NO972028L - Kjemiske forbindelser og antikonsepsjonsmidler inneholdende disse - Google Patents

Kjemiske forbindelser og antikonsepsjonsmidler inneholdende disse

Info

Publication number
NO972028L
NO972028L NO972028A NO972028A NO972028L NO 972028 L NO972028 L NO 972028L NO 972028 A NO972028 A NO 972028A NO 972028 A NO972028 A NO 972028A NO 972028 L NO972028 L NO 972028L
Authority
NO
Norway
Prior art keywords
chemical compounds
contraceptives containing
contraceptives
antiprogestatlonal
substituents
Prior art date
Application number
NO972028A
Other languages
English (en)
Other versions
NO972028D0 (no
Inventor
Eckhardt Ottow
Guenter Neef
Walter Elger
Martin Schneider
Karl-Heinrich Fritzemeier
Original Assignee
Schering Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Publication of NO972028L publication Critical patent/NO972028L/no
Application filed by Schering Ag filed Critical Schering Ag
Publication of NO972028D0 publication Critical patent/NO972028D0/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J53/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by condensation with a carbocyclic rings or by formation of an additional ring by means of a direct link between two ring carbon atoms, including carboxyclic rings fused to the cyclopenta(a)hydrophenanthrene skeleton are included in this class
    • C07J53/002—Carbocyclic rings fused
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/04—Drugs for genital or sexual disorders; Contraceptives for inducing labour or abortion; Uterotonics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/36—Antigestagens
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J63/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by expansion of only one ring by one or two atoms
    • C07J63/008—Expansion of ring D by one atom, e.g. D homo steroids

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Diabetes (AREA)
  • Urology & Nephrology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pregnancy & Childbirth (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Orthopedics, Nursing, And Contraception (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

Abstract

Beskrevet er 8-en-19,l1β-broede steroider av generell formel I (I) som har et nytt strukturtrykk i form av en dobbeltbinding mellom 8-stilling og 9-stilling. Også beskrevet er en metode for fremstilling av disse. Substi- tuentene r', R^-y, R^'-Y' og Z er som definert i beskrivelsen. De nye forbindelser har i særdeleshet en sterk antiprogestatlonal aktivitet og er egnet som antikonsepsjonsmidler.
NO972028A 1990-11-27 1997-04-30 Kjemiske forbindelser og antikonsepsjonsmidler inneholdende disse NO972028D0 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE4038128A DE4038128A1 (de) 1990-11-27 1990-11-27 8-en-19, 11(beta)-ueberbrueckte steroide, deren herstellung und diese enthaltende pharmazeutische praeparate
PCT/EP1991/002239 WO1992009618A1 (de) 1990-11-27 1991-11-27 8-EN-19, 11β-ÜBERBRÜCKTE STEROIDE, DEREN HERSTELLUNG UND DIESE ENTHALTENDE PHARMAZEUTISCHE PRÄPARATE

Publications (2)

Publication Number Publication Date
NO972028L true NO972028L (no) 1993-05-26
NO972028D0 NO972028D0 (no) 1997-04-30

Family

ID=6419242

Family Applications (2)

Application Number Title Priority Date Filing Date
NO93931905A NO931905L (no) 1990-11-27 1993-05-26 8-en-19, 11beta-broede steroider, deres fremstilling og farmasoeytiske preparater inneholdende disse
NO972028A NO972028D0 (no) 1990-11-27 1997-04-30 Kjemiske forbindelser og antikonsepsjonsmidler inneholdende disse

Family Applications Before (1)

Application Number Title Priority Date Filing Date
NO93931905A NO931905L (no) 1990-11-27 1993-05-26 8-en-19, 11beta-broede steroider, deres fremstilling og farmasoeytiske preparater inneholdende disse

Country Status (14)

Country Link
US (1) US5478956A (no)
EP (1) EP0559690B1 (no)
JP (1) JP3202229B2 (no)
AT (1) ATE154031T1 (no)
AU (1) AU661831B2 (no)
CA (1) CA2097079A1 (no)
DE (2) DE4038128A1 (no)
DK (1) DK0559690T3 (no)
ES (1) ES2106091T3 (no)
FI (1) FI932388L (no)
GR (1) GR3024611T3 (no)
HU (1) HUT64363A (no)
NO (2) NO931905L (no)
WO (1) WO1992009618A1 (no)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE4235220A1 (de) * 1992-10-13 1994-06-16 Schering Ag Gestagen wirksame 19,11ß-überbrückte 4-Estrene
US6090798A (en) * 1997-12-19 2000-07-18 Alcon Laboratories, Inc. Treatment of GLC1A glaucoma with glucocorticoid antagonists
ATE473759T1 (de) 1998-05-22 2010-07-15 Univ Leland Stanford Junior Bifunktionelle moleküle sowie darauf basierende therapien.
WO2001032604A1 (en) * 1999-11-05 2001-05-10 University College London Activators of soluble guanylate cyclase
US7191438B2 (en) * 2001-02-23 2007-03-13 Lenovo (Singapore) Pte, Ltd. Computer functional architecture and a locked down environment in a client-server architecture
CN102379684B (zh) 2005-04-28 2014-11-19 普罗透斯数字保健公司 药物信息系统
US9062126B2 (en) 2005-09-16 2015-06-23 Raptor Pharmaceuticals Inc. Compositions comprising receptor-associated protein (RAP) variants specific for CR-containing proteins and uses thereof
ES2643318T3 (es) 2006-10-24 2017-11-22 Repros Therapeutics Inc. Composiciones y métodos para suprimir la proliferación endometrial
TWI539953B (zh) 2008-04-28 2016-07-01 瑞波若斯治療學公司 用於治療乳癌之組成物和方法
EP2398500B1 (en) 2009-02-20 2019-03-13 2-BBB Medicines B.V. Glutathione-based drug delivery system
ES2942923T3 (es) 2009-05-06 2023-06-07 Laboratory Skin Care Inc Composiciones de administración dérmica que comprenden complejos de agente activo-partículas de fosfato de calcio y métodos de uso de las mismas
BR112012023281A2 (pt) 2010-03-22 2016-05-17 Repros Therapeutics Inc composto ou sal do mesmo, composição farmacêutica, métodos para produzir efeito antiprogestacional em paciente e para tratar condição dependente de progesterona e usos de composto ou sal do mesmo farmaceuticamente aceitável do mesmo e de composição
US20110233118A1 (en) * 2010-03-29 2011-09-29 Nelson Steven D Sports bottle device with filter isolated from filtered fluid

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3127423A (en) * 1962-09-21 1964-03-31 Olin Mathieson Phenyl derivatives of methylsterols and process for production thereof
DE3708942A1 (de) * 1987-03-18 1988-09-29 Schering Ag 19,11ss-ueberbrueckte steroide, deren herstellung und diese enthaltende pharmazeutische praeparate
DE3717169A1 (de) * 1987-05-19 1988-12-01 Schering Ag 19,11ss-ueberbrueckte steroide, deren herstellung und diese enthaltende pharmazeutische praeparate
DE3832303A1 (de) * 1988-09-20 1990-04-12 Schering Ag 11ss-phenyl-14ssh-steroide
DE3917274A1 (de) * 1989-05-24 1990-11-29 Schering Ag 9(alpha)-hydroxy-19, 11(beta)-ueberbrueckte steroide, deren herstellung und diese enthaltende pharmazeutische praeparate
US5041434A (en) * 1991-08-17 1991-08-20 Virginia Lubkin Drugs for topical application of sex steroids in the treatment of dry eye syndrome, and methods of preparation and application

Also Published As

Publication number Publication date
FI932388A7 (fi) 1993-05-26
HUT64363A (en) 1993-12-28
EP0559690B1 (de) 1997-06-04
NO972028D0 (no) 1997-04-30
US5478956A (en) 1995-12-26
FI932388A0 (fi) 1993-05-26
FI932388L (fi) 1993-05-26
GR3024611T3 (en) 1997-12-31
EP0559690A1 (de) 1993-09-15
CA2097079A1 (en) 1992-05-28
NO931905D0 (no) 1993-05-26
AU661831B2 (en) 1995-08-10
HU9301542D0 (en) 1993-09-28
NO931905L (no) 1993-05-26
DE4038128A1 (de) 1992-06-04
JP3202229B2 (ja) 2001-08-27
ES2106091T3 (es) 1997-11-01
JPH06502631A (ja) 1994-03-24
AU8946091A (en) 1992-06-25
DK0559690T3 (da) 1997-12-29
ATE154031T1 (de) 1997-06-15
DE59108744D1 (de) 1997-07-10
WO1992009618A1 (de) 1992-06-11

Similar Documents

Publication Publication Date Title
CA1258859A (en) CARBOSTYRILE DERIVATIVE, AND ITS PREPARATION
ATE151764T1 (de) Neue benzopyran-derivate, verfahren zu ihrer herstellung und ihre verwendung sowie die verbindungen enthaltenden zubereitungen
IE890906L (en) Method of lowering the blood pressure
IE832529L (en) ß-CARBOLINES, PROCESS FOR THEIR PRODUCTION AND¹PHARMACEUTICAL PREPARATIONS CONTAINING THEM
NO911158L (no) Hydantoinderivater.
IT1264563B1 (it) Composti fotocromatici e metodo per la loro preparazione
NO931905L (no) 8-en-19, 11beta-broede steroider, deres fremstilling og farmasoeytiske preparater inneholdende disse
HU9203761D0 (en) Method for producing substituted pyridine derivatives
ES2000368A6 (es) Un procedimiento para preparar di-t-butilfenoles sustituidos
CA2013166A1 (en) Suppression of parathyroid hormone synthesis and secretion
NO981393L (no) Guanidinoproteasehemmere
EP0472733A4 (en) Phenanthrene derivative
EP0757987A4 (en) PYRAZOLECARBOXYLIC ACID DERIVATIVE AND PLANT DISEASE CONTROL AGENT
ES8301928A1 (es) Un procedimiento para preparar 4-(2-4-dicloro-3-metilbenzoil)-1,3-dimetil-5-fenaciloxipirazol).
NO904191L (no) Nye fremgangsmaate.
ES8302733A1 (es) Un procedimiento para preparar nuevos derivados de antraci- clina
ES8303393A1 (es) Un procedimiento para preparar derivados del acido ascorbico.
GR3021686T3 (en) METHOD OF PREPARING -g(b)-CARBOLINES.
EP0031388A4 (en) METHOD FOR PRODUCING IMIDAZOLE DERIVATIVES.
NO962620L (no) Nye mellomprodukter for syntese av L-aspartyl-D--aminoalkanoyl-(S)-N--alkylbenzylamider anvendbare son kunstige sötningsmidler
HU9904686D0 (en) New hydroxy-bicyclolactam derivatives, their use and medicaments containing them
AU5388879A (en) Isoxazole derivatives and their use as bronchodilating agent
JPS5424856A (en) 1-(3 or 4-methyl-3-cyclohexenyl)-2-methyl-1-penten-3-ol
NZ332245A (en) Substituted benzo-oxazolol carboxylic acid derivatives, process for their production and medicaments containing them
EP0392015A4 (en) Novel derivatives of physiologically active substance ml-236b and process for their preparation