PL375935A1 - Pochodne skondensowanych azolopirymidyn - Google Patents

Pochodne skondensowanych azolopirymidyn

Info

Publication number: PL375935A1
Authority: PL; Poland
Prior art keywords: pyrimidine derivatives; fused azole; azole; fused; pyrimidine
Prior art date: 2002-09-30

Application number

PL03375935A

Other languages

English (en)

Other versions

PL226562B1 (pl

Inventor

Mitsuyuki Shimada

Toshiki Murata

Kinji Fuchikami

Hideki Tsujishita

Naoki Omori

Issei Kato

Mami Miura

Klaus Urbahns

Florian Gantner

Kevin Bacon

Original Assignee

Bayer Pharmaceuticals Corporation

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2002-09-30

Filing date

2003-09-18

Publication date

2005-12-12

2003-09-18 Application filed by Bayer Pharmaceuticals Corporation filed Critical Bayer Pharmaceuticals Corporation

2005-12-12 Publication of PL375935A1 publication Critical patent/PL375935A1/pl

2017-08-31 Publication of PL226562B1 publication Critical patent/PL226562B1/pl

Links

DDWJFSYHYPDQEL-UHFFFAOYSA-N pyrimidine;1h-pyrrole Chemical class C=1C=CNC=1.C1=CN=CN=C1 DDWJFSYHYPDQEL-UHFFFAOYSA-N 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
- C07D471/14—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/02—Nasal agents, e.g. decongestants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/14—Drugs for disorders of the endocrine system of the thyroid hormones, e.g. T3, T4
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Life Sciences & Earth Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Immunology (AREA)
Cardiology (AREA)
Diabetes (AREA)
Heart & Thoracic Surgery (AREA)
Pulmonology (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Hospice & Palliative Care (AREA)
Endocrinology (AREA)
Urology & Nephrology (AREA)
Rheumatology (AREA)
Hematology (AREA)
Emergency Medicine (AREA)
Obesity (AREA)
Pain & Pain Management (AREA)
Vascular Medicine (AREA)
Psychiatry (AREA)
Otolaryngology (AREA)
Orthopedic Medicine & Surgery (AREA)
Physical Education & Sports Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

PL375935A 2002-09-30 2003-09-18 Skondensowane pochodne azolopirymidyn, leki zawierające takie pochodne oraz ich zastosowanie PL226562B1 (pl)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
EP02021861.6		2002-09-30
EP02021861		2002-09-30
PCT/EP2003/010377 WO2004029055A1 (en)	2002-09-30	2003-09-18	Fused azole-pyrimidine derivatives

Publications (2)

Publication Number	Publication Date
PL375935A1 true PL375935A1 (pl)	2005-12-12
PL226562B1 PL226562B1 (pl)	2017-08-31

Family

ID=32039115

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
PL375935A PL226562B1 (pl)	2002-09-30	2003-09-18	Skondensowane pochodne azolopirymidyn, leki zawierające takie pochodne oraz ich zastosowanie

Country Status (32)

Country	Link
US (2)	US7511041B2 (pl)
EP (2)	EP2042504B1 (pl)
JP (1)	JP4790266B2 (pl)
KR (1)	KR101059652B1 (pl)
CN (1)	CN100384846C (pl)
AR (2)	AR041426A1 (pl)
AT (2)	ATE411996T1 (pl)
AU (1)	AU2003293310B2 (pl)
BR (1)	BRPI0314830B8 (pl)
CA (1)	CA2499134C (pl)
CY (2)	CY1109790T1 (pl)
DE (1)	DE60324296D1 (pl)
DK (2)	DK1549652T3 (pl)
EC (2)	ECSP055768A (pl)
ES (2)	ES2312843T3 (pl)
HR (2)	HRP20050375B1 (pl)
IL (1)	IL166855A (pl)
MA (1)	MA27483A1 (pl)
MX (1)	MXPA05001808A (pl)
MY (1)	MY140756A (pl)
NO (1)	NO331457B1 (pl)
NZ (1)	NZ539062A (pl)
PE (1)	PE20050089A1 (pl)
PL (1)	PL226562B1 (pl)
PT (2)	PT1549652E (pl)
RU (1)	RU2326881C9 (pl)
SI (2)	SI1549652T1 (pl)
TW (1)	TWI327570B (pl)
UA (1)	UA82205C2 (pl)
UY (1)	UY28001A1 (pl)
WO (1)	WO2004029055A1 (pl)
ZA (1)	ZA200503306B (pl)

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Also Published As

Publication number	Publication date
HRP20050375A2 (en)	2006-05-31
KR20050067404A (ko)	2005-07-01
EP1549652A1 (en)	2005-07-06
PT2042504E (pt)	2011-09-07
BR0314830A (pt)	2005-08-16
ATE411996T1 (de)	2008-11-15
NO331457B1 (no)	2012-01-09
IL166855A (en)	2014-05-28
PT1549652E (pt)	2008-12-15
RU2326881C9 (ru)	2009-04-10
WO2004029055A1 (en)	2004-04-08
AU2003293310A1 (en)	2004-04-19
EP2042504A1 (en)	2009-04-01
CY1112174T1 (el)	2015-12-09
CN100384846C (zh)	2008-04-30
US8129386B2 (en)	2012-03-06
HRP20131159A2 (hr)	2014-05-23
CA2499134C (en)	2011-12-20
UY28001A1 (es)	2004-04-30
AU2003293310B2 (en)	2010-04-01
EP2042504B1 (en)	2011-06-01
ES2312843T3 (es)	2009-03-01
JP2006508063A (ja)	2006-03-09
BRPI0314830B1 (pt)	2018-03-27
CN1688582A (zh)	2005-10-26
DK2042504T3 (da)	2011-09-19
MXPA05001808A (es)	2005-08-16
AR041426A1 (es)	2005-05-18
HRP20050375B1 (hr)	2014-03-14
DE60324296D1 (de)	2008-12-04
US20060128732A1 (en)	2006-06-15
ECSP055768A (es)	2005-08-11
ECSP11005768A (es)	2011-03-31
TWI327570B (en)	2010-07-21
PE20050089A1 (es)	2005-04-20
NZ539062A (en)	2007-05-31
JP4790266B2 (ja)	2011-10-12
AR072458A2 (es)	2010-09-01
HRP20131159B1 (hr)	2019-11-01
HK1084393A1 (zh)	2006-07-28
US7511041B2 (en)	2009-03-31
NO20052076L (no)	2005-04-27
TW200413379A (en)	2004-08-01
EP1549652B1 (en)	2008-10-22
US20090270388A1 (en)	2009-10-29
ES2367141T3 (es)	2011-10-28
BRPI0314830B8 (pt)	2021-05-25
CA2499134A1 (en)	2004-04-08
MY140756A (en)	2010-01-15
ZA200503306B (en)	2006-07-26
UA82205C2 (en)	2008-03-25
DK1549652T3 (da)	2009-02-23
MA27483A1 (fr)	2005-08-01
SI1549652T1 (sl)	2009-04-30
PL226562B1 (pl)	2017-08-31
CY1109790T1 (el)	2014-09-10
SI2042504T1 (sl)	2011-10-28
ATE511510T1 (de)	2011-06-15
KR101059652B1 (ko)	2011-08-25
RU2005113165A (ru)	2005-10-10
RU2326881C2 (ru)	2008-06-20

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