DK2964229T3 - Benzoimidazol-2-yl-pyrimidinmodulatorer af histamin-h4 receptoren - Google Patents

Benzoimidazol-2-yl-pyrimidinmodulatorer af histamin-h4 receptoren Download PDF

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DK2964229T3
DK2964229T3 DK14760540.6T DK14760540T DK2964229T3 DK 2964229 T3 DK2964229 T3 DK 2964229T3 DK 14760540 T DK14760540 T DK 14760540T DK 2964229 T3 DK2964229 T3 DK 2964229T3
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histamin
benzoimidazole
receptor
modulators
pyrimidine
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DK14760540.6T
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Magali B Hickey
Stefan Horns
Susanne Lochner
Matteo Conza
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Janssen Pharmaceutica Nv
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    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
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DK14760540.6T 2013-03-06 2014-03-06 Benzoimidazol-2-yl-pyrimidinmodulatorer af histamin-h4 receptoren DK2964229T3 (da)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US201361773706P 2013-03-06 2013-03-06
US201361776260P 2013-03-11 2013-03-11
US201361784909P 2013-03-14 2013-03-14
PCT/US2014/021130 WO2014138368A1 (en) 2013-03-06 2014-03-06 Benzoimidazol-2-yl pyrimidine modulators of the histamine h4 receptor

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DK2964229T3 true DK2964229T3 (da) 2020-01-27

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US (4) US8859575B2 (da)
EP (2) EP2964229B1 (da)
JP (1) JP6471103B2 (da)
KR (1) KR102230383B1 (da)
CN (1) CN105025898B (da)
AU (1) AU2014225675B2 (da)
BR (1) BR112015021463A8 (da)
CA (1) CA2903737C (da)
CL (1) CL2015002434A1 (da)
CR (1) CR20150435A (da)
CY (1) CY1122545T1 (da)
DK (1) DK2964229T3 (da)
DO (1) DOP2016000027A (da)
EA (1) EA201591648A1 (da)
ES (1) ES2773543T3 (da)
GT (1) GT201500243A (da)
HR (1) HRP20200253T1 (da)
HU (1) HUE047681T2 (da)
IL (1) IL240247B (da)
JO (1) JO3516B1 (da)
LT (1) LT2964229T (da)
MX (1) MX373874B (da)
MY (1) MY180726A (da)
NZ (1) NZ710640A (da)
PE (1) PE20151536A1 (da)
PH (1) PH12015501731A1 (da)
PL (1) PL2964229T3 (da)
PT (1) PT2964229T (da)
RS (1) RS59909B1 (da)
SA (1) SA515360981B1 (da)
SG (1) SG11201507117XA (da)
SI (1) SI2964229T1 (da)
SM (1) SMT202000084T1 (da)
TW (1) TWI617554B (da)
UA (1) UA118754C2 (da)
UY (1) UY35370A (da)
WO (1) WO2014138368A1 (da)
ZA (1) ZA201507351B (da)

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PL2007752T3 (pl) 2006-03-31 2011-02-28 Janssen Pharmaceutica Nv Benzoimidazol-2-ilopirymidyny i pirazyny jako modulatory receptora histaminowego H4
US9371311B2 (en) 2008-06-30 2016-06-21 Janssen Pharmaceutica Nv Benzoimidazol-2-yl pyrimidine derivatives
SMT202000084T1 (it) 2013-03-06 2020-03-13 Janssen Pharmaceutica Nv Modulatori benzoimidazol-2-il pirimidinici del recettore h4 dell'istamina
JO3509B1 (ar) 2013-03-14 2020-07-05 Janssen Pharmaceutica Nv معدلات p2x7
US9040534B2 (en) 2013-03-14 2015-05-26 Janssen Pharmaceutica Nv [1,2,4]triazolo[4,3-a]pyrazines as P2X7 modulators
TWI644671B (zh) 2013-03-14 2018-12-21 比利時商健生藥品公司 Ｐ２ｘ７調節劑
US9604982B2 (en) 2013-03-14 2017-03-28 Janssen Pharmaceutica Nv P2X7 modulators
WO2016039977A1 (en) 2014-09-12 2016-03-17 Janssen Pharmaceutica Nv P2x7 modulators
AU2015315693B2 (en) 2014-09-12 2020-01-16 Janssen Pharmaceutica Nv P2X7 modulating n-acyl-triazolopyrazines
US20180325931A1 (en) 2017-01-21 2018-11-15 Ningbo Zhiming Biotechnology Co., Ltd. Use of paeoniflorin-6'-o-benzenesulfonate in treatment of sjögren's syndrome
KR20210069079A (ko) 2018-09-28 2021-06-10 얀센 파마슈티카 엔.브이. 모노아실글리세롤 리파아제 조절제
MY205440A (en) 2018-09-28 2024-10-21 Janssen Pharmaceutica Nv Monoacylglycerol lipase modulators
JP7697934B2 (ja) 2019-09-30 2025-06-24 ヤンセン ファーマシューティカ エヌ．ベー． 放射線標識されたｍｇｌ ｐｅｔリガンド
BR112022019077A2 (pt) 2020-03-26 2022-12-27 Janssen Pharmaceutica Nv Moduladores da monoacilglicerol lipase

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