SK12752003A3 - Prípravky užitočné na liečbu patológií odpovedajúce na aktiváciu PPAR-gamma receptora - Google Patents

Prípravky užitočné na liečbu patológií odpovedajúce na aktiváciu PPAR-gamma receptora Download PDF

Info

Publication number: SK12752003A3
Authority: SK; Slovakia
Prior art keywords: formula; treatment; ppar; spirolaxin; activation
Prior art date: 2001-03-16

Application number

SK1275-2003A

Other languages

English (en)

Slovak (sk)

Inventor

Claudio Pisano

Teresa Riccioni

Original Assignee

Sigma-Tau Industrie Farmaceutiche Riunite S.P.A.

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2001-03-16

Filing date

2002-03-01

Publication date

2004-01-08

2002-03-01 Application filed by Sigma-Tau Industrie Farmaceutiche Riunite S.P.A. filed Critical Sigma-Tau Industrie Farmaceutiche Riunite S.P.A.

2004-01-08 Publication of SK12752003A3 publication Critical patent/SK12752003A3/sk

Links

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CZIMFHQXGMXDMO-DGROVODQSA-N (3r)-5-hydroxy-7-methoxy-3-[5-[(2r,5r,7r)-2-methyl-1,6-dioxaspiro[4.5]decan-7-yl]pentyl]-3h-2-benzofuran-1-one Chemical compound C([C@H](O1)CCCCC[C@@H]2C=3C=C(O)C=C(C=3C(=O)O2)OC)CC[C@@]21CC[C@@H](C)O2 CZIMFHQXGMXDMO-DGROVODQSA-N 0.000 claims abstract description 29
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Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/365—Lactones
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/48—Drugs for disorders of the endocrine system of the pancreatic hormones
- A61P5/50—Drugs for disorders of the endocrine system of the pancreatic hormones for increasing or potentiating the activity of insulin
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid

Landscapes

Health & Medical Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Chemical & Material Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Medicinal Chemistry (AREA)
General Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Diabetes (AREA)
Epidemiology (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Hematology (AREA)
Endocrinology (AREA)
Emergency Medicine (AREA)
Obesity (AREA)
Oncology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Peptides Or Proteins (AREA)

SK1275-2003A 2001-03-16 2002-03-01 Prípravky užitočné na liečbu patológií odpovedajúce na aktiváciu PPAR-gamma receptora SK12752003A3 (sk)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
IT2001RM000136A ITRM20010136A1 (it)	2001-03-16	2001-03-16	Composti utili per il trattamento di patologie che rispondono all'attivazione del recettore ppar-gamma.
PCT/IT2002/000127 WO2002074291A2 (en)	2001-03-16	2002-03-01	Compositions useful for the treatment of pathologies responding to the activation of ppar-gamma receptor

Publications (1)

Publication Number	Publication Date
SK12752003A3 true SK12752003A3 (sk)	2004-01-08

Family

ID=11455333

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
SK1275-2003A SK12752003A3 (sk)	2001-03-16	2002-03-01	Prípravky užitočné na liečbu patológií odpovedajúce na aktiváciu PPAR-gamma receptora

Country Status (19)

Country	Link
US (4)	US6897235B2 (cs)
EP (1)	EP1368025B1 (cs)
JP (1)	JP4276842B2 (cs)
KR (1)	KR100851678B1 (cs)
CN (2)	CN1286456C (cs)
AT (1)	ATE308984T1 (cs)
AU (1)	AU2002247951B2 (cs)
BR (1)	BR0208157A (cs)
CA (1)	CA2440979C (cs)
CZ (1)	CZ20032523A3 (cs)
DE (1)	DE60207215T2 (cs)
DK (1)	DK1368025T3 (cs)
ES (1)	ES2249568T3 (cs)
HU (1)	HUP0303518A3 (cs)
IT (1)	ITRM20010136A1 (cs)
MX (1)	MXPA03008317A (cs)
PL (1)	PL369295A1 (cs)
SK (1)	SK12752003A3 (cs)
WO (1)	WO2002074291A2 (cs)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US7041691B1 (en)	1999-06-30	2006-05-09	Amgen Inc.	Compounds for the modulation of PPARγ activity
US20030171399A1 (en)	2000-06-28	2003-09-11	Tularik Inc.	Quinolinyl and benzothiazolyl modulators
WO2004100945A1 (en) *	2003-05-14	2004-11-25	Dsm Ip Assets B.V.	Use of phthalide derivatives for the treatment and prevention of diabetes mellitus
US7223761B2 (en)	2003-10-03	2007-05-29	Amgen Inc.	Salts and polymorphs of a potent antidiabetic compound
WO2008030604A2 (en)	2006-09-08	2008-03-13	Rhode Island Hospital	Treatment, prevention, and reversal of alcohol-induced brain disease

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
JPH07285862A (ja) *	1994-04-21	1995-10-31	Kokka Iyaku Kanrikyoku Shisen Kokinso Kogyo Kenkyusho	脂質低下剤
JPH107557A (ja) *	1996-06-17	1998-01-13	Banyu Pharmaceut Co Ltd	抗腫瘍性物質スピロラキシン
US6440961B1 (en) *	1997-10-27	2002-08-27	Dr. Reddy's Research Foundation	Tricyclic compounds and their use in medicine: process for their preparation and pharmaceutical compositions containing them
IT1317001B1 (it) *	2000-03-13	2003-05-26	Sigma Tau Ind Farmaceuti	Uso della spirolaxina per il trattamento di patologie associate ad unaalterata angiogenesi.

2001
- 2001-03-16 IT IT2001RM000136A patent/ITRM20010136A1/it unknown
2002
- 2002-03-01 KR KR1020037012030A patent/KR100851678B1/ko not_active Expired - Fee Related
- 2002-03-01 CZ CZ20032523A patent/CZ20032523A3/cs unknown
- 2002-03-01 AU AU2002247951A patent/AU2002247951B2/en not_active Ceased
- 2002-03-01 CN CNB028081382A patent/CN1286456C/zh not_active Expired - Fee Related
- 2002-03-01 JP JP2002572999A patent/JP4276842B2/ja not_active Expired - Fee Related
- 2002-03-01 ES ES02717031T patent/ES2249568T3/es not_active Expired - Lifetime
- 2002-03-01 AT AT02717031T patent/ATE308984T1/de not_active IP Right Cessation
- 2002-03-01 US US10/471,786 patent/US6897235B2/en not_active Expired - Fee Related
- 2002-03-01 CA CA2440979A patent/CA2440979C/en not_active Expired - Fee Related
- 2002-03-01 SK SK1275-2003A patent/SK12752003A3/sk unknown
- 2002-03-01 MX MXPA03008317A patent/MXPA03008317A/es active IP Right Grant
- 2002-03-01 EP EP02717031A patent/EP1368025B1/en not_active Expired - Lifetime
- 2002-03-01 DE DE60207215T patent/DE60207215T2/de not_active Expired - Lifetime
- 2002-03-01 PL PL02369295A patent/PL369295A1/xx not_active Application Discontinuation
- 2002-03-01 CN CNB2006100057819A patent/CN100462073C/zh not_active Expired - Fee Related
- 2002-03-01 BR BR0208157-1A patent/BR0208157A/pt not_active IP Right Cessation
- 2002-03-01 WO PCT/IT2002/000127 patent/WO2002074291A2/en not_active Ceased
- 2002-03-01 DK DK02717031T patent/DK1368025T3/da active
- 2002-03-01 HU HU0303518A patent/HUP0303518A3/hu unknown
2004
- 2004-07-13 US US10/889,030 patent/US20040242675A1/en not_active Abandoned
- 2004-07-13 US US10/889,029 patent/US7276533B2/en not_active Expired - Fee Related
- 2004-10-18 US US10/965,740 patent/US20050131060A1/en not_active Abandoned

Also Published As

Publication number	Publication date
CN1610545A (zh)	2005-04-27
MXPA03008317A (es)	2003-12-11
CZ20032523A3 (cs)	2004-05-12
PL369295A1 (en)	2005-04-18
JP2004523578A (ja)	2004-08-05
HK1075006A1 (en)	2005-12-02
US20050131060A1 (en)	2005-06-16
WO2002074291A3 (en)	2003-03-13
ATE308984T1 (de)	2005-11-15
ITRM20010136A0 (it)	2001-03-16
DE60207215T2 (de)	2006-07-20
DK1368025T3 (da)	2005-12-19
KR100851678B1 (ko)	2008-08-13
AU2002247951B2 (en)	2007-03-01
JP4276842B2 (ja)	2009-06-10
US6897235B2 (en)	2005-05-24
CN1286456C (zh)	2006-11-29
US20040242675A1 (en)	2004-12-02
HK1096850A1 (zh)	2007-06-15
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