|
EP0682027B1
(de)
*
|
1994-05-03 |
1997-10-15 |
Novartis AG |
Pyrrolopyrimidinderivate mit antiproliferativer Wirkung
|
|
TW321649B
(cs)
*
|
1994-11-12 |
1997-12-01 |
Zeneca Ltd |
|
|
GB9424233D0
(en)
*
|
1994-11-30 |
1995-01-18 |
Zeneca Ltd |
Quinazoline derivatives
|
|
ES2150113T3
(es)
*
|
1995-04-03 |
2000-11-16 |
Novartis Ag |
Derivados de pirazol y procedimientos para la preparacion de los mismos.
|
|
GB9508537D0
(en)
*
|
1995-04-27 |
1995-06-14 |
Zeneca Ltd |
Quinazoline derivatives
|
|
GB9508565D0
(en)
*
|
1995-04-27 |
1995-06-14 |
Zeneca Ltd |
Quiazoline derivative
|
|
GB9508538D0
(en)
*
|
1995-04-27 |
1995-06-14 |
Zeneca Ltd |
Quinazoline derivatives
|
|
GB9508535D0
(en)
*
|
1995-04-27 |
1995-06-14 |
Zeneca Ltd |
Quinazoline derivative
|
|
WO1996033977A1
(en)
*
|
1995-04-27 |
1996-10-31 |
Zeneca Limited |
Quinazoline derivatives
|
|
MX9800215A
(es)
*
|
1995-07-06 |
1998-03-31 |
Novartis Ag |
Pirrolopirimidas y procesos para su preparacion.
|
|
GB9624482D0
(en)
*
|
1995-12-18 |
1997-01-15 |
Zeneca Phaema S A |
Chemical compounds
|
|
ATE217873T1
(de)
*
|
1996-01-23 |
2002-06-15 |
Novartis Erfind Verwalt Gmbh |
Pyrrolopyrimidinen und verfahren zu deren herstellung
|
|
BR9707495A
(pt)
|
1996-02-13 |
1999-07-27 |
Zeneca Ltd |
Derivado de quinazolina processo para a preparação do mesmo composição farmacêutica e processo para a produç o de um efeito antiangiogênico e/ou de redução de permeabilidade vascular em um animal de sangue quente
|
|
GB9603097D0
(en)
*
|
1996-02-14 |
1996-04-10 |
Zeneca Ltd |
Quinazoline compounds
|
|
GB9603095D0
(en)
*
|
1996-02-14 |
1996-04-10 |
Zeneca Ltd |
Quinazoline derivatives
|
|
US6291455B1
(en)
|
1996-03-05 |
2001-09-18 |
Zeneca Limited |
4-anilinoquinazoline derivatives
|
|
HU228446B1
(en)
|
1996-04-12 |
2013-03-28 |
Warner Lambert Co |
Kinazoline derivatives as irreversible inhibitors of protein-kinase, pharmaceutical compositions containing these compounds and use thereof
|
|
GB9607729D0
(en)
*
|
1996-04-13 |
1996-06-19 |
Zeneca Ltd |
Quinazoline derivatives
|
|
AU3176297A
(en)
*
|
1996-06-25 |
1998-01-14 |
Novartis Ag |
Substituted 7-amino-pyrrolo{3,2-d}pyrimidines and the use thereof
|
|
WO1998007726A1
(en)
|
1996-08-23 |
1998-02-26 |
Novartis Ag |
Substituted pyrrolopyrimidines and processes for their preparation
|
|
US6251911B1
(en)
|
1996-10-02 |
2001-06-26 |
Novartis Ag |
Pyrimidine derivatives and processes for the preparation thereof
|
|
US6225318B1
(en)
|
1996-10-17 |
2001-05-01 |
Pfizer Inc |
4-aminoquinazolone derivatives
|
|
US6413971B1
(en)
|
1996-11-27 |
2002-07-02 |
Pfizer Inc |
Fused bicyclic pyrimidine derivatives
|
|
EP1012151B1
(en)
|
1997-09-02 |
2002-08-07 |
Bristol-Myers Squibb Pharma Company |
Heterocyclyl-substituted ring-fused pyridines and pyrimidines as corticotropin releasing hormone (crh) antagonists, useful for treating cns and stress-related disorders
|
|
CA2309690A1
(en)
|
1997-11-11 |
1999-05-20 |
Pfizer Products Inc. |
Thienopyrimidine and thienopyridine derivatives useful as anticancer agents
|
|
JPH11236333A
(ja)
*
|
1997-12-30 |
1999-08-31 |
Pfizer Prod Inc |
抗ガン剤として有用なイミダゾリン−4−オン誘導体
|
|
RS49779B
(sr)
|
1998-01-12 |
2008-06-05 |
Glaxo Group Limited, |
Biciklična heteroaromatična jedinjenja kao inhibitori protein tirozin kinaze
|
|
US6187777B1
(en)
|
1998-02-06 |
2001-02-13 |
Amgen Inc. |
Compounds and methods which modulate feeding behavior and related diseases
|
|
DE69943144D1
(de)
|
1998-03-31 |
2011-03-03 |
Kyowa Hakko Kirin Co Ltd |
Stickstoffenthaltende heterocyclische verbindungen
|
|
BR9911365A
(pt)
|
1998-06-19 |
2001-03-13 |
Pfizer Prod Inc |
Compostos pirrolo[2,3-d]pirimidina
|
|
PA8474101A1
(es)
*
|
1998-06-19 |
2000-09-29 |
Pfizer Prod Inc |
Compuestos de pirrolo [2,3-d] pirimidina
|
|
WO2000023444A1
(en)
*
|
1998-10-21 |
2000-04-27 |
Abbott Laboratories |
5,7-disubstituted-4-aminopyrido[2,3-d]pyrimidine compounds
|
|
US6174903B1
(en)
|
1998-12-28 |
2001-01-16 |
Pfizer Inc. |
Imidazolidin-4-one derivatives useful as anticancer agents
|
|
JP3270834B2
(ja)
|
1999-01-27 |
2002-04-02 |
ファイザー・プロダクツ・インク |
抗がん剤として有用なヘテロ芳香族二環式誘導体
|
|
UA71945C2
(en)
*
|
1999-01-27 |
2005-01-17 |
Pfizer Prod Inc |
Substituted bicyclic derivatives being used as anticancer agents
|
|
US6933299B1
(en)
|
1999-07-09 |
2005-08-23 |
Smithkline Beecham Corporation |
Anilinoquinazolines as protein tyrosine kinase inhibitors
|
|
ATE377597T1
(de)
|
1999-07-09 |
2007-11-15 |
Glaxo Group Ltd |
Anilinochinazoline als protein-tyrosin- kinasehemmer
|
|
US6432979B1
(en)
|
1999-08-12 |
2002-08-13 |
American Cyanamid Company |
Method of treating or inhibiting colonic polyps and colorectal cancer
|
|
EP1409487A1
(en)
|
1999-09-15 |
2004-04-21 |
Warner-Lambert Company Llc |
Pteridinones as kinase inhibitors
|
|
RU2264404C2
(ru)
*
|
1999-10-21 |
2005-11-20 |
Ф.Хоффманн-Ля Рош Аг |
Алкиламинозамещенные бициклические азотсодержащие гетероциклы и фармацевтическая композиция на их основе
|
|
GB9925958D0
(en)
*
|
1999-11-02 |
1999-12-29 |
Bundred Nigel J |
Therapeutic use
|
|
CZ301689B6
(cs)
|
1999-11-05 |
2010-05-26 |
Astrazeneca Ab |
Derivát chinazolinu a farmaceutický prostredek, který ho obsahuje
|
|
JP2001142235A
(ja)
|
1999-11-17 |
2001-05-25 |
Fuji Denki Gazo Device Kk |
電子写真用感光体
|
|
EP1382339B1
(en)
|
1999-12-10 |
2007-12-05 |
Pfizer Products Inc. |
Compositions containing pyrrolo ¬2,3-d pyrimidine derivatives
|
|
JP2003535867A
(ja)
|
2000-06-06 |
2003-12-02 |
ファイザー プロダクツ インコーポレイテッド |
抗癌剤として有用なチオフェン誘導体
|
|
IL152771A0
(en)
|
2000-06-26 |
2003-06-24 |
Pfizer Prod Inc |
PYRROLO(2,3-d) PYRIMIDINE COMPOUNDS AS IMMUNOSUPPRESSIVE AGENTS
|
|
WO2002024667A1
(en)
|
2000-09-20 |
2002-03-28 |
Merck Patent Gmbh |
4-amino-quinazolines
|
|
DE60137273D1
(de)
|
2000-10-20 |
2009-02-12 |
Eisai R&D Man Co Ltd |
Verfahren zur Herstellung von 4-Phenoxy chinolin Derivaten
|
|
ES2263743T3
(es)
|
2001-04-13 |
2006-12-16 |
Pfizer Products Inc. |
Derivados de 4-aminopiridopirimidina sustituidos con un grupo biciclico.
|
|
AR035885A1
(es)
*
|
2001-05-14 |
2004-07-21 |
Novartis Ag |
Derivados de 4-amino-5-fenil-7-ciclobutilpirrolo (2,3-d)pirimidina, un proceso para su preparacion, una composicion farmaceutica y el uso de dichos derivados para la preparacion de una composicion farmaceutica
|
|
US7301023B2
(en)
|
2001-05-31 |
2007-11-27 |
Pfizer Inc. |
Chiral salt resolution
|
|
AU2002345792A1
(en)
|
2001-06-21 |
2003-01-08 |
Pfizer Inc. |
Thienopyridine and thienopyrimidine anticancer agents
|
|
CZ294535B6
(cs)
*
|
2001-08-02 |
2005-01-12 |
Ústav Experimentální Botaniky Avčr |
Heterocyklické sloučeniny na bázi N6-substituovaného adeninu, způsoby jejich přípravy, jejich použití pro přípravu léčiv, kosmetických přípravků a růstových regulátorů, farmaceutické přípravky, kosmetické přípravky a růstové regulátory tyto sloučeniny obsahující
|
|
GB0121033D0
(en)
*
|
2001-08-30 |
2001-10-24 |
Novartis Ag |
Organic compounds
|
|
US7829566B2
(en)
|
2001-09-17 |
2010-11-09 |
Werner Mederski |
4-amino-quinazolines
|
|
PY0228255A
(es)
*
|
2001-12-06 |
2004-06-01 |
Pfizer Prod Inc |
Compuestos cristalinos novedosos
|
|
RU2289583C2
(ru)
*
|
2001-12-27 |
2006-12-20 |
Ф.Хоффманн-Ля Рош Аг |
Пиримидотриазины, способ их получения, фармацевтическая композиция на их основе и применение
|
|
DE60320933D1
(de)
*
|
2002-01-10 |
2008-06-26 |
Bayer Healthcare Ag |
Rho-kinase inhibitoren
|
|
CN1627944A
(zh)
|
2002-01-17 |
2005-06-15 |
神经能质公司 |
取代的喹唑啉-4-基胺类似物作为辣椒辣素调节剂
|
|
MXPA04007196A
(es)
|
2002-01-23 |
2005-06-08 |
Bayer Pharmaceuticals Corp |
Inhibidores de rho-quinasa.
|
|
JP4469179B2
(ja)
|
2002-01-23 |
2010-05-26 |
バイエル ファーマセチカル コーポレーション |
Rhoキナーゼ阻害剤としてのピリミジン誘導体
|
|
JP2003238561A
(ja)
|
2002-02-13 |
2003-08-27 |
Fuji Denki Gazo Device Kk |
キノメタン化合物
|
|
BR0308162A
(pt)
|
2002-03-01 |
2004-12-07 |
Pfizer |
Derivados de indolil-uréia de tienopiridinas úteis como agentes antiangiogênicos e métodos para o seu uso
|
|
EP1485390B1
(en)
*
|
2002-03-07 |
2008-10-08 |
F. Hoffman-la Roche AG |
Bicyclic pyridine and pyrimidine p38 kinase inhibitors
|
|
UA77303C2
(en)
|
2002-06-14 |
2006-11-15 |
Pfizer |
Derivatives of thienopyridines substituted by benzocondensed heteroarylamide useful as therapeutic agents, pharmaceutical compositions and methods for their use
|
|
NZ539901A
(en)
|
2002-11-26 |
2007-09-28 |
Pfizer Prod Inc |
Method of treatment of transplant rejection
|
|
EP1592430A4
(en)
|
2003-01-17 |
2006-05-31 |
Threshold Pharmaceuticals Inc |
TREATMENT OF GOOD PROSTATE HYPERPLASIA BY MEANS OF ENERGYSTIC ACTIVE SUBSTANCES
|
|
FR2851248B1
(fr)
*
|
2003-02-18 |
2005-04-08 |
Aventis Pharma Sa |
Nouveaux derives de la purine, leur procede de preparation, leur application a titre de medicaments, compositions pharmaceutiques et nouvelle utilisation
|
|
PT1636236E
(pt)
|
2003-05-22 |
2013-12-16 |
Nerviano Medical Sciences Srl |
Derivados de pirazol-quinazolina, processo para sua preparação e sua utilização como inibidores de cinase
|
|
EP1656378A4
(en)
*
|
2003-08-15 |
2011-05-11 |
Irm Llc |
COMPOUNDS AND COMPOSITIONS INHIBITING TYROSINE KINASE RECEPTOR ACTIVITY
|
|
US7338957B2
(en)
*
|
2003-08-28 |
2008-03-04 |
Irm Llc |
Compounds and compositions as protein kinase inhibitors
|
|
EP1660504B1
(en)
|
2003-08-29 |
2008-10-29 |
Pfizer Inc. |
Thienopyridine-phenylacet amides and their derivatives useful as new anti-angiogenic agents
|
|
US7419978B2
(en)
|
2003-10-22 |
2008-09-02 |
Bristol-Myers Squibb Company |
Phenyl-aniline substituted bicyclic compounds useful as kinase inhibitors
|
|
US7683172B2
(en)
|
2003-11-11 |
2010-03-23 |
Eisai R&D Management Co., Ltd. |
Urea derivative and process for preparing the same
|
|
EA009994B1
(ru)
|
2003-12-23 |
2008-06-30 |
Пфайзер Инк. |
Новые хинолиновые производные
|
|
US20080269238A1
(en)
*
|
2004-04-01 |
2008-10-30 |
Takeda Pharmaceutical Company Limited |
Thiazolopyrimidine Derivative
|
|
MXPA06013805A
(es)
|
2004-05-27 |
2007-02-02 |
Pfizer Prod Inc |
Derivados de pirrolopirimidina de utilidad en el tratamiento contra el cancer.
|
|
CN1993362B
(zh)
*
|
2004-06-02 |
2010-12-15 |
武田药品工业株式会社 |
稠合的杂环化合物
|
|
WO2005118588A1
(ja)
*
|
2004-06-02 |
2005-12-15 |
Takeda Pharmaceutical Company Limited |
縮合複素環化合物
|
|
JP2007161585A
(ja)
*
|
2004-06-25 |
2007-06-28 |
Taisho Pharmaceut Co Ltd |
環状アミノ基で置換されているピロロピリミジン及びピロロピリジン誘導体
|
|
AU2005283422C1
(en)
|
2004-09-17 |
2017-02-02 |
Eisai R & D Management Co., Ltd. |
Medicinal composition
|
|
EP1838712B8
(en)
*
|
2004-12-14 |
2011-10-12 |
AstraZeneca AB |
Pyrazolopyrimidine compounds as antitumor agents
|
|
CA2596830A1
(en)
*
|
2005-02-03 |
2006-09-14 |
Vertex Pharmaceuticals Incorporated |
Pyrrolopyrimidines useful as inhibitors of protein kinase
|
|
US7423043B2
(en)
|
2005-02-18 |
2008-09-09 |
Lexicon Pharmaceuticals, Inc. |
4-Piperidin-1-yl-7H-pyrrolo[2,3-d]pyrimidine compounds
|
|
US20090111805A1
(en)
*
|
2005-02-24 |
2009-04-30 |
Pfizer Inc. |
Bicyclic heteroaromatic derivatives useful as anticancer agents
|
|
WO2006138714A2
(en)
*
|
2005-06-17 |
2006-12-28 |
Janssen Pharmaceutica N.V. |
Naphthyridine compounds
|
|
WO2007015578A1
(ja)
|
2005-08-02 |
2007-02-08 |
Eisai R & D Management Co., Ltd. |
血管新生阻害物質の効果を検定する方法
|
|
US7915411B2
(en)
|
2005-12-21 |
2011-03-29 |
Abbott Laboratories |
Anti-viral compounds
|
|
ATE475660T1
(de)
|
2005-12-21 |
2010-08-15 |
Abbott Lab |
Antivirale verbindungen
|
|
CN101443334A
(zh)
*
|
2005-12-21 |
2009-05-27 |
艾博特公司 |
抗病毒化合物
|
|
EP1979348B1
(en)
*
|
2005-12-21 |
2012-01-18 |
Abbott Laboratories |
Anti-viral compounds
|
|
JP5255559B2
(ja)
*
|
2006-03-31 |
2013-08-07 |
アボット・ラボラトリーズ |
インダゾール化合物
|
|
WO2007114926A2
(en)
*
|
2006-04-04 |
2007-10-11 |
The Regents Of The University Of California |
Kinase antagonists
|
|
RU2448708C3
(ru)
|
2006-05-18 |
2017-09-28 |
Эйсай Ар Энд Ди Менеджмент Ко., Лтд. |
Противоопухолевое средство против рака щитовидной железы
|
|
EP1889847A1
(en)
*
|
2006-07-10 |
2008-02-20 |
DeveloGen Aktiengesellschaft |
Pyrrolopyrimidines for pharmaceutical compositions
|
|
CN101511793B
(zh)
|
2006-08-28 |
2011-08-03 |
卫材R&D管理有限公司 |
针对未分化型胃癌的抗肿瘤剂
|
|
EP2103620A1
(en)
*
|
2006-12-12 |
2009-09-23 |
Takeda Pharmaceutical Company Limited |
Fused heterocyclic compound
|
|
US8236950B2
(en)
|
2006-12-20 |
2012-08-07 |
Abbott Laboratories |
Anti-viral compounds
|
|
CN101600694A
(zh)
|
2007-01-29 |
2009-12-09 |
卫材R&D管理有限公司 |
未分化型胃癌治疗用组合物
|
|
KR101513326B1
(ko)
|
2007-11-09 |
2015-04-17 |
에자이 알앤드디 매니지먼트 가부시키가이샤 |
혈관 신생 저해 물질과 항종양성 백금 착물의 병용
|
|
AR070874A1
(es)
|
2008-03-12 |
2010-05-12 |
Takeda Pharmaceutical |
Compuesto heterociclico fusionado, una composicion farmaceutica que lo comprende y su uso en el tratamiento del cancer.
|
|
AR073354A1
(es)
*
|
2008-07-31 |
2010-11-03 |
Genentech Inc |
Compuestos de pirimidina, composiciones farmaceuticas y su uso en el tratamiento del cancer.
|
|
JP4884570B2
(ja)
|
2008-08-20 |
2012-02-29 |
ファイザー・インク |
ピロロ[2,3−d]ピリミジン化合物
|
|
TW201014860A
(en)
*
|
2008-09-08 |
2010-04-16 |
Boehringer Ingelheim Int |
New chemical compounds
|
|
KR101126736B1
(ko)
*
|
2008-11-27 |
2012-04-12 |
주식회사 레고켐 바이오사이언스 |
티로신 키나아제 저해 화합물, 이의 이성질체 또는 이의 약학적으로 허용가능한 염 및 이를 포함하는 약학적 조성물
|
|
SG173014A1
(en)
|
2009-01-16 |
2011-08-29 |
Exelixis Inc |
Malate salt of n- (4- { [ 6, 7-bis (methyloxy) quin0lin-4-yl] oxy}phenyl)-n' - (4 -fluorophenyl) cyclopropane-1,1-dicarboxamide, and crystalline forms therof for the treatment of cancer
|
|
DE102009005193A1
(de)
*
|
2009-01-20 |
2010-07-22 |
Merck Patent Gmbh |
Neue heterocyclische Verbindungen als MetAP-2 Inhibitoren
|
|
JP5603883B2
(ja)
*
|
2009-02-17 |
2014-10-08 |
ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング |
B−Rafキナーゼを阻害するためのピリミドピリミジン誘導体
|
|
UA108618C2
(uk)
|
2009-08-07 |
2015-05-25 |
|
Застосування c-met-модуляторів в комбінації з темозоломідом та/або променевою терапією для лікування раку
|
|
DK2468281T3
(en)
|
2009-08-19 |
2016-03-21 |
Eisai R&D Man Co Ltd |
Quinolinderivatholdig pharmaceutical composition
|
|
WO2011058027A2
(en)
|
2009-11-12 |
2011-05-19 |
F. Hoffmann-La Roche Ag |
N-9-substituted purine compounds, compositions and methods of use
|
|
CN102712642B
(zh)
|
2009-11-12 |
2015-08-12 |
霍夫曼-拉罗奇有限公司 |
N-7取代的嘌呤和吡唑并嘧啶化合物、组合物和使用方法
|
|
JP2013518882A
(ja)
*
|
2010-02-05 |
2013-05-23 |
ファイザー・インク |
JAK阻害剤としてのピロロ[2,3−d]ピリミジン尿素化合物
|
|
WO2011162343A1
(ja)
|
2010-06-25 |
2011-12-29 |
エーザイ・アール・アンド・ディー・マネジメント株式会社 |
キナーゼ阻害作用を有する化合物の併用による抗腫瘍剤
|
|
AU2011295441B2
(en)
*
|
2010-08-27 |
2015-04-09 |
Merck Patent Gmbh |
Furopyridine derivatives
|
|
EP2614065B1
(en)
|
2010-12-17 |
2017-04-19 |
Nerviano Medical Sciences S.r.l. |
Substituted pyrazolo-quinazoline derivatives as kinase inhibitors
|
|
BR112013022552B1
(pt)
|
2011-03-04 |
2021-11-23 |
Newgen Therapeutics, Inc |
Compostos de quinazolina substituídos com alcino, seu uso, composição farmacêutica, e kit
|
|
CN103402519B
(zh)
|
2011-04-18 |
2015-11-25 |
卫材R&D管理有限公司 |
肿瘤治疗剂
|
|
JP6038128B2
(ja)
|
2011-06-03 |
2016-12-07 |
エーザイ・アール・アンド・ディー・マネジメント株式会社 |
レンバチニブ化合物に対する甲状腺癌対象及び腎臓癌対象の反応性を予測及び評価するためのバイオマーカー
|
|
AU2013224420B2
(en)
*
|
2012-02-21 |
2016-12-15 |
Merck Patent Gmbh |
Furopyridine derivatives
|
|
EP2900671A1
(en)
|
2012-09-26 |
2015-08-05 |
Bayer Pharma Aktiengesellschaft |
Substituted indazol-pyrrolopyrimidines useful in the treatment of hyperproliferative diseases
|
|
JP2015531361A
(ja)
|
2012-09-26 |
2015-11-02 |
バイエル・ファルマ・アクティエンゲゼルシャフト |
過剰増殖性疾患の治療に有用な置換インダゾール−ピロロピリミジン
|
|
AU2013364953A1
(en)
|
2012-12-21 |
2015-04-30 |
Eisai R&D Management Co., Ltd. |
Amorphous form of quinoline derivative, and method for producing same
|
|
JP2016506944A
(ja)
*
|
2013-02-01 |
2016-03-07 |
バイエル・ファルマ・アクティエンゲゼルシャフト |
置換ピラゾロピリミジニルアミノ−インダゾール
|
|
WO2014145576A2
(en)
|
2013-03-15 |
2014-09-18 |
Northwestern University |
Substituted pyrrolo(2,3-d)pyrimidines for the treatment of cancer
|
|
EP2997377B1
(en)
|
2013-05-14 |
2018-07-18 |
Eisai R&D Management Co., Ltd. |
Biomarkers for predicting and assessing responsiveness of endometrial cancer subjects to lenvatinib compounds
|
|
HRP20220522T1
(hr)
|
2014-08-04 |
2022-06-10 |
Nuevolution A/S |
Proizvoljno kondenzirani heterociklil-supstituirani derivati pirimidina koji su korisni za liječenje upalnih, metaboličkih, onkoloških i autoimunih bolesti
|
|
PT3524595T
(pt)
|
2014-08-28 |
2022-09-19 |
Eisai R&D Man Co Ltd |
Derivado de quinolina altamente puro e método para produção do mesmo
|
|
AU2016224583B2
(en)
|
2015-02-25 |
2021-06-03 |
Eisai R&D Management Co., Ltd. |
Method for suppressing bitterness of quinoline derivative
|
|
KR102662228B1
(ko)
|
2015-03-04 |
2024-05-02 |
머크 샤프 앤드 돔 코포레이션 |
암을 치료하기 위한 pd-1 길항제 및 vegfr/fgfr/ret 티로신 키나제 억제제의 조합
|
|
BR112017027227B1
(pt)
|
2015-06-16 |
2023-12-12 |
Eisai R&D Management Co., Ltd |
Agente anti-câncer
|
|
JP6553726B2
(ja)
|
2015-08-20 |
2019-07-31 |
エーザイ・アール・アンド・ディー・マネジメント株式会社 |
腫瘍治療剤
|
|
GB201520499D0
(en)
*
|
2015-11-20 |
2016-01-06 |
Medical Res Council Technology |
Compounds
|
|
CN106831779B
(zh)
*
|
2015-11-28 |
2019-07-19 |
南昌弘益药业有限公司 |
一类jak激酶抑制剂的新化合物
|
|
JP6581320B2
(ja)
|
2017-02-08 |
2019-09-25 |
エーザイ・アール・アンド・ディー・マネジメント株式会社 |
腫瘍治療用医薬組成物
|
|
EP3624800A4
(en)
|
2017-05-16 |
2021-02-17 |
Eisai R&D Management Co., Ltd. |
TREATMENT OF HEPATOCELLULAR CARCINOMA
|
|
NL2022471B1
(en)
|
2019-01-29 |
2020-08-18 |
Vationpharma B V |
Solid state forms of oclacitinib
|
|
CN111825674A
(zh)
*
|
2019-04-22 |
2020-10-27 |
上海仕谱生物科技有限公司 |
嘧啶并五元杂环类化合物及其作为突变型idh2抑制剂的用途
|
|
MX2022007265A
(es)
|
2019-12-20 |
2022-09-09 |
Nuevolution As |
Compuestos activos frente a receptores nucleares.
|
|
US11685727B2
(en)
|
2019-12-20 |
2023-06-27 |
Nuevolution A/S |
Compounds active towards nuclear receptors
|
|
EP4126874A1
(en)
|
2020-03-31 |
2023-02-08 |
Nuevolution A/S |
Compounds active towards nuclear receptors
|
|
CA3174176A1
(en)
|
2020-03-31 |
2021-10-07 |
Sanne Schroder Glad |
Compounds active towards nuclear receptors
|
|
EP4323356A1
(en)
|
2021-04-13 |
2024-02-21 |
Nuvalent, Inc. |
Amino-substituted heterocycles for treating cancers with egfr mutations
|