PL2964229T3 - Benzoimidazol-2-ilo pirymidynowe modulatory receptora histaminowego H<sub>4</sub> - Google Patents

Benzoimidazol-2-ilo pirymidynowe modulatory receptora histaminowego H<sub>4</sub>

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Publication number
PL2964229T3
PL2964229T3 PL14760540T PL14760540T PL2964229T3 PL 2964229 T3 PL2964229 T3 PL 2964229T3 PL 14760540 T PL14760540 T PL 14760540T PL 14760540 T PL14760540 T PL 14760540T PL 2964229 T3 PL2964229 T3 PL 2964229T3
Authority
PL
Poland
Prior art keywords
benzoimidazol
histamine
receptor
modulators
pyrimidine
Prior art date
Application number
PL14760540T
Other languages
English (en)
Inventor
Magali B. Hickey
Stefan Horns
Susanne Lochner
Matteo CONZA
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of PL2964229T3 publication Critical patent/PL2964229T3/pl

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    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
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PL14760540T 2013-03-06 2014-03-06 Benzoimidazol-2-ilo pirymidynowe modulatory receptora histaminowego H<sub>4</sub> PL2964229T3 (pl)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201361773706P 2013-03-06 2013-03-06
US201361776260P 2013-03-11 2013-03-11
US201361784909P 2013-03-14 2013-03-14
PCT/US2014/021130 WO2014138368A1 (en) 2013-03-06 2014-03-06 Benzoimidazol-2-yl pyrimidine modulators of the histamine h4 receptor
EP14760540.6A EP2964229B1 (en) 2013-03-06 2014-03-06 Benzoimidazol-2-yl pyrimidine modulators of the histamine h4 receptor

Publications (1)

Publication Number Publication Date
PL2964229T3 true PL2964229T3 (pl) 2020-05-18

Family

ID=51488591

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Application Number Title Priority Date Filing Date
PL14760540T PL2964229T3 (pl) 2013-03-06 2014-03-06 Benzoimidazol-2-ilo pirymidynowe modulatory receptora histaminowego H<sub>4</sub>

Country Status (38)

Country Link
US (4) US8859575B2 (pl)
EP (2) EP2964229B1 (pl)
JP (1) JP6471103B2 (pl)
KR (1) KR102230383B1 (pl)
CN (1) CN105025898B (pl)
AU (1) AU2014225675B2 (pl)
BR (1) BR112015021463A8 (pl)
CA (1) CA2903737C (pl)
CL (1) CL2015002434A1 (pl)
CR (1) CR20150435A (pl)
CY (1) CY1122545T1 (pl)
DK (1) DK2964229T3 (pl)
DO (1) DOP2016000027A (pl)
EA (1) EA201591648A1 (pl)
ES (1) ES2773543T3 (pl)
GT (1) GT201500243A (pl)
HR (1) HRP20200253T1 (pl)
HU (1) HUE047681T2 (pl)
IL (1) IL240247B (pl)
JO (1) JO3516B1 (pl)
LT (1) LT2964229T (pl)
MX (1) MX373874B (pl)
MY (1) MY180726A (pl)
NZ (1) NZ710640A (pl)
PE (1) PE20151536A1 (pl)
PH (1) PH12015501731B1 (pl)
PL (1) PL2964229T3 (pl)
PT (1) PT2964229T (pl)
RS (1) RS59909B1 (pl)
SA (1) SA515360981B1 (pl)
SG (1) SG11201507117XA (pl)
SI (1) SI2964229T1 (pl)
SM (1) SMT202000084T1 (pl)
TW (1) TWI617554B (pl)
UA (1) UA118754C2 (pl)
UY (1) UY35370A (pl)
WO (1) WO2014138368A1 (pl)
ZA (1) ZA201507351B (pl)

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US9371311B2 (en) 2008-06-30 2016-06-21 Janssen Pharmaceutica Nv Benzoimidazol-2-yl pyrimidine derivatives
RS59909B1 (sr) 2013-03-06 2020-03-31 Janssen Pharmaceutica Nv Benzoimidazol-2-il pirimidinski modulatori histaminskog h4 receptora
US9040534B2 (en) 2013-03-14 2015-05-26 Janssen Pharmaceutica Nv [1,2,4]triazolo[4,3-a]pyrazines as P2X7 modulators
TWI627174B (zh) 2013-03-14 2018-06-21 比利時商健生藥品公司 Ｐ２ｘ７調控劑
TWI599567B (zh) 2013-03-14 2017-09-21 健生藥品公司 Ｐ２ｘ７調節劑
EP2970271B1 (en) 2013-03-14 2017-11-08 Janssen Pharmaceutica NV P2x7 modulators
WO2016039977A1 (en) 2014-09-12 2016-03-17 Janssen Pharmaceutica Nv P2x7 modulators
JP6625616B2 (ja) 2014-09-12 2019-12-25 ヤンセン ファーマシューティカ エヌ．ベー． Ｐ２ｘ７調節ｎ−アシル−トリアゾロピラジン
US20180325931A1 (en) 2017-01-21 2018-11-15 Ningbo Zhiming Biotechnology Co., Ltd. Use of paeoniflorin-6'-o-benzenesulfonate in treatment of sjögren's syndrome
TW202035409A (zh) 2018-09-28 2020-10-01 比利時商健生藥品公司 單醯基甘油脂肪酶調節劑
MY205440A (en) 2018-09-28 2024-10-21 Janssen Pharmaceutica Nv Monoacylglycerol lipase modulators
AU2020358948A1 (en) 2019-09-30 2022-05-26 Janssen Pharmaceutica Nv Radiolabelled MGL PET ligands
BR112022019077A2 (pt) 2020-03-26 2022-12-27 Janssen Pharmaceutica Nv Moduladores da monoacilglicerol lipase

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