PL353989A1 - Sposób wytwarzania odmiany polimorficznej I olanzaSposób wytwarzania odmiany polimorficznej I olanzapinypiny - Google Patents
Sposób wytwarzania odmiany polimorficznej I olanzaSposób wytwarzania odmiany polimorficznej I olanzapinypinyInfo
- Publication number
- PL353989A1 PL353989A1 PL02353989A PL35398902A PL353989A1 PL 353989 A1 PL353989 A1 PL 353989A1 PL 02353989 A PL02353989 A PL 02353989A PL 35398902 A PL35398902 A PL 35398902A PL 353989 A1 PL353989 A1 PL 353989A1
- Authority
- PL
- Poland
- Prior art keywords
- olansapine
- obtaining
- polymorphous form
- polymorphous
- obtaining polymorphous
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Psychiatry (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Priority Applications (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| PL353989A PL196814B1 (pl) | 2002-05-17 | 2002-05-17 | Sposób wytwarzania odmiany polimorficznej I olanzapiny i jej solwaty |
| US10/514,520 US7538213B2 (en) | 2002-05-17 | 2003-05-16 | Methods for preparation of olanzapine polymorphic form I |
| EP03752952A EP1509531A1 (en) | 2002-05-17 | 2003-05-16 | Methods for preparation of olanzapine polymorphic form i |
| AU2003251247A AU2003251247A1 (en) | 2002-05-17 | 2003-05-16 | Methods for preparation of olanzapine polymorphic form i |
| PCT/PL2003/000044 WO2003097650A1 (en) | 2002-05-17 | 2003-05-16 | Methods for preparation of olanzapine polymorphic form i |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| PL353989A PL196814B1 (pl) | 2002-05-17 | 2002-05-17 | Sposób wytwarzania odmiany polimorficznej I olanzapiny i jej solwaty |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| PL353989A1 true PL353989A1 (pl) | 2003-12-01 |
| PL196814B1 PL196814B1 (pl) | 2008-02-29 |
Family
ID=29546557
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PL353989A PL196814B1 (pl) | 2002-05-17 | 2002-05-17 | Sposób wytwarzania odmiany polimorficznej I olanzapiny i jej solwaty |
Country Status (5)
| Country | Link |
|---|---|
| US (1) | US7538213B2 (pl) |
| EP (1) | EP1509531A1 (pl) |
| AU (1) | AU2003251247A1 (pl) |
| PL (1) | PL196814B1 (pl) |
| WO (1) | WO2003097650A1 (pl) |
Families Citing this family (23)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PL196814B1 (pl) | 2002-05-17 | 2008-02-29 | Inst Farmaceutyczny | Sposób wytwarzania odmiany polimorficznej I olanzapiny i jej solwaty |
| ATE500258T1 (de) | 2002-05-31 | 2011-03-15 | Sandoz Ag | Verfahren zur herstellung von olanzapin form i |
| PL202856B1 (pl) * | 2002-12-20 | 2009-07-31 | Adamed Spo & Lstrok Ka Z Ogran | Sposób otrzymywania farmaceutycznie czystej polimorficznej postaci I olanzapiny |
| AU2003300324A1 (en) * | 2002-12-24 | 2004-07-22 | Teva Pharmaceutical Industries Ltd. | Novel crystal forms of olanzapine, methods for their preparation and method for the preparation of known olanzapine crystal forms |
| CA2551806A1 (en) | 2003-12-22 | 2005-07-14 | Teva Pharmaceutical Industries, Ltd. | Methods of preparing olanzapine |
| AR047459A1 (es) | 2004-01-27 | 2006-01-18 | Synthon Bv | Sales estables de 2-metil-4-(4-metil-1-piperazinil)-10h-tieno[2,3-b][1,5]benzodiazepina (olanzapina) |
| AR047460A1 (es) * | 2004-01-27 | 2006-01-18 | Synthon Bv | Proceso para la fabricacion de acetato de 2-metil-4-(4-metil-1-piperazinil)-10h-tieno[2,3-b][1,5]benzodiazepina (acetato de olanzapina) |
| WO2005107375A2 (en) * | 2004-05-06 | 2005-11-17 | Matrix Laboratories Ltd | Process for the preparation of olanzapine form-i |
| EP2264016B1 (en) | 2004-07-14 | 2013-05-01 | Jubilant Organosys Limited | A process for producing pure form form of 2-Methyl-4-(4-Methyl-1-Piperazinyl)-10h-thieno[2,3-B][1,5] benzodiazepine |
| ES2292333B1 (es) * | 2004-07-27 | 2008-12-16 | Inke, S.A. | Mejoras en el objeto de la patente principal n. 200401850, por "solvato mixto de olanzapina, procedimiento para su obtencion y procedimiento de obtencion de la forma i de olanzapina a partir del mismo". |
| ES2253091B1 (es) * | 2004-07-27 | 2007-02-01 | Inke, S.A. | Solvato mixto de olanzapina, procedimiento para su obtencion y procedimiento de obtencion de la forma i de olanzapina a partir del mismo. |
| WO2006025065A1 (en) * | 2004-08-31 | 2006-03-09 | Lee Pharma Private Limited | A process for the preparation of anhydrous olanzopine hydrochloride of form-1 |
| WO2006027800A1 (en) | 2004-09-06 | 2006-03-16 | Shasun Chemicals And Drugs Limited | A novel process for preparation of a pharmaceutically pure polymorphic form 1 of olanzapine |
| GB0522473D0 (en) * | 2005-11-03 | 2005-12-14 | Actavis Group | A pharmaceutical formulation |
| ES2279715B1 (es) | 2005-12-26 | 2008-06-01 | Laboratorios Lesvi, S.L. | Formulacion oral de olanzapina. |
| US8129522B2 (en) | 2006-01-05 | 2012-03-06 | Inke, S.A. | Method for preparing a mixed solvate of olanzapine |
| US7834176B2 (en) * | 2006-01-26 | 2010-11-16 | Sandoz Ag | Polymorph E of Olanzapine and preparation of anhydrous non-solvated crystalline polymorphic Form I of 2-methyl-4(4-methyl-1-piperazinyl)-10H-thieno[2,3-b][1,5] benzodiazepine (Olanzapine Form I) from the polymorphic Olanzapine Form E |
| WO2007102167A1 (en) * | 2006-03-06 | 2007-09-13 | Lee Pharma Limited | A process for the preparation of anhydrous polymorphic form of olanzapine |
| WO2007144901A1 (en) * | 2006-06-12 | 2007-12-21 | Jubilant Organosys Limited | Process for stabilization of olanzapine polymorphic form i |
| PL381564A1 (pl) | 2007-01-22 | 2008-08-04 | Koźluk Tomasz Nobilus Ent | Sposób wytwarzania zasadniczo czystej odmiany polimorficznej I olanzapiny |
| WO2008151430A1 (en) * | 2007-06-14 | 2008-12-18 | Apotex Pharmachem Inc. | Novel processes to form-i of olanzapine |
| CN106265571A (zh) * | 2016-08-31 | 2017-01-04 | 安徽省润生医药股份有限公司 | 一种奥氮平片剂的制备方法 |
| FI128719B (en) | 2019-05-02 | 2020-10-30 | Andritz Oy | Vortex cleaner reject chamber and vortex cleaner |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5229382A (en) | 1990-04-25 | 1993-07-20 | Lilly Industries Limited | 2-methyl-thieno-benzodiazepine |
| GB9009229D0 (en) | 1990-04-25 | 1990-06-20 | Lilly Industries Ltd | Pharmaceutical compounds |
| EG23659A (en) | 1995-03-24 | 2007-03-26 | Lilly Co Eli | Process and crystal forms of methyl-thieno-benzodiazepine |
| US5637584A (en) * | 1995-03-24 | 1997-06-10 | Eli Lilly And Company | Solvate of olanzapine |
| JPH11506096A (ja) | 1995-05-30 | 1999-06-02 | イーライ・リリー・アンド・カンパニー | 認識機能不全を処置する方法 |
| HK1041199B (en) | 1998-09-30 | 2005-03-18 | Eli Lilly & Company | 2-Methyl-thiophenone-benzodiazine formula |
| US6348458B1 (en) * | 1999-12-28 | 2002-02-19 | U & I Pharmaceuticals Ltd. | Polymorphic forms of olanzapine |
| SK2502003A3 (en) | 2000-08-31 | 2004-03-02 | Reddys Lab Ltd Dr | Process for preparation of hydrates of olanzapine and their conversion into crystalline forms of olanzapine |
| PL196814B1 (pl) | 2002-05-17 | 2008-02-29 | Inst Farmaceutyczny | Sposób wytwarzania odmiany polimorficznej I olanzapiny i jej solwaty |
-
2002
- 2002-05-17 PL PL353989A patent/PL196814B1/pl unknown
-
2003
- 2003-05-16 WO PCT/PL2003/000044 patent/WO2003097650A1/en not_active Ceased
- 2003-05-16 US US10/514,520 patent/US7538213B2/en not_active Expired - Fee Related
- 2003-05-16 AU AU2003251247A patent/AU2003251247A1/en not_active Abandoned
- 2003-05-16 EP EP03752952A patent/EP1509531A1/en not_active Withdrawn
Also Published As
| Publication number | Publication date |
|---|---|
| WO2003097650A1 (en) | 2003-11-27 |
| US7538213B2 (en) | 2009-05-26 |
| AU2003251247A1 (en) | 2003-12-02 |
| EP1509531A1 (en) | 2005-03-02 |
| US20050239772A1 (en) | 2005-10-27 |
| PL196814B1 (pl) | 2008-02-29 |
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