SK13082001A3 - Cyklický peptidový analóg a jeho výroba - Google Patents
Cyklický peptidový analóg a jeho výroba Download PDFInfo
- Publication number
- SK13082001A3 SK13082001A3 SK1308-2001A SK13082001A SK13082001A3 SK 13082001 A3 SK13082001 A3 SK 13082001A3 SK 13082001 A SK13082001 A SK 13082001A SK 13082001 A3 SK13082001 A3 SK 13082001A3
- Authority
- SK
- Slovakia
- Prior art keywords
- heteroaryl
- alkyl
- hydrogen
- heterocycloalkyl
- aryl
- Prior art date
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Classifications
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- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/665—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans derived from pro-opiomelanocortin, pro-enkephalin or pro-dynorphin
- C07K14/68—Melanocyte-stimulating hormone [MSH]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Organic Chemistry (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Endocrinology (AREA)
- Neurology (AREA)
- Toxicology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Molecular Biology (AREA)
- Genetics & Genomics (AREA)
- Biophysics (AREA)
- Biochemistry (AREA)
- Gastroenterology & Hepatology (AREA)
- Zoology (AREA)
- Diabetes (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Reproductive Health (AREA)
- Gynecology & Obstetrics (AREA)
- Hematology (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Physical Education & Sports Medicine (AREA)
- Psychology (AREA)
- Pregnancy & Childbirth (AREA)
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Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US12667399P | 1999-03-29 | 1999-03-29 | |
| PCT/US2000/007473 WO2000058361A1 (fr) | 1999-03-29 | 2000-03-21 | Ligands du recepteur de melanocortine |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| SK13082001A3 true SK13082001A3 (sk) | 2002-03-05 |
Family
ID=22426131
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SK1308-2001A SK13082001A3 (sk) | 1999-03-29 | 2000-03-21 | Cyklický peptidový analóg a jeho výroba |
Country Status (34)
| Country | Link |
|---|---|
| US (2) | US6613874B1 (fr) |
| EP (1) | EP1165613B1 (fr) |
| JP (1) | JP2002542159A (fr) |
| KR (2) | KR100519201B1 (fr) |
| CN (1) | CN1249086C (fr) |
| AR (1) | AR023201A1 (fr) |
| AT (1) | ATE393783T1 (fr) |
| AU (1) | AU763510B2 (fr) |
| BR (1) | BR0009497A (fr) |
| CA (1) | CA2368431C (fr) |
| CO (1) | CO5170531A1 (fr) |
| CZ (1) | CZ20013407A3 (fr) |
| DE (1) | DE60038734T2 (fr) |
| DK (1) | DK1165613T3 (fr) |
| ES (1) | ES2304345T3 (fr) |
| HK (1) | HK1044954B (fr) |
| HU (1) | HUP0202203A3 (fr) |
| ID (1) | ID30262A (fr) |
| IL (1) | IL145406A0 (fr) |
| MA (1) | MA25403A1 (fr) |
| MX (1) | MXPA01009881A (fr) |
| MY (1) | MY126585A (fr) |
| NO (1) | NO20014568L (fr) |
| NZ (1) | NZ514141A (fr) |
| PE (1) | PE20001641A1 (fr) |
| PL (1) | PL350095A1 (fr) |
| PT (1) | PT1165613E (fr) |
| RU (1) | RU2213098C2 (fr) |
| SA (1) | SA00210192B1 (fr) |
| SK (1) | SK13082001A3 (fr) |
| TR (1) | TR200102765T2 (fr) |
| TW (1) | TWI250990B (fr) |
| WO (1) | WO2000058361A1 (fr) |
| ZA (1) | ZA200107411B (fr) |
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| US7192713B1 (en) | 1999-05-18 | 2007-03-20 | President And Fellows Of Harvard College | Stabilized compounds having secondary structure motifs |
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| US7235625B2 (en) | 1999-06-29 | 2007-06-26 | Palatin Technologies, Inc. | Multiple agent therapy for sexual dysfunction |
| US6693165B2 (en) | 2000-01-18 | 2004-02-17 | Merck & Co., Inc. | Cyclic peptides as potent and selective melanocortin-4 receptor antagonists |
| PL366630A1 (en) | 2000-08-30 | 2005-02-07 | F.Hoffmann-La Roche Ag | Selective cyclic peptides |
| NZ524190A (en) * | 2000-09-27 | 2004-09-24 | Procter & Gamble | Melanocortin receptor ligands |
| AU2002238106A1 (en) | 2001-02-13 | 2002-08-28 | Palatin Technologies, Inc. | Melanocortin metallopeptides for treatment of sexual dysfunction |
| CA2453515A1 (fr) | 2001-07-11 | 2003-01-23 | Palatin Technologies, Inc. | Peptides lineaires et cycliques specifiques du recepteur de melanocortine |
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| BR112012000867A2 (pt) | 2009-07-13 | 2019-09-24 | Harvard College | "polipeptídeos bifuncional costurado e uso do mesmo" |
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| BR112012011780A2 (pt) | 2009-11-23 | 2019-09-24 | Palatin Technologies, Inc | peptídeo linear,composição farmacêutica,métodopara tratamento de umadoença,indicação,condição ou sídrome mediadsa por receptor de melanocortina emum mamífero humano ou não humano e método para tratamento de uma condição responsiva ás alterações em função de receptor de melanocortina em um mamifero humano ou não humano |
| CN101824415A (zh) * | 2010-03-31 | 2010-09-08 | 华东师范大学 | 黑素皮质1型受体基因的snp及其应用 |
| KR102104762B1 (ko) | 2010-08-13 | 2020-04-24 | 에일러론 테라퓨틱스 인코포레이티드 | 펩티도미메틱 거대고리 |
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| PT3773558T (pt) | 2019-05-10 | 2022-09-13 | Synact Pharma Aps | Tratamento combinado de doença artrítica |
| CN110681362B (zh) * | 2019-09-26 | 2020-09-11 | 浙江大学 | 以羧基和吲哚基为功能基团的混合模式层析介质 |
| US11590209B2 (en) | 2020-01-21 | 2023-02-28 | Palatin Technologies, Inc. | Use of bremelanotide in patients with controlled hypertension |
| US11932628B2 (en) | 2021-01-04 | 2024-03-19 | Regents Of The University Of Minnesota | Selective small molecule peptidomimetic melanocortin ligands |
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| US5462927A (en) | 1985-04-30 | 1995-10-31 | The Administrators Of The Tulane Educational Fund | Peptides aiding nerve regeneration |
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| US5731408A (en) * | 1995-04-10 | 1998-03-24 | Arizona Board Of Regents On Behalf Of The University Of Arizona | Peptides having potent antagonist and agonist bioactivities at melanocortin receptors |
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| US5770380A (en) | 1996-09-13 | 1998-06-23 | University Of Pittsburgh | Synthetic antibody mimics--multiple peptide loops attached to a molecular scaffold |
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-
2000
- 2000-03-21 DK DK00919500T patent/DK1165613T3/da active
- 2000-03-21 PT PT00919500T patent/PT1165613E/pt unknown
- 2000-03-21 IL IL14540600A patent/IL145406A0/xx unknown
- 2000-03-21 KR KR10-2001-7012436A patent/KR100519201B1/ko not_active Expired - Fee Related
- 2000-03-21 HU HU0202203A patent/HUP0202203A3/hu unknown
- 2000-03-21 MX MXPA01009881A patent/MXPA01009881A/es active IP Right Grant
- 2000-03-21 EP EP00919500A patent/EP1165613B1/fr not_active Expired - Lifetime
- 2000-03-21 CA CA002368431A patent/CA2368431C/fr not_active Expired - Fee Related
- 2000-03-21 DE DE60038734T patent/DE60038734T2/de not_active Expired - Fee Related
- 2000-03-21 PL PL00350095A patent/PL350095A1/xx not_active Application Discontinuation
- 2000-03-21 WO PCT/US2000/007473 patent/WO2000058361A1/fr not_active Ceased
- 2000-03-21 AU AU40179/00A patent/AU763510B2/en not_active Ceased
- 2000-03-21 SK SK1308-2001A patent/SK13082001A3/sk unknown
- 2000-03-21 TR TR2001/02765T patent/TR200102765T2/xx unknown
- 2000-03-21 AT AT00919500T patent/ATE393783T1/de not_active IP Right Cessation
- 2000-03-21 RU RU2001128890/04A patent/RU2213098C2/ru not_active IP Right Cessation
- 2000-03-21 JP JP2000608653A patent/JP2002542159A/ja active Pending
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- 2000-03-21 ES ES00919500T patent/ES2304345T3/es not_active Expired - Lifetime
- 2000-03-21 BR BR0009497-8A patent/BR0009497A/pt not_active IP Right Cessation
- 2000-03-21 NZ NZ514141A patent/NZ514141A/xx unknown
- 2000-03-21 HK HK02104687.8A patent/HK1044954B/en not_active IP Right Cessation
- 2000-03-21 CN CNB008057540A patent/CN1249086C/zh not_active Expired - Fee Related
- 2000-03-21 ID IDW00200102111A patent/ID30262A/id unknown
- 2000-03-21 CZ CZ20013407A patent/CZ20013407A3/cs unknown
- 2000-03-27 MY MYPI20001220A patent/MY126585A/en unknown
- 2000-03-28 CO CO00022068A patent/CO5170531A1/es not_active Application Discontinuation
- 2000-03-28 TW TW089105726A patent/TWI250990B/zh not_active IP Right Cessation
- 2000-03-29 PE PE2000000267A patent/PE20001641A1/es not_active Application Discontinuation
- 2000-03-29 US US09/537,789 patent/US6613874B1/en not_active Expired - Fee Related
- 2000-03-29 AR ARP000101405A patent/AR023201A1/es active IP Right Grant
- 2000-06-26 SA SA00210192A patent/SA00210192B1/ar unknown
-
2001
- 2001-09-07 ZA ZA200107411A patent/ZA200107411B/xx unknown
- 2001-09-20 NO NO20014568A patent/NO20014568L/no not_active Application Discontinuation
- 2001-09-26 MA MA26340A patent/MA25403A1/fr unknown
-
2003
- 2003-07-02 US US10/612,104 patent/US6951916B2/en not_active Expired - Fee Related
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