PT1530457E - Composições farmacêuticas de fármacos na forma semi-ordenada e de polímeros - Google Patents

Composições farmacêuticas de fármacos na forma semi-ordenada e de polímeros Download PDF

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Publication number
PT1530457E
PT1530457E PT03784384T PT03784384T PT1530457E PT 1530457 E PT1530457 E PT 1530457E PT 03784384 T PT03784384 T PT 03784384T PT 03784384 T PT03784384 T PT 03784384T PT 1530457 E PT1530457 E PT 1530457E
Authority
PT
Portugal
Prior art keywords
drugs
polymers
semi
pharmaceutical compositions
ordered form
Prior art date
Application number
PT03784384T
Other languages
English (en)
Inventor
Marshall David Crew
Dwayne Thomas Friesen
Walter Christian Babcock
William Brett Caldwell
Daniel Tod Smithey
Ravi Mysore Shanker
Original Assignee
Bend Res Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=31715934&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PT1530457(E) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bend Res Inc filed Critical Bend Res Inc
Publication of PT1530457E publication Critical patent/PT1530457E/pt

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605—Excipients; Inactive ingredients
    • A61K9/1629—Organic macromolecular compounds
    • A61K9/1652—Polysaccharides, e.g. alginate, cellulose derivatives; Cyclodextrin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/141—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
    • A61K9/146—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic macromolecular compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605—Excipients; Inactive ingredients
    • A61K9/1629—Organic macromolecular compounds
    • A61K9/1635—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1682—Processes
    • A61K9/1694—Processes resulting in granules or microspheres of the matrix type containing more than 5% of excipient

Landscapes

  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
PT03784384T 2002-08-12 2003-07-31 Composições farmacêuticas de fármacos na forma semi-ordenada e de polímeros PT1530457E (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US40308702P 2002-08-12 2002-08-12

Publications (1)

Publication Number Publication Date
PT1530457E true PT1530457E (pt) 2009-11-06

Family

ID=31715934

Family Applications (1)

Application Number Title Priority Date Filing Date
PT03784384T PT1530457E (pt) 2002-08-12 2003-07-31 Composições farmacêuticas de fármacos na forma semi-ordenada e de polímeros

Country Status (24)

Country Link
US (2) US8257739B2 (pt)
EP (2) EP2111856A3 (pt)
JP (1) JP2006500349A (pt)
CN (1) CN1681479A (pt)
AR (1) AR040969A1 (pt)
AT (1) ATE442130T1 (pt)
AU (1) AU2003249474A1 (pt)
BR (1) BR0313428A (pt)
CA (1) CA2496441C (pt)
DE (1) DE60329188D1 (pt)
ES (1) ES2333318T3 (pt)
GT (1) GT200300170A (pt)
IL (1) IL166411A0 (pt)
MX (1) MXPA05000977A (pt)
NO (1) NO20050419L (pt)
PA (1) PA8579801A1 (pt)
PE (1) PE20040865A1 (pt)
PL (1) PL375345A1 (pt)
PT (1) PT1530457E (pt)
RU (1) RU2005103625A (pt)
TW (1) TW200406224A (pt)
UY (1) UY27929A1 (pt)
WO (1) WO2004014342A1 (pt)
ZA (1) ZA200500470B (pt)

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US8377952B2 (en) 2003-08-28 2013-02-19 Abbott Laboratories Solid pharmaceutical dosage formulation
US8025899B2 (en) * 2003-08-28 2011-09-27 Abbott Laboratories Solid pharmaceutical dosage form
JP2008511607A (ja) * 2004-08-31 2008-04-17 ファイザー・プロダクツ・インク 低溶解性薬物および重合体を含む医薬投与剤形
WO2006079921A2 (en) 2005-01-28 2006-08-03 Pfizer Products Inc. Drying of drug-containing particles
US8834929B2 (en) 2006-07-21 2014-09-16 Bend Research, Inc. Drying of drug-containing particles
CN101657216B (zh) * 2007-04-20 2012-11-21 大同化成工业株式会社 干式固体分散体用基剂、含有该基剂的固体分散体及含有该分散体的组合物
US20100048524A1 (en) 2008-03-14 2010-02-25 Angela Brodie Novel C-17-Heteroaryl Steroidal CYP17 Inhibitors/Antiandrogens;Synthesis In Vitro Biological Activities, Pharmacokinetics and Antitumor Activity
EP2393827B1 (en) 2009-02-05 2015-10-07 Tokai Pharmaceuticals, Inc. Novel prodrugs of steroidal cyp17 inhibitors/antiandrogens
EP2366378A1 (en) 2010-03-01 2011-09-21 Dexcel Pharma Technologies Ltd. Sustained-release donepezil formulations
WO2012122279A1 (en) 2011-03-08 2012-09-13 Zalicus Pharmaceuticals Ltd. Solid dispersion formulations and methods of use thereof
US9095585B2 (en) * 2011-07-21 2015-08-04 Bristol-Myers Squibb Company Bioavailable compositions of amorphous piperidinyl compounds
BR112015019807B1 (pt) 2013-03-07 2020-12-08 Dow Global Technologies Llc acetato succinato de hidroxipropil metilcelulose, composição, dispersão sólida, forma de dosagem e envoltório de cápsula
JP6334574B2 (ja) 2013-03-07 2018-05-30 ダウ グローバル テクノロジーズ エルエルシー 新規の超高分子量のエステル化セルロースエーテル
CN105025887B (zh) 2013-03-07 2017-07-28 陶氏环球技术有限责任公司 新颖极低粘度酯化纤维素醚
CA2904170A1 (en) 2013-03-14 2014-09-25 University Of Maryland, Baltimore Androgen receptor down-regulating agents and uses thereof
EP2832723B1 (en) * 2013-07-29 2017-02-15 Zentiva, a.s. Stabilised amorphous forms of Saxagliptin
KR20160058774A (ko) 2013-08-12 2016-05-25 토카이 파마슈티컬, 아이엔씨. 안드로겐-표적 치료제를 이용하는 종양 질환 치료를 위한 바이오마커
CA2962719A1 (en) 2014-10-31 2016-05-06 Bend Research Inc. Process for forming active domains dispersed in a matrix
US20200147032A1 (en) 2018-11-14 2020-05-14 Robert K. Prud'homme Dihydromyricetin hot melt extrusion formulations and methods for forming them
MX2021015457A (es) 2019-06-14 2022-04-06 Univ Princeton Formulaciones de dihidromiricetina y un permeabilizante.

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Also Published As

Publication number Publication date
PL375345A1 (en) 2005-11-28
EP1530457A1 (en) 2005-05-18
WO2004014342A1 (en) 2004-02-19
DE60329188D1 (de) 2009-10-22
GT200300170A (es) 2004-05-12
UY27929A1 (es) 2004-03-31
CN1681479A (zh) 2005-10-12
TW200406224A (en) 2004-05-01
AU2003249474A1 (en) 2004-02-25
US20040156905A1 (en) 2004-08-12
US8257739B2 (en) 2012-09-04
NO20050419L (no) 2005-04-04
JP2006500349A (ja) 2006-01-05
ZA200500470B (en) 2006-07-26
CA2496441C (en) 2010-03-16
PE20040865A1 (es) 2004-11-25
EP2111856A2 (en) 2009-10-28
AR040969A1 (es) 2005-04-27
RU2005103625A (ru) 2005-08-20
PA8579801A1 (es) 2004-02-16
US8491933B2 (en) 2013-07-23
ATE442130T1 (de) 2009-09-15
MXPA05000977A (es) 2005-05-16
ES2333318T3 (es) 2010-02-19
EP1530457B1 (en) 2009-09-09
IL166411A0 (en) 2006-01-15
US20120322805A1 (en) 2012-12-20
EP2111856A3 (en) 2014-09-10
CA2496441A1 (en) 2004-02-19
BR0313428A (pt) 2005-06-28

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