-20
ATE174343T1 (de)	1998-12-15
CZ322092A3 (en)	1993-02-17
AU1278392A (en)	1992-10-06
NO924076D0 (no)	1992-10-21
RO111369B1 (ro)	1996-09-30
DE69130605D1 (de)	1999-01-21
AU650954B2 (en)	1994-07-07
ES2037613B1 (es)	1994-03-16
CA2081471A1 (en)	1992-08-28
CZ280952B6 (cs)	1996-05-15
PL296625A1 (en)	1993-08-09
PT100148A (pt)	1993-05-31
FI924850A7 (fi)	1992-10-26
FI924850A0 (fi)	1992-10-26
ES2037613A1 (es)	1993-06-16
US5432159A (en)	1995-07-11
RU2098424C1 (ru)	1997-12-10
FI924850L (fi)	1992-10-26
HUT62313A (en)	1993-04-28
JPH05507295A (ja)	1993-10-21
EP0500989B1 (de)	1998-12-09
PL167915B1 (pl)	1995-12-30
PT100148B (pt)	1999-06-30

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NO924076L (no)	1992-12-21	Antihypertensive midler
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NO302070B1 (no)	1998-01-19	Pyridinkarboksimidamid-forbindelse og anvendelse av samme
HU9203431D0 (en)	1993-01-28	New phthalazines containing ehter- or thioether group in location 1 and method for producing them
ES8607953A1 (es)	1986-06-01	Un procedimiento para la preparacion de nuevos derivados de triazina
DE3370159D1 (en)	1987-04-16	Amide derivatives
GR3015047T3 (en)	1995-05-31	Heterocyclic acyl aminodiol beta-amino acid derivatives.
PT1021404E (pt)	2003-04-30	Derivados de azetidinona para o tratamento de infeccoes pelo hcmv
DE3787030D1 (de)	1993-09-16	1-carboxy-1-vinyloxyiminoaminothiazol-cephalosporin-derivate und deren herstellung.
ATE181327T1 (de)	1999-07-15	Indolderivate
EP0802179A4 (de)	2000-04-05	Derivate substituierter amidinonaphthylester
ES2103675A1 (es)	1997-09-16	Nuevas piperidinas sustituidas.
DE68910090D1 (de)	1993-11-25	Verwendung heterozyklischer Amide zur Verhinderung der Tumormetastasierung.
TR199800039T1 (xx)	1998-04-21	Pirimidin n�kleozit t�revleri.
NO951985L (no)	1995-07-19	Acetamidderivat